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Gene Set: D4 : CTD - Amiodarone


Collection D4 : CTD
Chemical Name Amiodarone ( From PubChem : AMIODARONE )
FDA NPC WHO Indian Australia China Traditional
Herbal
Clinical
Trail
ApprovedNotApprovedApprovedNotApprovedNotNot
Molecular
Weight
Hydrogen Bond
Donor Count
Hydrogen Bond
Acceptor Count
cLogP Lipinski Rule
645.312 g/mol 0 4 6.9362 False(2/4)
Structure
InChI InChI=1S/C25H29I2NO3/c1-4-7-11-22-23(18-10-8-9-12-21(18)31-22)24(29)17-15-19(26)25(20(27)16-17)30-14-13-28(5-2)6-3/h8-10,12,15-16H,4-7,11,13-14H2,1-3H3
InChIKey IYIKLHRQXLHMJQ-UHFFFAOYSA-N
Links

Gene (625 / 765)


⊖ Less

Source Type Unit Value Gene PMID Assay Other
CTDincreases(expression)ABCA2
D000638
CTDdecreases(reaction)ABCB1
D000638
CTDincreases(secretion)ABCB1
D000638
CTDdecreases(reaction)ABCB1
D000638
CTDincreases(transport)ABCB1
D000638
CTDdecreases(activity)ABCB1
D000638
CTDdecreases(reaction)ABCB11
D000638
CTDincreases(transport)ABCB11
D000638
CTDdecreases(activity)ABCB11
D000638
CTDincreases(expression)ABCC11
D000638
CTDincreases(expression)ABL1
D000638
CTDincreases(expression)ACACA
D000638
CTDincreases(expression)ACOT8
D000638
CTDincreases(expression)ACSF3
D000638
CTDincreases(expression)ACTR3B
D000638
CTDincreases(expression)ACVR1B
D000638
CTDincreases(expression)ACYP1
D000638
CTDincreases(expression)ADGRD1
D000638
CTDincreases(expression)ADORA3
D000638
CTDincreases(expression)ADRA2A
D000638
CTDdecreases(expression)ADRB1
D000638
CTDdecreases(expression)ADRB2
D000638
CTDincreases(expression)AGT
D000638
CTDdecreases(reaction)AGT
D000638
CTDaffects(cotreatment)AGT
D000638
CTDincreases(reaction)AGT
D000638
CTDincreases(expression)AHNAK
D000638
CTDincreases(expression)AKR1C1
D000638
CTDdecreases(phosphorylation)AKT1
D000638
CTDincreases(expression)ALAS1
D000638
CTDincreases(expression)ALB
D000638
CTDincreases(expression)ALG12
D000638
CTDincreases(expression)ALG2
D000638
CTDincreases(expression)ALK
D000638
CTDincreases(expression)AMIGO1
D000638
CTDincreases(expression)ANXA4
D000638
CTDdecreases(expression)AP1S1
D000638
CTDincreases(expression)ARC
D000638
CTDincreases(expression)ARHGAP15
D000638
CTDincreases(expression)ARHGAP35
D000638
CTDincreases(expression)ARHGAP4
D000638
CTDincreases(expression)ARHGAP9
D000638
CTDincreases(expression)ARHGEF10L
D000638
CTDincreases(expression)ARHGEF7
D000638
CTDincreases(expression)ARHGEF9
D000638
CTDincreases(expression)ARID5A
D000638
CTDincreases(expression)ARMC9
D000638
CTDincreases(expression)ARPC4
D000638
CTDincreases(expression)ASAH1
D000638
CTDincreases(expression)ASB7
D000638
CTDincreases(expression)ASNS
D000638
CTDincreases(expression)ATF3
D000638
CTDincreases(expression)ATF4
D000638
CTDincreases(expression)ATF6B
D000638
CTDincreases(expression)ATG7
D000638
CTDaffects(reaction)ATG7
D000638
CTDincreases(cleavage)ATG7
D000638
CTDaffects(response to substance)ATG7
D000638
CTDincreases(expression)ATOH1
D000638
CTDincreases(expression)ATP11C
D000638
CTDincreases(expression)BAG1
D000638
CTDincreases(expression)BAIAP2L1
D000638
CTDincreases(expression)BAX
D000638
CTDincreases(expression)BBOX1
D000638
