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Gene Set: D4 : CTD - Azacitidine


Collection D4 : CTD
Chemical Name Azacitidine ( From PubChem : 5-AZACYTIDINE )
FDA NPC WHO Indian Australia China Traditional
Herbal
Clinical
Trail
ApprovedNotNotNotNotNotNotNot
Molecular
Weight
Hydrogen Bond
Donor Count
Hydrogen Bond
Acceptor Count
cLogP Lipinski Rule
244.205 g/mol 4 9 -2.5868 True
Structure
InChI InChI=1S/C8H12N4O5/c9-7-10-2-12(8(16)11-7)6-5(15)4(14)3(1-13)17-6/h2-6,13-15H,1H2,(H2,9,11,16)/t3-,4-,5-,6-/m1/s1
InChIKey NMUSYJAQQFHJEW-KVTDHHQDSA-N
Links

Gene (352 / 576)


⊖ Less

Source Type Unit Value Gene PMID Assay Other
CTDdecreases(reaction)ACTA2
D001374
CTDincreases(expression)ACTA2
D001374
CTDdecreases(expression)ADAMTS1
D001374
CTDincreases(expression)AGGF1
D001374
CTDincreases(expression)AHR
D001374
CTDincreases(expression)AK5
D001374
CTDdecreases(reaction)AKT1
D001374
CTDincreases(phosphorylation)AKT1
D001374
CTDdecreases(expression)ALAD
D001374
CTDincreases(expression)APOBEC3F
D001374
CTDincreases(expression)APOBEC3G
D001374
CTDincreases(expression)AR
D001374
CTDincreases(response to substance)AR
D001374
CTDincreases(expression)ARHGAP35
D001374
CTDdecreases(expression)ARHGEF2
D001374
CTDincreases(expression)ART1
D001374
CTDincreases(expression)ASB2
D001374
CTDdecreases(expression)ATP2B1
D001374
CTDincreases(expression)ATP6V0C
D001374
CTDaffects(cotreatment)AURKA
D001374
CTDaffects(expression)AURKA
D001374
CTDincreases(expression)BAK1
D001374
CTDdecreases(expression)BAX
D001374
CTDincreases(reaction)BAX
D001374
CTDdecreases(expression)BCAT1
D001374
CTDdecreases(expression)BCL2
D001374
CTDdecreases(reaction)BCL2
D001374
CTDaffects(expression)BCL2L1
D001374
CTDaffects(cotreatment)BCL2L1
D001374
CTDdecreases(expression)BCL2L1
D001374
CTDincreases(expression)BCL2L13
D001374
CTDdecreases(expression)BICD1
D001374
CTDincreases(expression)BLK
D001374
CTDaffects(cotreatment)BUB1B
D001374
CTDaffects(expression)BUB1B
D001374
CTDincreases(expression)C3AR1
D001374
CTDincreases(expression)C6ORF62
D001374
CTDdecreases(methylation)CALCA
D001374
CTDincreases(expression)CALD1
D001374
CTDincreases(expression)CASP10
D001374
CTDaffects(expression)CASP3
D001374
CTDaffects(cotreatment)CASP3
D001374
CTDincreases(expression)CASP3
D001374
CTDincreases(expression)CASP5
D001374
CTDincreases(expression)CASP6
D001374
CTDincreases(expression)CASP8
D001374
CTDaffects(binding)CCNA1
D001374
CTDdecreases(reaction)CCNA1
D001374
CTDincreases(reaction)CCNA1
D001374
CTDdecreases(expression)CCNA1
D001374
CTDaffects(cotreatment)CCNA2
D001374
CTDaffects(expression)CCNA2
D001374
CTDdecreases(expression)CCNA2
D001374
CTDaffects(cotreatment)CCNB1
D001374
CTDaffects(expression)CCNB1
D001374
CTDdecreases(expression)CCNB1
D001374
CTDincreases(expression)CCNB1
D001374
CTDdecreases(reaction)CCNB1
D001374
CTDincreases(expression)CCND1
D001374
CTDaffects(methylation)CCND2
