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Gene Set: D4 : CTD - Sirolimus


Collection D4 : CTD
Chemical Name Sirolimus ( From PubChem : RAPAMYCIN )
FDA NPC WHO Indian Australia China Traditional
Herbal
Clinical
Trail
NotNotNotNotNotNotNotNot
Molecular
Weight
Hydrogen Bond
Donor Count
Hydrogen Bond
Acceptor Count
cLogP Lipinski Rule
914.172 g/mol 3 14 6.1185 False(1/4)
Structure
InChI InChI=1S/C51H79NO13/c1-30-16-12-11-13-17-31(2)42(61-8)28-38-21-19-36(7)51(60,65-38)48(57)49(58)52-23-15-14-18-39(52)50(59)64-43(33(4)26-37-20-22-40(53)44(27-37)62-9)29-41(54)32(3)25-35(6)46(56)47(63-10)45(55)34(5)24-30/h11-13,16-17,25,30,32-34,36-40,42-44,46-47,53,56,60H,14-15,18-24,26-29H2,1-10H3
InChIKey QFJCIRLUMZQUOT-UHFFFAOYSA-N
Links

Gene (247 / 907)


⊖ Less

Source Type Unit Value Gene PMID Assay Other
CTDaffects(cotreatment)ABCA1
D020123
CTDdecreases(expression)ABCA1
D020123
CTDincreases(expression)ABCA1
D020123
CTDaffects(metabolic processing)ABCB1
D020123
CTDaffects(transport)ABCB1
D020123
CTDdecreases(expression)ACER2
D020123
CTDdecreases(reaction)ACER2
D020123
CTDaffects(cotreatment)ACTA2
D020123
CTDincreases(expression)ACTA2
D020123
CTDaffects(cotreatment)AIFM1
D020123
CTDaffects(localization)AIFM1
D020123
CTDdecreases(reaction)AIFM1
D020123
CTDdecreases(reaction)AKT1
D020123
CTDincreases(phosphorylation)AKT1
D020123
CTDincreases(expression)AKT1
D020123
CTDaffects(cotreatment)AKT1
D020123
CTDdecreases(phosphorylation)AKT1
D020123
CTDdecreases(reaction)AKT1
D020123
CTDincreases(phosphorylation)AKT1
D020123
CTDdecreases(reaction)AKT1
D020123
CTDincreases(phosphorylation)AKT1
D020123
CTDdecreases(phosphorylation)AKT1
D020123
CTDincreases(activity)AKT2
D020123
CTDincreases(expression)AKT2
D020123
CTDincreases(phosphorylation)AKT2
D020123
CTDdecreases(expression)APP
D020123
CTDincreases(expression)APP
D020123
CTDdecreases(reaction)AR
D020123
CTDincreases(activity)AR
D020123
CTDaffects(reaction)AR
D020123
CTDincreases(expression)AR
D020123
CTDaffects(expression)AR
D020123
CTDincreases(reaction)AR
D020123
CTDaffects(binding)AR
D020123
CTDdecreases(activity)AR
D020123
CTDincreases(expression)AR
D020123
CTDaffects(reaction)ATG5
D020123
CTDdecreases(reaction)ATG5
D020123
CTDincreases(cleavage)ATG5
D020123
CTDaffects(cotreatment)AURKB
D020123
CTDdecreases(expression)AURKB
D020123
CTDaffects(cotreatment)BAX
D020123
CTDincreases(expression)BAX
D020123
CTDaffects(localization)BAX
D020123
CTDincreases(expression)BAX
D020123
CTDaffects(cotreatment)BBC3
D020123
CTDincreases(expression)BBC3
D020123
CTDincreases(expression)BBC3
D020123
CTDincreases(reaction)BBC3
D020123
CTDaffects(cotreatment)BCL2
D020123
CTDdecreases(expression)BCL2
D020123
CTDdecreases(reaction)BCL2
D020123
CTDincreases(expression)BCL2
D020123
CTDincreases(expression)BCL2
D020123
CTDincreases(reaction)BCL2
D020123
CTDdecreases(expression)BCL2
D020123
CTDdecreases(expression)BCL2
D020123
CTDaffects(cotreatment)BCL2L1
D020123
CTDdecreases(expression)BCL2L1
D020123
CTDdecreases(reaction)BCL2L1
D020123
CTDincreases(expression)BCL2L1
D020123
CTDdecreases(expression)BCL2L1
D020123
CTDdecreases(reaction)BCL2L11
D020123
CTDincreases(expression)BCL2L11
D020123
CTDincreases(phosphorylation)BCL2L11
D020123
CTDincreases(reaction)BCL2L11
D020123
CTDdecreases(reaction)BECN1
D020123
CTDincreases(degradation)BECN1
D020123
CTDaffects(cotreatment)BID
D020123
CTDincreases(cleavage)BID
D020123
CTDdecreases(reaction)BIRC2
D020123
CTDincreases(expression)BIRC2
D020123
CTDaffects(cotreatment)BIRC5
D020123
CTDdecreases(expression)BIRC5
D020123
CTDdecreases(expression)BIRC5
D020123
CTDincreases(reaction)BIRC5
D020123
CTDdecreases(expression)BIRC5
D020123
CTDdecreases(reaction)BTBD11
D020123
CTDincreases(expression)BTBD11
D020123
CTDaffects(cotreatment)BUB1
D020123
CTDdecreases(expression)BUB1
D020123
CTDaffects(cotreatment)BUB1B
D020123
CTDdecreases(expression)BUB1B
D020123
CTDdecreases(reaction)C9ORF3
D020123
CTDincreases(expression)C9ORF3
D020123
CTDaffects(cotreatment)CALD1
D020123
CTDincreases(expression)CALD1
D020123
CTDincreases(activity)CALD1
D020123
CTDaffects(cotreatment)CASP2
D020123
CTDincreases(cleavage)CASP2
D020123
CTDdecreases(reaction)CASP2
D020123
CTDaffects(cotreatment)CASP3
D020123
CTDincreases(cleavage)CASP3
D020123
CTDdecreases(reaction)CASP3
D020123
CTDaffects(cotreatment)CASP3
D020123
CTDincreases(activity)CASP3
D020123
