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Gene Set: D4 : CTD - Cycloheximide


Collection D4 : CTD
Chemical Name Cycloheximide ( From PubChem : CYCLOHEXIMIDE )
FDA NPC WHO Indian Australia China Traditional
Herbal
Clinical
Trail
NotNotNotNotNotNotNotNot
Molecular
Weight
Hydrogen Bond
Donor Count
Hydrogen Bond
Acceptor Count
cLogP Lipinski Rule
281.347 g/mol 2 5 1.3703 True
Structure
InChI InChI=1S/C15H23NO4/c1-8-3-9(2)15(20)11(4-8)12(17)5-10-6-13(18)16-14(19)7-10/h8-12,17H,3-7H2,1-2H3,(H,16,18,19)/t8-,9-,11-,12+/m0/s1
InChIKey YPHMISFOHDHNIV-FSZOTQKASA-N
Links

Gene (324 / 894)


⊖ Less

Source Type Unit Value Gene PMID Assay Other
CTDincreases(expression)ABCB1
D003513
CTDincreases(reaction)ABCB1
D003513
CTDdecreases(expression)ABCB4
D003513
CTDdecreases(reaction)ABCB4
D003513
CTDaffects(cotreatment)ABCC3
D003513
CTDincreases(expression)ABCC3
D003513
CTDaffects(cotreatment)ABCC5
D003513
CTDdecreases(expression)ABCC5
D003513
CTDaffects(cotreatment)ACSL3
D003513
CTDaffects(expression)ACSL3
D003513
CTDdecreases(reaction)ADAM9
D003513
CTDincreases(expression)ADAM9
D003513
CTDincreases(expression)ADM
D003513
CTDincreases(reaction)ADM
D003513
CTDaffects(cotreatment)ADORA2B
D003513
CTDincreases(expression)ADORA2B
D003513
CTDaffects(cotreatment)ADRB2
D003513
CTDincreases(expression)ADRB2
D003513
CTDdecreases(expression)AHR
D003513
CTDdecreases(reaction)AHR
D003513
CTDdecreases(expression)AHR
D003513
CTDdecreases(reaction)AHR
D003513
CTDincreases(degradation)AHR
D003513
CTDincreases(reaction)AHR
D003513
CTDdecreases(expression)AKAP5
D003513
CTDdecreases(reaction)AKAP5
D003513
CTDdecreases(expression)AKAP6
D003513
CTDdecreases(reaction)AKAP6
D003513
CTDaffects(cotreatment)ALDH1A3
D003513
CTDincreases(expression)ALDH1A3
D003513
CTDaffects(cotreatment)ALDH3A2
D003513
CTDincreases(expression)ALDH3A2
D003513
CTDdecreases(expression)ALOX5AP
D003513
CTDdecreases(reaction)ALOX5AP
D003513
CTDdecreases(activity)ALPI
D003513
CTDdecreases(expression)AMHR2
D003513
CTDdecreases(reaction)AMHR2
D003513
CTDdecreases(expression)ANK2
D003513
CTDdecreases(reaction)ANK2
D003513
CTDaffects(cotreatment)ANKRD27
D003513
CTDincreases(expression)ANKRD27
D003513
CTDdecreases(expression)APAF1
D003513
CTDaffects(cotreatment)APAF1
D003513
CTDaffects(cotreatment)AREG
D003513
CTDincreases(expression)AREG
D003513
CTDincreases(expression)AREG
D003513
CTDaffects(cotreatment)ARMC5
D003513
CTDincreases(expression)ARMC5
D003513
CTDaffects(cotreatment)ASB1
D003513
CTDincreases(expression)ASB1
D003513
CTDdecreases(reaction)ATF4
D003513
CTDincreases(expression)ATF4
D003513
CTDdecreases(expression)AVPR1A
D003513
CTDdecreases(reaction)AVPR1A
D003513
CTDdecreases(expression)BBOX1
D003513
CTDdecreases(reaction)BBOX1
D003513
CTDdecreases(reaction)BCL2
D003513
CTDincreases(phosphorylation)BCL2
D003513
CTDincreases(expression)BCL2L1
D003513
CTDdecreases(reaction)BCL2L1
D003513
CTDaffects(cotreatment)BCL2L14
D003513
CTDincreases(expression)BCL2L14
D003513
CTDdecreases(expression)BDH1
D003513
CTDdecreases(reaction)BDH1
D003513
CTDdecreases(reaction)BECN1
D003513
CTDincreases(expression)BECN1
D003513
CTDaffects(cotreatment)BID
D003513
CTDincreases(cleavage)BID
D003513
CTDdecreases(reaction)BID
D003513
CTDincreases(cleavage)BID
D003513
CTDdecreases(reaction)BID
D003513
CTDincreases(reaction)BID
D003513
CTDdecreases(expression)BRCA1
D003513
CTDdecreases(reaction)BRCA1
D003513
CTDdecreases(expression)BRCA2
D003513
CTDdecreases(reaction)BRCA2
D003513
CTDdecreases(expression)CALB1
D003513
CTDdecreases(reaction)CALB1
D003513
CTDdecreases(reaction)CAMLG
D003513
CTDincreases(expression)CAMLG
D003513
CTDdecreases(reaction)CASP1
D003513
CTDincreases(expression)CASP1
D003513
CTDaffects(cotreatment)CASP3
D003513
CTDdecreases(reaction)CASP3
D003513
CTDincreases(activity)CASP3
D003513
CTDincreases(cleavage)CASP3
D003513
CTDaffects(cotreatment)CASP3
D003513
CTDincreases(activity)CASP3
D003513
CTDincreases(cleavage)CASP3
D003513
CTDincreases(activity)CASP3
D003513
CTDincreases(reaction)CASP3
D003513
CTDincreases(activity)CASP3
D003513
CTDdecreases(reaction)CASP3
D003513
CTDdecreases(reaction)CASP3
D003513
CTDdecreases(reaction)CASP4
D003513
CTDincreases(expression)CASP4
D003513
CTDdecreases(reaction)CASP7
D003513
CTDincreases(expression)CASP7
D003513
CTDincreases(activity)CASP7
D003513
