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Gene Set: D4 : CTD - Isotretinoin


Collection D4 : CTD
Chemical Name Isotretinoin ( From PubChem : VITINOIN )
FDA NPC WHO Indian Australia China Traditional
Herbal
Clinical
Trail
NotNotNotNotNotNotNotNot
Molecular
Weight
Hydrogen Bond
Donor Count
Hydrogen Bond
Acceptor Count
cLogP Lipinski Rule
300.435 g/mol 1 2 5.6026 False(3/4)
Structure
InChI InChI=1S/C20H28O2/c1-15(8-6-9-16(2)14-19(21)22)11-12-18-17(3)10-7-13-20(18,4)5/h6,8-9,11-12,14H,7,10,13H2,1-5H3,(H,21,22)/b9-6+,12-11+,15-8+,16-14+
InChIKey SHGAZHPCJJPHSC-YCNIQYBTSA-N
Links

Gene (780 / 861)


⊖ Less

Source Type Unit Value Gene PMID Assay Other
CTDincreases(expression)A2M
D015474
CTDdecreases(expression)AACS
D015474
CTDaffects(cotreatment)ABCB1
D015474
CTDincreases(expression)ABCB1
D015474
CTDdecreases(expression)ABHD5
D015474
CTDdecreases(expression)ACAA1
D015474
CTDdecreases(expression)ACAA2
D015474
CTDdecreases(expression)ACACA
D015474
CTDdecreases(expression)ACAD8
D015474
CTDdecreases(expression)ACADM
D015474
CTDdecreases(expression)ACADVL
D015474
CTDdecreases(expression)ACAT2
D015474
CTDdecreases(expression)ACLY
D015474
CTDdecreases(expression)ACO1
D015474
CTDdecreases(expression)ACOT13
D015474
CTDdecreases(expression)ACOT2
D015474
CTDdecreases(expression)ACOX2
D015474
CTDdecreases(expression)ACP6
D015474
CTDdecreases(expression)ACSBG1
D015474
CTDdecreases(expression)ACSL3
D015474
CTDdecreases(expression)ACSL5
D015474
CTDdecreases(expression)ACSM3
D015474
CTDdecreases(expression)ACY1
D015474
CTDincreases(expression)ADGRA2
D015474
CTDincreases(expression)ADGRE5
D015474
CTDdecreases(expression)ADGRG2
D015474
CTDincreases(expression)ADRA2A
D015474
CTDdecreases(expression)ADTRP
D015474
CTDdecreases(expression)AGA
D015474
CTDdecreases(expression)AGPAT3
D015474
CTDdecreases(expression)AGR2
D015474
CTDdecreases(expression)AHSP
D015474
CTDdecreases(expression)AIFM1
D015474
CTDdecreases(expression)AIP
D015474
CTDincreases(expression)AKAP11
D015474
CTDdecreases(expression)AKR1A1
D015474
CTDdecreases(expression)ALAS1
D015474
CTDdecreases(expression)ALCAM
D015474
CTDdecreases(expression)ALDH3B2
D015474
CTDdecreases(expression)ALG13
D015474
CTDdecreases(expression)ALOX15B
D015474
CTDdecreases(expression)AMACR
D015474
CTDincreases(expression)ANK2
D015474
CTDdecreases(expression)ANKHD1
D015474
CTDdecreases(expression)ANO10
D015474
CTDincreases(expression)AP2B1
D015474
CTDdecreases(expression)AP3S2
D015474
CTDdecreases(expression)APOC1
D015474
CTDaffects(response to substance)APOE
D015474
CTDdecreases(expression)APOOL
D015474
CTDdecreases(reaction)AREG
D015474
CTDincreases(expression)AREG
D015474
CTDdecreases(expression)ARF1P1
D015474
CTDdecreases(expression)ARG2
D015474
CTDincreases(expression)ARHGDIB
D015474
CTDincreases(expression)ARHGEF6
D015474
CTDaffects(cotreatment)ARTN
D015474
CTDincreases(expression)ARTN
D015474
CTDincreases(expression)ASAP3
D015474
CTDaffects(cotreatment)ATF5
D015474
CTDdecreases(expression)ATF5
D015474
CTDdecreases(expression)ATG4A
D015474
CTDincreases(expression)ATP2B4
D015474
CTDdecreases(expression)ATP5C1
D015474
CTDdecreases(expression)ATP5G3
D015474
CTDdecreases(expression)ATP5J2
D015474
CTDdecreases(expression)ATP6V0B
D015474
CTDdecreases(expression)ATP6V0C
D015474
CTDdecreases(expression)ATP6V1D
D015474
CTDincreases(expression)BASP1
D015474
CTDincreases(expression)BAX
D015474
CTDincreases(expression)BAX
D015474
CTDdecreases(expression)BCAP29
D015474
CTDdecreases(expression)BCAP31
D015474
CTDdecreases(expression)BCAT2
D015474
CTDdecreases(expression)BCKDHB
D015474
CTDdecreases(expression)BCL2
D015474
CTDdecreases(expression)BCL2
D015474
CTDincreases(expression)BCL2
D015474
CTDdecreases(expression)BCL2L1
D015474
CTDincreases(expression)BCL2L1
D015474
CTDdecreases(expression)BDH1
D015474
CTDdecreases(expression)BEAN1
D015474
CTDincreases(expression)BEND5
D015474
CTDincreases(expression)BGN
D015474
CTDincreases(expression)BHLHE40
D015474
CTDdecreases(expression)BIRC5
D015474
CTDdecreases(expression)BLVRB
D015474
CTDdecreases(expression)BPY2
D015474
CTDdecreases(expression)BRAF
D015474
CTDdecreases(expression)BSG
D015474
CTDincreases(expression)BTBD3
D015474
CTDdecreases(expression)BTD
D015474
CTDincreases(expression)BTN3A3
