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Gene Set: D4 : CTD - Rotenone


Collection D4 : CTD
Chemical Name Rotenone ( From PubChem : CUBE ROOT EXTRACT )
FDA NPC WHO Indian Australia China Traditional
Herbal
Clinical
Trail
NotNotNotNotNotNotNotNot
Molecular
Weight
Hydrogen Bond
Donor Count
Hydrogen Bond
Acceptor Count
cLogP Lipinski Rule
394.417 g/mol 0 6 3.7033 True
Structure
InChI InChI=1S/C23H22O6/c1-11(2)16-8-14-15(28-16)6-5-12-22(24)21-13-7-18(25-3)19(26-4)9-17(13)27-10-20(21)29-23(12)14/h5-7,9,16,20-21H,1,8,10H2,2-4H3/t16-,20+,21+/m0/s1
InChIKey JUVIOZPCNVVQFO-ZLGUVYLKSA-N
Links

Gene (211 / 526)


⊖ Less

Source Type Unit Value Gene PMID Assay Other
CTDaffects(activity)ABCB1
D012402
CTDaffects(cotreatment)ABCG5
D012402
CTDdecreases(expression)ABCG5
D012402
CTDaffects(cotreatment)ABCG8
D012402
CTDdecreases(expression)ABCG8
D012402
CTDdecreases(expression)ACAD9
D012402
CTDaffects(cotreatment)ACAT1
D012402
CTDdecreases(expression)ACAT1
D012402
CTDdecreases(activity)ACO1
D012402
CTDincreases(activity)ACO1
D012402
CTDdecreases(activity)ACO2
D012402
CTDdecreases(reaction)ACP5
D012402
CTDincreases(expression)ACP5
D012402
CTDdecreases(reaction)ACTA2
D012402
CTDincreases(expression)ACTA2
D012402
CTDdecreases(reaction)AGT
D012402
CTDincreases(phosphorylation)AGT
D012402
CTDincreases(reaction)AGT
D012402
CTDaffects(localization)AIFM1
D012402
CTDdecreases(reaction)AIFM1
D012402
CTDincreases(expression)ANPEP
D012402
CTDincreases(expression)APAF1
D012402
CTDdecreases(expression)ARL2
D012402
CTDincreases(expression)ATF4
D012402
CTDaffects(reaction)ATG5
D012402
CTDdecreases(reaction)ATG5
D012402
CTDincreases(cleavage)ATG5
D012402
CTDaffects(response to substance)ATG5
D012402
CTDincreases(expression)ATM
D012402
CTDincreases(expression)ATP5E
D012402
CTDincreases(expression)ATP5G3
D012402
CTDincreases(expression)ATP5I
D012402
CTDincreases(expression)ATP5J
D012402
CTDincreases(expression)ATP5L
D012402
CTDincreases(expression)ATP5O
D012402
CTDincreases(expression)ATR
D012402
CTDincreases(expression)ATXN3
D012402
CTDdecreases(reaction)BACE1
D012402
CTDincreases(expression)BACE1
D012402
CTDdecreases(phosphorylation)BAD
D012402
CTDdecreases(reaction)BAD
D012402
CTDincreases(expression)BARD1
D012402
CTDdecreases(reaction)BAX
D012402
CTDincreases(expression)BAX
D012402
CTDincreases(expression)BAX
D012402
CTDdecreases(reaction)BAX
D012402
CTDincreases(expression)BAX
D012402
CTDdecreases(response to substance)BCL2
D012402
CTDdecreases(reaction)BCL2
D012402
CTDdecreases(expression)BCL2
D012402
CTDdecreases(reaction)BCL2
D012402
CTDdecreases(expression)BCL2
D012402
CTDincreases(expression)BCL2
D012402
CTDdecreases(expression)BCL2
D012402
CTDdecreases(reaction)BCL2
D012402
CTDdecreases(reaction)BECN1
D012402
CTDincreases(expression)BECN1
D012402
CTDaffects(response to substance)BECN1
D012402
CTDaffects(cotreatment)BIRC3
D012402
CTDdecreases(reaction)BIRC3
D012402
CTDincreases(expression)BIRC3
D012402
CTDincreases(expression)BRCA1
D012402
CTDincreases(expression)BRCA2
D012402
CTDaffects(localization)BUB1B
D012402