D001374
CTDaffects(expression)CCND2
D001374
CTDaffects(methylation)CCND2
D001374
CTDdecreases(expression)CCNG2
D001374
CTDaffects(cotreatment)CDC20
D001374
CTDaffects(expression)CDC20
D001374
CTDdecreases(expression)CDC42BPA
D001374
CTDdecreases(methylation)CDH1
D001374
CTDincreases(expression)CDH1
D001374
CTDincreases(expression)CDK1
D001374
CTDaffects(cotreatment)CDK1
D001374
CTDaffects(expression)CDK1
D001374
CTDdecreases(expression)CDK2
D001374
CTDdecreases(expression)CDK4
D001374
CTDincreases(expression)CDKN1A
D001374
CTDincreases(expression)CDKN1A
D001374
CTDincreases(expression)CDKN1A
D001374
CTDaffects(cotreatment)CDKN1A
D001374
CTDincreases(expression)CDKN1A
D001374
CTDdecreases(reaction)CDKN1A
D001374
CTDincreases(expression)CDKN1C
D001374
CTDaffects(methylation)CDKN2A
D001374
CTDdecreases(metabolic processing)CDKN2A
D001374
CTDdecreases(methylation)CDKN2A
D001374
CTDincreases(expression)CDKN2A
D001374
CTDdecreases(reaction)CDKN2A
D001374
CTDdecreases(methylation)CDKN2B
D001374
CTDaffects(response to substance)CDKN2B
D001374
CTDaffects(cotreatment)CDKN2B
D001374
CTDincreases(expression)CDKN2B
D001374
CTDdecreases(methylation)CEBPA
D001374
CTDaffects(cotreatment)CENPA
D001374
CTDaffects(expression)CENPA
D001374
CTDaffects(cotreatment)CENPF
D001374
CTDaffects(expression)CENPF
D001374
CTDincreases(expression)CENPO
D001374
CTDdecreases(expression)CHGA
D001374
CTDincreases(expression)CHIT1
D001374
CTDincreases(expression)CIITA
D001374
CTDincreases(reaction)CIITA
D001374
CTDdecreases(methylation)CIITA
D001374
CTDincreases(expression)CIITA
D001374
CTDincreases(reaction)CIITA
D001374
CTDincreases(expression)CIITA
D001374
CTDdecreases(expression)CLDN10
D001374
CTDdecreases(methylation)CLDN6
D001374
CTDincreases(expression)CLDN6
D001374
CTDaffects(cotreatment)CLDN6
D001374
CTDincreases(expression)CLDN8
D001374
CTDdecreases(methylation)CLDN9
D001374
CTDincreases(expression)CLDN9
D001374
CTDaffects(cotreatment)CLDN9
D001374
CTDdecreases(expression)CNNM2
D001374
CTDincreases(expression)COL14A1
D001374
CTDdecreases(reaction)COL1A1
D001374
CTDincreases(expression)COL1A1
D001374
CTDdecreases(expression)COL6A3
D001374
CTDincreases(expression)COX6A2
D001374
CTDincreases(expression)CPE
D001374
CTDincreases(expression)CPLX1
D001374
CTDaffects(binding)CREB1
D001374
CTDincreases(reaction)CREB1
D001374
CTDdecreases(expression)CREM
D001374
CTDincreases(expression)CSN1S1
D001374
CTDincreases(expression)CST3
D001374
CTDincreases(expression)CST4
D001374
CTDdecreases(methylation)CXCL12
D001374
CTDincreases(expression)CXCL12
D001374
CTDincreases(activity)CYP1A1
D001374
CTDincreases(reaction)CYP1A1
D001374
CTDincreases(expression)CYP1A1
D001374
CTDincreases(reaction)CYP1A1
D001374
CTDincreases(expression)CYP1A2
D001374
CTDincreases(reaction)CYP1A2
D001374
CTDincreases(expression)CYP1B1
D001374
CTDincreases(reaction)CYP1B1
D001374
