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Gene Set: D4 : CTD - Estazolam

Collection D4 : CTD
Chemical Name Estazolam ( From PubChem : ESTAZOLAM )
FDA NPC WHO Indian Australia China Traditional
Herbal		 Clinical
Trail
ApprovedNotNotNotNotNotNot4
Molecular
Weight		 Hydrogen Bond
Donor Count		 Hydrogen Bond
Acceptor Count		 cLogP Lipinski Rule
294.738 g/mol 0 4 2.7073 True
Structure
InChI InChI=1S/C16H11ClN4/c17-12-6-7-14-13(8-12)16(11-4-2-1-3-5-11)18-9-15-20-19-10-21(14)15/h1-8,10H,9H2
InChIKey CDCHDCWJMGXXRH-UHFFFAOYSA-N
Links

Gene (7 / 9)


⊖ Less
Source Type Unit Value Gene PMID Assay Other
CTDdecreases(activity)AKR1C1
D004949
CTDdecreases(activity)AKR1C2
D004949
CTDdecreases(activity)AKR1C3
D004949
CTDincreases(hydroxylation)CYP3A4
D004949
ChEMBLActivity-BRD3
-Target : CHEMBL1795186
ChEMBLActivity-BRD3
-Target : CHEMBL1795186
ChEMBLActivity-BRD4
-Target : CHEMBL1163125
ChEMBLActivity-BRD4
-Target : CHEMBL1163125
ChEMBLActivity-CREBBP
-Target : CHEMBL5747
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