CTDincreases(expression)BUB1B
D012402
CTDdecreases(reaction)CASP3
D012402
CTDincreases(activity)CASP3
D012402
CTDincreases(activity)CASP3
D012402
CTDincreases(reaction)CASP3
D012402
CTDdecreases(reaction)CASP3
D012402
CTDincreases(activity)CASP3
D012402
CTDdecreases(reaction)CASP3
D012402
CTDincreases(activity)CASP3
D012402
CTDincreases(cleavage)CASP3
D012402
CTDdecreases(reaction)CASP3
D012402
CTDincreases(cleavage)CASP3
D012402
CTDdecreases(reaction)CASP3
D012402
CTDincreases(cleavage)CASP3
D012402
CTDincreases(activity)CASP3
D012402
CTDincreases(activity)CASP3
D012402
CTDincreases(cleavage)CASP3
D012402
CTDincreases(cleavage)CASP3
D012402
CTDdecreases(reaction)CASP3
D012402
CTDincreases(cleavage)CASP3
D012402
CTDdecreases(reaction)CASP3
D012402
CTDincreases(activity)CASP3
D012402
CTDincreases(cleavage)CASP3
D012402
CTDdecreases(reaction)CASP7
D012402
CTDincreases(activity)CASP7
D012402
CTDdecreases(reaction)CASP9
D012402
CTDincreases(activity)CASP9
D012402
CTDdecreases(reaction)CASP9
D012402
CTDincreases(cleavage)CASP9
D012402
CTDdecreases(reaction)CASP9
D012402
CTDincreases(cleavage)CASP9
D012402
CTDincreases(cleavage)CASP9
D012402
CTDdecreases(reaction)CASP9
D012402
CTDincreases(cleavage)CASP9
D012402
CTDdecreases(reaction)CAT
D012402
CTDincreases(activity)CAT
D012402
CTDincreases(expression)CAT
D012402
CTDdecreases(reaction)CCND1
D012402
CTDincreases(expression)CCND1
D012402
CTDincreases(expression)CCNH
D012402
CTDincreases(expression)CD14
D012402
CTDdecreases(reaction)CD36
D012402
CTDincreases(abundance)CD36
D012402
CTDincreases(expression)CD36
D012402
CTDincreases(expression)CD38
D012402
CTDincreases(expression)CD38
D012402
CTDdecreases(expression)CDH1
D012402
CTDdecreases(reaction)CDH1
D012402
CTDdecreases(reaction)CDKN1A
D012402
CTDincreases(expression)CDKN1A
D012402
CTDincreases(expression)CDKN1A
D012402
CTDincreases(expression)CHEK1
D012402
CTDincreases(expression)CNOT7
D012402
CTDdecreases(reaction)CNTF
D012402
CTDincreases(activity)CNTF
D012402
CTDincreases(phosphorylation)CNTF
D012402
CTDdecreases(reaction)CNTF
D012402
CTDincreases(phosphorylation)CNTF
D012402
CTDincreases(reaction)CNTF
D012402
CTDdecreases(activity)CNTF
D012402
CTDdecreases(activity)CNTF
D012402
CTDaffects(cotreatment)COL6A3
D012402
CTDdecreases(reaction)COL6A3
D012402
CTDincreases(response to substance)COL6A3
D012402
CTDincreases(reaction)COL6A3
D012402
CTDaffects(cotreatment)COX1
D012402
CTDincreases(expression)COX1
D012402
CTDincreases(expression)COX4I1
D012402
CTDincreases(expression)COX5A
D012402
CTDincreases(expression)COX5B
D012402
CTDincreases(expression)COX7A2
D012402
CTDincreases(expression)COX7B
D012402
CTDdecreases(expression)CP
D012402
CTDincreases(degradation)CP
D012402
CTDdecreases(reaction)CXCL8
D012402
CTDincreases(expression)CXCL8
D012402
CTDdecreases(activity)CYP19A1
D012402
CTDincreases(expression)DDIT3
D012402
CTDaffects(response to substance)DFFB
D012402
CTDdecreases(response to substance)DPP3
D012402
CTDdecreases(reaction)EDN1
D012402
CTDincreases(expression)EDN1
D012402
CTDincreases(phosphorylation)EIF2AK3
D012402