CTDincreases(expression)CYTH1
D001374
CTDaffects(methylation)DAPK1
D001374
CTDaffects(cotreatment)DCN
D001374
CTDincreases(expression)DCN
D001374
CTDincreases(reaction)DCN
D001374
CTDdecreases(expression)DCN
D001374
CTDincreases(expression)DES
D001374
CTDaffects(cotreatment)DES
D001374
CTDdecreases(expression)DHX9
D001374
CTDdecreases(expression)DIO2
D001374
CTDdecreases(methylation)DLK1
D001374
CTDincreases(expression)DLX6
D001374
CTDdecreases(expression)DNMT1
D001374
CTDdecreases(reaction)DNMT1
D001374
CTDdecreases(expression)DNMT1
D001374
CTDincreases(uptake)DNMT1
D001374
CTDincreases(reaction)DNMT1
D001374
CTDdecreases(expression)DNMT3A
D001374
CTDdecreases(reaction)DNMT3A
D001374
CTDincreases(reaction)DNMT3A
D001374
CTDdecreases(methylation)DPYD
D001374
CTDdecreases(methylation)DPYD
D001374
CTDincreases(expression)DPYD
D001374
CTDdecreases(response to substance)DPYD
D001374
CTDincreases(expression)DUSP1
D001374
CTDincreases(expression)DUSP6
D001374
CTDaffects(reaction)E2F1
D001374
CTDdecreases(activity)E2F1
D001374
CTDdecreases(expression)E2F1
D001374
CTDdecreases(expression)EEF1A1
D001374
CTDincreases(expression)EFNA3
D001374
CTDincreases(expression)EGR2
D001374
CTDdecreases(expression)EIF3LP3
D001374
CTDdecreases(expression)ENO2
D001374
CTDincreases(expression)ENTPD1
D001374
CTDincreases(expression)ESR1
D001374
CTDaffects(binding)ETS1
D001374
CTDincreases(reaction)ETS1
D001374
CTDdecreases(expression)EYA1
D001374
CTDdecreases(expression)FADS2
D001374
CTDincreases(expression)FAM129A
D001374
CTDincreases(reaction)FAM129A
D001374
CTDincreases(expression)FAM8A1
D001374
CTDincreases(response to substance)FASLG
D001374
CTDincreases(expression)FBLN1
D001374
CTDaffects(cotreatment)FEN1
D001374
CTDaffects(expression)FEN1
D001374
CTDdecreases(expression)FGF7
D001374
CTDdecreases(expression)FILIP1L
D001374
CTDaffects(cotreatment)FOXO1
D001374
CTDincreases(expression)FOXO1
D001374
CTDincreases(expression)FYN
D001374
CTDincreases(expression)GABARAPL3
D001374
CTDincreases(expression)GABRB1
D001374
CTDdecreases(methylation)GADD45A
D001374
CTDincreases(expression)GADD45A
D001374
CTDincreases(expression)GADD45A
D001374
CTDincreases(response to substance)GADD45A
D001374
CTDdecreases(reaction)GADD45A
D001374
CTDincreases(expression)GADD45A
D001374
CTDincreases(reaction)GADD45A
D001374
CTDincreases(expression)GADD45B
D001374
CTDincreases(reaction)GADD45B
D001374
CTDdecreases(expression)GBP2
D001374
CTDdecreases(expression)GCNT2
D001374
CTDdecreases(expression)GJA1
D001374
CTDaffects(methylation)GNG7
D001374
CTDincreases(expression)GPKOW
D001374
CTDdecreases(expression)GPNMB
D001374
CTDincreases(expression)GUK1
D001374
CTDdecreases(reaction)GZMB
D001374
CTDincreases(secretion)GZMB
D001374
CTDincreases(expression)H1F0
D001374
CTDincreases(expression)H2AFX
D001374
CTDincreases(expression)HGD
D001374
CTDincreases(expression)HGF
D001374
