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Gene Set: D4 : CTD - Medroxyprogesterone Acetate


Collection D4 : CTD
Chemical Name Medroxyprogesterone Acetate ( From PubChem : MEDROXYPROGESTERONE ACETATE )
FDA NPC WHO Indian Australia China Traditional
Herbal
Clinical
Trail
ApprovedNotApprovedApprovedNotApprovedApprovedNot
Molecular
Weight
Hydrogen Bond
Donor Count
Hydrogen Bond
Acceptor Count
cLogP Lipinski Rule
386.524 g/mol 0 4 4.6552 True
Structure
InChI InChI=1S/C24H34O4/c1-14-12-18-19(22(4)9-6-17(27)13-21(14)22)7-10-23(5)20(18)8-11-24(23,15(2)25)28-16(3)26/h13-14,18-20H,6-12H2,1-5H3/t14-,18+,19-,20-,22+,23-,24-/m0/s1
InChIKey PSGAAPLEWMOORI-PEINSRQWSA-N
Links

Gene (389 / 759)


⊖ Less

Source Type Unit Value Gene PMID Assay Other
CTDdecreases(activity)ABCB11
D017258
CTDincreases(expression)ACKR1
D017258
CTDdecreases(expression)ACPP
D017258
CTDincreases(expression)ACSL1
D017258
CTDaffects(cotreatment)ADAMTS1
D017258
CTDdecreases(expression)ADAMTS1
D017258
CTDincreases(expression)ADORA3
D017258
CTDincreases(expression)AIF1
D017258
CTDaffects(cotreatment)AK5
D017258
CTDincreases(expression)AK5
D017258
CTDdecreases(activity)AKR1C1
D017258
CTDdecreases(expression)AKR1C1
D017258
CTDincreases(expression)AKR1C1
D017258
CTDdecreases(activity)AKR1C2
D017258
CTDincreases(metabolic processing)AKR1C2
D011372
CTDaffects(cotreatment)AKR1C3
D017258
CTDdecreases(reaction)AKR1C3
D017258
CTDincreases(reduction)AKR1C3
D017258
CTDdecreases(reaction)AKR1C3
D017258
CTDincreases(abundance)AKR1C3
D017258
CTDincreases(metabolic processing)AKR1C3
D017258
CTDdecreases(activity)AKR1C3
D017258
CTDaffects(cotreatment)AKR1C4
D017258
CTDaffects(response to substance)AKR1C4
D017258
CTDdecreases(activity)AKR1C4
D017258
CTDincreases(expression)ALCAM
D017258
CTDincreases(expression)ALOX5AP
D017258
CTDaffects(cotreatment)ANTXR1
D017258
CTDincreases(expression)ANTXR1
D017258
CTDaffects(cotreatment)ANXA2
D017258
CTDdecreases(expression)ANXA2
D017258
CTDaffects(cotreatment)ANXA2P3
D017258
CTDdecreases(expression)ANXA2P3
D017258
CTDincreases(expression)APOD
D017258
CTDincreases(expression)AQP3
D017258
CTDaffects(binding)AR
D017258
CTDincreases(activity)AR
D017258
CTDincreases(expression)ARHGEF19
D017258
CTDaffects(cotreatment)ARHGEF2
D017258
CTDdecreases(expression)ARHGEF2
D017258
CTDaffects(cotreatment)ATP11A
D017258
CTDincreases(expression)ATP11A
D017258
CTDincreases(expression)ATP1A1
D017258
CTDaffects(cotreatment)ATP2B1
D017258
CTDdecreases(expression)ATP2B1
D017258
CTDdecreases(expression)ATP2B4
D017258
CTDaffects(cotreatment)ATP6V0C
D017258
CTDincreases(expression)ATP6V0C
D017258
CTDincreases(expression)AZGP1
D017258
CTDaffects(cotreatment)BAX
D017258
CTDincreases(expression)BAX
D017258
CTDaffects(cotreatment)BCAT1
D017258
CTDdecreases(expression)BCAT1
D017258
CTDaffects(cotreatment)BCKDK
D017258
CTDincreases(expression)BCKDK
D017258
CTDaffects(cotreatment)BCL2L11
D017258
CTDincreases(expression)BCL2L11
D017258
CTDaffects(cotreatment)BCL2L13
D017258
CTDincreases(expression)BCL2L13
D017258
CTDdecreases(expression)BDKRB1
D017258
CTDaffects(cotreatment)BET1L
D017258
CTDincreases(expression)BET1L
D017258
CTDaffects(cotreatment)BICD1
D017258
CTDdecreases(expression)BICD1
D017258
CTDaffects(cotreatment)BSND
D017258
CTDincreases(expression)BSND
D017258
CTDincreases(expression)C10ORF10
D017258
CTDdecreases(expression)C15ORF48
D017258
CTDincreases(expression)C1ORF162
D017258
CTDincreases(expression)C1QA
D017258
CTDincreases(expression)C1QB
D017258
CTDincreases(expression)C1QC
D017258
CTDaffects(cotreatment)C1R
D017258
CTDincreases(expression)C1R
D017258
CTDdecreases(expression)C2CD4B
D017258
CTDincreases(expression)CA2
D017258
CTDincreases(expression)CA8
D017258
CTDaffects(cotreatment)CALM1