CTDincreases(expression)EIF2S1
D012402
CTDincreases(phosphorylation)EIF2S1
D012402
CTDincreases(expression)EXO1
D012402
CTDincreases(expression)FANCA
D012402
CTDincreases(expression)FANCC
D012402
CTDincreases(expression)FANCD2
D012402
CTDincreases(expression)FANCE
D012402
CTDincreases(expression)FANCF
D012402
CTDincreases(expression)FANCG
D012402
CTDdecreases(expression)FAS
D012402
CTDdecreases(reaction)FN1
D012402
CTDincreases(secretion)FN1
D012402
CTDdecreases(expression)FN1
D012402
CTDdecreases(secretion)FN1
D012402
CTDdecreases(reaction)FOS
D012402
CTDincreases(expression)FOS
D012402
CTDincreases(expression)FTH1
D012402
CTDincreases(activity)GPX1
D012402
CTDincreases(expression)GPX1
D012402
CTDaffects(expression)HAX1
D012402
CTDdecreases(degradation)HIF1A
D012402
CTDdecreases(reaction)HIF1A
D012402
CTDdecreases(reaction)HIF1A
D012402
CTDincreases(activity)HIF1A
D012402
CTDdecreases(reaction)HIF1A
D012402
CTDincreases(expression)HIF1A
D012402
CTDdecreases(expression)HIF1A
D012402
CTDaffects(cotreatment)HMGCR
D012402
CTDdecreases(expression)HMGCR
D012402
CTDdecreases(reaction)HMOX1
D012402
CTDincreases(expression)HMOX1
D012402
CTDdecreases(expression)HNRNPH1
D012402
CTDaffects(splicing)HNRNPH1
D012402
CTDdecreases(expression)HSPA9
D012402
CTDdecreases(expression)HTRA2
D012402
CTDincreases(expression)HTRA2
D012402
CTDincreases(expression)HUS1
D012402
CTDdecreases(reaction)ICAM1
D012402
CTDincreases(expression)ICAM1
D012402
CTDdecreases(expression)IDH3A
D012402
CTDincreases(expression)IDH3A
D012402
CTDaffects(localization)IFNG
D012402
CTDdecreases(reaction)IFNG
D012402
CTDincreases(activity)IFNG
D012402
CTDincreases(phosphorylation)IFNG
D012402
CTDdecreases(activity)IFNG
D012402
CTDdecreases(reaction)IGF1
D012402
CTDincreases(activity)IGF1
D012402
CTDdecreases(reaction)IL6
D012402
CTDincreases(expression)IL6
D012402
CTDdecreases(activity)IL6
D012402
CTDdecreases(reaction)JAK1
D012402
CTDincreases(activity)JAK1
D012402
CTDincreases(phosphorylation)JAK1
D012402
CTDdecreases(phosphorylation)JAK1
D012402
CTDdecreases(reaction)JAK2
D012402
CTDincreases(activity)JAK2
D012402
CTDincreases(phosphorylation)JAK2
D012402
CTDdecreases(reaction)JAK2
D012402
CTDincreases(phosphorylation)JAK2
D012402
CTDincreases(reaction)JAK2
D012402
CTDdecreases(phosphorylation)JAK2
D012402
CTDdecreases(reaction)JUN
D012402
CTDincreases(phosphorylation)JUN
D012402
CTDincreases(activity)JUN
D012402
CTDincreases(phosphorylation)JUN
D012402
CTDincreases(phosphorylation)JUN
D012402
CTDdecreases(reaction)KCNA5
D012402
CTDincreases(expression)KCNA5
D012402
CTDdecreases(activity)KCNH2
D012402
CTDdecreases(reaction)LEP
D012402
CTDincreases(chemical synthesis)LEP
D012402
CTDdecreases(response to substance)LEP
D012402
CTDincreases(response to substance)LRRK2
D012402
CTDdecreases(response to substance)LRRK2
D012402
CTDincreases(response to substance)LRRK2
D012402
CTDdecreases(reaction)LRRK2
D012402
CTDdecreases(reaction)MAPK1
D012402
CTDincreases(phosphorylation)MAPK1
D012402
CTDdecreases(reaction)MAPK1
D012402
CTDincreases(activity)MAPK1
D012402