CTDaffects(binding)HIST3H3
D001374
CTDincreases(reaction)HIST3H3
D001374
CTDaffects(binding)HIST4H4
D001374
CTDincreases(reaction)HIST4H4
D001374
CTDincreases(expression)HLA-DRA
D001374
CTDincreases(reaction)HLA-DRA
D001374
CTDincreases(expression)HMGA1
D001374
CTDincreases(expression)HMGA2
D001374
CTDincreases(reaction)HMGA2
D001374
CTDaffects(cotreatment)HOXA1
D001374
CTDdecreases(expression)HOXA1
D001374
CTDdecreases(reaction)HOXA1
D001374
CTDincreases(expression)HOXA1
D001374
CTDdecreases(methylation)HPGD
D001374
CTDincreases(expression)HPGD
D001374
CTDincreases(reaction)HPGD
D001374
CTDincreases(expression)HRK
D001374
CTDincreases(expression)HSPA6
D001374
CTDincreases(expression)ID1
D001374
CTDincreases(expression)ID3
D001374
CTDincreases(expression)IFNG
D001374
CTDincreases(reaction)IFNG
D001374
CTDdecreases(methylation)IFNG
D001374
CTDincreases(expression)IFNG
D001374
CTDincreases(secretion)IFNG
D001374
CTDaffects(cotreatment)IGFBP1
D001374
CTDdecreases(reaction)IGFBP1
D001374
CTDincreases(expression)IGFBP1
D001374
CTDincreases(reaction)IGFBP1
D001374
CTDincreases(expression)IGFBP4
D001374
CTDincreases(expression)IL12B
D001374
CTDdecreases(reaction)IL2
D001374
CTDincreases(secretion)IL2
D001374
CTDaffects(methylation)IL4
D001374
CTDaffects(methylation)IL6
D001374
CTDaffects(secretion)IL6
D001374
CTDaffects(expression)IL6R
D001374
CTDaffects(phosphorylation)IL6R
D001374
CTDincreases(expression)ISCA1
D001374
CTDdecreases(expression)ITGB1
D001374
CTDdecreases(expression)ITGB2
D001374
CTDaffects(cotreatment)KIF2C
D001374
CTDaffects(expression)KIF2C
D001374
CTDdecreases(methylation)KIR2DL1
D001374
CTDincreases(expression)KIR2DL1
D001374
CTDincreases(expression)KIR2DL1
D001374
CTDaffects(binding)KIR2DL2
D001374
CTDincreases(reaction)KIR2DL2
D001374
CTDdecreases(methylation)KIR2DL2
D001374
CTDincreases(expression)KIR2DL2
D001374
CTDdecreases(methylation)KIR2DL3
D001374
CTDincreases(expression)KIR2DL3
D001374
CTDincreases(expression)KIR2DL3
D001374
CTDaffects(binding)KIR2DL4
D001374
CTDincreases(reaction)KIR2DL4
D001374
CTDdecreases(methylation)KIR2DL4
D001374
CTDincreases(expression)KIR2DL4
D001374
CTDincreases(secretion)KIR2DL4
D001374
CTDincreases(expression)KIR2DS4
D001374
CTDdecreases(methylation)KIR3DL1
D001374
CTDincreases(expression)KIR3DL1
D001374
CTDincreases(expression)KIR3DL1
D001374
CTDincreases(expression)KLF6
D001374
CTDincreases(reaction)KLF6
D001374
CTDincreases(expression)KLK3
D001374
CTDincreases(expression)KRT19
D001374
CTDincreases(expression)KRT32
D001374
CTDaffects(cotreatment)KRT8
D001374
CTDdecreases(expression)KRT8
D001374
CTDdecreases(reaction)KRT8
D001374
CTDincreases(expression)KRT8
D001374
CTDdecreases(methylation)L1RE1
D001374
CTDdecreases(reaction)L1RE1
D001374
CTDincreases(expression)LAMB2
D001374
CTDincreases(expression)LDHB
D001374
CTDincreases(expression)LIMS1
D001374
CTDdecreases(expression)LITAF