D017258
CTDdecreases(expression)CALM1
D017258
CTDaffects(cotreatment)CAPN2
D017258
CTDdecreases(expression)CAPN2
D017258
CTDaffects(cotreatment)CAST
D017258
CTDincreases(expression)CAST
D017258
CTDaffects(cotreatment)CAT
D017258
CTDincreases(expression)CAT
D017258
CTDaffects(cotreatment)CAV2
D017258
CTDdecreases(expression)CAV2
D017258
CTDincreases(expression)CCL23
D017258
CTDaffects(cotreatment)CCNB1
D017258
CTDincreases(expression)CCNB1
D017258
CTDaffects(cotreatment)CCND1
D017258
CTDaffects(expression)CCND1
D017258
CTDdecreases(expression)CCND1
D017258
CTDincreases(expression)CCND1
D011372
CTDincreases(expression)CD163
D017258
CTDaffects(cotreatment)CD40LG
D017258
CTDdecreases(activity)CD40LG
D017258
CTDaffects(cotreatment)CDC42BPA
D017258
CTDdecreases(expression)CDC42BPA
D017258
CTDincreases(activity)CDK2
D011372
CTDincreases(expression)CDK2
D011372
CTDaffects(cotreatment)CDKN1A
D017258
CTDincreases(expression)CDKN1A
D017258
CTDaffects(cotreatment)CDKN1A
D017258
CTDincreases(expression)CDKN1A
D017258
CTDincreases(expression)CDKN1B
D017258
CTDincreases(reaction)CDKN1B
D017258
CTDaffects(cotreatment)CDKN1B
D017258
CTDdecreases(reaction)CDKN1B
D017258
CTDaffects(cotreatment)CEBPZ
D017258
CTDdecreases(expression)CEBPZ
D017258
CTDaffects(cotreatment)CFLAR
D017258
CTDincreases(expression)CFLAR
D017258
CTDdecreases(expression)CILP
D017258
CTDincreases(expression)CLDN5
D017258
CTDaffects(cotreatment)CNGB1
D017258
CTDincreases(expression)CNGB1
D017258
CTDincreases(expression)CNR1
D017258
CTDaffects(cotreatment)COL6A2
D017258
CTDdecreases(expression)COL6A2
D017258
CTDaffects(cotreatment)COL6A3
D017258
CTDdecreases(expression)COL6A3
D017258
CTDaffects(cotreatment)COX6A2
D017258
CTDincreases(expression)COX6A2
D017258
CTDaffects(cotreatment)CPLX1
D017258
CTDincreases(expression)CPLX1
D017258
CTDaffects(binding)CREBBP
D017258
CTDincreases(reaction)CREBBP
D017258
CTDaffects(cotreatment)CREM
D017258
CTDdecreases(expression)CREM
D017258
CTDaffects(cotreatment)CRP
D017258
CTDincreases(expression)CRP
D017258
CTDaffects(cotreatment)CTGF
D017258
CTDincreases(expression)CTGF
D017258
CTDaffects(cotreatment)CTPS2
D017258
CTDdecreases(expression)CTPS2
D017258
CTDincreases(expression)CTSD
D017258
CTDaffects(cotreatment)CYB5D1
D017258
CTDincreases(expression)CYB5D1
D017258
CTDdecreases(reaction)CYP1A1
D017258
CTDincreases(expression)CYP1A1
D017258
CTDincreases(expression)CYP1A1
D017258
CTDaffects(cotreatment)CYP1B1
D017258
CTDaffects(response to substance)CYP1B1
D017258
CTDdecreases(expression)CYP27B1
D017258
CTDincreases(expression)CYP3A4
D017258
CTDaffects(cotreatment)DCN
D017258
CTDincreases(expression)DCN
D017258
CTDincreases(reaction)DCN
D017258
CTDaffects(cotreatment)DDX27
D017258
CTDincreases(expression)DDX27
D017258
CTDaffects(cotreatment)DES
D017258
CTDincreases(expression)DES
D017258
CTDaffects(cotreatment)DHX9
D017258
CTDdecreases(expression)DHX9
D017258
CTDaffects(cotreatment)DIO2
D017258
CTDdecreases(expression)DIO2
D017258
CTDdecreases(expression)DIO2
D017258
CTDincreases(expression)DKK1
D017258
CTDincreases(expression)DLG5
D017258
CTDincreases(expression)DNER
D017258
CTDaffects(cotreatment)DTYMK
D017258
CTDdecreases(expression)DTYMK
D017258
CTDincreases(expression)DUSP23
D017258
CTDaffects(cotreatment)EDA
D017258
CTDincreases(expression)EDA
D017258
CTDaffects(cotreatment)EEF1A1
D017258
CTDdecreases(expression)EEF1A1
D017258
CTDaffects(cotreatment)EFEMP1
D017258
CTDincreases(expression)EFEMP1
D017258
CTDincreases(expression)EFHD1
D017258
CTDaffects(cotreatment)EGR2
D017258
CTDincreases(expression)EGR2
D017258
CTDaffects(cotreatment)EIF3LP3
D017258
CTDdecreases(expression)EIF3LP3
D017258
CTDincreases(expression)ELF3
D017258
CTDincreases(expression)ENPP2