CTDaffects(cotreatment)BCL2
D000638
CTDdecreases(expression)BCL2
D000638
CTDincreases(expression)BCL2L11
D000638
CTDincreases(expression)BHLHE40
D000638
CTDaffects(cotreatment)BID
D000638
CTDincreases(cleavage)BID
D000638
CTDincreases(expression)BMP2K
D000638
CTDincreases(expression)BOLA2
D000638
CTDincreases(expression)BOLL
D000638
CTDincreases(expression)BRCC3
D000638
CTDincreases(expression)BRPF1
D000638
CTDincreases(expression)BSG
D000638
CTDincreases(expression)C10ORF10
D000638
CTDincreases(expression)C11ORF16
D000638
CTDincreases(expression)C16ORF74
D000638
CTDincreases(expression)C1ORF95
D000638
CTDincreases(expression)C21ORF67
D000638
CTDincreases(expression)C21ORF91
D000638
CTDincreases(expression)C2CD4B
D000638
CTDincreases(expression)C3ORF18
D000638
CTDincreases(expression)C3ORF33
D000638
CTDincreases(expression)C6ORF141
D000638
CTDincreases(expression)C7ORF31
D000638
CTDincreases(expression)CAMK2A
D000638
CTDincreases(expression)CAPN11
D000638
CTDincreases(expression)CAPN3
D000638
CTDincreases(expression)CARD9
D000638
CTDincreases(expression)CASKIN2
D000638
CTDincreases(cleavage)CASP3
D000638
CTDincreases(reaction)CASP3
D000638
CTDincreases(activity)CASP3
D000638
CTDincreases(reaction)CASP3
D000638
CTDincreases(activity)CASP3
D000638
CTDincreases(expression)CASP3
D000638
CTDaffects(reaction)CASP3
D000638
CTDaffects(cotreatment)CASP3
D000638
CTDincreases(cleavage)CASP3
D000638
CTDincreases(activity)CASP7
D000638
CTDincreases(reaction)CASP7
D000638
CTDincreases(activity)CASP7
D000638
CTDaffects(cotreatment)CASP8
D000638
CTDincreases(cleavage)CASP8
D000638
CTDincreases(expression)CASP9
D000638
CTDaffects(cotreatment)CASP9
D000638
CTDincreases(cleavage)CASP9
D000638
CTDincreases(expression)CAV3
D000638
CTDincreases(expression)CCDC134
D000638
CTDincreases(expression)CCDC17
D000638
CTDincreases(expression)CCDC9
D000638
CTDincreases(expression)CCDC96
D000638
CTDdecreases(reaction)CCL2
D000638
CTDincreases(expression)CCL2
D000638
CTDincreases(expression)CCL2
D000638
CTDincreases(expression)CCNT1
D000638
CTDincreases(expression)CCR9
D000638
CTDincreases(expression)CD320
D000638
CTDaffects(cotreatment)CD86
D000638
CTDincreases(expression)CD86
D000638
CTDincreases(expression)CDC25A
D000638
CTDincreases(expression)CDC42SE1
D000638
CTDincreases(expression)CDH15
D000638
CTDincreases(expression)CDH26
D000638
CTDincreases(expression)CDK17
D000638
CTDincreases(expression)CEBPB
D000638
CTDincreases(expression)CECR1
D000638
CTDincreases(expression)CELF6
D000638
CTDincreases(expression)CES1
D000638
CTDincreases(expression)CHAC1
D000638
CTDincreases(expression)CHGA
D000638
CTDincreases(expression)CHRNB3
D000638
CTDincreases(expression)CHST6
D000638
CTDincreases(expression)CLCN5
D000638
CTDincreases(expression)CLCN6
D000638
CTDincreases(expression)CLTCL1
D000638
CTDincreases(expression)CLVS2
D000638
CTDincreases(expression)CMTM7
D000638
CTDincreases(expression)CMYA5
D000638
CTDincreases(expression)CNIH3
D000638
CTDincreases(expression)CNNM2
D000638
CTDincreases(expression)CNOT7
D000638
CTDincreases(expression)CNP
D000638
CTDincreases(expression)COL11A1
D000638
CTDincreases(expression)COL27A1