D001374
CTDdecreases(expression)LTB4R
D001374
CTDincreases(expression)LYZ
D001374
CTDdecreases(expression)MAD1L1
D001374
CTDdecreases(methylation)MAGEA1
D001374
CTDdecreases(reaction)MAGEA1
D001374
CTDdecreases(methylation)MAGEA3
D001374
CTDdecreases(methylation)MAGEA3
D001374
CTDincreases(expression)MAGEA3
D001374
CTDincreases(expression)MAGEA3
D001374
CTDincreases(reaction)MAGEA3
D001374
CTDdecreases(expression)MAP1A
D001374
CTDdecreases(expression)MAP2K5
D001374
CTDdecreases(expression)MAPT
D001374
CTDaffects(cotreatment)MCM5
D001374
CTDaffects(expression)MCM5
D001374
CTDincreases(expression)MDC1
D001374
CTDincreases(expression)MDM2
D001374
CTDaffects(binding)MECP2
D001374
CTDdecreases(reaction)MECP2
D001374
CTDdecreases(expression)MEGF6
D001374
CTDdecreases(expression)MFAP2
D001374
CTDdecreases(methylation)MGMT
D001374
CTDincreases(expression)MGMT
D001374
CTDaffects(cotreatment)MKI67
D001374
CTDaffects(expression)MKI67
D001374
CTDincreases(expression)MMP1
D001374
CTDdecreases(reaction)MMP9
D001374
CTDincreases(expression)MMP9
D001374
CTDdecreases(expression)MORF4L2
D001374
CTDincreases(expression)MOV10L1
D001374
CTDincreases(expression)MSRB2
D001374
CTDdecreases(expression)MTHFD2
D001374
CTDdecreases(expression)MYC
D001374
CTDaffects(reaction)MYC
D001374
CTDdecreases(activity)MYC
D001374
CTDdecreases(expression)MYC
D001374
CTDincreases(expression)NEFL
D001374
CTDincreases(expression)NFATC1
D001374
CTDincreases(expression)NHP2L1
D001374
CTDincreases(expression)NKX2-5
D001374
CTDincreases(expression)NLGN3
D001374
CTDincreases(expression)NMI
D001374
CTDdecreases(expression)NOM1
D001374
CTDincreases(expression)NPHP1
D001374
CTDaffects(cotreatment)NR4A1
D001374
CTDincreases(expression)NR4A1
D001374
CTDdecreases(expression)NRIP1
D001374
CTDdecreases(expression)NRN1
D001374
CTDincreases(expression)NT5E
D001374
CTDdecreases(expression)NTS
D001374
CTDaffects(cotreatment)NUSAP1
D001374
CTDaffects(expression)NUSAP1
D001374
CTDincreases(expression)NXT2
D001374
CTDincreases(expression)OCLN
D001374
CTDincreases(expression)OGFRL1
D001374
CTDincreases(expression)OR8B8
D001374
CTDincreases(expression)OXR1
D001374
CTDdecreases(expression)OXTR
D001374
CTDincreases(expression)P4HB
D001374
CTDdecreases(expression)PAEP
D001374
CTDincreases(expression)PAK1
D001374
CTDdecreases(expression)PANK3
D001374
CTDincreases(expression)PAX4
D001374
CTDdecreases(expression)PCDH18
D001374
CTDdecreases(expression)PCDHB14
D001374
CTDdecreases(expression)PCDHB4
D001374
CTDincreases(expression)PDK1
D001374
CTDincreases(expression)PFN1
D001374
CTDincreases(expression)PHACTR2
D001374
CTDdecreases(expression)PIP5K1A
D001374
CTDdecreases(expression)PITPNC1
D001374
CTDincreases(expression)PJA1
D001374
CTDincreases(expression)PKD2L1
D001374
CTDincreases(expression)PKM
D001374
CTDdecreases(methylation)PLCB1
D001374
CTDincreases(expression)PLCB1
D001374