D015474
CTDdecreases(expression)C14ORF1
D015474
CTDdecreases(expression)C14ORF2
D015474
CTDincreases(expression)C16ORF45
D015474
CTDincreases(expression)C1ORF21
D015474
CTDdecreases(expression)C1ORF27
D015474
CTDincreases(expression)C1R
D015474
CTDincreases(expression)C1S
D015474
CTDdecreases(expression)C20ORF24
D015474
CTDdecreases(expression)C21ORF33
D015474
CTDincreases(expression)C3
D015474
CTDdecreases(expression)C9ORF16
D015474
CTDincreases(expression)CALD1
D015474
CTDdecreases(expression)CALML3
D015474
CTDincreases(cleavage)CASP3
D015474
CTDincreases(expression)CASP3
D015474
CTDincreases(expression)CASP3
D015474
CTDincreases(cleavage)CASP8
D015474
CTDdecreases(expression)CBX3
D015474
CTDdecreases(expression)CCDC86
D015474
CTDdecreases(reaction)CCL5
D015474
CTDincreases(expression)CCL5
D015474
CTDincreases(secretion)CCL5
D015474
CTDdecreases(expression)CCL5
D015474
CTDdecreases(expression)CCND1
D015474
CTDincreases(expression)CD2
D015474
CTDincreases(expression)CD247
D015474
CTDincreases(expression)CD34
D015474
CTDincreases(expression)CD37
D015474
CTDincreases(expression)CD38
D015474
CTDincreases(expression)CD3D
D015474
CTDincreases(expression)CD52
D015474
CTDaffects(cotreatment)CD69
D015474
CTDaffects(reaction)CD69
D015474
CTDincreases(expression)CD69
D015474
CTDincreases(expression)CD81
D015474
CTDdecreases(expression)CDA
D015474
CTDincreases(expression)CDC14B
D015474
CTDincreases(expression)CDH5
D015474
CTDdecreases(expression)CDK5
D015474
CTDdecreases(expression)CDK5RAP1
D015474
CTDdecreases(expression)CDKN1A
D015474
CTDincreases(expression)CDKN1A
D015474
CTDaffects(cotreatment)CDKN1A
D015474
CTDincreases(expression)CDKN1A
D015474
CTDdecreases(expression)CDKN1C
D015474
CTDdecreases(expression)CEACAM1
D015474
CTDaffects(cotreatment)CEACAM5
D015474
CTDincreases(expression)CEACAM5
D015474
CTDincreases(expression)CECR1
D015474
CTDincreases(expression)CEL
D015474
CTDincreases(expression)CELF2
D015474
CTDdecreases(expression)CERS4
D015474
CTDdecreases(expression)CFAP45
D015474
CTDdecreases(expression)CHI3L1
D015474
CTDdecreases(expression)CHI3L2
D015474
CTDdecreases(expression)CHP1
D015474
CTDincreases(expression)CHST6
D015474
CTDdecreases(expression)CIDEA
D015474
CTDdecreases(expression)CKB
D015474
CTDincreases(expression)CKM
D015474
CTDdecreases(expression)CKMT1B
D015474
CTDdecreases(expression)CLCN3
D015474
CTDdecreases(expression)CLPX
D015474
CTDdecreases(expression)CLSTN3
D015474
CTDdecreases(expression)CNDP2
D015474
CTDincreases(expression)COCH
D015474
CTDincreases(expression)COL14A1
D015474
CTDdecreases(expression)COL17A1
D015474
CTDincreases(expression)COL4A2
D015474
CTDincreases(expression)COL5A1
D015474
CTDincreases(expression)COL5A2
D015474
CTDdecreases(expression)COL6A1
D015474
CTDincreases(expression)COL6A1
D015474
CTDincreases(expression)COL6A2
D015474
CTDincreases(expression)COL6A3
D015474
CTDdecreases(expression)COL8A2
D015474
CTDdecreases(expression)COX5A
D015474
CTDdecreases(expression)COX5B
D015474
CTDdecreases(expression)COX6A1
D015474
CTDdecreases(expression)COX7A2
D015474
CTDdecreases(expression)COX7B
D015474
CTDdecreases(expression)COX7BP1
D015474
CTDdecreases(expression)CPD
D015474
CTDdecreases(expression)CPT2
D015474
CTDincreases(expression)CRABP2
D015474
CTDincreases(reaction)CRABP2
D015474
CTDdecreases(expression)CRAT
D015474
CTDincreases(phosphorylation)CREB1
D015474
CTDdecreases(expression)CRIPT
D015474
CTDincreases(expression)CRTC3
D015474
CTDincreases(expression)CSF1R
D015474
CTDincreases(expression)CST3
D015474
CTDdecreases(expression)CSTB
D015474
CTDdecreases(expression)CTH
D015474
CTDdecreases(expression)CTTN
D015474
CTDdecreases(expression)CUX2
D015474
CTDdecreases(expression)CXCL1
D015474
CTDdecreases(expression)CXCL10
D015474
CTDincreases(expression)CXCL12
D015474
CTDdecreases(expression)CYB5A
D015474
CTDincreases(expression)CYP26A1
D015474
CTDincreases(expression)CYP26B1
D015474
CTDincreases(expression)CYP26B1
D015474
CTDincreases(reaction)CYP26B1
D015474
CTDdecreases(expression)CYP27A1
D015474
CTDaffects(binding)CYP3A4
D015474
CTDincreases(expression)CYP3A4
D015474
CTDincreases(reaction)CYP3A4
D015474
CTDincreases(activity)CYP3A4
D015474
CTDdecreases(expression)CYP3A7
D015474
CTDdecreases(expression)CYP4A11