D017258
CTDaffects(cotreatment)EPB41L4A
D017258
CTDincreases(expression)EPB41L4A
D017258
CTDaffects(cotreatment)EPHA3
D017258
CTDincreases(expression)EPHA3
D017258
CTDincreases(expression)EPHX1
D017258
CTDincreases(reaction)EPHX1
D017258
CTDincreases(expression)ESR1
D017258
CTDincreases(reaction)ESR1
D017258
CTDdecreases(expression)ESR1
D017258
CTDaffects(cotreatment)EYA1
D017258
CTDdecreases(expression)EYA1
D017258
CTDaffects(cotreatment)EZH2
D017258
CTDdecreases(expression)EZH2
D017258
CTDdecreases(reaction)EZH2
D017258
CTDincreases(expression)EZH2
D017258
CTDincreases(expression)F13A1
D017258
CTDincreases(expression)F2
D017258
CTDincreases(reaction)F2
D017258
CTDincreases(expression)F2
D017258
CTDincreases(expression)F2
D011372
CTDincreases(expression)F2R
D017258
CTDincreases(expression)F3
D017258
CTDincreases(reaction)F3
D017258
CTDincreases(expression)F3
D017258
CTDdecreases(expression)F7
D017258
CTDdecreases(reaction)F7
D011372
CTDincreases(activity)F7
D011372
CTDincreases(expression)F7
D011372
CTDincreases(expression)F9
D017258
CTDaffects(cotreatment)FADS2
D017258
CTDdecreases(expression)FADS2
D017258
CTDincreases(expression)FAM107A
D017258
CTDincreases(expression)FAM84B
D017258
CTDincreases(expression)FAS
D017258
CTDaffects(cotreatment)FASLG
D017258
CTDincreases(expression)FASLG
D017258
CTDincreases(expression)FBLN1
D017258
CTDdecreases(reaction)FBLN1
D017258
CTDaffects(cotreatment)FBXO11
D017258
CTDincreases(expression)FBXO11
D017258
CTDaffects(cotreatment)FBXW5
D017258
CTDincreases(expression)FBXW5
D017258
CTDincreases(expression)FCGBP
D017258
CTDaffects(cotreatment)FGD1
D017258
CTDdecreases(expression)FGD1
D017258
CTDdecreases(expression)FGF7
D017258
CTDincreases(expression)FIBIN
D017258
CTDaffects(cotreatment)FILIP1L
D017258
CTDdecreases(expression)FILIP1L
D017258
CTDincreases(expression)FKBP5
D017258
CTDaffects(cotreatment)FN1
D017258
CTDdecreases(expression)FN1
D017258
CTDaffects(cotreatment)FN1
D017258
CTDincreases(expression)FN1
D017258
CTDincreases(expression)FOLR2
D017258
CTDaffects(cotreatment)FOXO1
D017258
CTDincreases(expression)FOXO1
D017258
CTDaffects(cotreatment)FOXO1
D017258
CTDaffects(reaction)FOXO1
D017258
CTDdecreases(expression)FOXO1
D017258
CTDincreases(expression)FOXO1
D017258
CTDincreases(secretion)FOXO1
D017258
CTDdecreases(reaction)FOXO1
D017258
CTDaffects(cotreatment)FOXO3
D017258
CTDaffects(reaction)FOXO3
D017258
CTDdecreases(expression)FOXO3
D017258
CTDdecreases(reaction)FOXO3
D017258
CTDincreases(expression)FOXO3
D017258
CTDincreases(expression)FPR1
D017258
CTDaffects(cotreatment)FSCN2
D017258
CTDincreases(expression)FSCN2
D017258
CTDaffects(cotreatment)FSHB
D017258
CTDdecreases(expression)FSHB
D017258
CTDincreases(expression)FXYD3
D017258
CTDaffects(cotreatment)GADD45A
D017258
CTDincreases(expression)GADD45A
D017258
CTDaffects(cotreatment)GARS
D017258
CTDdecreases(expression)GARS
D017258
CTDaffects(cotreatment)GBE1
D017258
CTDincreases(expression)GBE1
D017258
CTDaffects(cotreatment)GBP2
D017258
CTDdecreases(expression)GBP2
D017258
CTDaffects(cotreatment)GCNT2
D017258
CTDdecreases(expression)GCNT2
D017258
CTDdecreases(expression)GDF10
D017258
CTDaffects(cotreatment)GIPC1
D017258
CTDincreases(expression)GIPC1
D017258
CTDdecreases(expression)GJA1
D017258
CTDincreases(expression)GLRX
D017258
CTDaffects(cotreatment)GPKOW
D017258
CTDincreases(expression)GPKOW
D017258
CTDaffects(cotreatment)GPNMB
D017258
CTDdecreases(expression)GPNMB
D017258
CTDincreases(expression)GPR34
D017258
CTDdecreases(expression)GPR83
D017258
CTDincreases(expression)GPX3
D017258
CTDincreases(expression)GSN
D017258
CTDincreases(expression)GSTM3
D017258
CTDincreases(expression)HAVCR2
D017258
CTDdecreases(expression)HBEGF
D017258
CTDaffects(cotreatment)HOXA1