D000638
CTDincreases(expression)COL8A2
D000638
CTDincreases(expression)CORO2A
D000638
CTDincreases(expression)CPLX2
D000638
CTDincreases(expression)CRB3
D000638
CTDdecreases(reaction)CRP
D000638
CTDincreases(expression)CRP
D000638
CTDincreases(expression)CST6
D000638
CTDincreases(expression)CST7
D000638
CTDincreases(expression)CTC1
D000638
CTDincreases(expression)CTLA4
D000638
CTDaffects(cotreatment)CXCL8
D000638
CTDincreases(expression)CXCL8
D000638
CTDincreases(secretion)CXCL8
D000638
CTDdecreases(reaction)CXCL8
D000638
CTDdecreases(activity)CYP1A2
D000638
CTDincreases(expression)CYP26A1
D000638
CTDdecreases(activity)CYP2C8
D000638
CTDincreases(metabolic processing)CYP2C8
D000638
CTDdecreases(reaction)CYP2C8
D000638
CTDaffects(metabolic processing)CYP2C9
D000638
CTDdecreases(reaction)CYP2C9
D000638
CTDincreases(reaction)CYP2C9
D000638
CTDincreases(metabolic processing)CYP2C9
D000638
CTDincreases(reaction)CYP2C9
D000638
CTDdecreases(activity)CYP2C9
D000638
CTDdecreases(activity)CYP2C9
D000638
CTDdecreases(chemical synthesis)CYP2C9
D000638
CTDdecreases(activity)CYP2D6
D000638
CTDincreases(expression)CYP2D6
D000638
CTDaffects(reaction)CYP2D6
D000638
CTDincreases(abundance)CYP2D6
D000638
CTDincreases(expression)CYP2J2
D000638
CTDincreases(expression)CYP2R1
D000638
CTDdecreases(ethylation)CYP3A
D000638
CTDaffects(cotreatment)CYP3A4
D000638
CTDincreases(expression)CYP3A4
D000638
CTDincreases(secretion)CYP3A4
D000638
CTDdecreases(reaction)CYP3A4
D000638
CTDincreases(hydroxylation)CYP3A4
D000638
CTDdecreases(reaction)CYP3A4
D000638
CTDincreases(oxidation)CYP3A4
D000638
CTDdecreases(activity)CYP3A4
D000638
CTDdecreases(ethylation)CYP3A4
D000638
CTDincreases(metabolic processing)CYP3A4
D000638
CTDincreases(response to substance)CYP3A4
D000638
CTDdecreases(reaction)CYP3A4
D000638
CTDdecreases(reaction)CYP3A4
D000638
CTDincreases(metabolic processing)CYP3A4
D000638
CTDincreases(expression)DAPK2
D000638
CTDincreases(expression)DBN1
D000638
CTDincreases(expression)DBNDD1
D000638
CTDincreases(expression)DCST2
D000638
CTDincreases(expression)DCTN1
D000638
CTDincreases(expression)DDIT3
D000638
CTDincreases(expression)DDIT3
D000638
CTDdecreases(reaction)DDIT3
D000638
CTDincreases(expression)DDIT4
D000638
CTDincreases(expression)DDX17
D000638
CTDincreases(expression)DDX31
D000638
CTDincreases(expression)DDX39A
D000638
CTDincreases(expression)DDX49
D000638
CTDincreases(expression)DEDD
D000638
CTDincreases(expression)DEPTOR
D000638
CTDincreases(expression)DHRS2
D000638
CTDincreases(expression)DHX57
D000638
CTDdecreases(activity)DIO1
D000638
CTDincreases(expression)DLG4
D000638
CTDincreases(expression)DLK2
D000638
CTDincreases(expression)DNAAF3
D000638
CTDincreases(expression)DNAH7
D000638
CTDincreases(expression)DNAJB12
D000638
CTDincreases(expression)DNAJB7
D000638
CTDincreases(expression)DNAJB9
D000638
CTDincreases(expression)DNASE1
D000638
CTDincreases(expression)DOCK5
D000638
CTDincreases(expression)DPM2
D000638
CTDincreases(expression)DRC7
D000638
CTDincreases(expression)DUSP1
D000638
CTDincreases(expression)DUSP10
D000638
CTDincreases(expression)DUT
D000638
CTDincreases(expression)EAF2