D015474
CTDdecreases(expression)CYP4F2
D015474
CTDdecreases(expression)CYP4F3
D015474
CTDdecreases(expression)CYP4F8
D015474
CTDdecreases(expression)CYP51A1
D015474
CTDdecreases(expression)CYP51A1P2
D015474
CTDdecreases(expression)DBI
D015474
CTDincreases(expression)DBN1
D015474
CTDdecreases(expression)DBT
D015474
CTDdecreases(expression)DCXR
D015474
CTDdecreases(expression)DDC
D015474
CTDdecreases(expression)DDO
D015474
CTDdecreases(expression)DDT
D015474
CTDincreases(expression)DENND5A
D015474
CTDdecreases(expression)DESI1
D015474
CTDdecreases(expression)DHCR24
D015474
CTDdecreases(expression)DHCR7
D015474
CTDdecreases(expression)DHFR
D015474
CTDdecreases(expression)DHRS11
D015474
CTDincreases(expression)DHRS3
D015474
CTDdecreases(expression)DHRS7B
D015474
CTDdecreases(expression)DHRS9
D015474
CTDaffects(cotreatment)DHRS9
D015474
CTDincreases(expression)DHRS9
D015474
CTDdecreases(expression)DIRAS3
D015474
CTDincreases(expression)DIXDC1
D015474
CTDdecreases(expression)DLD
D015474
CTDincreases(expression)DLG5
D015474
CTDincreases(expression)DLST
D015474
CTDdecreases(expression)DNAJA3
D015474
CTDdecreases(expression)DNAJC15
D015474
CTDdecreases(expression)DNAJC3
D015474
CTDincreases(expression)DNASE1
D015474
CTDdecreases(expression)DNASE1L2
D015474
CTDincreases(expression)DNM1
D015474
CTDdecreases(expression)DOPEY2
D015474
CTDdecreases(expression)DPP3
D015474
CTDincreases(expression)DPYSL2
D015474
CTDdecreases(expression)DRP2
D015474
CTDdecreases(expression)DSC1
D015474
CTDdecreases(expression)DSC2
D015474
CTDincreases(expression)DUSP10
D015474
CTDdecreases(expression)DUSP11
D015474
CTDdecreases(expression)DUSP4
D015474
CTDdecreases(expression)E2F8
D015474
CTDdecreases(expression)EBP
D015474
CTDdecreases(expression)ECH1
D015474
CTDdecreases(expression)ECHDC1
D015474
CTDdecreases(expression)ECI1
D015474
CTDincreases(expression)EFEMP2
D015474
CTDdecreases(expression)EGFR
D015474
CTDdecreases(expression)EGR3
D015474
CTDdecreases(expression)EI24
D015474
CTDdecreases(expression)EIF2B3
D015474
CTDdecreases(expression)EIF4E
D015474
CTDdecreases(expression)EIF4EBP2
D015474
CTDdecreases(expression)ELL2
D015474
CTDdecreases(expression)ELOVL1
D015474
CTDdecreases(expression)ELOVL4
D015474
CTDdecreases(expression)ELOVL5
D015474
CTDincreases(expression)EMP1
D015474
CTDdecreases(expression)ERCC1
D015474
CTDdecreases(expression)ETFDH
D015474
CTDdecreases(expression)ETNK1
D015474
CTDdecreases(expression)EXOC7
D015474
CTDdecreases(expression)FA2H
D015474
CTDdecreases(expression)FABP5
D015474
CTDdecreases(expression)FABP6
D015474
CTDdecreases(expression)FABP7
D015474
CTDdecreases(expression)FADS1
D015474
CTDdecreases(expression)FADS2
D015474
CTDdecreases(expression)FAM134B
D015474
CTDincreases(expression)FAM149A
D015474
CTDdecreases(expression)FAM3C
D015474
CTDincreases(expression)FAM3C
D015474
CTDdecreases(expression)FAM46C
D015474
CTDdecreases(expression)FAR2
D015474
CTDdecreases(expression)FASN
D015474
CTDdecreases(expression)FASTK
D015474
CTDincreases(expression)FBLN1
D015474
CTDdecreases(expression)FBP1
D015474
CTDdecreases(expression)FBP2
D015474
CTDincreases(expression)FBXL7
D015474
CTDdecreases(expression)FBXO9
D015474
CTDdecreases(expression)FDFT1
D015474
CTDdecreases(expression)FDPS
D015474
CTDincreases(expression)FEZ2
D015474
CTDdecreases(expression)FGF1
D015474
CTDincreases(expression)FGFR1
D015474
CTDincreases(expression)FGFR3
D015474
CTDdecreases(expression)FH
D015474
CTDincreases(expression)FKBP10
D015474
CTDdecreases(expression)FKBP8
D015474
CTDdecreases(expression)FLG
D015474
CTDincreases(expression)FLNA
D015474
CTDincreases(expression)FLT3LG
D015474
CTDincreases(expression)FN1
D015474
CTDdecreases(expression)FOSB
D015474
CTDincreases(expression)FOXD1
D015474
CTDincreases(expression)FUT8
D015474
CTDincreases(expression)FYB
D015474
CTDdecreases(expression)FZD5
D015474
CTDdecreases(expression)G6PD
D015474
CTDincreases(expression)G6PD
D015474
CTDdecreases(expression)GABRA4
D015474
CTDdecreases(expression)GAGE5
D015474
CTDdecreases(expression)GAL
D015474
CTDaffects(cotreatment)GATA3
D015474
CTDincreases(expression)GATA3
D015474
CTDdecreases(expression)GBA
D015474
CTDdecreases(expression)GBE1
D015474
CTDdecreases(expression)GCLM
D015474