CTDincreases(reaction)CASP7
D003513
CTDaffects(cotreatment)CASP8
D003513
CTDdecreases(reaction)CASP8
D003513
CTDincreases(activity)CASP8
D003513
CTDincreases(cleavage)CASP8
D003513
CTDaffects(cotreatment)CASP8
D003513
CTDincreases(activity)CASP8
D003513
CTDincreases(cleavage)CASP8
D003513
CTDincreases(activity)CASP8
D003513
CTDincreases(reaction)CASP8
D003513
CTDincreases(activity)CASP8
D003513
CTDdecreases(reaction)CASP8
D003513
CTDaffects(cotreatment)CASP9
D003513
CTDincreases(activity)CASP9
D003513
CTDaffects(cotreatment)CASP9
D003513
CTDincreases(activity)CASP9
D003513
CTDincreases(cleavage)CASP9
D003513
CTDdecreases(reaction)CASP9
D003513
CTDdecreases(reaction)CAV1
D003513
CTDincreases(expression)CAV1
D003513
CTDaffects(cotreatment)CBX1
D003513
CTDincreases(expression)CBX1
D003513
CTDincreases(expression)CCL2
D003513
CTDincreases(reaction)CCL2
D003513
CTDdecreases(reaction)CCL2
D003513
CTDincreases(expression)CCL5
D003513
CTDincreases(reaction)CCL5
D003513
CTDdecreases(reaction)CCL5
D003513
CTDaffects(cotreatment)CCNA2
D003513
CTDincreases(expression)CCNA2
D003513
CTDdecreases(expression)CCNA2
D003513
CTDdecreases(reaction)CCND1
D003513
CTDincreases(expression)CCND1
D003513
CTDaffects(cotreatment)CCND1
D003513
CTDincreases(degradation)CCND1
D003513
CTDaffects(cotreatment)CCT5
D003513
CTDdecreases(expression)CCT5
D003513
CTDaffects(reaction)CD38
D003513
CTDincreases(expression)CD38
D003513
CTDdecreases(expression)CD3E
D003513
CTDdecreases(reaction)CD3E
D003513
CTDdecreases(expression)CD47
D003513
CTDdecreases(reaction)CD47
D003513
CTDdecreases(reaction)CD63
D003513
CTDincreases(expression)CD63
D003513
CTDaffects(cotreatment)CD8A
D003513
CTDincreases(expression)CD8A
D003513
CTDincreases(expression)CDC42SE2
D003513
CTDaffects(cotreatment)CDC42SE2
D003513
CTDaffects(expression)CDC42SE2
D003513
CTDincreases(expression)CDCA5
D003513
CTDaffects(cotreatment)CDCA5
D003513
CTDdecreases(expression)CDK2
D003513
CTDdecreases(reaction)CDK2
D003513
CTDdecreases(reaction)CDKN1A
D003513
CTDincreases(expression)CDKN1A
D003513
CTDdecreases(reaction)CDKN1A
D003513
CTDincreases(expression)CDKN1A
D003513
CTDdecreases(expression)CDKN1A
D003513
CTDincreases(expression)CDKN2A
D003513
CTDdecreases(expression)CFLAR
D003513
CTDdecreases(expression)CFLAR
D003513
CTDdecreases(expression)CHRM1
D003513
CTDdecreases(reaction)CHRM1
D003513
CTDaffects(cotreatment)CITED2
D003513
CTDaffects(expression)CITED2
D003513
CTDaffects(cotreatment)CLCN3
D003513
CTDincreases(expression)CLCN3
D003513
CTDdecreases(reaction)CNR1
D003513
CTDincreases(expression)CNR1
D003513
CTDdecreases(reaction)CNR1
D003513
CTDincreases(expression)CNR1
D003513
CTDaffects(cotreatment)CRYL1
D003513
CTDincreases(expression)CRYL1
D003513
CTDdecreases(reaction)CSF2
D003513
CTDincreases(secretion)CSF2
D003513
CTDdecreases(reaction)CSF2
D003513
CTDincreases(secretion)CSF2
D003513
CTDdecreases(expression)CSNK1D
D003513
CTDincreases(reaction)CSNK1D
D003513
CTDincreases(expression)CTGF
D003513
CTDaffects(cotreatment)CTGF
D003513
CTDdecreases(expression)CTGF
D003513
CTDdecreases(reaction)CXCL8
D003513
CTDincreases(secretion)CXCL8
D003513
CTDaffects(secretion)CXCL8
D003513
CTDdecreases(reaction)CXCL8
D003513
CTDdecreases(reaction)CXCL8
D003513
CTDincreases(expression)CXCL8
D003513
CTDdecreases(reaction)CXCL8
D003513
CTDincreases(expression)CXCL8
D003513
CTDdecreases(reaction)CXCL8
D003513
CTDincreases(expression)CXCL8
D003513
CTDdecreases(expression)CXCL8
D003513
CTDdecreases(reaction)CXCL8
D003513
CTDincreases(expression)CXCL8
D003513
CTDincreases(expression)CXCL8
D003513
CTDaffects(cotreatment)CXCL8
D003513
CTDincreases(secretion)CXCL8
D003513
CTDincreases(reaction)CXCL8
D003513
CTDdecreases(reaction)CXCL8
D003513
CTDdecreases(expression)CYCS
D003513
CTDdecreases(reaction)CYCS
D003513
CTDdecreases(activity)CYP19A1
D003513
CTDdecreases(reaction)CYP1A1
D003513
CTDincreases(expression)CYP1A1
D003513
CTDincreases(expression)CYP1A1
D003513
CTDincreases(reaction)CYP1A1
D003513
CTDaffects(cotreatment)CYP1A1
D003513
CTDdecreases(expression)CYP1A1
D003513
CTDdecreases(reaction)CYP1A1
D003513
CTDaffects(cotreatment)CYP1A1
D003513
CTDdecreases(reaction)CYP1A1
D003513
CTDincreases(expression)CYP1A1
D003513
CTDdecreases(reaction)CYP1A1
D003513
CTDincreases(expression)CYP1A1
D003513
CTDincreases(expression)CYP1A1