CTDincreases(expression)CASP3
D020123
CTDincreases(reaction)CASP3
D020123
CTDaffects(cotreatment)CASP3
D020123
CTDaffects(cotreatment)CASP3
D020123
CTDincreases(cleavage)CASP3
D020123
CTDdecreases(reaction)CASP3
D020123
CTDincreases(cleavage)CASP3
D020123
CTDdecreases(reaction)CASP3
D020123
CTDincreases(cleavage)CASP3
D020123
CTDincreases(cleavage)CASP3
D020123
CTDincreases(reaction)CASP3
D020123
CTDincreases(activity)CASP3
D020123
CTDincreases(reaction)CASP3
D020123
CTDincreases(activity)CASP3
D020123
CTDincreases(cleavage)CASP3
D020123
CTDaffects(cotreatment)CASP7
D020123
CTDincreases(activity)CASP7
D020123
CTDaffects(cotreatment)CASP7
D020123
CTDincreases(cleavage)CASP7
D020123
CTDaffects(cotreatment)CASP8
D020123
CTDincreases(cleavage)CASP8
D020123
CTDdecreases(reaction)CASP8
D020123
CTDincreases(cleavage)CASP8
D020123
CTDincreases(reaction)CASP8
D020123
CTDaffects(cotreatment)CASP8
D020123
CTDincreases(cleavage)CASP8
D020123
CTDaffects(cotreatment)CASP9
D020123
CTDincreases(cleavage)CASP9
D020123
CTDaffects(cotreatment)CASP9
D020123
CTDincreases(activity)CASP9
D020123
CTDaffects(cotreatment)CASP9
D020123
CTDincreases(activity)CASP9
D020123
CTDaffects(cotreatment)CASP9
D020123
CTDincreases(cleavage)CASP9
D020123
CTDincreases(cleavage)CASP9
D020123
CTDincreases(reaction)CASP9
D020123
CTDaffects(cotreatment)CASP9
D020123
CTDincreases(cleavage)CASP9
D020123
CTDdecreases(reaction)CAV3
D020123
CTDincreases(expression)CAV3
D020123
CTDaffects(cotreatment)CCNA2
D020123
CTDdecreases(expression)CCNA2
D020123
CTDdecreases(expression)CCNA2
D020123
CTDdecreases(expression)CCNA2
D020123
CTDaffects(cotreatment)CCNB2
D020123
CTDdecreases(expression)CCNB2
D020123
CTDaffects(cotreatment)CCND1
D020123
CTDdecreases(expression)CCND1
D020123
CTDdecreases(reaction)CCND1
D020123
CTDincreases(expression)CCND1
D020123
CTDdecreases(activity)CCND1
D020123
CTDdecreases(expression)CCND1
D020123
CTDdecreases(reaction)CCND1
D020123
CTDaffects(cotreatment)CCND1
D020123
CTDdecreases(expression)CCND1
D020123
CTDaffects(cotreatment)CCND1
D020123
CTDdecreases(expression)CCND1
D020123
CTDaffects(cotreatment)CCND1
D020123
CTDdecreases(expression)CCND1
D020123
CTDdecreases(expression)CCND1
D020123
CTDincreases(activity)CCND1
D020123
CTDincreases(degradation)CCND1
D020123
CTDincreases(phosphorylation)CCND1
D020123
CTDaffects(cotreatment)CCND2
D020123
CTDdecreases(reaction)CCND2
D020123
CTDincreases(expression)CCND2
D020123
CTDdecreases(expression)CCND2
D020123
CTDaffects(cotreatment)CCND3
D020123
CTDdecreases(reaction)CCND3
D020123
CTDincreases(expression)CCND3
D020123
CTDdecreases(expression)CCND3
D020123
CTDdecreases(expression)CCND3
D020123
CTDdecreases(stability)CCND3
D020123
CTDaffects(cotreatment)CCNE2
D020123
CTDdecreases(expression)CCNE2
D020123
CTDaffects(cotreatment)CCNG2
D020123
CTDincreases(expression)CCNG2
D020123
CTDdecreases(reaction)CCNG2
D020123
CTDincreases(expression)CCNG2
D020123
CTDincreases(expression)CCNG2
D020123
CTDaffects(expression)CD36
D020123
CTDdecreases(reaction)CD36
D020123
CTDincreases(expression)CD36
D020123
CTDdecreases(expression)CD68
D020123
CTDincreases(expression)CD84
D020123
CTDaffects(cotreatment)CDC20
D020123
CTDdecreases(expression)CDC20
D020123
CTDaffects(cotreatment)CDK1
D020123
CTDdecreases(expression)CDK1
D020123
CTDaffects(cotreatment)CDK1
D020123
CTDdecreases(expression)CDK1
D020123
CTDaffects(cotreatment)CDK1
D020123
CTDdecreases(phosphorylation)CDK1
D020123
CTDaffects(cotreatment)CDK1
D020123
CTDdecreases(expression)CDK1
D020123
CTDdecreases(expression)CDK1
D020123
CTDaffects(cotreatment)CDK2
D020123
CTDaffects(localization)CDK2
D020123
CTDaffects(binding)CDK2
D020123
CTDincreases(reaction)CDK2
D020123
CTDdecreases(activity)CDK2
D020123
CTDaffects(binding)CDK2
D020123
CTDaffects(cotreatment)CDK2
D020123
CTDdecreases(reaction)CDK2
D020123
CTDincreases(reaction)CDK2
D020123
CTDdecreases(activity)CDK2
D020123
CTDdecreases(phosphorylation)CDK2
D020123
CTDincreases(expression)CDKN1A
D020123
CTDincreases(reaction)CDKN1A
D020123
CTDaffects(cotreatment)CDKN1A
D020123
CTDaffects(binding)CDKN1A
D020123
CTDaffects(cotreatment)CDKN1A
D020123
CTDincreases(reaction)CDKN1A
D020123
CTDincreases(expression)CDKN1A
D020123
CTDincreases(expression)CDKN1A
D020123
CTDincreases(expression)CDKN1A
D020123
CTDaffects(binding)CDKN1A
D020123
CTDaffects(cotreatment)CDKN1A
D020123