CTDincreases(expression)GCNT3
D015474
CTDdecreases(expression)GCSH
D015474
CTDdecreases(expression)GDAP1L1
D015474
CTDincreases(expression)GDF15
D015474
CTDincreases(expression)GDF2
D015474
CTDdecreases(expression)GGCX
D015474
CTDdecreases(expression)GGPS1
D015474
CTDdecreases(expression)GHITM
D015474
CTDdecreases(expression)GINS1
D015474
CTDdecreases(expression)GK
D015474
CTDdecreases(expression)GK6P
D015474
CTDdecreases(expression)GLDC
D015474
CTDdecreases(expression)GLRX2
D015474
CTDdecreases(expression)GLRX5
D015474
CTDincreases(expression)GLUL
D015474
CTDdecreases(expression)GNG4
D015474
CTDdecreases(expression)GNPAT
D015474
CTDdecreases(expression)GPR143
D015474
CTDincreases(expression)GPX2
D015474
CTDdecreases(expression)GPX3
D015474
CTDdecreases(expression)GRB7
D015474
CTDdecreases(expression)GRPEL1
D015474
CTDdecreases(expression)GSTM1
D015474
CTDaffects(metabolic processing)GSTP1
D015474
CTDdecreases(reaction)GSTP1
D015474
CTDdecreases(expression)GSTZ1
D015474
CTDdecreases(expression)H2AFX
D015474
CTDdecreases(expression)H2BFS
D015474
CTDdecreases(expression)HADH
D015474
CTDdecreases(expression)HAO2
D015474
CTDincreases(expression)HBEGF
D015474
CTDincreases(expression)HCLS1
D015474
CTDdecreases(expression)HCN3
D015474
CTDdecreases(expression)HGD
D015474
CTDdecreases(expression)HIBCH
D015474
CTDdecreases(expression)HILPDA
D015474
CTDincreases(expression)HIP1
D015474
CTDdecreases(expression)HIST1H1C
D015474
CTDdecreases(expression)HIST1H2AE
D015474
CTDdecreases(expression)HIST1H2AG
D015474
CTDdecreases(expression)HIST1H2BC
D015474
CTDdecreases(expression)HIST1H2BD
D015474
CTDdecreases(expression)HIST1H2BE
D015474
CTDdecreases(expression)HIST1H2BG
D015474
CTDdecreases(expression)HIST1H2BH
D015474
CTDdecreases(expression)HIST1H2BK
D015474
CTDdecreases(expression)HIST2H2BE
D015474
CTDdecreases(expression)HIST3H2A
D015474
CTDincreases(expression)HLA-DPA1
D015474
CTDincreases(expression)HLA-DPB1
D015474
CTDincreases(expression)HLA-DQB1
D015474
CTDincreases(expression)HLA-DQB2
D015474
CTDincreases(expression)HLA-E
D015474
CTDincreases(expression)HLA-F
D015474
CTDincreases(expression)HLA-G
D015474
CTDdecreases(expression)HLCS
D015474
CTDdecreases(expression)HMGCR
D015474
CTDdecreases(expression)HMGCS1
D015474
CTDdecreases(expression)HRSP12
D015474
CTDdecreases(expression)HSD11B1
D015474
CTDdecreases(expression)HSD17B12
D015474
CTDdecreases(expression)HSD17B7
D015474
CTDdecreases(expression)HSD3B1
D015474
CTDdecreases(expression)HSP90B1
D015474
CTDdecreases(expression)HSPA9
D015474
CTDdecreases(expression)HSPD1
D015474
CTDincreases(expression)HTRA1
D015474
CTDdecreases(expression)HUS1
D015474
CTDincreases(expression)ICAM2
D015474
CTDdecreases(expression)IDH1
D015474
CTDdecreases(expression)IDI1
D015474
CTDdecreases(expression)IDI2-AS1
D015474
CTDdecreases(expression)IER3
D015474
CTDincreases(expression)IFI35
D015474
CTDincreases(expression)IFITM1
D015474
CTDaffects(cotreatment)IFNA2
D015474
CTDaffects(reaction)IFNA2
D015474
CTDincreases(expression)IFNA2
D015474
CTDdecreases(expression)IFRD1
D015474
CTDdecreases(expression)IFT20
D015474
CTDincreases(expression)IGF1
D015474
CTDincreases(expression)IGFBP3
D015474
CTDincreases(expression)IGFBP4
D015474
CTDincreases(expression)IGFBP5
D015474
CTDdecreases(expression)IL10RA
D015474
CTDdecreases(expression)IL13RA1
D015474
CTDdecreases(expression)IL1B
D015474
CTDincreases(expression)IL1B
D015474
CTDaffects(cotreatment)IL1B
D015474
CTDincreases(expression)IL1B
D015474
CTDdecreases(expression)IL1R2
D015474
CTDdecreases(expression)IL24
D015474
CTDincreases(expression)IL32
D015474
CTDdecreases(expression)IL6
D015474
CTDdecreases(expression)INPP4B
D015474
CTDdecreases(expression)INSIG1
D015474
CTDincreases(expression)IRF1
D015474
CTDincreases(reaction)IRF1
D015474
CTDdecreases(expression)ISCA1
D015474
CTDincreases(expression)ISLR
D015474
CTDdecreases(expression)ISOC1
D015474
CTDincreases(expression)ITGA4
D015474
CTDincreases(expression)ITGAV
D015474
CTDincreases(expression)ITGB2
D015474
CTDincreases(expression)JAK1
D015474
CTDincreases(expression)KANK2
D015474
CTDdecreases(expression)KCNJ15
D015474
CTDdecreases(expression)KCNK1
D015474
CTDincreases(expression)KCTD12
D015474
CTDdecreases(expression)KLHDC4
D015474