D003513
CTDincreases(reaction)CYP1A1
D003513
CTDincreases(expression)CYP1A1
D003513
CTDincreases(reaction)CYP1A1
D003513
CTDincreases(expression)CYP1A1
D003513
CTDaffects(cotreatment)CYP1A1
D003513
CTDincreases(expression)CYP1A1
D003513
CTDdecreases(reaction)CYP1B1
D003513
CTDincreases(expression)CYP1B1
D003513
CTDincreases(expression)CYP1B1
D003513
CTDaffects(cotreatment)CYP1B1
D003513
CTDdecreases(reaction)CYP24A1
D003513
CTDincreases(expression)CYP24A1
D003513
CTDincreases(reaction)CYP24A1
D003513
CTDdecreases(expression)CYP2A6
D003513
CTDdecreases(reaction)CYP2A6
D003513
CTDdecreases(reaction)CYP2E1
D003513
CTDincreases(degradation)CYP2E1
D003513
CTDincreases(reaction)CYP2E1
D003513
CTDdecreases(reaction)CYP2E1
D003513
CTDincreases(oxidation)CYP2E1
D003513
CTDincreases(oxidation)CYP2E1
D003513
CTDincreases(degradation)CYP2E1
D003513
CTDincreases(reaction)CYP2E1
D003513
CTDdecreases(reaction)CYP2E1
D003513
CTDincreases(oxidation)CYP2E1
D003513
CTDdecreases(reaction)CYP2F1
D003513
CTDincreases(expression)CYP2F1
D003513
CTDdecreases(expression)CYP3A4
D003513
CTDdecreases(reaction)CYR61
D003513
CTDincreases(expression)CYR61
D003513
CTDdecreases(expression)DAG1
D003513
CTDdecreases(reaction)DAG1
D003513
CTDdecreases(expression)DCN
D003513
CTDdecreases(reaction)DCN
D003513
CTDaffects(cotreatment)DEAF1
D003513
CTDincreases(expression)DEAF1
D003513
CTDdecreases(expression)DEGS1
D003513
CTDdecreases(reaction)DEGS1
D003513
CTDdecreases(activity)DIO2
D003513
CTDdecreases(reaction)DIO2
D003513
CTDaffects(cotreatment)DLEU2
D003513
CTDincreases(expression)DLEU2
D003513
CTDdecreases(expression)DNAJB5
D003513
CTDdecreases(reaction)DNAJB5
D003513
CTDincreases(expression)DNM1L
D003513
CTDaffects(cotreatment)DNM1L
D003513
CTDaffects(cotreatment)EDN1
D003513
CTDincreases(expression)EDN1
D003513
CTDincreases(expression)EGFR
D003513
CTDdecreases(reaction)EGR1
D003513
CTDincreases(expression)EGR1
D003513
CTDincreases(expression)EGR2
D003513
CTDdecreases(reaction)EIF2A
D003513
CTDincreases(phosphorylation)EIF2A
D003513
CTDincreases(expression)EIF2S1
D003513
CTDaffects(cotreatment)EIF2S1
D003513
CTDdecreases(reaction)EIF4G3
D003513
CTDincreases(expression)EIF4G3
D003513
CTDaffects(cotreatment)EIF5
D003513
CTDdecreases(expression)EIF5
D003513
CTDdecreases(reaction)ELF4
D003513
CTDincreases(expression)ELF4
D003513
CTDincreases(expression)ELK1
D003513
CTDaffects(cotreatment)ELK1
D003513
CTDaffects(cotreatment)ENC1
D003513
CTDdecreases(expression)ENC1
D003513
CTDdecreases(expression)ENDOG
D003513
CTDdecreases(reaction)ENDOG
D003513
CTDdecreases(expression)EPYC
D003513
CTDdecreases(reaction)EPYC
D003513
CTDaffects(cotreatment)ERBB2
D003513
CTDdecreases(expression)ERBB2
D003513
CTDdecreases(expression)ERBB2
D003513
CTDdecreases(expression)ERBB2
D003513
CTDincreases(reaction)ERBB2
D003513
CTDdecreases(expression)ERBB3
D003513
CTDincreases(expression)EREG
D003513
CTDdecreases(expression)ESR1
D003513
CTDincreases(reaction)ESR1
D003513
CTDdecreases(reaction)ESR1
D003513
CTDincreases(expression)ESR2
D003513
CTDincreases(reaction)ESR2
D003513
CTDdecreases(reaction)ESR2
D003513
CTDdecreases(expression)EXT2
D003513
CTDdecreases(reaction)EXT2
D003513
CTDdecreases(expression)F12
D003513
CTDdecreases(reaction)F12
D003513
CTDdecreases(activity)F2
D003513
CTDdecreases(reaction)F2
D003513
CTDdecreases(expression)F3
D003513
CTDdecreases(reaction)F3
D003513
CTDincreases(activity)FAS
D003513
CTDincreases(reaction)FAS
D003513
CTDdecreases(expression)FASLG
D003513
CTDdecreases(reaction)FASLG
D003513
CTDdecreases(expression)FASN
D003513
CTDdecreases(reaction)FASN
D003513
CTDaffects(cotreatment)FBL
D003513
CTDincreases(expression)FBL
D003513
CTDdecreases(expression)FGL2
D003513
CTDdecreases(reaction)FGL2
D003513
CTDaffects(cotreatment)FHIT
D003513
CTDincreases(expression)FHIT
D003513
CTDdecreases(expression)FIGF
D003513
CTDdecreases(reaction)FIGF
D003513
CTDaffects(cotreatment)FMR1
D003513
CTDincreases(expression)FMR1
D003513
CTDdecreases(reaction)FOS
D003513
CTDincreases(expression)FOS
D003513
CTDdecreases(expression)FRK
D003513
CTDdecreases(reaction)FRK
D003513
CTDdecreases(reaction)FST
D003513
CTDincreases(expression)FST
D003513
CTDdecreases(reaction)FUT4
D003513
CTDincreases(expression)FUT4
D003513
CTDdecreases(expression)FZD7
D003513
CTDdecreases(reaction)FZD7
