DSigDB Home
Search Gene
Collections
Browse Gene Sets
Download
Help

Gene Set: D4 : TTD - INCB13739

Collection D4 : TTD
Chemical Name INCB13739 ( From PubChem : PHENYLARSINE OXIDE )
FDA NPC WHO Indian Australia China Traditional
Herbal		 Clinical
Trail
NotNotNotNotNotNotNotNot
Molecular
Weight		 Hydrogen Bond
Donor Count		 Hydrogen Bond
Acceptor Count		 cLogP Lipinski Rule
169.033 g/mol 1 1 0.4741 True
Structure
InChI InChI=1S/C6H5AsO/c8-7-6-4-2-1-3-5-6/h1-5H
InChIKey BQVCCPGCDUSGOE-UHFFFAOYSA-N
Links

Gene (8 / 14)


⊖ Less
Source Type Unit Value Gene PMID Assay Other
TTDInhibitorHSD11B1Clinical trial target
TTDDrug(s)HSD11B1Clinical trial target
TTDInhibitorPTPDC1Research target
PubChem AR Potency (uM)uM0.295AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.306AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.347AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.306CYP19A1-GI(Protien) :
PubChem Ratio Potency (uM)uM0.905ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM3.090ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM4.364ESR1-GI(Protien) :
PubChem Ratio Potency (uM)uM5.495ESR1-GI(Protien) :
PubChem Ratio Potency (uM)uM0.666HSPB1-GI(Protien) :
PubChem NoneuMPPARD-GI(Protien) :
PubChem Potency-Replicate_1uM0.245VDR-GI(Protien) :
Download gene sets gmt, text, Detailed text
Contact us
Tan Lab , Mail Stop 8117
12801 East 17th Avenue
Division of Medical Oncology , Department of Medicine
University of Colorado School of Medicine
Aurora, CO 80045, USA

* Best viewed in the latest version of Chrome (42+), Safari (8+), IE (11+) or Firefox (35+).