CTDdecreases(expression)KRAS
D015474
CTDdecreases(expression)KRT1
D015474
CTDdecreases(expression)KRT10
D015474
CTDdecreases(expression)KRT14
D015474
CTDincreases(expression)KRT15
D015474
CTDdecreases(expression)KRT16
D015474
CTDdecreases(expression)KRT17
D015474
CTDdecreases(expression)KRT17
D015474
CTDincreases(expression)KRT19
D015474
CTDdecreases(expression)KRT5
D015474
CTDdecreases(expression)KRT6A
D015474
CTDincreases(expression)KRT7
D015474
CTDdecreases(expression)KRT75
D015474
CTDdecreases(expression)LACTB2
D015474
CTDdecreases(expression)LAGE3
D015474
CTDdecreases(expression)LAMA2
D015474
CTDincreases(expression)LAMA2
D015474
CTDdecreases(expression)LAMA3
D015474
CTDincreases(expression)LAMC1
D015474
CTDincreases(expression)LAMC3
D015474
CTDincreases(expression)LAPTM5
D015474
CTDdecreases(expression)LARP4
D015474
CTDincreases(expression)LCK
D015474
CTDincreases(expression)LCN2
D015474
CTDincreases(expression)LCP2
D015474
CTDdecreases(expression)LDLR
D015474
CTDincreases(expression)LHFP
D015474
CTDincreases(expression)LIMCH1
D015474
CTDincreases(expression)LIPC
D015474
CTDincreases(expression)LMNB1
D015474
CTDincreases(expression)LMO2
D015474
CTDincreases(expression)LOXL2
D015474
CTDdecreases(expression)LPCAT3
D015474
CTDdecreases(expression)LPIN1
D015474
CTDincreases(expression)LRAT
D015474
CTDincreases(expression)LTBP1
D015474
CTDincreases(expression)LYN
D015474
CTDdecreases(expression)MAFF
D015474
CTDincreases(expression)MAN1A1
D015474
CTDincreases(expression)MAP4
D015474
CTDdecreases(expression)MBOAT2
D015474
CTDdecreases(expression)MC5R
D015474
CTDdecreases(expression)MCAT
D015474
CTDdecreases(expression)MCCC1
D015474
CTDdecreases(expression)MCCC2
D015474
CTDdecreases(expression)MCFD2
D015474
CTDdecreases(expression)MCTS1
D015474
CTDdecreases(expression)MCUR1
D015474
CTDdecreases(expression)MDH1
D015474
CTDdecreases(expression)ME1
D015474
CTDdecreases(expression)MECR
D015474
CTDdecreases(expression)MED8
D015474
CTDincreases(expression)MEF2C
D015474
CTDdecreases(expression)MFAP2
D015474
CTDincreases(expression)MFAP2
D015474
CTDdecreases(expression)MFAP3L
D015474
CTDincreases(expression)MFAP4
D015474
CTDdecreases(expression)MINA
D015474
CTDincreases(expression)MKL2
D015474
CTDdecreases(expression)MLANA
D015474
CTDdecreases(expression)MMP10
D015474
CTDdecreases(reaction)MMP13
D015474
CTDincreases(expression)MMP13
D015474
CTDincreases(secretion)MMP13
D015474
CTDdecreases(expression)MMP13
D015474
CTDdecreases(reaction)MMP2
D015474
CTDincreases(expression)MMP2
D015474
CTDincreases(secretion)MMP2
D015474
CTDincreases(expression)MMP2
D015474
CTDincreases(expression)MMP23B
D015474
CTDdecreases(reaction)MMP9
D015474
CTDincreases(expression)MMP9
D015474
CTDincreases(secretion)MMP9
D015474
CTDdecreases(expression)MMP9
D015474
CTDdecreases(expression)MOCOS
D015474
CTDdecreases(expression)MOSPD1
D015474
CTDdecreases(expression)MPC1
D015474
CTDdecreases(expression)MPC2
D015474
CTDdecreases(expression)MRPL33
D015474
CTDdecreases(expression)MRPS16
D015474
CTDdecreases(expression)MRPS18A
D015474
CTDdecreases(expression)MRPS33
D015474
CTDdecreases(expression)MRS2
D015474
CTDincreases(expression)MSMB
D015474
CTDdecreases(expression)MSMO1
D015474
CTDdecreases(expression)MSRB1
D015474
CTDdecreases(expression)MTCH2
D015474
CTDdecreases(expression)MTO1
D015474
CTDdecreases(expression)MTX1
D015474
CTDdecreases(expression)MUC1
D015474
CTDdecreases(expression)MVD
D015474
CTDdecreases(expression)MVK
D015474
CTDdecreases(expression)MYCBP
D015474
CTDdecreases(expression)MYCN
D015474
CTDincreases(reaction)MYCN
D015474
CTDdecreases(expression)MYL4
D015474
CTDdecreases(expression)MYOD1
D015474
CTDdecreases(expression)NADK
D015474
CTDdecreases(expression)NAMPT
D015474
CTDdecreases(expression)NBN
D015474
CTDdecreases(expression)NDUFA3
D015474
CTDdecreases(expression)NDUFAF1
D015474
CTDdecreases(expression)NDUFB3
D015474
CTDdecreases(expression)NDUFC2
D015474
CTDdecreases(expression)NDUFS1
D015474
CTDdecreases(expression)NDUFS3
D015474
CTDdecreases(expression)NDUFS7
D015474
CTDdecreases(expression)NDUFS8
D015474
CTDdecreases(expression)NDUFV2
D015474
CTDincreases(expression)NEDD9
D015474
CTDdecreases(expression)NEFL
D015474
CTDdecreases(expression)NIT2
D015474
CTDdecreases(expression)NOP16