D003513
CTDaffects(cotreatment)GALNT1
D003513
CTDdecreases(expression)GALNT1
D003513
CTDdecreases(expression)GAS1
D003513
CTDdecreases(reaction)GAS1
D003513
CTDaffects(expression)GDF15
D003513
CTDdecreases(reaction)GDF15
D003513
CTDdecreases(reaction)GDF15
D003513
CTDincreases(expression)GDF15
D003513
CTDincreases(expression)GPAA1
D003513
CTDaffects(cotreatment)GPAA1
D003513
CTDdecreases(reaction)GPR37
D003513
CTDincreases(expression)GPR37
D003513
CTDaffects(cotreatment)GRN
D003513
CTDdecreases(expression)GRN
D003513
CTDdecreases(expression)GSK3B
D003513
CTDdecreases(reaction)GSK3B
D003513
CTDincreases(expression)HBEGF
D003513
CTDdecreases(reaction)HIF1A
D003513
CTDincreases(expression)HIF1A
D003513
CTDdecreases(reaction)HIF1A
D003513
CTDincreases(expression)HIF1A
D003513
CTDdecreases(reaction)HIF1A
D003513
CTDincreases(stability)HIF1A
D003513
CTDdecreases(reaction)HIF1A
D003513
CTDincreases(expression)HIF1A
D003513
CTDincreases(degradation)HIF1A
D003513
CTDdecreases(reaction)HMOX1
D003513
CTDincreases(expression)HMOX1
D003513
CTDdecreases(reaction)HMOX1
D003513
CTDincreases(expression)HMOX1
D003513
CTDdecreases(reaction)HMOX1
D003513
CTDincreases(expression)HMOX1
D003513
CTDdecreases(reaction)HMOX1
D003513
CTDincreases(expression)HMOX1
D003513
CTDdecreases(response to substance)HMOX1
D003513
CTDincreases(expression)HMOX1
D003513
CTDincreases(expression)HNRNPH2
D003513
CTDdecreases(expression)HTATIP2
D003513
CTDdecreases(reaction)HTATIP2
D003513
CTDdecreases(reaction)ICAM1
D003513
CTDincreases(expression)ICAM1
D003513
CTDdecreases(expression)ICAM1
D003513
CTDaffects(cotreatment)IER3
D003513
CTDincreases(expression)IER3
D003513
CTDdecreases(reaction)IFI6
D003513
CTDincreases(activity)IFI6
D003513
CTDaffects(cotreatment)IFNA2
D003513
CTDincreases(expression)IFNA2
D003513
CTDaffects(cotreatment)IFNG
D003513
CTDincreases(expression)IFNG
D003513
CTDdecreases(reaction)IFNG
D003513
CTDincreases(expression)IFNG
D003513
CTDdecreases(expression)IFT27
D003513
CTDdecreases(reaction)IFT27
D003513
CTDaffects(cotreatment)IGFBP4
D003513
CTDincreases(expression)IGFBP4
D003513
CTDincreases(expression)IL1A
D003513
CTDaffects(cotreatment)IL1A
D003513
CTDaffects(secretion)IL1B
D003513
CTDdecreases(reaction)IL1B
D003513
CTDdecreases(reaction)IL1B
D003513
CTDincreases(expression)IL1B
D003513
CTDincreases(reaction)IL1B
D003513
CTDdecreases(reaction)IL1B
D003513
CTDincreases(secretion)IL1B
D003513
CTDincreases(expression)IL1B
D003513
CTDaffects(cotreatment)IL1B
D003513
CTDaffects(secretion)IL6
D003513
CTDdecreases(reaction)IL6
D003513
CTDdecreases(secretion)IL6
D003513
CTDincreases(expression)IL6
D003513
CTDincreases(secretion)IL6
D003513
CTDincreases(reaction)IL6
D003513
CTDdecreases(reaction)IL6
D003513
CTDdecreases(reaction)IL6ST
D003513
CTDincreases(expression)IL6ST
D003513
CTDdecreases(reaction)IQGAP1
D003513
CTDincreases(expression)IQGAP1
D003513
CTDaffects(cotreatment)IRS1
D003513
CTDincreases(expression)IRS1
D003513
CTDdecreases(expression)IRS1
D003513
CTDdecreases(reaction)ITGB3
D003513
CTDincreases(expression)ITGB3
D003513
CTDdecreases(reaction)ITGB6
D003513
CTDincreases(expression)ITGB6
D003513
CTDdecreases(reaction)ITGB6
D003513
CTDincreases(expression)ITGB6
D003513
CTDaffects(cotreatment)ITPK1
D003513
CTDdecreases(reaction)ITPK1
D003513
CTDincreases(activity)ITPK1
D003513
CTDincreases(cleavage)ITPK1
D003513
CTDincreases(reaction)ITPK1
D003513
CTDincreases(response to substance)ITPK1
D003513
CTDdecreases(reaction)ITPR1
D003513
CTDincreases(expression)ITPR1
D003513
CTDdecreases(reaction)ITPR1
D003513
CTDincreases(expression)ITPR1
D003513
CTDaffects(cotreatment)KANK1
D003513
CTDincreases(expression)KANK1
D003513
CTDaffects(cotreatment)KIAA0930
D003513
CTDincreases(expression)KIAA0930
D003513
CTDdecreases(reaction)KRAS
D003513
CTDincreases(expression)KRAS
D003513
CTDaffects(cotreatment)KRT13
D003513
CTDincreases(expression)KRT13
D003513
CTDaffects(cotreatment)KRTCAP2
D003513
CTDincreases(expression)KRTCAP2
D003513
CTDdecreases(reaction)LCK
D003513
CTDincreases(expression)LCK
D003513
CTDdecreases(reaction)LGALS3
D003513
CTDincreases(expression)LGALS3
D003513
CTDincreases(expression)LINC00152
D003513
CTDdecreases(reaction)LMO7
D003513
CTDincreases(expression)LMO7
D003513
CTDdecreases(reaction)LPXN
D003513
CTDincreases(expression)LPXN