CTDincreases(reaction)CDKN1A
D020123
CTDaffects(cotreatment)CDKN1A
D020123
CTDincreases(expression)CDKN1A
D020123
CTDdecreases(reaction)CDKN1B
D020123
CTDincreases(expression)CDKN1B
D020123
CTDincreases(phosphorylation)CDKN1B
D020123
CTDaffects(cotreatment)CDKN1B
D020123
CTDincreases(expression)CDKN1B
D020123
CTDaffects(cotreatment)CDKN1B
D020123
CTDaffects(localization)CDKN1B
D020123
CTDincreases(reaction)CDKN1B
D020123
CTDdecreases(degradation)CDKN1B
D020123
CTDincreases(expression)CDKN1B
D020123
CTDaffects(binding)CDKN1B
D020123
CTDaffects(cotreatment)CDKN1B
D020123
CTDincreases(reaction)CDKN1B
D020123
CTDdecreases(reaction)CHRNB3
D020123
CTDincreases(expression)CHRNB3
D020123
CTDdecreases(reaction)COL1A2
D020123
CTDincreases(expression)COL1A2
D020123
CTDdecreases(activity)CRTC2
D020123
CTDdecreases(reaction)CXCL8
D020123
CTDincreases(phosphorylation)CXCL8
D020123
CTDaffects(cotreatment)CYP27A1
D020123
CTDdecreases(activity)CYP27A1
D020123
CTDaffects(metabolic processing)CYP3A
D020123
CTDaffects(metabolic processing)CYP3A4
D020123
CTDaffects(metabolic processing)CYP3A4
D020123
CTDdecreases(reaction)DDIT3
D020123
CTDincreases(expression)DDIT3
D020123
CTDdecreases(activity)DDIT3
D020123
CTDdecreases(expression)DDIT3
D020123
CTDdecreases(reaction)DEPTOR
D020123
CTDincreases(expression)DEPTOR
D020123
CTDaffects(cotreatment)DIABLO
D020123
CTDaffects(localization)DIABLO
D020123
CTDdecreases(reaction)DIABLO
D020123
CTDaffects(cotreatment)DNMT1
D020123
CTDdecreases(expression)DNMT1
D020123
CTDdecreases(expression)DPYD
D020123
CTDincreases(expression)DUSP10
D020123
CTDaffects(cotreatment)E2F1
D020123
CTDdecreases(expression)E2F1
D020123
CTDaffects(binding)E2F4
D020123
CTDaffects(cotreatment)E2F4
D020123
CTDdecreases(reaction)E2F4
D020123
CTDdecreases(reaction)EGF
D020123
CTDincreases(phosphorylation)EGF
D020123
CTDdecreases(reaction)EGFR
D020123
CTDincreases(phosphorylation)EGFR
D020123
CTDdecreases(expression)EIF4E
D020123
CTDdecreases(reaction)EIF4E
D020123
CTDdecreases(activity)EIF4E
D020123
CTDdecreases(phosphorylation)EIF4EBP1
D020123
CTDincreases(reaction)EIF4EBP1
D020123
CTDaffects(reaction)EIF4EBP1
D020123
CTDincreases(phosphorylation)EIF4EBP1
D020123
CTDaffects(cotreatment)EIF4EBP1
D020123
CTDdecreases(phosphorylation)EIF4EBP1
D020123
CTDaffects(cotreatment)EIF4EBP1
D020123
CTDdecreases(phosphorylation)EIF4EBP1
D020123
CTDdecreases(reaction)EIF4EBP1
D020123
CTDincreases(phosphorylation)EIF4EBP1
D020123
CTDdecreases(reaction)EIF4EBP1
D020123
CTDincreases(phosphorylation)EIF4EBP1
D020123
CTDdecreases(phosphorylation)EIF4EBP1
D020123
CTDincreases(reaction)EIF4EBP1
D020123
CTDdecreases(phosphorylation)EIF4EBP1
D020123
CTDincreases(reaction)EIF4EBP1
D020123
CTDdecreases(phosphorylation)EIF4EBP1
D020123
CTDincreases(reaction)EIF4EBP1
D020123
CTDdecreases(activity)EIF4EBP1
D020123
CTDdecreases(phosphorylation)EIF4EBP1
D020123
CTDdecreases(phosphorylation)EIF4EBP1
D020123
CTDincreases(expression)EIF4G2
D020123
CTDaffects(cotreatment)ESPL1
D020123
CTDdecreases(expression)ESPL1
D020123
CTDincreases(expression)ESR1
D020123
CTDincreases(phosphorylation)ESR1
D020123
CTDincreases(expression)EVI2A
D020123
CTDdecreases(expression)EWSR1
D020123
CTDincreases(expression)F3
D020123
CTDincreases(reaction)F3
D020123
CTDdecreases(secretion)FASLG
D020123
CTDdecreases(reaction)FAXDC2
D020123
CTDincreases(expression)FAXDC2
D020123
CTDdecreases(reaction)FBXO32
D020123
CTDincreases(expression)FBXO32
D020123
CTDincreases(expression)FBXO32
D020123
CTDaffects(cotreatment)FBXO5
D020123
CTDdecreases(expression)FBXO5
D020123
CTDdecreases(reaction)FGF7
D020123
CTDincreases(expression)FGF7
D020123
CTDaffects(binding)FKBP1A
D020123
CTDaffects(binding)FKBP1A
D020123
CTDincreases(activity)FKBP1A
D020123
CTDaffects(binding)FKBP1A
D020123
CTDdecreases(reaction)FKBP1A
D020123
CTDdecreases(reaction)FOLR1
D020123
CTDincreases(expression)FOLR1
D020123
CTDaffects(cotreatment)FOXM1
D020123
CTDdecreases(expression)FOXM1
D020123
CTDincreases(phosphorylation)FOXO1
D020123
CTDdecreases(reaction)FOXO3
D020123
CTDincreases(phosphorylation)FOXO3
D020123
CTDincreases(expression)FOXO3
D020123
CTDaffects(cotreatment)FOXO3
D020123
CTDincreases(response to substance)FOXO3
D020123
CTDincreases(activity)FOXO3
D020123
CTDincreases(localization)FOXO3
D020123
CTDincreases(reaction)FOXO3
D020123
CTDdecreases(degradation)FOXO3
D020123