D017258
CTDdecreases(expression)HOXA1
D017258
CTDdecreases(reaction)HOXA1
D017258
CTDaffects(cotreatment)HOXA10
D017258
CTDincreases(expression)HOXA10
D017258
CTDincreases(expression)HOXA10
D017258
CTDdecreases(reaction)HOXA10
D017258
CTDincreases(expression)HOXA11
D017258
CTDaffects(cotreatment)HSD11B1
D017258
CTDincreases(activity)HSD11B1
D017258
CTDincreases(expression)HSD11B1
D017258
CTDaffects(cotreatment)HSD11B2
D017258
CTDincreases(expression)HSD11B2
D017258
CTDdecreases(expression)HSD17B2
D017258
CTDaffects(cotreatment)HTR1A
D017258
CTDincreases(expression)HTR1A
D017258
CTDdecreases(reaction)ICAM1
D017258
CTDincreases(expression)ICAM1
D017258
CTDincreases(expression)IDH1
D017258
CTDaffects(cotreatment)IFNG
D017258
CTDdecreases(secretion)IFNG
D017258
CTDaffects(cotreatment)IFRD2
D017258
CTDincreases(expression)IFRD2
D017258
CTDaffects(cotreatment)IGFBP1
D017258
CTDincreases(expression)IGFBP1
D017258
CTDaffects(cotreatment)IGFBP1
D017258
CTDdecreases(reaction)IGFBP1
D017258
CTDincreases(expression)IGFBP1
D017258
CTDincreases(reaction)IGFBP1
D017258
CTDaffects(cotreatment)IGFBP1
D017258
CTDincreases(expression)IGFBP1
D017258
CTDaffects(cotreatment)IGFBP1
D017258
CTDincreases(expression)IGFBP1
D017258
CTDdecreases(expression)IGFBP1
D017258
CTDincreases(reaction)IGFBP1
D017258
CTDdecreases(reaction)IGFBP1
D017258
CTDaffects(cotreatment)IGFBP1
D017258
CTDaffects(reaction)IGFBP1
D017258
CTDincreases(secretion)IGFBP1
D017258
CTDincreases(expression)IGFBP1
D017258
CTDaffects(cotreatment)IGFBP3
D017258
CTDincreases(expression)IGFBP3
D017258
CTDaffects(cotreatment)IGFBP4
D017258
CTDincreases(expression)IGFBP4
D017258
CTDdecreases(expression)IGFBP5
D017258
CTDdecreases(expression)IL11
D017258
CTDaffects(cotreatment)IL12B
D017258
CTDincreases(expression)IL12B
D017258
CTDdecreases(expression)IL1B
D017258
CTDaffects(cotreatment)IL2
D017258
CTDdecreases(secretion)IL2
D017258
CTDaffects(cotreatment)IL23A
D017258
CTDdecreases(expression)IL23A
D017258
CTDdecreases(expression)IL24
D017258
CTDdecreases(expression)IL6
D017258
CTDaffects(cotreatment)IL6
D017258
CTDdecreases(expression)IL6
D017258
CTDaffects(cotreatment)INTS7
D017258
CTDincreases(expression)INTS7
D017258
CTDaffects(cotreatment)IRF9
D017258
CTDincreases(expression)IRF9
D017258
CTDincreases(expression)IRS2
D017258
CTDaffects(cotreatment)ISG20L2
D017258
CTDdecreases(expression)ISG20L2
D017258
CTDdecreases(expression)ITGA1
D017258
CTDdecreases(expression)ITGA11
D017258
CTDdecreases(expression)ITGA2
D017258
CTDaffects(cotreatment)ITGB1
D017258
CTDdecreases(expression)ITGB1
D017258
CTDdecreases(expression)ITGB5
D017258
CTDaffects(cotreatment)ITIH5
D017258
CTDdecreases(expression)ITIH5
D017258
CTDincreases(expression)KCNB1
D017258
CTDaffects(cotreatment)KCNC4
D017258
CTDdecreases(expression)KCNC4
D017258
CTDdecreases(expression)KDR
D017258
CTDincreases(expression)KLF4
D017258
CTDaffects(cotreatment)KRT8
D017258
CTDdecreases(expression)KRT8
D017258
CTDdecreases(reaction)KRT8
D017258
CTDdecreases(expression)LAMA4
D017258
CTDaffects(cotreatment)LAMB2
D017258
CTDincreases(expression)LAMB2
D017258
CTDaffects(cotreatment)LCN2
D017258
CTDdecreases(expression)LCN2
D017258
CTDaffects(cotreatment)LDHA
D017258
CTDincreases(expression)LDHA
D017258
CTDdecreases(expression)LEFTY2
D017258
CTDaffects(cotreatment)LGALS3
D017258
CTDdecreases(expression)LGALS3
D017258
CTDincreases(expression)LINC00312
D017258
CTDdecreases(expression)LOXL4
D017258
CTDaffects(cotreatment)LPAR3
D017258
CTDincreases(expression)LPAR3
D017258
CTDaffects(cotreatment)LPL
D011372
CTDincreases(expression)LPL
D011372
CTDaffects(cotreatment)LTBP1
D017258
CTDincreases(expression)LTBP1
D017258
CTDincreases(expression)LYVE1
D017258
CTDaffects(cotreatment)MAP1A