D003513
CTDincreases(phosphorylation)MAPK1
D003513
CTDaffects(reaction)MAPK1
D003513
CTDdecreases(phosphorylation)MAPK14
D003513
CTDdecreases(reaction)MAPK14
D003513
CTDincreases(phosphorylation)MAPK3
D003513
CTDaffects(reaction)MAPK3
D003513
CTDdecreases(reaction)MAPK7
D003513
CTDincreases(expression)MAPK7
D003513
CTDincreases(expression)MAPK7
D003513
CTDaffects(cotreatment)MAPK7
D003513
CTDaffects(cotreatment)MCL1
D003513
CTDincreases(response to substance)MCL1
D003513
CTDdecreases(expression)MCL1
D003513
CTDdecreases(expression)MDK
D003513
CTDincreases(reaction)MDK
D003513
CTDdecreases(reaction)MIR21
D003513
CTDincreases(expression)MIR21
D003513
CTDdecreases(expression)MIR21
D003513
CTDdecreases(reaction)MIR21
D003513
CTDincreases(expression)MIR22HG
D003513
CTDincreases(stability)MIR22HG
D003513
CTDdecreases(reaction)MMP1
D003513
CTDincreases(expression)MMP1
D003513
CTDdecreases(reaction)MMP1
D003513
CTDincreases(expression)MMP1
D003513
CTDincreases(expression)MMP13
D003513
CTDaffects(cotreatment)MMP13
D003513
CTDdecreases(expression)MNX1
D003513
CTDdecreases(reaction)MNX1
D003513
CTDdecreases(reaction)MPG
D003513
CTDincreases(expression)MPG
D003513
CTDdecreases(expression)MRPS7
D003513
CTDaffects(cotreatment)MRPS7
D003513
CTDaffects(expression)MRPS7
D003513
CTDdecreases(expression)MSH3
D003513
CTDdecreases(reaction)MSH3
D003513
CTDdecreases(reaction)MSR1
D003513
CTDincreases(expression)MSR1
D003513
CTDaffects(cotreatment)MTCH2
D003513
CTDincreases(expression)MTCH2
D003513
CTDincreases(expression)MTMR7
D003513
CTDaffects(cotreatment)MTMR7
D003513
CTDdecreases(reaction)MXD1
D003513
CTDincreases(expression)MXD1
D003513
CTDaffects(cotreatment)MXD3
D003513
CTDincreases(expression)MXD3
D003513
CTDdecreases(reaction)MYLK
D003513
CTDincreases(expression)MYLK
D003513
CTDincreases(expression)NBR1
D003513
CTDaffects(cotreatment)NBR1
D003513
CTDdecreases(expression)NEK2
D003513
CTDdecreases(reaction)NEK2
D003513
CTDaffects(localization)NFE2L2
D003513
CTDaffects(reaction)NFE2L2
D003513
CTDdecreases(reaction)NFE2L2
D003513
CTDaffects(cotreatment)NFE2L2
D003513
CTDincreases(expression)NFE2L2
D003513
CTDdecreases(reaction)NFE2L2
D003513
CTDincreases(expression)NFE2L2
D003513
CTDdecreases(expression)NFE2L2
D003513
CTDaffects(localization)NFKB1
D003513
CTDaffects(binding)NFKB1
D003513
CTDdecreases(expression)NFKB1
D003513
CTDincreases(expression)NFKB1
D003513
CTDincreases(reaction)NFKB1
D003513
CTDdecreases(reaction)NFKB1
D003513
CTDdecreases(reaction)NFKBIA
D003513
CTDincreases(expression)NFKBIA
D003513
CTDdecreases(reaction)NFKBIA
D003513
CTDincreases(expression)NFKBIA
D003513
CTDdecreases(expression)NFKBIA
D003513
CTDincreases(reaction)NFKBIA
D003513
CTDincreases(degradation)NFKBIA
D003513
CTDdecreases(expression)NFKBIA
D003513
CTDaffects(reaction)NFKBIA
D003513
CTDincreases(expression)NFKBIA
D003513
CTDincreases(reaction)NFKBIA
D003513
CTDdecreases(reaction)NOS2
D003513
CTDincreases(expression)NOS2
D003513
CTDdecreases(reaction)NOS2
D003513
CTDincreases(expression)NOS2
D003513
CTDdecreases(reaction)NOS3
D003513
CTDincreases(expression)NOS3
D003513
CTDaffects(cotreatment)NOV
D003513
CTDdecreases(expression)NOV
D003513
CTDincreases(expression)NOV
D003513
CTDdecreases(expression)NPY1R
D003513
CTDdecreases(reaction)NPY1R
D003513
CTDincreases(expression)NR1H3
D003513
CTDaffects(cotreatment)NR1H3
D003513
CTDaffects(cotreatment)NUCKS1
D003513
CTDincreases(expression)NUCKS1
D003513
CTDincreases(expression)OPRK1
D003513
CTDaffects(cotreatment)OPRK1
D003513
CTDdecreases(reaction)OPRM1
D003513
CTDincreases(expression)OPRM1
D003513
CTDdecreases(expression)PA2G4
D003513
CTDincreases(reaction)PA2G4
D003513
CTDincreases(expression)PAPPA
D003513
CTDaffects(cotreatment)PAPPA
D003513
CTDaffects(cotreatment)PARP1
D003513
CTDincreases(cleavage)PARP1
D003513
CTDaffects(cotreatment)PARP1
D003513
CTDincreases(cleavage)PARP1
D003513
CTDincreases(cleavage)PARP1
D003513
CTDdecreases(reaction)PARP1
D003513
CTDincreases(reaction)PARP1
D003513
CTDdecreases(expression)PAX3
D003513
CTDdecreases(reaction)PAX3
D003513
CTDaffects(cotreatment)PCGF1
D003513
CTDincreases(expression)PCGF1
D003513
CTDdecreases(expression)PCNA
D003513
CTDdecreases(reaction)PCNA
D003513
CTDdecreases(reaction)PDCD2
D003513
CTDincreases(expression)PDCD2
D003513
CTDdecreases(expression)PI4KA