D015474
CTDdecreases(expression)NPC1
D015474
CTDdecreases(expression)NPL
D015474
CTDdecreases(expression)NQO2
D015474
CTDaffects(binding)NR1I2
D015474
CTDincreases(expression)NR1I2
D015474
CTDincreases(reaction)NR1I2
D015474
CTDincreases(expression)NR2F1
D015474
CTDdecreases(expression)NSDHL
D015474
CTDdecreases(expression)NTAN1
D015474
CTDincreases(expression)NTRK2
D015474
CTDdecreases(expression)NUDT21
D015474
CTDdecreases(expression)NUDT4
D015474
CTDdecreases(expression)NUS1P3
D015474
CTDdecreases(expression)OAS1
D015474
CTDdecreases(expression)ODC1
D015474
CTDdecreases(expression)OLAH
D015474
CTDdecreases(expression)OR7E12P
D015474
CTDdecreases(expression)ORMDL2
D015474
CTDdecreases(expression)OTUB2
D015474
CTDdecreases(expression)PAFAH2
D015474
CTDdecreases(expression)PANK3
D015474
CTDdecreases(expression)PAQR3
D015474
CTDdecreases(expression)PAWR
D015474
CTDdecreases(expression)PCCB
D015474
CTDaffects(cotreatment)PCDH1
D015474
CTDincreases(expression)PCDH1
D015474
CTDincreases(expression)PCOLCE
D015474
CTDdecreases(expression)PCTP
D015474
CTDdecreases(expression)PDE6A
D015474
CTDincreases(expression)PDGFRB
D015474
CTDdecreases(expression)PDHA1
D015474
CTDdecreases(expression)PDHB
D015474
CTDdecreases(expression)PDHX
D015474
CTDdecreases(expression)PDXK
D015474
CTDdecreases(expression)PDZK1
D015474
CTDdecreases(expression)PECR
D015474
CTDdecreases(expression)PEX11A
D015474
CTDdecreases(expression)PEX13
D015474
CTDdecreases(expression)PEX16
D015474
CTDdecreases(expression)PEX19
D015474
CTDdecreases(expression)PEX3
D015474
CTDdecreases(expression)PEX7
D015474
CTDdecreases(expression)PGD
D015474
CTDdecreases(expression)PGM1
D015474
CTDdecreases(expression)PGRMC1
D015474
CTDincreases(expression)PHGDH
D015474
CTDaffects(cotreatment)PHLDA1
D015474
CTDincreases(expression)PHLDA1
D015474
CTDdecreases(expression)PHLDA2
D015474
CTDdecreases(expression)PIK3C2G
D015474
CTDdecreases(expression)PIR
D015474
CTDincreases(expression)PIR
D015474
CTDdecreases(expression)PKLR
D015474
CTDincreases(expression)PKP1
D015474
CTDdecreases(expression)PLA2G7
D015474
CTDincreases(expression)PLAT
D015474
CTDincreases(expression)PLCL2
D015474
CTDdecreases(expression)PLIN2
D015474
CTDincreases(expression)PLTP
D015474
CTDdecreases(expression)PMEL
D015474
CTDdecreases(expression)PMPCB
D015474
CTDdecreases(expression)PMVK
D015474
CTDdecreases(expression)PNPLA3
D015474
CTDincreases(expression)POLR2M
D015474
CTDdecreases(expression)PON3
D015474
CTDdecreases(expression)POPDC2
D015474
CTDincreases(expression)PPAP2B
D015474
CTDdecreases(expression)PPIF
D015474
CTDdecreases(expression)PPM1B
D015474
CTDincreases(expression)PPP1R16B
D015474
CTDdecreases(expression)PRDX2
D015474
CTDdecreases(expression)PREPL
D015474
CTDincreases(expression)PROS1
D015474
CTDdecreases(expression)PRSS8
D015474
CTDdecreases(expression)PSMA1
D015474
CTDdecreases(expression)PSMA3
D015474
CTDdecreases(expression)PSMA4
D015474
CTDdecreases(expression)PSMA5
D015474
CTDdecreases(expression)PSMA7
D015474
CTDdecreases(expression)PSMB5
D015474
CTDdecreases(expression)PTGDR
D015474
CTDincreases(expression)PTGDS
D015474
CTDdecreases(expression)PTGS1
D015474
CTDdecreases(expression)PTGS2
D015474
CTDincreases(expression)PTPRB
D015474
CTDincreases(expression)PTPRC
D015474
CTDincreases(expression)PTPRG
D015474
CTDincreases(expression)PTPRM
D015474
CTDincreases(expression)PTRF
D015474
CTDdecreases(expression)PTRH2
D015474
CTDdecreases(expression)PTS
D015474
CTDdecreases(expression)PXMP2
D015474
CTDdecreases(expression)PXMP4
D015474
CTDincreases(expression)QKI
D015474
CTDdecreases(expression)RAB27A
D015474
CTDdecreases(expression)RAB38
D015474
CTDincreases(expression)RAC2
D015474
CTDincreases(expression)RARA
D015474
CTDincreases(expression)RARB
D015474
CTDaffects(cotreatment)RARB
D015474
CTDincreases(acetylation)RARB
D015474
CTDincreases(expression)RARB
D015474
CTDincreases(reaction)RARB
D015474
CTDdecreases(reaction)RARRES1
D015474
CTDincreases(expression)RARRES1
D015474
CTDdecreases(expression)RASAL1
D015474
CTDincreases(expression)RASSF2
D015474
CTDdecreases(expression)RBKS
D015474
CTDdecreases(expression)RBM47
D015474
CTDincreases(expression)RBPMS
D015474
CTDdecreases(expression)RC3H2
D015474
CTDdecreases(expression)RDH11