D017258
CTDdecreases(expression)MAP1A
D017258
CTDaffects(cotreatment)MAP4K4
D017258
CTDincreases(expression)MAP4K4
D017258
CTDdecreases(expression)MAP7
D017258
CTDincreases(expression)MARCO
D017258
CTDaffects(cotreatment)MGAT4B
D017258
CTDincreases(expression)MGAT4B
D017258
CTDincreases(expression)MGST1
D017258
CTDincreases(expression)MIR142
D017258
CTDincreases(expression)MIR146B
D017258
CTDdecreases(expression)MIR193B
D017258
CTDincreases(expression)MIR21
D017258
CTDdecreases(expression)MIR29C
D017258
CTDincreases(expression)MIR625
D017258
CTDdecreases(expression)MIR633
D017258
CTDdecreases(expression)MMP1
D017258
CTDaffects(cotreatment)MMP2
D017258
CTDincreases(expression)MMP2
D017258
CTDdecreases(expression)MMP9
D017258
CTDincreases(expression)MMRN1
D017258
CTDincreases(expression)MS4A6A
D017258
CTDincreases(expression)MT1G
D017258
CTDincreases(expression)MT1H
D017258
CTDincreases(expression)MT1L
D017258
CTDaffects(cotreatment)MTHFD2
D017258
CTDdecreases(expression)MTHFD2
D017258
CTDaffects(cotreatment)MTR
D017258
CTDdecreases(expression)MTR
D017258
CTDincreases(expression)MTSS1
D017258
CTDincreases(expression)MUC1
D017258
CTDaffects(cotreatment)MUC12
D017258
CTDdecreases(expression)MUC12
D017258
CTDdecreases(expression)MYB
D017258
CTDaffects(cotreatment)MYH9
D017258
CTDdecreases(expression)MYH9
D017258
CTDaffects(cotreatment)MYL12A
D017258
CTDdecreases(expression)MYL12A
D017258
CTDaffects(cotreatment)MYL12B
D017258
CTDdecreases(expression)MYL12B
D017258
CTDaffects(cotreatment)MYLK
D017258
CTDdecreases(expression)MYLK
D017258
CTDaffects(cotreatment)MYOF
D017258
CTDdecreases(expression)MYOF
D017258
CTDaffects(cotreatment)NCF1
D017258
CTDdecreases(expression)NCF1
D017258
CTDaffects(binding)NCOA1
D017258
CTDincreases(reaction)NCOA1
D017258
CTDaffects(cotreatment)NDST1
D017258
CTDincreases(expression)NDST1
D017258
CTDdecreases(expression)NEFM
D017258
CTDaffects(cotreatment)NEXN
D017258
CTDdecreases(expression)NEXN
D017258
CTDincreases(expression)NFE2L2
D017258
CTDincreases(expression)NLGN4X
D017258
CTDaffects(cotreatment)NOM1
D017258
CTDdecreases(expression)NOM1
D017258
CTDdecreases(reaction)NOS3
D017258
CTDincreases(activity)NOS3
D017258
CTDincreases(expression)NOS3
D017258
CTDaffects(cotreatment)NPHP1
D017258
CTDincreases(expression)NPHP1
D017258
CTDincreases(expression)NPTX2
D017258
CTDaffects(cotreatment)NPTXR
D017258
CTDdecreases(expression)NPTXR
D017258
CTDdecreases(reaction)NPY1R
D017258
CTDincreases(expression)NPY1R
D017258
CTDdecreases(expression)NPY1R
D017258
CTDincreases(activity)NR1I2
D017258
CTDaffects(cotreatment)NR2F1
D017258
CTDdecreases(expression)NR2F1
D017258
CTDaffects(cotreatment)NR3C1
D017258
CTDdecreases(expression)NR3C1
D017258
CTDaffects(response to substance)NR3C1
D017258
CTDaffects(cotreatment)NR3C2
D017258
CTDincreases(expression)NR3C2
D017258
CTDdecreases(expression)NR4A2
D017258
CTDaffects(cotreatment)NRIP1
D017258
CTDdecreases(expression)NRIP1
D017258
CTDaffects(cotreatment)NT5E
D017258
CTDincreases(expression)NT5E
D017258
CTDdecreases(expression)NT5E
D017258
CTDaffects(cotreatment)NTS
D017258
CTDdecreases(expression)NTS
D017258
CTDaffects(cotreatment)NUP155
D017258
CTDdecreases(expression)NUP155
D017258
CTDaffects(cotreatment)OGFRL1
D017258
CTDincreases(expression)OGFRL1
D017258
CTDaffects(cotreatment)OR8B8
D017258
CTDincreases(expression)OR8B8
D017258
CTDaffects(cotreatment)P4HB
D017258
CTDincreases(expression)P4HB
D017258
CTDaffects(cotreatment)PAEP
D017258
CTDdecreases(expression)PAEP
D017258
CTDaffects(cotreatment)PALM2-AKAP2
D017258
CTDincreases(expression)PALM2-AKAP2
D017258
CTDdecreases(expression)PCDH17
D017258
CTDaffects(cotreatment)PCDH18
D017258
CTDdecreases(expression)PCDH18
D017258
CTDdecreases(expression)PCDH20