D000638
CTDincreases(expression)EED
D000638
CTDincreases(expression)EEPD1
D000638
CTDincreases(expression)EFCAB5
D000638
CTDincreases(expression)EFCC1
D000638
CTDincreases(expression)EGFL6
D000638
CTDincreases(expression)EGR1
D000638
CTDincreases(expression)EGR2
D000638
CTDincreases(expression)EHMT1
D000638
CTDincreases(phosphorylation)EIF2A
D000638
CTDincreases(expression)EIF2AK3
D000638
CTDaffects(binding)EIF4E
D000638
CTDincreases(reaction)EIF4E
D000638
CTDdecreases(reaction)EIF4EBP1
D000638
CTDincreases(phosphorylation)EIF4EBP1
D000638
CTDaffects(binding)EIF4EBP1
D000638
CTDincreases(reaction)EIF4EBP1
D000638
CTDdecreases(phosphorylation)EIF4EBP1
D000638
CTDincreases(expression)EIF5
D000638
CTDincreases(expression)ELMO3
D000638
CTDincreases(expression)ENPP7
D000638
CTDincreases(expression)EPC1
D000638
CTDincreases(expression)EPC2
D000638
CTDincreases(expression)ERI2
D000638
CTDincreases(expression)ERMN
D000638
CTDincreases(expression)ETV7
D000638
CTDincreases(expression)EXO1
D000638
CTDdecreases(reaction)F2
D000638
CTDincreases(activity)F2
D000638
CTDincreases(expression)F2
D000638
CTDdecreases(reaction)F3
D000638
CTDincreases(activity)F3
D000638
CTDincreases(expression)F3
D000638
CTDincreases(expression)FABP1
D000638
CTDdecreases(activity)FADS2
D000638
CTDdecreases(reaction)FADS2
D000638
CTDincreases(expression)FADS2
D000638
CTDaffects(reaction)FADS2
D000638
CTDincreases(uptake)FADS2
D000638
CTDincreases(expression)FAM129A
D000638
CTDincreases(expression)FAM150A
D000638
CTDincreases(expression)FAM153A
D000638
CTDincreases(expression)FAM212B
D000638
CTDincreases(expression)FAM81A
D000638
CTDincreases(expression)FAM89A
D000638
CTDincreases(expression)FANCA
D000638
CTDincreases(expression)FARP2
D000638
CTDincreases(expression)FBXO16
D000638
CTDincreases(expression)FBXO32
D000638
CTDincreases(expression)FCRL1
D000638
CTDincreases(expression)FCRL2
D000638
CTDincreases(expression)FCRL3
D000638
CTDincreases(expression)FFAR3
D000638
CTDincreases(expression)FGD4
D000638
CTDincreases(expression)FGD5
D000638
CTDincreases(expression)FGFR1OP2
D000638
CTDincreases(expression)FIBCD1
D000638
CTDincreases(expression)FKBP10
D000638
CTDincreases(expression)FLCN
D000638
CTDincreases(expression)FNDC4
D000638
CTDincreases(expression)FOS
D000638
CTDaffects(cotreatment)FOS
D000638
CTDincreases(expression)FOS
D000638
CTDincreases(reaction)FOS
D000638
CTDincreases(expression)FOSB
D000638
CTDincreases(expression)FOXP3
D000638
CTDincreases(expression)FRAS1
D000638
CTDincreases(expression)FRMD3
D000638
CTDincreases(expression)FRMD5
D000638
CTDincreases(expression)FUNDC2
D000638
CTDincreases(expression)FUZ
D000638
CTDincreases(expression)FXYD1
D000638
CTDincreases(expression)G6PD
D000638
CTDincreases(expression)GADD45A
D000638
CTDincreases(expression)GADD45G
D000638
CTDincreases(expression)GAL3ST3
D000638
CTDincreases(expression)GBP2
D000638
CTDincreases(expression)GDF15
D000638
CTDincreases(expression)GDF5
D000638
CTDincreases(expression)GDPD3
D000638
CTDincreases(expression)GEM
D000638
CTDincreases(expression)GFOD1
D000638
CTDincreases(expression)GINS1
D000638
CTDincreases(expression)GJA5