CTDincreases(response to substance)PLCB1
D001374
CTDdecreases(response to substance)PLCB1
D001374
CTDdecreases(expression)PLS3
D001374
CTDincreases(expression)PML
D001374
CTDincreases(expression)PPAP2A
D001374
CTDaffects(binding)PPP2CA
D001374
CTDincreases(reaction)PPP2CA
D001374
CTDdecreases(methylation)PPP2CA
D001374
CTDincreases(expression)PPP2CA
D001374
CTDincreases(expression)PPP2R4
D001374
CTDdecreases(reaction)PRF1
D001374
CTDincreases(secretion)PRF1
D001374
CTDaffects(cotreatment)PRL
D001374
CTDincreases(expression)PRL
D001374
CTDdecreases(expression)PRSS12
D001374
CTDincreases(expression)PSG1
D001374
CTDdecreases(expression)PTEN
D001374
CTDdecreases(reaction)PTEN
D001374
CTDincreases(methylation)PTEN
D001374
CTDdecreases(expression)PTHLH
D001374
CTDincreases(expression)PTPRC
D001374
CTDdecreases(methylation)RAB13
D001374
CTDincreases(expression)RAB1B
D001374
CTDincreases(expression)RACGAP1
D001374
CTDincreases(expression)RANBP2
D001374
CTDincreases(expression)RASA3
D001374
CTDdecreases(expression)RCN1
D001374
CTDaffects(localization)RELA
D001374
CTDdecreases(expression)RET
D001374
CTDaffects(cotreatment)RFC3
D001374
CTDaffects(expression)RFC3
D001374
CTDincreases(expression)RHOB
D001374
CTDincreases(reaction)RHOB
D001374
CTDaffects(cotreatment)RHOB
D001374
CTDincreases(expression)RIN1
D001374
CTDincreases(expression)RIPK2
D001374
CTDdecreases(expression)RPL5P29
D001374
CTDincreases(expression)RPP21
D001374
CTDdecreases(phosphorylation)RPS6
D001374
CTDdecreases(expression)RPSA
D001374
CTDdecreases(expression)RPSAP12
D001374
CTDdecreases(expression)RPSAP28
D001374
CTDdecreases(expression)RPSAP3
D001374
CTDdecreases(expression)RPSAP31
D001374
CTDaffects(cotreatment)RRM2
D001374
CTDaffects(expression)RRM2
D001374
CTDincreases(expression)RRM2B
D001374
CTDaffects(binding)RUNX1
D001374
CTDincreases(reaction)RUNX1
D001374
CTDaffects(methylation)RUNX3
D001374
CTDdecreases(expression)S100A14
D001374
CTDincreases(expression)S100A9
D001374
CTDincreases(expression)S100P
D001374
CTDaffects(methylation)SALL4
D001374
CTDincreases(expression)SCAMP4
D001374
CTDdecreases(expression)SDCBP
D001374
CTDincreases(expression)SEMA3A
D001374
CTDincreases(expression)SEMA6C
D001374
CTDincreases(expression)SENP3
D001374
CTDdecreases(expression)SIRPB1
D001374
CTDincreases(expression)SKIV2L2
D001374
CTDincreases(response to substance)SLC28A1
D001374
CTDincreases(uptake)SLC28A1
D001374
CTDdecreases(expression)SLC28A1
D001374
CTDaffects(reaction)SLC28A1
D001374
CTDdecreases(expression)SLC29A2
D001374
CTDaffects(cotreatment)SLC5A5
D001374
CTDaffects(expression)SLC5A5
D001374
CTDincreases(expression)SLC5A5
D001374
CTDaffects(expression)SOCS3
D001374
CTDdecreases(expression)SOX13
D001374
CTDaffects(binding)SP1
D001374
CTDincreases(reaction)SP1
D001374
CTDdecreases(expression)SP1
D001374
CTDaffects(cotreatment)SPAG5
D001374
CTDaffects(expression)SPAG5