D003513
CTDincreases(reaction)PI4KA
D003513
CTDdecreases(expression)PIGH
D003513
CTDdecreases(reaction)PIGH
D003513
CTDdecreases(expression)PIGK
D003513
CTDdecreases(reaction)PIGK
D003513
CTDdecreases(expression)PIK3C3
D003513
CTDdecreases(reaction)PIK3C3
D003513
CTDdecreases(expression)PIK3CG
D003513
CTDdecreases(reaction)PIK3CG
D003513
CTDaffects(cotreatment)PILRB
D003513
CTDincreases(expression)PILRB
D003513
CTDdecreases(reaction)PLA2G1B
D003513
CTDincreases(expression)PLA2G1B
D003513
CTDaffects(cotreatment)PLAUR
D003513
CTDincreases(expression)PLAUR
D003513
CTDincreases(expression)PLD3
D003513
CTDaffects(cotreatment)PLD3
D003513
CTDdecreases(expression)PLN
D003513
CTDdecreases(reaction)PLN
D003513
CTDdecreases(reaction)PMAIP1
D003513
CTDincreases(expression)PMAIP1
D003513
CTDdecreases(reaction)PNPLA6
D003513
CTDincreases(activity)PNPLA6
D003513
CTDaffects(cotreatment)PNPLA6
D003513
CTDaffects(cotreatment)PPAN
D003513
CTDincreases(expression)PPAN
D003513
CTDdecreases(expression)PPP3CB
D003513
CTDdecreases(reaction)PPP3CB
D003513
CTDdecreases(reaction)PRDX4
D003513
CTDincreases(expression)PRDX4
D003513
CTDdecreases(expression)PRKCB
D003513
CTDaffects(cotreatment)PRKCB
D003513
CTDincreases(expression)PRKCB
D003513
CTDdecreases(reaction)PRKCZ
D003513
CTDincreases(expression)PRKCZ
D003513
CTDdecreases(reaction)PTEN
D003513
CTDincreases(expression)PTEN
D003513
CTDdecreases(reaction)PTGS2
D003513
CTDincreases(expression)PTGS2
D003513
CTDincreases(reaction)PTGS2
D003513
CTDdecreases(reaction)PTGS2
D003513
CTDincreases(activity)PTGS2
D003513
CTDincreases(expression)PTGS2
D003513
CTDdecreases(reaction)PTGS2
D003513
CTDincreases(expression)PTGS2
D003513
CTDincreases(expression)PTN
D003513
CTDaffects(cotreatment)PTN
D003513
CTDdecreases(reaction)PTP4A1
D003513
CTDincreases(expression)PTP4A1
D003513
CTDincreases(reaction)PTP4A1
D003513
CTDaffects(cotreatment)PTP4A3
D003513
CTDincreases(expression)PTP4A3
D003513
CTDaffects(cotreatment)RAPGEF1
D003513
CTDincreases(expression)RAPGEF1
D003513
CTDincreases(expression)RARRES2
D003513
CTDaffects(cotreatment)RARRES2
D003513
CTDdecreases(reaction)RBL1
D003513
CTDincreases(expression)RBL1
D003513
CTDaffects(localization)RELA
D003513
CTDaffects(binding)RELA
D003513
CTDaffects(cotreatment)RELA
D003513
CTDincreases(reaction)RELA
D003513
CTDdecreases(expression)RELA
D003513
CTDdecreases(reaction)REN
D003513
CTDincreases(secretion)REN
D003513
CTDaffects(cotreatment)RPS27L
D003513
CTDincreases(expression)RPS27L
D003513
CTDdecreases(expression)S100A12
D003513
CTDdecreases(reaction)S100A12
D003513
CTDdecreases(expression)S100A4
D003513
CTDdecreases(reaction)S100A4
D003513
CTDdecreases(expression)S100A7
D003513
CTDdecreases(reaction)S100A7
D003513
CTDaffects(binding)SAT1
D003513
CTDaffects(cotreatment)SAT1
D003513
CTDincreases(reaction)SAT1
D003513
CTDincreases(expression)SAT1
D003513
CTDaffects(reaction)SAT1
D003513
CTDaffects(cotreatment)SEC11C
D003513
CTDaffects(expression)SEC11C
D003513
CTDincreases(expression)SERPINB9
D003513
CTDincreases(reaction)SERPINB9
D003513
CTDdecreases(reaction)SERPINE1
D003513
CTDincreases(expression)SERPINE1
D003513
CTDincreases(expression)SERPINE2
D003513
CTDaffects(cotreatment)SERPINE2
D003513
CTDincreases(expression)SERTAD2
D003513
CTDaffects(cotreatment)SERTAD2
D003513
CTDdecreases(expression)SIRPA
D003513
CTDdecreases(reaction)SIRPA
D003513
CTDdecreases(reaction)SLA
D003513
CTDincreases(expression)SLA
D003513
CTDaffects(cotreatment)SLC16A1
D003513
CTDincreases(expression)SLC16A1
D003513
CTDincreases(expression)SLC22A4
D003513
CTDaffects(cotreatment)SLC22A4
D003513
CTDincreases(expression)SLC25A27
D003513
CTDaffects(cotreatment)SLC2A1
D003513
CTDincreases(expression)SLC2A1
D003513
CTDincreases(expression)SLC5A5
D003513
CTDaffects(cotreatment)SLC7A5
D003513
CTDincreases(expression)SLC7A5
D003513
CTDaffects(cotreatment)SMEK2
D003513
CTDincreases(expression)SMEK2
D003513
CTDdecreases(reaction)SMN1
D003513
CTDincreases(expression)SMN1
D003513
CTDincreases(expression)SNHG15
D003513
CTDincreases(stability)SNHG15
D003513
CTDaffects(cotreatment)SNW1
D003513
CTDincreases(expression)SNW1
D003513
CTDaffects(cotreatment)SOCS1
D003513
CTDincreases(expression)SOCS1
D003513
CTDincreases(expression)SOD2
D003513
CTDincreases(reaction)SOD2
D003513
CTDdecreases(reaction)SOS1
D003513