D000638
CTDincreases(expression)GJD3
D000638
CTDincreases(expression)GK5
D000638
CTDincreases(expression)GKAP1
D000638
CTDincreases(expression)GNAS
D000638
CTDincreases(expression)GON4L
D000638
CTDincreases(expression)GPRC5C
D000638
CTDincreases(activity)GPT
D000638
CTDincreases(expression)GPT
D000638
CTDincreases(expression)GRM2
D000638
CTDincreases(expression)GSTO2
D000638
CTDincreases(expression)GSTZ1
D000638
CTDincreases(expression)GUCY1A2
D000638
CTDincreases(expression)GUCY1B3
D000638
CTDincreases(expression)H2AFJ
D000638
CTDincreases(expression)HCN1
D000638
CTDincreases(expression)HDX
D000638
CTDincreases(expression)HELB
D000638
CTDincreases(expression)HERPUD1
D000638
CTDincreases(expression)HEXIM1
D000638
CTDincreases(expression)HGFAC
D000638
CTDincreases(expression)HIRA
D000638
CTDincreases(expression)HIST1H2AM
D000638
CTDincreases(expression)HIST1H2BE
D000638
CTDincreases(expression)HIST1H3I
D000638
CTDincreases(expression)HIST1H3J
D000638
CTDincreases(expression)HIST1H4H
D000638
CTDincreases(expression)HLA-DPB1
D000638
CTDincreases(expression)HMGXB4
D000638
CTDincreases(expression)HMHA1
D000638
CTDincreases(expression)HMOX1
D000638
CTDincreases(expression)HNF4G
D000638
CTDincreases(expression)HNRNPA1
D000638
CTDincreases(expression)HOXB6
D000638
CTDincreases(expression)HOXC4
D000638
CTDincreases(expression)HPN
D000638
CTDincreases(expression)HRK
D000638
CTDincreases(expression)HUS1
D000638
CTDaffects(cotreatment)ICAM1
D000638
CTDincreases(expression)ICAM1
D000638
CTDincreases(expression)ICAM1
D000638
CTDincreases(expression)ID2
D000638
CTDincreases(expression)IGFALS
D000638
CTDincreases(expression)IGSF8
D000638
CTDincreases(expression)IKBKAP
D000638
CTDincreases(expression)IL10RA
D000638
CTDincreases(expression)IL1A
D000638
CTDaffects(cotreatment)IL1A
D000638
CTDincreases(response to substance)IL1A
D000638
CTDincreases(expression)IL6
D000638
CTDincreases(secretion)IL6
D000638
CTDaffects(cotreatment)IL6
D000638
CTDincreases(response to substance)IL6
D000638
CTDdecreases(reaction)IL6
D000638
CTDincreases(expression)INHBE
D000638
CTDincreases(expression)IPPK
D000638
CTDincreases(expression)IRAK2
D000638
CTDincreases(expression)IRF1
D000638
CTDincreases(expression)ISX
D000638
CTDdecreases(expression)ITGB5
D000638
CTDincreases(expression)ITIH2
D000638
CTDincreases(expression)JAKMIP3
D000638
CTDincreases(expression)JRKL
D000638
CTDaffects(cotreatment)JUN
D000638
CTDincreases(expression)JUN
D000638
CTDincreases(reaction)JUN
D000638
CTDincreases(expression)KCNE5
D000638
CTDaffects(activity)KCNH2
D000638
CTDaffects(binding)KCNH2
D000638
CTDdecreases(activity)KCNH2
D000638
CTDdecreases(reaction)KCNH2
D000638
CTDincreases(transport)KCNH2
D000638
CTDdecreases(activity)KCNH2
D000638
CTDincreases(reaction)KCNH2
D000638
CTDdecreases(activity)KCNH2
D000638
CTDdecreases(activity)KCNH2
D000638
CTDdecreases(reaction)KCNH2
D000638
CTDincreases(expression)KCNJ2
D000638
CTDincreases(expression)KCNK12
D000638
CTDincreases(expression)KCNMA1
D000638
CTDincreases(expression)KCTD14
D000638
CTDincreases(expression)KIF16B
D000638
CTDincreases(expression)KIF17
D000638