D001374
CTDdecreases(expression)SRPX
D001374
CTDdecreases(expression)SRSF7
D001374
CTDincreases(expression)SSFA2
D001374
CTDincreases(expression)SSX2IP
D001374
CTDincreases(expression)ST3GAL6
D001374
CTDdecreases(expression)ST8SIA2
D001374
CTDaffects(expression)STAT3
D001374
CTDaffects(phosphorylation)STAT3
D001374
CTDdecreases(expression)STC2
D001374
CTDdecreases(expression)STK38
D001374
CTDdecreases(expression)SULF1
D001374
CTDincreases(expression)SULT1C2
D001374
CTDdecreases(expression)TBC1D4
D001374
CTDdecreases(expression)TCEA1
D001374
CTDincreases(expression)TECPR2
D001374
CTDdecreases(expression)TERT
D001374
CTDdecreases(activity)TERT
D001374
CTDdecreases(expression)TERT
D001374
CTDdecreases(methylation)TERT
D001374
CTDaffects(reaction)TERT
D001374
CTDincreases(expression)TFE3
D001374
CTDdecreases(expression)TGFB1
D001374
CTDdecreases(reaction)TGFB1
D001374
CTDincreases(expression)TGFB1
D001374
CTDincreases(methylation)TGFB1
D001374
CTDincreases(phosphorylation)TGFB1
D001374
CTDincreases(expression)THUMPD1
D001374
CTDincreases(expression)TIMP1
D001374
CTDincreases(expression)TJP1
D001374
CTDincreases(expression)TMED3
D001374
CTDaffects(cotreatment)TMPO
D001374
CTDaffects(expression)TMPO
D001374
CTDdecreases(expression)TNC
D001374
CTDincreases(response to substance)TNF
D001374
CTDincreases(expression)TNFRSF1B
D001374
CTDincreases(response to substance)TNFSF10
D001374
CTDaffects(cotreatment)TOP2A
D001374
CTDaffects(expression)TOP2A
D001374
CTDaffects(cotreatment)TOP2A
D001374
CTDdecreases(expression)TOP2A
D001374
CTDincreases(expression)TP53
D001374
CTDdecreases(reaction)TP53
D001374
CTDdecreases(expression)TP53
D001374
CTDincreases(reaction)TP53
D001374
CTDincreases(response to substance)TP53
D001374
CTDincreases(expression)TP73
D001374
CTDincreases(reaction)TP73
D001374
CTDincreases(expression)TPM2
D001374
CTDincreases(expression)TPO
D001374
CTDdecreases(expression)TPSG1
D001374
CTDdecreases(expression)TRH
D001374
CTDdecreases(expression)TRIB1
D001374
CTDincreases(expression)TRIM8
D001374
CTDaffects(expression)TSC1
D001374
CTDaffects(methylation)TSC1
D001374
CTDaffects(expression)TSC2
D001374
CTDaffects(methylation)TSC2
D001374
CTDdecreases(methylation)TSC2
D001374
CTDincreases(expression)TSC2
D001374
CTDincreases(expression)TSHR
D001374
CTDdecreases(expression)TSPAN32
D001374
CTDaffects(cotreatment)TTK
D001374
CTDaffects(expression)TTK
D001374
CTDaffects(cotreatment)UBE2C
D001374
CTDaffects(expression)UBE2C
D001374
CTDincreases(expression)UHMK1
D001374
CTDincreases(expression)USH2A
D001374
CTDdecreases(expression)USHBP1
D001374
CTDaffects(cotreatment)VIM
D001374
CTDincreases(expression)VIM
D001374
CTDdecreases(expression)WDR47
D001374
CTDincreases(expression)WNT5A
D001374
CTDincreases(expression)WWTR1
D001374
CTDdecreases(expression)XAF1
D001374
CTDdecreases(methylation)XAF1
D001374
CTDincreases(expression)XAF1