CTDaffects(cotreatment)FOXP3
D020123
CTDincreases(expression)FOXP3
D020123
CTDincreases(expression)FRAT1
D020123
CTDdecreases(reaction)FTL
D020123
CTDincreases(expression)FTL
D020123
CTDaffects(activity)GCM2
D020123
CTDincreases(reaction)GCM2
D020123
CTDincreases(expression)GPR18
D020123
CTDdecreases(activity)GSK3B
D020123
CTDdecreases(expression)GSK3B
D020123
CTDdecreases(reaction)GSK3B
D020123
CTDdecreases(activity)GSK3B
D020123
CTDincreases(phosphorylation)GSK3B
D020123
CTDincreases(activity)GSK3B
D020123
CTDincreases(degradation)GSK3B
D020123
CTDincreases(phosphorylation)GSK3B
D020123
CTDincreases(response to substance)GSTT1
D020123
CTDdecreases(expression)GZMB
D020123
CTDdecreases(expression)HES1
D020123
CTDdecreases(reaction)HIF1A
D020123
CTDincreases(expression)HIF1A
D020123
CTDdecreases(reaction)HIF1A
D020123
CTDincreases(expression)HIF1A
D020123
CTDaffects(binding)HIF1A
D020123
CTDdecreases(reaction)HIF1A
D020123
CTDincreases(activity)HIF1A
D020123
CTDincreases(expression)HIF1A
D020123
CTDdecreases(reaction)HIF1A
D020123
CTDincreases(expression)HIF1A
D020123
CTDdecreases(reaction)HIF1A
D020123
CTDincreases(expression)HIF1A
D020123
CTDdecreases(reaction)HIF1A
D020123
CTDincreases(expression)HIF1A
D020123
CTDdecreases(expression)HIF1A
D020123
CTDincreases(expression)HMGCR
D020123
CTDaffects(activity)HOXA9
D020123
CTDdecreases(reaction)HOXA9
D020123
CTDdecreases(expression)HSPA1B
D020123
CTDdecreases(expression)HSPA5
D020123
CTDdecreases(expression)HSPB8
D020123
CTDincreases(expression)ID1
D020123
CTDdecreases(phosphorylation)IFNG
D020123
CTDdecreases(reaction)IFNG
D020123
CTDdecreases(secretion)IFNG
D020123
CTDaffects(cotreatment)IGF1
D020123
CTDdecreases(reaction)IGF1
D020123
CTDincreases(phosphorylation)IGF1
D020123
CTDdecreases(activity)IGF1
D020123
CTDaffects(cotreatment)IGF1
D020123
CTDincreases(expression)IGF1
D020123
CTDdecreases(reaction)IGF1
D020123
CTDincreases(expression)IGF1
D020123
CTDdecreases(reaction)IGF1
D020123
CTDincreases(phosphorylation)IGF1
D020123
CTDdecreases(reaction)IGF1
D020123
CTDincreases(secretion)IGF1
D020123
CTDincreases(response to substance)IGF1
D020123
CTDaffects(activity)IGF1R
D020123
CTDaffects(binding)IGF1R
D020123
CTDincreases(phosphorylation)IGF1R
D020123
CTDincreases(reaction)IGF1R
D020123
CTDdecreases(reaction)IGFBP3
D020123
CTDincreases(secretion)IGFBP3
D020123
CTDdecreases(reaction)IL10
D020123
CTDincreases(expression)IL10
D020123
CTDdecreases(expression)IL10
D020123
CTDaffects(cotreatment)IL17RB
D020123
CTDdecreases(expression)IL17RB
D020123
CTDaffects(cotreatment)IL2
D020123
CTDdecreases(reaction)IL2
D020123
CTDincreases(expression)IL2
D020123
CTDincreases(phosphorylation)IL2
D020123
CTDdecreases(reaction)IL2
D020123
CTDincreases(phosphorylation)IL2
D020123
CTDdecreases(response to substance)IL2
D020123
CTDaffects(cotreatment)IL2RA
D020123
CTDdecreases(reaction)IL2RA
D020123
CTDincreases(secretion)IL2RA
D020123
CTDaffects(cotreatment)IL6
D020123
CTDdecreases(reaction)IL6
D020123
CTDincreases(phosphorylation)IL6
D020123
CTDdecreases(activity)IL6
D020123
CTDincreases(expression)IL6
D020123
CTDaffects(cotreatment)IL6
D020123
CTDdecreases(expression)IL6
D020123
CTDdecreases(reaction)ING4
D020123
CTDincreases(expression)ING4
D020123
CTDaffects(phosphorylation)IRS1
D020123
CTDaffects(binding)IRS1
D020123
CTDincreases(phosphorylation)IRS1
D020123
CTDincreases(reaction)IRS1
D020123
CTDaffects(binding)IRS1
D020123
CTDincreases(reaction)IRS1
D020123
CTDdecreases(activity)IRS1
D020123
CTDincreases(activity)IRS1
D020123
CTDdecreases(degradation)IRS1
D020123
CTDdecreases(phosphorylation)IRS1
D020123
CTDincreases(expression)ITGAM
D020123
CTDincreases(localization)ITGAM
D020123
CTDincreases(reaction)ITGAM
D020123
CTDdecreases(expression)JAG1
D020123
CTDdecreases(expression)JMY
D020123
CTDdecreases(reaction)JMY
D020123
CTDdecreases(phosphorylation)KIT
D020123
CTDincreases(reaction)KIT
D020123
CTDincreases(expression)KLF2
D020123
CTDincreases(expression)KLHL24
D020123
CTDincreases(expression)KLK2
D020123
CTDincreases(reaction)KLK2
D020123
CTDdecreases(reaction)KLK3
D020123
CTDincreases(expression)KLK3
D020123
CTDaffects(response to substance)L1CAM
D020123
CTDaffects(cotreatment)MAD2L1
D020123
CTDdecreases(expression)MAD2L1
D020123
CTDaffects(binding)MAP1LC3A
D020123
CTDdecreases(reaction)MAP1LC3A
D020123
CTDincreases(expression)MAP1LC3A