CTDincreases(expression)KIFC1
D000638
CTDincreases(expression)KIR2DL5B
D000638
CTDincreases(expression)KITLG
D000638
CTDincreases(expression)KLF10
D000638
CTDincreases(expression)KLF15
D000638
CTDincreases(expression)KLF16
D000638
CTDincreases(expression)KLF4
D000638
CTDincreases(expression)KLHL28
D000638
CTDincreases(expression)KLK14
D000638
CTDincreases(expression)KRT17
D000638
CTDincreases(expression)L3MBTL1
D000638
CTDincreases(expression)LACRT
D000638
CTDincreases(expression)LCTL
D000638
CTDincreases(expression)LDLR
D000638
CTDincreases(reaction)LDLR
D000638
CTDdecreases(expression)LDLR
D000638
CTDincreases(expression)LELP1
D000638
CTDincreases(expression)LHCGR
D000638
CTDincreases(expression)LIF
D000638
CTDincreases(expression)LIMS3
D000638
CTDincreases(expression)LIN7A
D000638
CTDincreases(expression)LINC00472
D000638
CTDincreases(expression)LINC00521
D000638
CTDincreases(expression)LRP5
D000638
CTDincreases(expression)LSS
D000638
CTDincreases(expression)LYZ
D000638
CTDincreases(expression)MACROD2
D000638
CTDincreases(expression)MAFG
D000638
CTDincreases(expression)MAGED4B
D000638
CTDincreases(expression)MASP1
D000638
CTDincreases(expression)MCAM
D000638
CTDincreases(expression)MCF2
D000638
CTDincreases(expression)MED11
D000638
CTDincreases(expression)MEF2C
D000638
CTDincreases(expression)MFHAS1
D000638
CTDincreases(expression)MGAT4A
D000638
CTDincreases(expression)MGST1
D000638
CTDincreases(expression)MICALL2
D000638
CTDincreases(expression)MID2
D000638
CTDincreases(expression)MITF
D000638
CTDincreases(expression)MMP23A
D000638
CTDincreases(expression)MORN5
D000638
CTDincreases(expression)MPI
D000638
CTDincreases(expression)MRPL10
D000638
CTDincreases(expression)MS4A14
D000638
CTDincreases(expression)MT1F
D000638
CTDincreases(expression)MT1G
D000638
CTDincreases(expression)MT1X
D000638
CTDdecreases(reaction)MTOR
D000638
CTDincreases(phosphorylation)MTOR
D000638
CTDincreases(expression)MXD1
D000638
CTDincreases(expression)MYEF2
D000638
CTDincreases(expression)MYH11
D000638
CTDincreases(expression)MYL4
D000638
CTDincreases(expression)MYLK2
D000638
CTDincreases(expression)MYO3A
D000638
CTDincreases(expression)N4BP3
D000638
CTDincreases(expression)NAA16
D000638
CTDincreases(expression)NANOS1
D000638
CTDincreases(expression)NBPF3
D000638
CTDincreases(expression)NEK8
D000638
CTDincreases(expression)NF2
D000638
CTDincreases(expression)NFIC
D000638
CTDincreases(expression)NFKBIA
D000638
CTDincreases(expression)NFKBIZ
D000638
CTDincreases(expression)NME8
D000638
CTDincreases(expression)NOL6
D000638
CTDincreases(expression)NOS1AP
D000638
CTDincreases(chemical synthesis)NOS3
D000638
CTDincreases(reaction)NOS3
D000638
CTDincreases(expression)NPSR1
D000638
CTDincreases(expression)NPTXR
D000638
CTDincreases(expression)NR4A2
D000638
CTDincreases(expression)NT5M
D000638
CTDincreases(expression)NTRK3
D000638
CTDincreases(expression)NUPR1
D000638
CTDincreases(expression)OCM
D000638
CTDincreases(expression)OPHN1
D000638
CTDincreases(expression)OR14I1
D000638
CTDincreases(expression)OR2B2
D000638
CTDincreases(expression)OR2D2
D000638
CTDincreases(expression)OR4C16
D000638