CTDincreases(phosphorylation)MAPK1
D012402
CTDdecreases(activity)MAPK1
D012402
CTDdecreases(phosphorylation)MAPK1
D012402
CTDdecreases(reaction)MAPK14
D012402
CTDincreases(phosphorylation)MAPK14
D012402
CTDincreases(activity)MAPK14
D012402
CTDincreases(phosphorylation)MAPK14
D012402
CTDincreases(phosphorylation)MAPK14
D012402
CTDdecreases(reaction)MAPK3
D012402
CTDincreases(phosphorylation)MAPK3
D012402
CTDdecreases(reaction)MAPK3
D012402
CTDincreases(activity)MAPK3
D012402
CTDincreases(phosphorylation)MAPK3
D012402
CTDdecreases(activity)MAPK3
D012402
CTDdecreases(phosphorylation)MAPK3
D012402
CTDincreases(activity)MAPK8
D012402
CTDincreases(activity)MAPK8
D012402
CTDincreases(phosphorylation)MAPK8
D012402
CTDdecreases(reaction)MAPK8
D012402
CTDdecreases(expression)MAPT
D012402
CTDincreases(expression)MEF2D
D012402
CTDincreases(expression)MIR195
D012402
CTDincreases(abundance)MMP2
D012402
CTDincreases(activity)MMP2
D012402
CTDincreases(expression)MRE11A
D012402
CTDincreases(expression)MRPS9
D012402
CTDdecreases(reaction)MSR1
D012402
CTDincreases(expression)MSR1
D012402
CTDdecreases(reaction)MT1B
D012402
CTDincreases(activity)MT1B
D012402
CTDdecreases(reaction)MT2A
D012402
CTDincreases(abundance)MT2A
D012402
CTDincreases(activity)MT2A
D012402
CTDincreases(expression)MT2A
D012402
CTDincreases(expression)MUS81
D012402
CTDdecreases(activity)NAMPT
D012402
CTDdecreases(response to substance)ND6
D012402
CTDincreases(expression)NDUFA10
D012402
CTDincreases(expression)NDUFA3
D012402
CTDincreases(expression)NDUFA4
D012402
CTDincreases(expression)NDUFA6
D012402
CTDincreases(expression)NDUFA9
D012402
CTDincreases(expression)NDUFB1
D012402
CTDaffects(splicing)NDUFB11
D012402
CTDdecreases(expression)NDUFB11
D012402
CTDincreases(expression)NDUFB2
D012402
CTDincreases(expression)NDUFB3
D012402
CTDincreases(expression)NDUFB4
D012402
CTDincreases(expression)NDUFB5
D012402
CTDincreases(expression)NDUFB6
D012402
CTDincreases(expression)NDUFB7
D012402
CTDincreases(expression)NDUFB8
D012402
CTDincreases(expression)NDUFS4
D012402
CTDincreases(expression)NDUFS6
D012402
CTDincreases(expression)NDUFS8
D012402
CTDdecreases(reaction)NFAT5
D012402
CTDincreases(activity)NFAT5
D012402
CTDdecreases(reaction)NFATC1
D012402
CTDincreases(expression)NFATC1
D012402
CTDdecreases(response to substance)NFE2L2
D012402
CTDaffects(cotreatment)NFE2L2
D012402
CTDincreases(expression)NFE2L2
D012402
CTDaffects(binding)NFKB1
D012402
CTDdecreases(reaction)NFKB1
D012402
CTDincreases(reaction)NFKB1
D012402
CTDdecreases(reaction)NOS3
D012402
CTDincreases(activity)NOS3
D012402
CTDincreases(phosphorylation)NOS3
D012402
CTDaffects(cotreatment)NPC1L1
D012402
CTDincreases(expression)NPC1L1
D012402
CTDdecreases(reaction)NPPB
D012402
CTDincreases(secretion)NPPB
D012402
CTDaffects(cotreatment)NQO1
D012402
CTDincreases(expression)NQO1
D012402
CTDincreases(expression)NUDT1
D012402
CTDdecreases(reaction)ODC1
D012402
CTDincreases(activity)ODC1
D012402
CTDincreases(expression)OPA1
D012402
CTDdecreases(reaction)OSCAR
D012402
CTDincreases(expression)OSCAR
D012402