D020123
CTDincreases(expression)MAP1LC3B
D020123
CTDincreases(expression)MAP1LC3B
D020123
CTDaffects(cotreatment)MAP2K1
D020123
CTDdecreases(expression)MAP2K1
D020123
CTDdecreases(phosphorylation)MAP2K1
D020123
CTDaffects(cotreatment)MAP2K2
D020123
CTDdecreases(phosphorylation)MAP2K2
D020123
CTDaffects(cotreatment)MAPK1
D020123
CTDdecreases(phosphorylation)MAPK1
D020123
CTDdecreases(reaction)MAPK1
D020123
CTDincreases(phosphorylation)MAPK1
D020123
CTDdecreases(reaction)MAPK1
D020123
CTDincreases(activity)MAPK1
D020123
CTDincreases(phosphorylation)MAPK1
D020123
CTDdecreases(phosphorylation)MAPK1
D020123
CTDaffects(cotreatment)MAPK3
D020123
CTDdecreases(phosphorylation)MAPK3
D020123
CTDdecreases(reaction)MAPK3
D020123
CTDincreases(phosphorylation)MAPK3
D020123
CTDdecreases(reaction)MAPK3
D020123
CTDincreases(activity)MAPK3
D020123
CTDincreases(phosphorylation)MAPK3
D020123
CTDdecreases(phosphorylation)MAPK3
D020123
CTDaffects(cotreatment)MAPK8
D020123
CTDincreases(phosphorylation)MAPK8
D020123
CTDdecreases(reaction)MAPK8
D020123
CTDdecreases(reaction)MBNL2
D020123
CTDincreases(expression)MBNL2
D020123
CTDaffects(cotreatment)MCL1
D020123
CTDdecreases(expression)MCL1
D020123
CTDdecreases(expression)MDM2
D020123
CTDdecreases(reaction)MDM2
D020123
CTDdecreases(reaction)MDM2
D020123
CTDincreases(phosphorylation)MDM2
D020123
CTDaffects(binding)MDM2
D020123
CTDincreases(reaction)MDM2
D020123
CTDincreases(expression)MIR151A
D020123
CTDincreases(reaction)MIR151A
D020123
CTDdecreases(expression)MIR181A2
D020123
CTDdecreases(reaction)MIR181A2
D020123
CTDincreases(expression)MIR190A
D020123
CTDincreases(reaction)MIR190A
D020123
CTDincreases(expression)MIR29C
D020123
CTDincreases(reaction)MIR29C
D020123
CTDincreases(expression)MIR324
D020123
CTDincreases(reaction)MIR324
D020123
CTDincreases(expression)MIR379
D020123
CTDincreases(reaction)MIR379
D020123
CTDincreases(expression)MIR433
D020123
CTDincreases(reaction)MIR433
D020123
CTDincreases(expression)MIR503
D020123
CTDincreases(reaction)MIR503
D020123
CTDincreases(expression)MIR508
D020123
CTDincreases(reaction)MIR508
D020123
CTDincreases(expression)MIR650
D020123
CTDincreases(reaction)MIR650
D020123
CTDincreases(expression)MIR654
D020123
CTDincreases(reaction)MIR654
D020123
CTDincreases(expression)MIR758
D020123
CTDincreases(reaction)MIR758
D020123
CTDincreases(expression)MIR760
D020123
CTDincreases(reaction)MIR760
D020123
CTDaffects(cotreatment)MKI67
D020123
CTDdecreases(expression)MKI67
D020123
CTDaffects(binding)MLST8
D020123
CTDdecreases(activity)MLST8
D020123
CTDincreases(expression)MMP1
D020123
CTDincreases(secretion)MMP1
D020123
CTDdecreases(expression)MSR1
D020123
CTDdecreases(activity)MTOR
D020123
CTDdecreases(reaction)MTOR
D020123
CTDaffects(cotreatment)MTOR
D020123
CTDdecreases(expression)MTOR
D020123
CTDaffects(cotreatment)MTOR
D020123
CTDaffects(phosphorylation)MTOR
D020123
CTDdecreases(reaction)MTOR
D020123
CTDincreases(phosphorylation)MTOR
D020123
CTDdecreases(reaction)MTOR
D020123
CTDincreases(phosphorylation)MTOR
D020123
CTDaffects(binding)MTOR
D020123
CTDdecreases(reaction)MTOR
D020123
CTDincreases(expression)MTOR
D020123
CTDdecreases(reaction)MTOR
D020123
CTDincreases(expression)MTOR
D020123
CTDdecreases(phosphorylation)MTOR
D020123
CTDincreases(reaction)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDaffects(binding)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDaffects(binding)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDincreases(activity)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDdecreases(reaction)MTOR
D020123
CTDincreases(activity)MTOR
D020123
CTDincreases(phosphorylation)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDdecreases(expression)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDdecreases(expression)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDdecreases(phosphorylation)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDdecreases(phosphorylation)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDdecreases(phosphorylation)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDdecreases(phosphorylation)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDincreases(phosphorylation)MTOR
D020123
CTDdecreases(activity)MTOR
D020123
CTDincreases(response to substance)MTOR
D020123
CTDdecreases(expression)MTOR
D020123
CTDdecreases(phosphorylation)MTOR