CTDincreases(expression)SOS1
D003513
CTDincreases(expression)SSBP1
D003513
CTDaffects(cotreatment)SSBP1
D003513
CTDincreases(expression)ST8SIA1
D003513
CTDaffects(cotreatment)ST8SIA1
D003513
CTDdecreases(expression)STK3
D003513
CTDdecreases(reaction)STK3
D003513
CTDdecreases(expression)STX2
D003513
CTDdecreases(reaction)STX2
D003513
CTDdecreases(reaction)SULT1A1
D003513
CTDincreases(expression)SULT1A1
D003513
CTDdecreases(reaction)SULT2B1
D003513
CTDincreases(expression)SULT2B1
D003513
CTDdecreases(expression)SUPT4H1
D003513
CTDdecreases(reaction)SUPT4H1
D003513
CTDincreases(expression)SYNPO
D003513
CTDaffects(cotreatment)SYNPO
D003513
CTDaffects(cotreatment)TACC1
D003513
CTDdecreases(expression)TACC1
D003513
CTDincreases(expression)TACC1
D003513
CTDaffects(cotreatment)TFF1
D003513
CTDincreases(expression)TFF1
D003513
CTDdecreases(reaction)TFF1
D003513
CTDincreases(expression)TFF1
D003513
CTDincreases(expression)TGFA
D003513
CTDdecreases(reaction)TGFB1
D003513
CTDincreases(expression)TGFB1
D003513
CTDdecreases(expression)TGFB1
D003513
CTDdecreases(reaction)TGFB1
D003513
CTDincreases(expression)TGFB1
D003513
CTDdecreases(expression)THBD
D003513
CTDdecreases(reaction)THBD
D003513
CTDdecreases(expression)THY1
D003513
CTDdecreases(reaction)THY1
D003513
CTDdecreases(expression)TIMM17A
D003513
CTDincreases(degradation)TIMM17A
D003513
CTDdecreases(reaction)TIMM17A
D003513
CTDdecreases(reaction)TJP1
D003513
CTDincreases(expression)TJP1
D003513
CTDdecreases(expression)TJP1
D003513
CTDaffects(cotreatment)TM7SF3
D003513
CTDincreases(expression)TM7SF3
D003513
CTDincreases(expression)TMEM263
D003513
CTDaffects(cotreatment)TMEM263
D003513
CTDaffects(cotreatment)TNF
D003513
CTDincreases(cleavage)TNF
D003513
CTDincreases(activity)TNF
D003513
CTDaffects(secretion)TNF
D003513
CTDdecreases(reaction)TNF
D003513
CTDdecreases(reaction)TNF
D003513
CTDincreases(expression)TNF
D003513
CTDdecreases(reaction)TNF
D003513
CTDincreases(expression)TNF
D003513
CTDdecreases(reaction)TNF
D003513
CTDincreases(expression)TNF
D003513
CTDdecreases(reaction)TNF
D003513
CTDincreases(expression)TNF
D003513
CTDdecreases(reaction)TNF
D003513
CTDincreases(expression)TNF
D003513
CTDincreases(reaction)TNF
D003513
CTDdecreases(reaction)TNF
D003513
CTDincreases(reaction)TNF
D003513
CTDincreases(response to substance)TNF
D003513
CTDaffects(cotreatment)TNF
D003513
CTDincreases(expression)TNF
D003513
CTDincreases(secretion)TNF
D003513
CTDincreases(reaction)TNF
D003513
CTDincreases(response to substance)TNF
D003513
CTDdecreases(reaction)TNF
D003513
CTDaffects(cotreatment)TNFAIP3
D003513
CTDincreases(expression)TNFAIP3
D003513
CTDincreases(reaction)TNFAIP3
D003513
CTDdecreases(reaction)TNFRSF10A
D003513
CTDincreases(expression)TNFRSF10A
D003513
CTDdecreases(reaction)TNFRSF10B
D003513
CTDincreases(expression)TNFRSF10B
D003513
CTDincreases(expression)TNFRSF10B
D003513
CTDincreases(reaction)TNFRSF10B
D003513
CTDaffects(cotreatment)TNFRSF10B
D003513
CTDincreases(expression)TNFRSF10B
D003513
CTDincreases(localization)TNFRSF10B
D003513
CTDincreases(reaction)TNFRSF10B
D003513
CTDincreases(response to substance)TNFRSF10B
D003513
CTDaffects(cotreatment)TNFRSF11B
D003513
CTDdecreases(expression)TNFRSF11B
D003513
CTDdecreases(reaction)TNFRSF8
D003513
CTDincreases(expression)TNFRSF8
D003513
CTDaffects(cotreatment)TNFSF10
D003513
CTDdecreases(reaction)TNFSF10
D003513
CTDincreases(activity)TNFSF10
D003513
CTDincreases(cleavage)TNFSF10
D003513
CTDdecreases(expression)TNFSF10
D003513
CTDdecreases(reaction)TNFSF10
D003513
CTDincreases(expression)TNFSF10
D003513
CTDincreases(localization)TNFSF10
D003513
CTDincreases(reaction)TNFSF10
D003513
CTDincreases(response to substance)TNFSF10
D003513
CTDdecreases(expression)TNFSF11
D003513
CTDdecreases(reaction)TNFSF11
D003513
CTDdecreases(reaction)TNNC1
D003513
CTDincreases(expression)TNNC1
D003513
CTDdecreases(reaction)TP53
D003513
CTDincreases(expression)TP53
D003513
CTDincreases(response to substance)TP53
D003513
CTDdecreases(reaction)TP53I11
D003513
CTDincreases(expression)TP53I11
D003513
CTDdecreases(expression)TP53I11
D003513
CTDdecreases(reaction)TP63
D003513
CTDincreases(expression)TP63
D003513
CTDdecreases(expression)TUBGCP3
D003513
CTDdecreases(reaction)TUBGCP3
D003513
CTDdecreases(reaction)TXNRD1
D003513
CTDincreases(expression)TXNRD1
D003513