D015474
CTDdecreases(expression)RFK
D015474
CTDdecreases(expression)RHOA
D015474
CTDdecreases(expression)RHOB
D015474
CTDincreases(expression)RHOBTB3
D015474
CTDdecreases(expression)RMDN1
D015474
CTDincreases(expression)RNASET2
D015474
CTDdecreases(expression)RND3
D015474
CTDdecreases(expression)RNF128
D015474
CTDincreases(expression)RNF38
D015474
CTDdecreases(expression)RNF5
D015474
CTDincreases(expression)ROR1
D015474
CTDdecreases(expression)RORA
D015474
CTDdecreases(expression)RPP40
D015474
CTDdecreases(expression)RTCA
D015474
CTDincreases(expression)RTN1
D015474
CTDaffects(binding)RXRA
D015474
CTDincreases(expression)RXRA
D015474
CTDincreases(reaction)RXRA
D015474
CTDincreases(activity)RXRA
D015474
CTDdecreases(expression)S100A1
D015474
CTDincreases(expression)S100A4
D015474
CTDincreases(expression)S100A7
D015474
CTDincreases(expression)S100A8
D015474
CTDincreases(expression)S100A9
D015474
CTDdecreases(expression)SAMM50
D015474
CTDincreases(expression)SAMSN1
D015474
CTDdecreases(expression)SAR1B
D015474
CTDdecreases(expression)SC5D
D015474
CTDdecreases(expression)SCAMP1
D015474
CTDincreases(expression)SCNN1A
D015474
CTDdecreases(expression)SDF2L1
D015474
CTDdecreases(expression)SDHC
D015474
CTDincreases(expression)SELPLG
D015474
CTDdecreases(expression)SEPT11
D015474
CTDincreases(expression)SERHL2
D015474
CTDincreases(expression)SERPINA3
D015474
CTDdecreases(expression)SERPINB2
D015474
CTDdecreases(expression)SERPINB8
D015474
CTDdecreases(expression)SERPINB9
D015474
CTDincreases(expression)SERPING1
D015474
CTDdecreases(expression)SGK2
D015474
CTDincreases(expression)SHC1P1
D015474
CTDdecreases(expression)SHMT1
D015474
CTDincreases(expression)SIRPA
D015474
CTDincreases(expression)SLA
D015474
CTDdecreases(expression)SLC11A2
D015474
CTDdecreases(expression)SLC15A1
D015474
CTDdecreases(expression)SLC16A1
D015474
CTDdecreases(expression)SLC16A7
D015474
CTDdecreases(expression)SLC22A18
D015474
CTDdecreases(expression)SLC25A11
D015474
CTDdecreases(expression)SLC25A15
D015474
CTDdecreases(expression)SLC25A16
D015474
CTDdecreases(expression)SLC25A17
D015474
CTDdecreases(expression)SLC26A3
D015474
CTDdecreases(expression)SLC27A2
D015474
CTDdecreases(expression)SLC30A1
D015474
CTDdecreases(expression)SLC30A10
D015474
CTDdecreases(expression)SLC31A1
D015474
CTDdecreases(expression)SLC35A2
D015474
CTDdecreases(expression)SLC35B1
D015474
CTDincreases(expression)SLC39A14
D015474
CTDdecreases(expression)SLC39A8
D015474
CTDdecreases(expression)SLC46A3
D015474
CTDdecreases(expression)SLC50A1
D015474
CTDdecreases(expression)SLC5A6
D015474
CTDdecreases(expression)SLC7A5
D015474
CTDdecreases(expression)SLCO4C1
D015474
CTDincreases(expression)SLIT3
D015474
CTDincreases(expression)SMYD3
D015474
CTDincreases(expression)SNED1
D015474
CTDdecreases(expression)SNX13
D015474
CTDdecreases(expression)SOAT1
D015474
CTDdecreases(expression)SOCS1
D015474
CTDincreases(expression)SOCS2
D015474
CTDdecreases(expression)SOD2
D015474
CTDdecreases(expression)SORBS1
D015474
CTDdecreases(expression)SORD
D015474
CTDdecreases(expression)SORT1
D015474
CTDdecreases(localization)SOX17
D015474
CTDdecreases(expression)SPCS3
D015474
CTDincreases(expression)SPP1
D015474
CTDincreases(expression)SPRED2
D015474
CTDincreases(expression)SPRR1B
D015474
CTDdecreases(expression)SPRR3
D015474
CTDdecreases(expression)SRD5A1
D015474
CTDdecreases(expression)SRPX2
D015474
CTDdecreases(expression)ST13
D015474
CTDdecreases(expression)ST6GALNAC4
D015474
CTDdecreases(expression)STAMBP
D015474
CTDdecreases(expression)STAP2
D015474
CTDdecreases(expression)SUCLG1
D015474
CTDincreases(expression)SULT2A1
D015474
CTDincreases(expression)SUSD5
D015474
CTDdecreases(expression)SYN2
D015474
CTDdecreases(expression)SYNGR1
D015474
CTDincreases(expression)TACSTD2
D015474
CTDincreases(expression)TAGLN
D015474
CTDaffects(cotreatment)TAGLN
D015474
CTDdecreases(expression)TAGLN3
D015474
CTDdecreases(expression)TALDO1
D015474
CTDincreases(expression)TBC1D1
D015474
CTDincreases(expression)TBL1XR1
D015474
CTDdecreases(expression)TCTA
D015474
CTDdecreases(expression)TECR
D015474
CTDdecreases(expression)TFDP2
D015474
CTDdecreases(expression)TFF2
D015474
CTDdecreases(expression)TFRC
D015474
CTDincreases(expression)TGFB1I1
D015474