D001374
CTDincreases(expression)XAF1
D001374
CTDaffects(methylation)ZFP64
D001374
CTDdecreases(expression)ZNF189
D001374
CTDincreases(expression)ZP3
D001374
PubChem PotencyuM22.387ALDH1A1-GI(Protien) :
PubChem Potency-Replicate_1uM1.096AR-GI(Protien) :
PubChem AR Potency (uM)uM2.342AR-GI(Protien) :
PubChem Potency-Replicate_1uM2.731AR-GI(Protien) :
PubChem Potency-Replicate_1uM3.378AR-GI(Protien) :
PubChem Potency-Replicate_1uM5.956AR-GI(Protien) :
PubChem PotencyuM1.254ATAD5-GI(Protien) :
PubChem PotencyuM2.818ATAD5-GI(Protien) :
PubChem PotencyuM5.601ATAD5-GI(Protien) :
PubChem PotencyuM8.196ATAD5-GI(Protien) :
PubChem PotencyuM15.785ATAD5-GI(Protien) :
PubChem Potency-Replicate_1uM8.635CYP19A1-GI(Protien) :
PubChem Potency-Replicate_1uM13.333CYP19A1-GI(Protien) :
PubChem PotencyuM3.162GMNN-GI(Protien) :
PubChem PotencyuM1.259HBB-GI(Protien) :
PubChem PotencyuM12.589HTT-GI(Protien) :
PubChem PotencyuM1.636IDH1-GI(Protien) :
PubChem NoneuMMDM2-GI(Protien) :
PubChem NoneuMMDM2-GI(Protien) :
PubChem NoneuMMDM4-GI(Protien) :
PubChem NoneuMMDM4-GI(Protien) :
PubChem NoneuMMITF-GI(Protien) :
PubChem NoneuMNCOA1-GI(Protien) :
PubChem NoneuMNCOA3-GI(Protien) :
PubChem NoneuMNCOA3-GI(Protien) :
PubChem PotencyuM1.369NFE2L2-GI(Protien) :
PubChem Potency-Replicate_1uM1.536NFE2L2-GI(Protien) :
PubChem Ratio Potency (uM)uM1.790NFE2L2-GI(Protien) :
PubChem PotencyuM1.883NFE2L2-GI(Protien) :
PubChem Potency-Replicate_1uM2.660NFE2L2-GI(Protien) :
PubChem Ratio Potency (uM)uM3.223NFE2L2-GI(Protien) :
PubChem NoneuMNR1H4-GI(Protien) :
PubChem Potency-Replicate_1uM1.738NR3C1-GI(Protien) :
PubChem Potency-Replicate_1uM3.011NR3C1-GI(Protien) :
PubChem PotencyuM5.623NR3C1-GI(Protien) :
PubChem PotencyuM7.943NR3C1-GI(Protien) :
PubChem NoneuMNR3C1-GI(Protien) :
PubChem NoneuMNR5A1-GI(Protien) :
PubChem NoneuMNR5A2-GI(Protien) :
PubChem NoneuMNR5A2-GI(Protien) :
PubChem NoneuMPRNP-GI(Protien) :
PubChem PotencyuM11.220SMAD3-GI(Protien) :
PubChem PotencyuM2.512TDP1-GI(Protien) :
PubChem PotencyuM3.162TDP1-GI(Protien) :
PubChem PotencyuM6.684TDP1-GI(Protien) :
PubChem PotencyuM7.308TDP1-GI(Protien) :
PubChem PotencyuM7.499TDP1-GI(Protien) :
PubChem PotencyuM8.200TDP1-GI(Protien) :
PubChem PotencyuM3.162THPO-GI(Protien) :
ChEMBLPotencynM22387.200ALDH1A1
-Target : CHEMBL3577
ChEMBLPotencynM2818.400ATAD5
-Target : CHEMBL1741209
ChEMBLPotencynM8196.100ATAD5
-Target : CHEMBL1741209
ChEMBLPotencynM3162.300GMNN
-Target : CHEMBL1293278
ChEMBLPotencynM1258.900HBB
-Target : CHEMBL4331
ChEMBLPotencynM12589.300HTT
-Target : CHEMBL5514
ChEMBLPotencynM3162.300THPO
-Target : CHEMBL1293256
Download gene sets gmt, text, Detailed text
Contact us
Tan Lab , Mail Stop 8117
12801 East 17th Avenue
Division of Medical Oncology , Department of Medicine
University of Colorado School of Medicine
Aurora, CO 80045, USA

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