CTDincreases(response to substance)PARK2
D012402
CTDaffects(response to substance)PARK2
D012402
CTDdecreases(reaction)PARK2
D012402
CTDincreases(response to substance)PARK2
D012402
CTDdecreases(response to substance)PARK2
D012402
CTDdecreases(reaction)PARK7
D012402
CTDincreases(expression)PARK7
D012402
CTDdecreases(reaction)PARK7
D012402
CTDincreases(expression)PARK7
D012402
CTDaffects(localization)PARK7
D012402
CTDdecreases(reaction)PARK7
D012402
CTDaffects(response to substance)PARK7
D012402
CTDdecreases(response to substance)PARK7
D012402
CTDaffects(localization)PARK7
D012402
CTDincreases(expression)PARK7
D012402
CTDdecreases(reaction)PARP1
D012402
CTDincreases(cleavage)PARP1
D012402
CTDdecreases(reaction)PARP1
D012402
CTDincreases(cleavage)PARP1
D012402
CTDaffects(reaction)PARP1
D012402
CTDdecreases(reaction)PARP1
D012402
CTDincreases(cleavage)PARP1
D012402
CTDdecreases(reaction)PARP1
D012402
CTDincreases(cleavage)PARP1
D012402
CTDincreases(cleavage)PARP1
D012402
CTDdecreases(reaction)PARP1
D012402
CTDincreases(cleavage)PARP1
D012402
CTDincreases(expression)PDHB
D012402
CTDaffects(cotreatment)PDK1
D012402
CTDdecreases(reaction)PDK1
D012402
CTDincreases(expression)PDK1
D012402
CTDaffects(response to substance)PINK1
D012402
CTDdecreases(response to substance)PINK1
D012402
CTDincreases(expression)POLA1
D012402
CTDincreases(expression)POLE2
D012402
CTDaffects(cotreatment)PPARG
D012402
CTDincreases(expression)PPARG
D012402
CTDaffects(cotreatment)PPARGC1A
D012402
CTDincreases(expression)PPARGC1A
D012402
CTDincreases(expression)PPID
D012402
CTDincreases(expression)PRKAA1
D012402
CTDincreases(expression)PROM1
D012402
CTDincreases(expression)RAD1
D012402
CTDincreases(expression)RAD17
D012402
CTDincreases(expression)RAD18
D012402
CTDincreases(expression)RAD50
D012402
CTDincreases(expression)RAD51
D012402
CTDincreases(expression)RAD51AP1
D012402
CTDincreases(expression)RAD54B
D012402
CTDincreases(expression)RAD9A
D012402
CTDaffects(binding)RELA
D012402
CTDdecreases(reaction)RELA
D012402
CTDincreases(reaction)RELA
D012402
CTDincreases(expression)RFC4
D012402
CTDincreases(expression)RFC5
D012402
CTDaffects(cotreatment)SDHA
D012402
CTDincreases(expression)SDHA
D012402
CTDdecreases(reaction)SLC2A1
D012402
CTDincreases(expression)SLC2A1
D012402
CTDdecreases(reaction)SLC2A1
D012402
CTDincreases(activity)SLC2A1
D012402
CTDdecreases(response to substance)SLC2A1
D012402
CTDdecreases(reaction)SLC6A12
D012402
CTDincreases(expression)SLC6A12
D012402
CTDincreases(response to substance)SLC6A3
D012402
CTDincreases(expression)SMN1
D012402
CTDdecreases(reaction)SNAI1
D012402
CTDincreases(expression)SNAI1
D012402
CTDdecreases(reaction)SNCA
D012402
CTDincreases(response to substance)SNCA
D012402
CTDincreases(reaction)SNCA
D012402
CTDaffects(cotreatment)SNCA
D012402
CTDdecreases(reaction)SNCA
D012402
CTDincreases(expression)SNCA
D012402
CTDdecreases(reaction)SNCA
D012402
CTDincreases(expression)SNCA
D012402
CTDaffects(localization)SNCA
D012402
CTDaffects(binding)SNCA
D012402
CTDincreases(reaction)SNCA
D012402
CTDaffects(binding)SNCA
D012402