D017258
CTDaffects(cotreatment)PCDHB4
D017258
CTDdecreases(expression)PCDHB4
D017258
CTDaffects(binding)PDGFA
D017258
CTDaffects(cotreatment)PDGFA
D017258
CTDdecreases(secretion)PDGFA
D017258
CTDaffects(binding)PDGFB
D017258
CTDaffects(cotreatment)PDGFB
D017258
CTDdecreases(secretion)PDGFB
D017258
CTDaffects(cotreatment)PDK1
D017258
CTDincreases(expression)PDK1
D017258
CTDdecreases(expression)PENK
D017258
CTDaffects(binding)PGR
D017258
CTDincreases(reaction)PGR
D017258
CTDdecreases(expression)PGR
D017258
CTDdecreases(expression)PGR
D017258
CTDdecreases(reaction)PGR
D011372
CTDincreases(activity)PGR
D011372
CTDincreases(expression)PGR
D011372
CTDaffects(localization)PGR
D011372
CTDincreases(activity)PGR
D011372
CTDincreases(phosphorylation)PGR
D011372
CTDaffects(cotreatment)PGRMC2
D017258
CTDincreases(expression)PGRMC2
D017258
CTDaffects(cotreatment)PITPNC1
D017258
CTDdecreases(expression)PITPNC1
D017258
CTDaffects(cotreatment)PKD2L1
D017258
CTDincreases(expression)PKD2L1
D017258
CTDaffects(cotreatment)PLAT
D017258
CTDincreases(expression)PLAT
D017258
CTDdecreases(expression)PLAU
D017258
CTDincreases(expression)PLCXD3
D017258
CTDaffects(cotreatment)PLEKHG3
D017258
CTDincreases(expression)PLEKHG3
D017258
CTDincreases(expression)PLG
D017258
CTDdecreases(expression)PLOD2
D017258
CTDaffects(cotreatment)PLS3
D017258
CTDdecreases(expression)PLS3
D017258
CTDdecreases(expression)PPBP
D017258
CTDaffects(cotreatment)PPIA
D017258
CTDdecreases(expression)PPIA
D017258
CTDaffects(cotreatment)PPIAL4A
D017258
CTDdecreases(expression)PPIAL4A
D017258
CTDaffects(cotreatment)PPP2R4
D017258
CTDincreases(expression)PPP2R4
D017258
CTDaffects(cotreatment)PRL
D017258
CTDincreases(expression)PRL
D017258
CTDaffects(cotreatment)PRL
D017258
CTDincreases(expression)PRL
D017258
CTDincreases(reaction)PRL
D017258
CTDaffects(cotreatment)PRL
D017258
CTDincreases(expression)PRL
D017258
CTDdecreases(reaction)PRL
D017258
CTDaffects(cotreatment)PRL
D017258
CTDaffects(reaction)PRL
D017258
CTDincreases(secretion)PRL
D017258
CTDincreases(expression)PRL
D017258
CTDdecreases(reaction)PRL
D017258
CTDdecreases(expression)PRRX1
D017258
CTDaffects(cotreatment)PRSS12
D017258
CTDdecreases(expression)PRSS12
D017258
CTDdecreases(expression)PTGS2
D017258
CTDaffects(cotreatment)PTK7
D017258
CTDincreases(expression)PTK7
D017258
CTDdecreases(reaction)PTP4A1
D017258
CTDincreases(expression)PTP4A1
D017258
CTDaffects(cotreatment)RAB1B
D017258
CTDincreases(expression)RAB1B
D017258
CTDaffects(cotreatment)RAB31
D017258
CTDincreases(expression)RAB31
D017258
CTDaffects(cotreatment)RAN
D017258
CTDdecreases(expression)RAN
D017258
CTDaffects(localization)RELA
D017258
CTDdecreases(reaction)RELA
D017258
CTDaffects(cotreatment)RET
D017258
CTDdecreases(expression)RET
D017258
CTDaffects(cotreatment)RGS10
D017258
CTDdecreases(expression)RGS10
D017258
CTDaffects(cotreatment)RHOBTB3
D017258
CTDdecreases(expression)RHOBTB3
D017258
CTDaffects(cotreatment)RIN1
D017258
CTDincreases(expression)RIN1
D017258
CTDincreases(expression)RNASE1
D017258
CTDincreases(expression)RPGR
D017258
CTDaffects(cotreatment)RPL5P29
D017258
CTDdecreases(expression)RPL5P29
D017258
CTDaffects(cotreatment)RPN1
D017258
CTDincreases(expression)RPN1
D017258
CTDaffects(cotreatment)RPS6KB1
D017258
CTDincreases(expression)RPS6KB1
D017258
CTDaffects(cotreatment)RPSA
D017258
CTDdecreases(expression)RPSA
D017258
CTDaffects(cotreatment)RPSAP12
D017258
CTDdecreases(expression)RPSAP12
D017258
CTDaffects(cotreatment)RPSAP28
D017258
CTDdecreases(expression)RPSAP28
D017258
CTDaffects(cotreatment)RPSAP3
D017258
CTDdecreases(expression)RPSAP3
D017258
CTDaffects(cotreatment)RPSAP31
D017258
CTDdecreases(expression)RPSAP31
D017258
CTDincreases(expression)RUNX1
D017258