D020123
CTDdecreases(chemical synthesis)MTOR
D020123
CTDdecreases(phosphorylation)MTOR
D020123
CTDincreases(activity)MTOR
D020123
CTDincreases(phosphorylation)MTOR
D020123
CTDdecreases(reaction)MTURN
D020123
CTDincreases(expression)MTURN
D020123
CTDaffects(cotreatment)MYC
D020123
CTDdecreases(expression)MYC
D020123
CTDaffects(cotreatment)MYH11
D020123
CTDincreases(expression)MYH11
D020123
CTDincreases(activity)MYH11
D020123
CTDdecreases(reaction)MYLK
D020123
CTDincreases(expression)MYLK
D020123
CTDdecreases(reaction)MYOF
D020123
CTDincreases(expression)MYOF
D020123
CTDaffects(cotreatment)NDC80
D020123
CTDdecreases(expression)NDC80
D020123
CTDaffects(cotreatment)NEK2
D020123
CTDdecreases(expression)NEK2
D020123
CTDdecreases(reaction)NFKB1
D020123
CTDincreases(activity)NFKB1
D020123
CTDdecreases(expression)NFKBIA
D020123
CTDdecreases(reaction)NFKBIA
D020123
CTDincreases(degradation)NFKBIA
D020123
CTDdecreases(reaction)NFKBIA
D020123
CTDincreases(phosphorylation)NFKBIA
D020123
CTDaffects(activity)NHLH1
D020123
CTDdecreases(reaction)NHLH1
D020123
CTDaffects(cotreatment)NME1
D020123
CTDdecreases(expression)NME1
D020123
CTDdecreases(reaction)NMU
D020123
CTDincreases(expression)NMU
D020123
CTDdecreases(expression)NOS3
D020123
CTDdecreases(reaction)NOS3
D020123
CTDdecreases(expression)NOS3
D020123
CTDaffects(expression)NR1H3
D020123
CTDdecreases(expression)NR1H4
D020123
CTDdecreases(reaction)NR1H4
D020123
CTDaffects(expression)OLR1
D020123
CTDdecreases(reaction)OXA1L
D020123
CTDincreases(expression)OXA1L
D020123
CTDaffects(reaction)PARP1
D020123
CTDdecreases(reaction)PARP1
D020123
CTDincreases(cleavage)PARP1
D020123
CTDdecreases(reaction)PARP1
D020123
CTDincreases(cleavage)PARP1
D020123
CTDaffects(activity)PAX8
D020123
CTDincreases(reaction)PAX8
D020123
CTDaffects(cotreatment)PCNA
D020123
CTDdecreases(expression)PCNA
D020123
CTDdecreases(expression)PCNA
D020123
CTDincreases(expression)PDCD4
D020123
CTDincreases(reaction)PDCD4
D020123
CTDincreases(expression)PDCD4
D020123
CTDdecreases(reaction)PDGFB
D020123
CTDincreases(activity)PDGFB
D020123
CTDincreases(phosphorylation)PDGFB
D020123
CTDdecreases(activity)PDGFB
D020123
CTDdecreases(response to substance)PIK3CA
D020123
CTDincreases(activity)PIK3CA
D020123
CTDdecreases(reaction)PIK3CA
D020123
CTDaffects(binding)PIK3R1
D020123
CTDincreases(reaction)PIK3R1
D020123
CTDdecreases(activity)PKM
D020123
CTDdecreases(expression)PKM
D020123
CTDincreases(expression)PLCL1
D020123
CTDaffects(cotreatment)PMAIP1
D020123
CTDincreases(expression)PMAIP1
D020123
CTDdecreases(response to substance)PML
D020123
CTDincreases(expression)PML
D020123
CTDincreases(localization)PML
D020123
CTDincreases(expression)PNRC1
D020123
CTDaffects(expression)PPARG
D020123
CTDaffects(cotreatment)PPARG
D020123
CTDdecreases(expression)PPARG
D020123
CTDincreases(expression)PPARG
D020123
CTDdecreases(expression)PRF1
D020123
CTDdecreases(reaction)PRKCA
D020123
CTDincreases(phosphorylation)PRKCA
D020123
CTDaffects(localization)PRKCD
D020123
CTDdecreases(phosphorylation)PRKCD
D020123
CTDincreases(reaction)PRKCD
D020123
CTDaffects(binding)PRKCG
D020123
CTDdecreases(reaction)PRKCG
D020123
CTDincreases(degradation)PRKCG
D020123
CTDdecreases(response to substance)PRKCH
D020123
CTDdecreases(phosphorylation)PRKCH
D020123
CTDdecreases(reaction)PRKCH
D020123
CTDincreases(activity)PRKCH
D020123
CTDdecreases(expression)PSMD11
D020123
CTDaffects(cotreatment)PTEN
D020123
CTDincreases(expression)PTEN
D020123
CTDdecreases(response to substance)PTEN
D020123
CTDaffects(binding)PTGER1
D020123
CTDdecreases(reaction)PTGER1
D020123
CTDincreases(activity)PTGER1
D020123
CTDincreases(expression)PTGER1
D020123
CTDaffects(cotreatment)PTTG1
D020123
CTDdecreases(expression)PTTG1
D020123
CTDaffects(cotreatment)RAD51
D020123
CTDdecreases(expression)RAD51
D020123
CTDaffects(cotreatment)RAF1
D020123
CTDdecreases(expression)RAF1
D020123
CTDaffects(cotreatment)RB1
D020123
CTDdecreases(reaction)RB1
D020123
CTDincreases(phosphorylation)RB1
D020123
CTDaffects(cotreatment)RB1
D020123
CTDdecreases(expression)RB1
D020123
CTDaffects(cotreatment)RB1
D020123
CTDdecreases(phosphorylation)RB1
D020123
CTDdecreases(reaction)RB1
D020123
CTDincreases(phosphorylation)RB1
D020123
CTDdecreases(phosphorylation)RB1
D020123
CTDaffects(cotreatment)RB1
D020123
CTDdecreases(phosphorylation)RB1
D020123
CTDaffects(cotreatment)RB1