CTDincreases(reaction)SNCA
D012402
CTDincreases(expression)SNCA
D012402
CTDincreases(expression)SNCA
D012402
CTDincreases(response to substance)SNCA
D012402
CTDincreases(response to substance)SNCA
D012402
CTDdecreases(response to substance)SNCA
D012402
CTDincreases(response to substance)SNCA
D012402
CTDaffects(binding)SNCA
D012402
CTDaffects(cotreatment)SNCA
D012402
CTDincreases(reaction)SNCA
D012402
CTDaffects(cotreatment)SOD1
D012402
CTDincreases(expression)SOD1
D012402
CTDdecreases(reaction)SOD2
D012402
CTDincreases(activity)SOD2
D012402
CTDincreases(expression)SOD2
D012402
CTDincreases(abundance)SOD2
D012402
CTDincreases(expression)SOD2
D012402
CTDdecreases(reaction)SOD2
D012402
CTDincreases(expression)SOD2
D012402
CTDdecreases(response to substance)SOD2
D012402
CTDdecreases(response to substance)SQSTM1
D012402
CTDincreases(expression)SREBF1
D012402
CTDincreases(expression)SSBP1
D012402
CTDdecreases(reaction)STAT1
D012402
CTDincreases(activity)STAT1
D012402
CTDincreases(phosphorylation)STAT1
D012402
CTDdecreases(reaction)STAT1
D012402
CTDincreases(phosphorylation)STAT1
D012402
CTDaffects(localization)STAT1
D012402
CTDincreases(reaction)STAT1
D012402
CTDdecreases(reaction)STAT3
D012402
CTDincreases(activity)STAT3
D012402
CTDincreases(phosphorylation)STAT3
D012402
CTDdecreases(reaction)STAT3
D012402
CTDincreases(phosphorylation)STAT3
D012402
CTDincreases(reaction)STAT3
D012402
CTDaffects(cotreatment)TFAM
D012402
CTDincreases(expression)TFAM
D012402
CTDincreases(expression)TK2
D012402
CTDdecreases(reaction)TNF
D012402
CTDincreases(abundance)TNF
D012402
CTDincreases(cleavage)TNF
D012402
CTDdecreases(expression)TNFRSF11B
D012402
CTDdecreases(secretion)TNFRSF11B
D012402
CTDdecreases(reaction)TNFSF11
D012402
CTDincreases(expression)TNFSF11
D012402
CTDaffects(localization)TP53
D012402
CTDincreases(expression)TP53
D012402
CTDincreases(phosphorylation)TP53
D012402
CTDincreases(expression)TP53
D012402
CTDincreases(oxidation)TXN2
D012402
CTDincreases(response to substance)TXN2
D012402
CTDincreases(expression)UBE2N
D012402
CTDincreases(expression)UQCRB
D012402
CTDincreases(expression)UQCRC1
D012402
CTDdecreases(reaction)VDAC1
D012402
CTDincreases(expression)VDAC1
D012402
CTDincreases(activity)VDR
D012402
CTDaffects(cotreatment)VEGFA
D012402
CTDdecreases(reaction)VEGFA
D012402
CTDincreases(expression)VEGFA
D012402
CTDdecreases(reaction)VEGFA
D012402
CTDincreases(expression)VEGFA
D012402
CTDdecreases(reaction)VEGFA
D012402
CTDincreases(expression)VEGFA
D012402
CTDdecreases(reaction)VEGFA
D012402
CTDincreases(expression)VEGFA
D012402
CTDdecreases(reaction)VEGFA
D012402
CTDincreases(secretion)VEGFA
D012402
CTDdecreases(activity)XDH
D012402
CTDaffects(binding)YWHAB
D012402
CTDincreases(reaction)YWHAB
D012402
CTDdecreases(response to substance)YWHAG
D012402
PubChem PotencyuM6.310CYP3A4-GI(Protien) :
PubChem PotencyuM0.052TDP1-GI(Protien) :
PubChem PotencyuM0.103TDP1-GI(Protien) :
PubChem NoneuMABCB1-GI(Protien) :