CTDincreases(expression)OR4F5
D000638
CTDincreases(expression)OR52N2
D000638
CTDincreases(expression)OR6T1
D000638
CTDincreases(expression)OR9Q2
D000638
CTDincreases(expression)OSBP2
D000638
CTDincreases(expression)OXSM
D000638
CTDaffects(cotreatment)PARP1
D000638
CTDincreases(cleavage)PARP1
D000638
CTDaffects(cotreatment)PARP1
D000638
CTDincreases(cleavage)PARP1
D000638
CTDincreases(expression)PAX3
D000638
CTDincreases(expression)PCDH1
D000638
CTDincreases(expression)PCDH7
D000638
CTDincreases(expression)PCDH8
D000638
CTDincreases(expression)PCDHAC2
D000638
CTDincreases(expression)PCDHGC3
D000638
CTDincreases(expression)PCSK9
D000638
CTDincreases(expression)PDCD10
D000638
CTDincreases(expression)PDE6G
D000638
CTDincreases(expression)PDE7B
D000638
CTDincreases(expression)PDF
D000638
CTDincreases(expression)PDGFRL
D000638
CTDincreases(expression)PDLIM2
D000638
CTDincreases(expression)PDYN
D000638
CTDincreases(expression)PER1
D000638
CTDincreases(expression)PGK2
D000638
CTDincreases(expression)PHF20L1
D000638
CTDincreases(expression)PHF5A
D000638
CTDincreases(expression)PHKA1
D000638
CTDincreases(expression)PIFO
D000638
CTDincreases(expression)PIGA
D000638
CTDincreases(expression)PIP5K1A
D000638
CTDincreases(expression)PLAA
D000638
CTDincreases(expression)PLAC8L1
D000638
CTDincreases(expression)PLEKHG4
D000638
CTDincreases(expression)PLS1
D000638
CTDincreases(expression)PODN
D000638
CTDincreases(expression)POLL
D000638
CTDincreases(expression)POTEH
D000638
CTDdecreases(activity)PPARG
D000638
CTDdecreases(reaction)PPARG
D000638
CTDincreases(expression)PPARG
D000638
CTDincreases(uptake)PPARG
D000638
CTDincreases(expression)PPM1B
D000638
CTDincreases(expression)PPP1R15A
D000638
CTDincreases(expression)PPP2R5C
D000638
CTDincreases(expression)PPP3R1
D000638
CTDincreases(expression)PRDM2
D000638
CTDincreases(expression)PRDM8
D000638
CTDincreases(expression)PRIM2
D000638
CTDincreases(phosphorylation)PRKAA1
D000638
CTDincreases(phosphorylation)PRKAA2
D000638
CTDincreases(expression)PRMT1
D000638
CTDincreases(expression)PROSER2
D000638
CTDincreases(expression)PROX1
D000638
CTDincreases(expression)PRR19
D000638
CTDincreases(expression)PSEN1
D000638
CTDincreases(expression)PSIP1
D000638
CTDincreases(expression)PSMD11
D000638
CTDincreases(expression)PTGR1
D000638
CTDincreases(expression)PTGS2
D000638
CTDincreases(expression)PTPN3
D000638
CTDincreases(expression)PTPRF
D000638
CTDincreases(expression)PTPRN
D000638
CTDincreases(expression)PYGO1
D000638
CTDincreases(expression)RAB39B
D000638
CTDincreases(expression)RAB9B
D000638
CTDincreases(expression)RAC3
D000638
CTDincreases(expression)RBBP8
D000638
CTDincreases(expression)RBKS
D000638
CTDincreases(expression)RBM33
D000638
CTDincreases(expression)RBPMS
D000638
CTDincreases(expression)RCN3
D000638
CTDincreases(expression)RDH8
D000638
CTDincreases(expression)RELB
D000638
CTDincreases(expression)REPIN1
D000638
CTDincreases(expression)RGS6
D000638
CTDincreases(expression)RHEBL1
D000638
CTDincreases(expression)RIN3
D000638
CTDincreases(expression)RNF146
D000638
CTDincreases(expression)RNF19A
D000638
CTDincreases(expression)RNF212
D000638