CTDaffects(cotreatment)S100A14
D017258
CTDdecreases(expression)S100A14
D017258
CTDincreases(expression)S100P
D017258
CTDaffects(cotreatment)SARAF
D017258
CTDincreases(expression)SARAF
D017258
CTDaffects(cotreatment)SCAMP4
D017258
CTDincreases(expression)SCAMP4
D017258
CTDaffects(cotreatment)SDCBP
D017258
CTDdecreases(expression)SDCBP
D017258
CTDaffects(cotreatment)SEMA3A
D017258
CTDincreases(expression)SEMA3A
D017258
CTDincreases(expression)SEPP1
D017258
CTDaffects(cotreatment)SEPT11
D017258
CTDdecreases(expression)SEPT11
D017258
CTDincreases(expression)SERPINC1
D017258
CTDdecreases(expression)SERPINC1
D011372
CTDincreases(expression)SERPINE1
D017258
CTDincreases(expression)SERPINE1
D017258
CTDaffects(cotreatment)SFN
D017258
CTDincreases(expression)SFN
D017258
CTDincreases(expression)SGK1
D017258
CTDaffects(cotreatment)SIRPB1
D017258
CTDdecreases(expression)SIRPB1
D017258
CTDaffects(cotreatment)SIRT1
D017258
CTDincreases(expression)SIRT1
D017258
CTDincreases(expression)SLC1A3
D017258
CTDdecreases(expression)SLC46A2
D017258
CTDdecreases(expression)SLC47A1
D017258
CTDdecreases(expression)SLC5A3
D017258
CTDincreases(expression)SLC7A2
D017258
CTDincreases(expression)SLC7A8
D017258
CTDincreases(expression)SLC9A9
D017258
CTDincreases(expression)SLN
D017258
CTDdecreases(expression)SMOX
D017258
CTDaffects(cotreatment)SOD1
D017258
CTDincreases(activity)SOD1
D017258
CTDincreases(expression)SOD1
D017258
CTDaffects(cotreatment)SOD1
D017258
CTDdecreases(activity)SOD1
D017258
CTDdecreases(expression)SOD1
D017258
CTDincreases(activity)SOD1
D017258
CTDincreases(reaction)SOD1
D017258
CTDaffects(cotreatment)SOD1
D017258
CTDincreases(expression)SOD1
D017258
CTDincreases(expression)SOD1
D017258
CTDaffects(cotreatment)SOD2
D017258
CTDincreases(activity)SOD2
D017258
CTDincreases(expression)SOD2
D017258
CTDaffects(cotreatment)SOD2
D017258
CTDaffects(reaction)SOD2
D017258
CTDincreases(expression)SOD2
D017258
CTDaffects(binding)SOD2
D017258
CTDincreases(reaction)SOD2
D017258
CTDincreases(activity)SOD2
D017258
CTDincreases(expression)SOD2
D017258
CTDdecreases(reaction)SOD2
D017258
CTDincreases(expression)SOD2
D017258
CTDdecreases(reaction)SOD2
D017258
CTDaffects(reaction)SOD2
D017258
CTDincreases(abundance)SOD2
D017258
CTDincreases(expression)SPP1
D017258
CTDincreases(expression)SPRY1
D017258
CTDincreases(expression)SRPX
D017258
CTDaffects(cotreatment)SRSF7
D017258
CTDdecreases(expression)SRSF7
D017258
CTDaffects(cotreatment)STK38
D017258
CTDdecreases(expression)STK38
D017258
CTDincreases(expression)STOM
D017258
CTDaffects(cotreatment)SULF1
D017258
CTDdecreases(expression)SULF1
D017258
CTDaffects(cotreatment)TAGLN
D017258
CTDdecreases(expression)TAGLN
D017258
CTDincreases(expression)TBXAS1
D017258
CTDaffects(cotreatment)TCEA1
D017258
CTDdecreases(expression)TCEA1
D017258
CTDaffects(cotreatment)TERT
D017258
CTDincreases(expression)TERT
D017258
CTDincreases(expression)TFPI
D017258
CTDdecreases(expression)TFPI2
D017258
CTDdecreases(expression)TGFB3
D017258
CTDincreases(expression)TGFBR2
D017258
CTDdecreases(expression)THBS1
D017258
CTDdecreases(expression)TIMP3
D017258
CTDdecreases(expression)TMEM158
D017258
CTDaffects(cotreatment)TNC
D017258
CTDdecreases(expression)TNC
D017258
CTDaffects(cotreatment)TNF
D017258
CTDdecreases(secretion)TNF
D017258
CTDaffects(cotreatment)TNF
D017258
CTDdecreases(expression)TNF
D017258
CTDincreases(expression)TOX2
D017258
CTDaffects(cotreatment)TP53
D017258
CTDincreases(expression)TP53
D017258
CTDdecreases(reaction)TP53
D011372
CTDincreases(expression)TP53
D011372
CTDincreases(expression)TPD52
D017258
CTDaffects(cotreatment)TPI1
D017258
CTDincreases(expression)TPI1
D017258
CTDaffects(cotreatment)TPSG1
D017258
CTDdecreases(expression)TPSG1
D017258