PubChem Potency-Replicate_1uM0.010AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.025AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.188AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.279AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.756AR-GI(Protien) :
PubChem PotencyuM35.481CBX1-GI(Protien) :
PubChem Potency-Replicate_1uM14.960CYP19A1-GI(Protien) :
PubChem Potency-Replicate_1uM34.376CYP19A1-GI(Protien) :
PubChem Potency-Replicate_1uM34.831CYP19A1-GI(Protien) :
PubChem NoneuMCYP1A2-GI(Protien) :
PubChem PotencyuM1.000CYP2C19-GI(Protien) :
PubChem PotencyuM15.849CYP3A4-GI(Protien) :
PubChem Potency-Replicate_1uM0.015ESR1-GI(Protien) :
PubChem ER Potency (uM)uM0.031ESR1-GI(Protien) :
PubChem ER Potency (uM)uM0.031ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM0.039ESR1-GI(Protien) :
PubChem ER Potency (uM)uM0.144ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM0.150ESR1-GI(Protien) :
PubChem Ratio Potency (uM)uM40.417ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM48.966ESR1-GI(Protien) :
PubChem PotencyuM11.220GLS-GI(Protien) :
PubChem PotencyuM0.755GMNN-GI(Protien) :
PubChem PotencyuM0.920GMNN-GI(Protien) :
PubChem PotencyuM1.066GMNN-GI(Protien) :
PubChem PotencyuM1.413GMNN-GI(Protien) :
PubChem PotencyuM3.933GMNN-GI(Protien) :
PubChem PotencyuM0.046MTOR-GI(Protien) :
PubChem PotencyuM0.059MTOR-GI(Protien) :
PubChem Potency-Replicate_1uM0.008NFE2L2-GI(Protien) :
PubChem Ratio Potency (uM)uM0.018NFE2L2-GI(Protien) :
PubChem Ratio Potency (uM)uM0.020NFE2L2-GI(Protien) :
PubChem Ratio Potency (uM)uM0.046NFE2L2-GI(Protien) :
PubChem Potency-Replicate_1uM0.750NR1H4-GI(Protien) :
PubChem NoneuMNR1H4-GI(Protien) :
PubChem Potency-Replicate_1uM4.897PPARD-GI(Protien) :
PubChem Potency-Replicate_1uM13.332PPARG-GI(Protien) :
PubChem PotencyuM44.668PPARG-GI(Protien) :
PubChem NoneuMPPARG-GI(Protien) :
PubChem PotencyuM19.953RXRA-GI(Protien) :
PubChem PotencyuM0.150TDP1-GI(Protien) :
PubChem PotencyuM0.188TDP1-GI(Protien) :
PubChem PotencyuM0.237TDP1-GI(Protien) :
PubChem PotencyuM0.237TDP1-GI(Protien) :
ChEMBLPotencynM35481.300CBX1
-Target : CHEMBL1741193
ChEMBLActivity-CDK1
-Target : CHEMBL308
ChEMBLActivity-CDK1
-Target : CHEMBL308
ChEMBLActivity-CFL1
-Target : CHEMBL1075129
ChEMBLPotencynM1000.000CYP2C19
-Target : CHEMBL3622
ChEMBLPotencynM15848.900CYP3A4
-Target : CHEMBL340
ChEMBLPotencynM1412.500GMNN
-Target : CHEMBL1293278
ChEMBLPotencynM1065.900GMNN
-Target : CHEMBL1293278
ChEMBLPotencynM754.600GMNN
-Target : CHEMBL1293278
ChEMBLPotencynM920.000GMNN
-Target : CHEMBL1293278
ChEMBLActivity-JUN
-Target : CHEMBL4977
ChEMBLPotencynM58.500MTOR
-Target : CHEMBL2842
ChEMBLInhibition-MTOR
-Target : CHEMBL2842
ChEMBLActivity-MTOR
-Target : CHEMBL2842
ChEMBLActivity-MTOR
-Target : CHEMBL2842
ChEMBLActivity-MTOR
-Target : CHEMBL2842
ChEMBLPotencynM46.500MTOR
-Target : CHEMBL2842
ChEMBLActivity-TP53
-Target : CHEMBL4096
Download gene sets gmt, text, Detailed text
Contact us
Tan Lab , Mail Stop 8117
12801 East 17th Avenue
Division of Medical Oncology , Department of Medicine
University of Colorado School of Medicine
Aurora, CO 80045, USA

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