D020123
CTDdecreases(phosphorylation)RB1
D020123
CTDaffects(binding)RBL1
D020123
CTDaffects(cotreatment)RBL1
D020123
CTDdecreases(reaction)RBL1
D020123
CTDdecreases(reaction)RBL2
D020123
CTDincreases(phosphorylation)RBL2
D020123
CTDaffects(binding)RBL2
D020123
CTDaffects(cotreatment)RBL2
D020123
CTDdecreases(reaction)RBL2
D020123
CTDdecreases(reaction)RELA
D020123
CTDincreases(activity)RELA
D020123
CTDaffects(localization)RELA
D020123
CTDdecreases(reaction)RELA
D020123
CTDdecreases(reaction)RELA
D020123
CTDincreases(localization)RELA
D020123
CTDincreases(phosphorylation)RELA
D020123
CTDaffects(activity)REST
D020123
CTDincreases(reaction)REST
D020123
CTDdecreases(expression)RICTOR
D020123
CTDdecreases(expression)RPL7P26
D020123
CTDdecreases(reaction)RPL7P26
D020123
CTDaffects(binding)RPS27L
D020123
CTDincreases(reaction)RPS27L
D020123
CTDdecreases(reaction)RPS6
D020123
CTDincreases(phosphorylation)RPS6
D020123
CTDdecreases(reaction)RPS6
D020123
CTDincreases(phosphorylation)RPS6
D020123
CTDdecreases(reaction)RPS6
D020123
CTDincreases(phosphorylation)RPS6
D020123
CTDdecreases(reaction)RPS6
D020123
CTDincreases(phosphorylation)RPS6
D020123
CTDdecreases(activity)RPS6
D020123
CTDdecreases(phosphorylation)RPS6
D020123
CTDdecreases(phosphorylation)RPS6
D020123
CTDdecreases(phosphorylation)RPS6
D020123
CTDdecreases(reaction)RPS6
D020123
CTDincreases(activity)RPS6
D020123
CTDincreases(phosphorylation)RPS6KA1
D020123
CTDaffects(cotreatment)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDaffects(cotreatment)RPS6KB1
D020123
CTDdecreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(activity)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(activity)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(activity)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(reaction)RPS6KB1
D020123
CTDincreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(phosphorylation)RPS6KB1
D020123
CTDincreases(reaction)RPS6KB1
D020123
CTDdecreases(activity)RPS6KB1
D020123
CTDdecreases(activity)RPS6KB1
D020123
CTDdecreases(activity)RPS6KB1
D020123
CTDdecreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(activity)RPS6KB1
D020123
CTDdecreases(abundance)RPS6KB1
D020123
CTDdecreases(activity)RPS6KB1
D020123
CTDincreases(abundance)RPS6KB1
D020123
CTDdecreases(activity)RPS6KB1
D020123
CTDincreases(activity)RPS6KB1
D020123
CTDdecreases(activity)RPS6KB1
D020123
CTDdecreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(phosphorylation)RPS6KB1
D020123
CTDdecreases(activity)RPS6KB2
D020123
CTDdecreases(reaction)RPS6KB2
D020123
CTDincreases(activity)RPS6KB2
D020123
CTDdecreases(reaction)RPTOR
D020123
CTDincreases(activity)RPTOR
D020123
CTDaffects(binding)RPTOR
D020123
CTDdecreases(reaction)RPTOR
D020123
CTDincreases(expression)RPTOR
D020123
CTDdecreases(phosphorylation)RPTOR
D020123
CTDdecreases(reaction)RPTOR
D020123
CTDaffects(binding)RPTOR
D020123
CTDdecreases(activity)RPTOR
D020123
CTDaffects(binding)RPTOR
D020123
CTDdecreases(activity)RPTOR
D020123
CTDaffects(binding)RRAD
D020123
CTDincreases(reaction)RRAD
D020123
CTDincreases(expression)S1PR1
D020123
CTDdecreases(expression)SCARB2
D020123
CTDdecreases(expression)SCD
D020123
CTDdecreases(reaction)SCD
D020123
CTDdecreases(reaction)SEMA3C
D020123
CTDincreases(expression)SEMA3C
D020123
CTDaffects(localization)SERPINA1
D020123
CTDdecreases(expression)SERPINE1
D020123
CTDdecreases(reaction)SERPINE1
D020123
CTDincreases(expression)SHISA2
D020123
CTDdecreases(expression)SIRT1
D020123
CTDdecreases(reaction)SIRT1
D020123
CTDdecreases(reaction)SIRT2
D020123
CTDincreases(expression)SIRT2
D020123
CTDdecreases(expression)SKP2
D020123
CTDdecreases(reaction)SLC15A1
D020123
CTDincreases(activity)SLC15A1
D020123
CTDincreases(expression)SLC15A1
D020123
CTDdecreases(reaction)SMIM14
D020123
CTDincreases(expression)SMIM14
D020123
CTDdecreases(expression)SQSTM1
D020123
CTDdecreases(reaction)STARD10
D020123
CTDincreases(expression)STARD10
D020123
CTDdecreases(phosphorylation)STAT3
D020123
CTDdecreases(reaction)STAT3
D020123
CTDdecreases(phosphorylation)STAT3
D020123
CTDdecreases(reaction)STS
D020123
CTDincreases(activity)STS
D020123
CTDdecreases(reaction)SYT1
D020123
CTDincreases(expression)SYT1
D020123
CTDaffects(activity)TAL1
D020123
CTDdecreases(reaction)TAL1
D020123
CTDaffects(cotreatment)TCF19
D020123
CTDdecreases(expression)TCF19
D020123
CTDaffects(activity)TEAD1