CTDincreases(expression)TSC22D3
D017258
CTDdecreases(expression)TSKU
D017258
CTDaffects(cotreatment)TXN
D017258
CTDincreases(expression)TXN
D017258
CTDaffects(cotreatment)UBE2D4
D017258
CTDincreases(expression)UBE2D4
D017258
CTDaffects(cotreatment)UGCG
D017258
CTDdecreases(expression)UGCG
D017258
CTDaffects(cotreatment)UGT2B15
D017258
CTDdecreases(expression)UGT2B15
D017258
CTDaffects(cotreatment)USP12
D017258
CTDincreases(expression)USP12
D017258
CTDdecreases(reaction)VCAM1
D017258
CTDincreases(expression)VCAM1
D017258
CTDaffects(cotreatment)VDR
D017258
CTDaffects(response to substance)VDR
D017258
CTDincreases(expression)VEGFA
D017258
CTDdecreases(reaction)VEGFA
D017258
CTDincreases(expression)VEGFA
D017258
CTDdecreases(reaction)VEGFA
D011372
CTDincreases(expression)VEGFA
D011372
CTDdecreases(reaction)VEGFA
D011372
CTDincreases(activity)VEGFA
D011372
CTDincreases(expression)VEGFA
D011372
CTDaffects(cotreatment)VIM
D017258
CTDincreases(expression)VIM
D017258
CTDdecreases(expression)VMO1
D017258
CTDaffects(cotreatment)VPS39
D017258
CTDincreases(expression)VPS39
D017258
CTDincreases(expression)VSIG4
D017258
CTDaffects(cotreatment)WNT5A
D017258
CTDincreases(expression)WNT5A
D017258
CTDincreases(expression)WNT5A
D017258
CTDaffects(reaction)WNT5A
D017258
CTDincreases(abundance)WNT5A
D017258
CTDaffects(cotreatment)WWTR1
D017258
CTDincreases(expression)WWTR1
D017258
CTDincreases(expression)ZBTB16
D017258
CTDaffects(cotreatment)ZBTB45
D017258
CTDincreases(expression)ZBTB45
D017258
CTDincreases(expression)ZFP36
D017258
CTDaffects(cotreatment)ZFP36L1
D017258
CTDincreases(expression)ZFP36L1
D017258
CTDaffects(cotreatment)ZNF135
D017258
CTDincreases(expression)ZNF135
D017258
CTDaffects(cotreatment)ZNF530
D017258
CTDincreases(expression)ZNF530
D017258
CTDincreases(expression)ZPLD1
D017258
CTDaffects(cotreatment)ZSCAN10
D017258
CTDincreases(expression)ZSCAN10
D017258
CTDaffects(cotreatment)ZSCAN20
D017258
CTDincreases(expression)ZSCAN20
D017258
PubChem PotencyuM31.623ALDH1A1-GI(Protien) :
PubChem Potency-Replicate_1uM0.009AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.011AR-GI(Protien) :
PubChem Ratio Potency (uM)uM0.123AR-GI(Protien) :
PubChem Ratio Potency (uM)uM0.151AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.245AR-GI(Protien) :
PubChem Ratio Potency (uM)uM0.258AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.301AR-GI(Protien) :
PubChem Ratio Potency (uM)uM0.436AR-GI(Protien) :
PubChem PotencyuM1.585AR-GI(Protien) :
PubChem NoneuMCFTR-GI(Protien) :
PubChem PotencyuM15.849CYP3A4-GI(Protien) :
PubChem PotencyuM25.119ERG-GI(Protien) :
PubChem PotencyuM0.184NFE2L2-GI(Protien) :
PubChem PotencyuM0.259NFE2L2-GI(Protien) :
PubChem Ratio Potency (uM)uM27.278NFE2L2-GI(Protien) :
PubChem PotencyuM27.306NFE2L2-GI(Protien) :
PubChem PotencyuM2.512NPSR1-GI(Protien) :
PubChem Potency-Replicate_1uM0.022NR3C1-GI(Protien) :
PubChem Ratio Potency (uM)uM0.034NR3C1-GI(Protien) :
PubChem Potency-Replicate_1uM0.038NR3C1-GI(Protien) :
PubChem Ratio Potency (uM)uM0.105NR3C1-GI(Protien) :
PubChem NoneuMNR3C1-GI(Protien) :
PubChem PotencyuM31.623PARK2-GI(Protien) :
PubChem PotencyuM16.360TDP1-GI(Protien) :
PubChem PotencyuM18.356TDP1-GI(Protien) :
ChEMBLPotencynM31622.800ALDH1A1
-Target : CHEMBL3577
ChEMBLPotencynM15848.900CYP3A4
-Target : CHEMBL340
ChEMBLPotencynM259.300NFE2L2
-Target : CHEMBL1075094
ChEMBLPotencynM183.600NFE2L2
-Target : CHEMBL1075094
ChEMBLPotencynM2511.900NPSR1
-Target : CHEMBL5162
Download gene sets gmt, text, Detailed text
Contact us
Tan Lab , Mail Stop 8117
12801 East 17th Avenue
Division of Medical Oncology , Department of Medicine
University of Colorado School of Medicine
Aurora, CO 80045, USA

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