CTDincreases(expression)TGFBR2
D015474
CTDdecreases(expression)TGM1
D015474
CTDdecreases(expression)THBS1
D015474
CTDincreases(expression)THBS4
D015474
CTDdecreases(expression)TIMM13
D015474
CTDdecreases(expression)TIMM23
D015474
CTDincreases(expression)TIMP3
D015474
CTDincreases(expression)TJP3
D015474
CTDdecreases(expression)TKT
D015474
CTDdecreases(expression)TM7SF2
D015474
CTDdecreases(expression)TMBIM6
D015474
CTDdecreases(expression)TMED3
D015474
CTDdecreases(expression)TMED5
D015474
CTDdecreases(expression)TMEM164
D015474
CTDdecreases(expression)TMEM208
D015474
CTDdecreases(expression)TMEM254
D015474
CTDdecreases(expression)TMEM33
D015474
CTDdecreases(expression)TMEM41B
D015474
CTDdecreases(expression)TMEM53
D015474
CTDdecreases(expression)TMEM97
D015474
CTDdecreases(expression)TMPRSS11E
D015474
CTDdecreases(reaction)TNF
D015474
CTDincreases(expression)TNF
D015474
CTDincreases(secretion)TNF
D015474
CTDincreases(expression)TNFSF10
D015474
CTDincreases(expression)TNN
D015474
CTDincreases(expression)TNXB
D015474
CTDincreases(expression)TOB2
D015474
CTDdecreases(expression)TOMM70A
D015474
CTDdecreases(expression)TPD52L1
D015474
CTDincreases(expression)TPSB2
D015474
CTDincreases(expression)TRAF3IP3
D015474
CTDincreases(expression)TRBC1
D015474
CTDincreases(expression)TRIM22
D015474
CTDincreases(expression)TRIM31
D015474
CTDdecreases(expression)TROVE2
D015474
CTDdecreases(expression)TSPAN6
D015474
CTDdecreases(expression)TST
D015474
CTDincreases(expression)TXK
D015474
CTDaffects(cotreatment)TXK
D015474
CTDdecreases(expression)UBE2A
D015474
CTDdecreases(expression)UBE2K
D015474
CTDdecreases(expression)UBE2S
D015474
CTDdecreases(expression)UBE2W
D015474
CTDdecreases(expression)UBIAD1
D015474
CTDdecreases(expression)UGT2A1
D015474
CTDdecreases(expression)UGT2B28
D015474
CTDdecreases(expression)ULK4
D015474
CTDdecreases(expression)UNC5B
D015474
CTDdecreases(expression)UNG
D015474
CTDdecreases(expression)UPB1
D015474
CTDdecreases(expression)UQCRC1
D015474
CTDdecreases(expression)UQCRC2
D015474
CTDdecreases(expression)UQCRQ
D015474
CTDdecreases(expression)USP2
D015474
CTDdecreases(expression)USP3
D015474
CTDdecreases(expression)UVRAG
D015474
CTDincreases(expression)VCAN
D015474
CTDincreases(expression)VEGFA
D015474
CTDdecreases(expression)VEGFC
D015474
CTDdecreases(expression)VMP1
D015474
CTDincreases(expression)VOPP1
D015474
CTDdecreases(expression)WASL
D015474
CTDdecreases(expression)WDR61
D015474
CTDincreases(expression)WIF1
D015474
CTDdecreases(expression)YARS2
D015474
CTDdecreases(expression)ZBTB16
D015474
CTDdecreases(expression)ZNF117
D015474
CTDdecreases(expression)ZNF165
D015474
CTDdecreases(expression)ZNF254
D015474
CTDdecreases(expression)ZNF43
D015474
CTDdecreases(expression)ZNF430
D015474
CTDincreases(expression)ZNF532
D015474
CTDdecreases(expression)ZNF675
D015474
CTDdecreases(expression)ZNF91
D015474
PubChem NoneuMABCB1-GI(Protien) :
PubChem Potency-Replicate_1uM48.706AR-GI(Protien) :
PubChem IC50_CF-PAF_MeanuM0.640CFTR-GI(Protien) :
PubChem NoneuMCFTR-GI(Protien) :
PubChem IC50_CF-PAF_MeanuMCFTR-GI(Protien) :
PubChem NoneuMCFTR-GI(Protien) :
PubChem ER Potency (uM)uM0.043ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM0.244ESR1-GI(Protien) :
PubChem NoneuMKCNK9-GI(Protien) :
PubChem NoneuMMDM2-GI(Protien) :
PubChem NoneuMMDM2-GI(Protien) :
PubChem NoneuMMDM4-GI(Protien) :
PubChem NoneuMMDM4-GI(Protien) :
PubChem NoneuMNR0B1-GI(Protien) :
PubChem NoneuMNR0B1-GI(Protien) :
PubChem Potency-Replicate_1uM49.110NR1H4-GI(Protien) :
PubChem Ratio Potency (uM)uM49.110NR1H4-GI(Protien) :
PubChem NoneuMNR5A1-GI(Protien) :
PubChem NoneuMPLA2G7-GI(Protien) :
PubChem Ratio Potency (uM)uM0.335PPARG-GI(Protien) :
PubChem PotencyuM23.109TDP1-GI(Protien) :
PubChem PotencyuM22.387THRB-GI(Protien) :
PubChem PotencyuM28.184THRB-GI(Protien) :
PubChem PotencyuM50.119VDR-GI(Protien) :
ChEMBLPotencynM28183.800THRB
-Target : CHEMBL1947
ChEMBLPotencynM22387.200THRB
-Target : CHEMBL1947
Download gene sets gmt, text, Detailed text
Contact us
Tan Lab , Mail Stop 8117
12801 East 17th Avenue
Division of Medical Oncology , Department of Medicine
University of Colorado School of Medicine
Aurora, CO 80045, USA

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