CTDdecreases(reaction)TXNRD1
D003513
CTDincreases(expression)TXNRD1
D003513
CTDdecreases(expression)TYMS
D003513
CTDdecreases(reaction)TYMS
D003513
CTDdecreases(reaction)TYR
D003513
CTDincreases(activity)TYR
D003513
CTDaffects(cotreatment)UGT1A1
D003513
CTDdecreases(expression)UGT1A1
D003513
CTDincreases(expression)UGT2B15
D003513
CTDdecreases(reaction)VEGFA
D003513
CTDincreases(expression)VEGFA
D003513
CTDincreases(expression)VEGFA
D003513
CTDincreases(reaction)VEGFA
D003513
CTDdecreases(expression)VLDLR
D003513
CTDdecreases(reaction)VLDLR
D003513
CTDdecreases(expression)VSNL1
D003513
CTDdecreases(reaction)VSNL1
D003513
CTDaffects(cotreatment)YAP1
D003513
CTDincreases(expression)YAP1
D003513
CTDdecreases(reaction)YME1L1
D003513
CTDincreases(degradation)YME1L1
D003513
PubChem Potency-Replicate_1uM0.668AHR-GI(Protien) :
PubChem AR Potency (uM)uM0.207AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.216AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.298AR-GI(Protien) :
PubChem AR Potency (uM)uM0.390AR-GI(Protien) :
PubChem Potency-Replicate_1uM0.434AR-GI(Protien) :
PubChem Potency-Replicate_1uM1.068AR-GI(Protien) :
PubChem PotencyuM0.291ATAD5-GI(Protien) :
PubChem NoneuMCFTR-GI(Protien) :
PubChem IC50_CF-PAF_MeanuMCFTR-GI(Protien) :
PubChem NoneuMCFTR-GI(Protien) :
PubChem Potency-Replicate_1uM0.383CYP19A1-GI(Protien) :
PubChem Potency-Replicate_1uM0.750CYP19A1-GI(Protien) :
PubChem NoneuMCYP19A1-GI(Protien) :
PubChem NoneuMEPAS1-GI(Protien) :
PubChem ER Potency (uM)uM0.293ESR1-GI(Protien) :
PubChem ER Potency (uM)uM0.511ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM0.541ESR1-GI(Protien) :
PubChem Potency-Replicate_1uM0.668ESR1-GI(Protien) :
PubChem PotencyuM0.794GLP1R-GI(Protien) :
PubChem AC50_uMuM0.195HSP90AA1-GI(Protien) :
PubChem PotencyuM0.731IDH1-GI(Protien) :
PubChem NoneuMIL1B-GI(Protien) :
PubChem NoneuMMDM2-GI(Protien) :
PubChem NoneuMMDM2-GI(Protien) :
PubChem NoneuMMDM2-GI(Protien) :
PubChem NoneuMMDM4-GI(Protien) :
PubChem NoneuMMDM4-GI(Protien) :
PubChem NoneuMMDM4-GI(Protien) :
PubChem NoneuMMITF-GI(Protien) :
PubChem NoneuMNCOA1-GI(Protien) :
PubChem NoneuMNCOA2-GI(Protien) :
PubChem NoneuMNCOA2-GI(Protien) :
PubChem NoneuMNCOA3-GI(Protien) :
PubChem PotencyuM0.581NFE2L2-GI(Protien) :
PubChem PotencyuM5.805NFE2L2-GI(Protien) :
PubChem NoneuMNLRP3-GI(Protien) :
PubChem NoneuMNLRP3-GI(Protien) :
PubChem NoneuMNLRP3-GI(Protien) :
PubChem NoneuMNLRP3-GI(Protien) :
PubChem NoneuMNOD2-GI(Protien) :
PubChem NoneuMNR2E3-GI(Protien) :
PubChem NoneuMNR2E3-GI(Protien) :
PubChem IC50uM1.315NR2F2-GI(Protien) :
PubChem NoneuMNR2F2-GI(Protien) :
PubChem NoneuMNR2F2-GI(Protien) :
PubChem PotencyuM3.162NR3C1-GI(Protien) :
PubChem Potency-Replicate_1uM4.772NR3C1-GI(Protien) :
PubChem Potency-Replicate_1uM12.232NR3C1-GI(Protien) :
PubChem NoneuMNR3C1-GI(Protien) :
PubChem NoneuMNR5A1-GI(Protien) :
PubChem NoneuMNR5A2-GI(Protien) :
PubChem NoneuMNR5A2-GI(Protien) :
PubChem PotencyuM0.200PPARD-GI(Protien) :
PubChem PotencyuM0.316PPARD-GI(Protien) :
PubChem NoneuMPPARD-GI(Protien) :
PubChem NoneuMPPARG-GI(Protien) :
PubChem NoneuMPRNP-GI(Protien) :
PubChem NoneuMPRNP-GI(Protien) :
PubChem NoneuMPRNP-GI(Protien) :
PubChem NoneuMRIPK2-GI(Protien) :
PubChem PotencyuM1.000SMAD3-GI(Protien) :
PubChem NoneuMSTK33-GI(Protien) :
PubChem PotencyuM0.047TDP1-GI(Protien) :
PubChem PotencyuM0.060TDP1-GI(Protien) :
PubChem PotencyuM0.119TDP1-GI(Protien) :
PubChem PotencyuM0.150TDP1-GI(Protien) :
PubChem PotencyuM0.164TDP1-GI(Protien) :
PubChem PotencyuM0.164TDP1-GI(Protien) :
PubChem NoneuMVDR-GI(Protien) :
ChEMBLPotencynM290.800ATAD5
-Target : CHEMBL1741209
ChEMBLInhibition-EEF2
-Target : CHEMBL1795108
ChEMBLInhibition-EEF2
-Target : CHEMBL1795108
ChEMBLInhibition-EEF2
-Target : CHEMBL1795108
ChEMBLActivity-HIF1A
-Target : CHEMBL4261
ChEMBLActivity-HIF1A
-Target : CHEMBL4261
ChEMBLActivity-HIF1A
-Target : CHEMBL4261
ChEMBLActivity-HIF1A
-Target : CHEMBL4261
ChEMBLActivity-HSF1
-Target : CHEMBL5869
ChEMBLPotencynM580.500NFE2L2
-Target : CHEMBL1075094
Download gene sets gmt, text, Detailed text
Contact us
Tan Lab , Mail Stop 8117
12801 East 17th Avenue
Division of Medical Oncology , Department of Medicine
University of Colorado School of Medicine
Aurora, CO 80045, USA

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