D020123
CTDincreases(reaction)TEAD1
D020123
CTDdecreases(expression)TERT
D020123
CTDdecreases(expression)TERT
D020123
CTDaffects(binding)TGFB1
D020123
CTDincreases(activity)TGFB1
D020123
CTDaffects(cotreatment)TGFB1
D020123
CTDaffects(localization)TGFB1
D020123
CTDaffects(binding)TGFB1
D020123
CTDincreases(reaction)TGFB1
D020123
CTDdecreases(phosphorylation)TGFB1
D020123
CTDincreases(expression)TGFB1
D020123
CTDaffects(cotreatment)TGFB1
D020123
CTDdecreases(reaction)TGFB1
D020123
CTDincreases(reaction)TGFB1
D020123
CTDdecreases(activity)TGFB1
D020123
CTDdecreases(expression)TGFB1
D020123
CTDdecreases(phosphorylation)TGFB1
D020123
CTDaffects(cotreatment)TGFB1
D020123
CTDdecreases(phosphorylation)TGFB1
D020123
CTDincreases(expression)TGFB1
D020123
CTDaffects(cotreatment)TGFB1
D020123
CTDdecreases(expression)TGFB1
D020123
CTDincreases(expression)TGFB1
D020123
CTDincreases(response to substance)TGFB1
D020123
CTDaffects(cotreatment)TIMELESS
D020123
CTDdecreases(expression)TIMELESS
D020123
CTDdecreases(expression)TIMP3
D020123
CTDdecreases(reaction)TMEM14C
D020123
CTDincreases(expression)TMEM14C
D020123
CTDdecreases(reaction)TNF
D020123
CTDincreases(phosphorylation)TNF
D020123
CTDincreases(expression)TNF
D020123
CTDincreases(reaction)TNF
D020123
CTDincreases(expression)TNF
D020123
CTDincreases(expression)TP53
D020123
CTDincreases(reaction)TP53
D020123
CTDdecreases(activity)TP53
D020123
CTDdecreases(phosphorylation)TP53
D020123
CTDdecreases(expression)TP63
D020123
CTDaffects(cotreatment)TP73
D020123
CTDincreases(expression)TP73
D020123
CTDaffects(activity)TP73
D020123
CTDdecreases(reaction)TP73
D020123
CTDdecreases(expression)TP73
D020123
CTDincreases(expression)TP73
D020123
CTDincreases(reaction)TP73
D020123
CTDaffects(binding)TP73
D020123
CTDincreases(response to substance)TP73
D020123
CTDaffects(cotreatment)TTK
D020123
CTDdecreases(expression)TTK
D020123
CTDdecreases(expression)TYMS
D020123
CTDdecreases(expression)TYMS
D020123
CTDdecreases(response to substance)URI1
D020123
CTDdecreases(reaction)VEGFA
D020123
CTDincreases(expression)VEGFA
D020123
CTDdecreases(reaction)VEGFA
D020123
CTDincreases(secretion)VEGFA
D020123
CTDdecreases(reaction)VEGFA
D020123
CTDincreases(expression)VEGFA
D020123
CTDdecreases(expression)VEGFA
D020123
CTDdecreases(expression)WT1
D020123
CTDdecreases(expression)WT1
D020123
CTDdecreases(reaction)XBP1
D020123
CTDincreases(splicing)XBP1
D020123
CTDdecreases(expression)XIAP
D020123
CTDincreases(reaction)XIAP
D020123
CTDdecreases(expression)YPEL1
D020123
CTDdecreases(reaction)YPEL1
D020123
CTDincreases(expression)ZBED8
D020123
CTDaffects(activity)ZIC2
D020123
CTDdecreases(reaction)ZIC2
D020123
CTDdecreases(expression)ZNF628
D020123
CTDdecreases(reaction)ZNRD1
D020123
CTDincreases(expression)ZNRD1
D020123
CTDaffects(cotreatment)ZWINT
D020123
CTDdecreases(expression)ZWINT
D020123
PubChem Ratio Potency (uM)uM9.893AR-GI(Protien) :
PubChem Potency-Replicate_1uM10.682AR-GI(Protien) :
PubChem Potency-Replicate_1uM21.132AR-GI(Protien) :
PubChem Potency-Replicate_1uM23.710AR-GI(Protien) :
PubChem Potency-Replicate_1uM26.832AR-GI(Protien) :
PubChem Ratio Potency (uM)uM26.832AR-GI(Protien) :
PubChem Potency-Replicate_1uM2.113CYP19A1-GI(Protien) :
PubChem NoneuMCYP19A1-GI(Protien) :
PubChem ER Potency (uM)uM0.003ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM0.004ESR1-GI(Protien) :
PubChem ER Potency (uM)uM0.005ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM0.007ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM16.930NR3C1-GI(Protien) :
PubChem Potency-Replicate_1uM23.915NR3C1-GI(Protien) :
PubChem PotencyuM0.002TDP1-GI(Protien) :
PubChem PotencyuM0.005TDP1-GI(Protien) :
PubChem PotencyuM0.008TDP1-GI(Protien) :
PubChem PotencyuM0.012TDP1-GI(Protien) :
PubChem PotencyuM4.467TDP1-GI(Protien) :
PubChem NoneuMSTK33-GI(Protien) :
ChEMBLActivity-MTOR
-Target : CHEMBL2842
ChEMBLActivity-MTOR
-Target : CHEMBL2842
ChEMBLActivity-MTOR
-Target : CHEMBL2842
ChEMBLActivity-MTOR
-Target : CHEMBL2842
ChEMBLActivity-MTOR
-Target : CHEMBL2842
ChEMBLActivity-MTOR
-Target : CHEMBL2842
Download gene sets gmt, text, Detailed text
Contact us
Tan Lab , Mail Stop 8117
12801 East 17th Avenue
Division of Medical Oncology , Department of Medicine
University of Colorado School of Medicine
Aurora, CO 80045, USA

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