CTDincreases(expression)RNF6
D000638
CTDincreases(expression)RNF8
D000638
CTDincreases(expression)RPL36A
D000638
CTDdecreases(phosphorylation)RPS6KB1
D000638
CTDincreases(expression)RUNDC3A
D000638
CTDincreases(expression)SARDH
D000638
CTDincreases(expression)SCAND2P
D000638
CTDdecreases(activity)SCD
D000638
CTDdecreases(reaction)SCD
D000638
CTDincreases(expression)SCD
D000638
CTDaffects(reaction)SCD
D000638
CTDincreases(uptake)SCD
D000638
CTDincreases(expression)SCIMP
D000638
CTDincreases(expression)SEMA3D
D000638
CTDincreases(expression)SEMA4D
D000638
CTDincreases(expression)SEMA6B
D000638
CTDincreases(expression)SEMG1
D000638
CTDincreases(expression)SERPINA10
D000638
CTDincreases(expression)SERTAD3
D000638
CTDincreases(expression)SESN2
D000638
CTDincreases(expression)SH2D1A
D000638
CTDincreases(expression)SIPA1L3
D000638
CTDincreases(expression)SIRT4
D000638
CTDincreases(expression)SIX1
D000638
CTDincreases(expression)SLC13A4
D000638
CTDincreases(expression)SLC14A2
D000638
CTDdecreases(reaction)SLC22A1
D000638
CTDincreases(uptake)SLC22A1
D000638
CTDdecreases(reaction)SLC22A5
D000638
CTDincreases(uptake)SLC22A5
D000638
CTDincreases(expression)SLC25A18
D000638
CTDincreases(expression)SLC25A25
D000638
CTDincreases(expression)SLC25A26
D000638
CTDincreases(expression)SLC25A30
D000638
CTDdecreases(expression)SLC26A4
D000638
CTDdecreases(expression)SLC2A3
D000638
CTDincreases(expression)SLC30A1
D000638
CTDincreases(expression)SLC35A2
D000638
CTDincreases(expression)SLC38A11
D000638
CTDincreases(expression)SLC3A2
D000638
CTDincreases(expression)SLC5A3
D000638
CTDdecreases(expression)SLC5A5
D000638
CTDincreases(uptake)SLCO2B1
D000638
CTDincreases(expression)SLCO4C1
D000638
CTDincreases(expression)SLCO5A1
D000638
CTDincreases(expression)SLFN5
D000638
CTDincreases(expression)SLITRK3
D000638
CTDincreases(expression)SLX4IP
D000638
CTDincreases(expression)SMG6
D000638
CTDincreases(expression)SMIM11
D000638
CTDincreases(expression)SMOX
D000638
CTDincreases(expression)SNRNP35
D000638
CTDincreases(expression)SNX18
D000638
CTDincreases(expression)SOCS6
D000638
CTDincreases(expression)SOD2
D000638
CTDincreases(expression)SPAG1
D000638
CTDincreases(expression)SPATA17
D000638
CTDincreases(expression)SPATA2L
D000638
CTDincreases(expression)SPEF2
D000638
CTDincreases(expression)SPHAR
D000638
CTDincreases(expression)SPOPL
D000638
CTDincreases(expression)SPR
D000638
CTDincreases(expression)SPTBN1
D000638
CTDincreases(expression)SQSTM1
D000638
CTDincreases(expression)SREK1IP1
D000638
CTDincreases(expression)SS18L1
D000638
CTDincreases(expression)STARD5
D000638
CTDincreases(expression)STK16
D000638
CTDincreases(expression)STX11
D000638
CTDincreases(expression)STXBP2
D000638
CTDincreases(expression)SULT1A3
D000638
CTDincreases(expression)SVIL
D000638
CTDincreases(expression)TAF5L
D000638
CTDdecreases(expression)TAGLN
D000638
CTDincreases(expression)TAPBPL
D000638
CTDincreases(expression)TAS2R10
D000638
CTDincreases(expression)TAZ
D000638
CTDincreases(expression)TBC1D3
D000638
CTDincreases(expression)TBX3
D000638
CTDincreases(expression)TBX4
D000638
CTDincreases(expression)TCAIM
D000638
CTDincreases(expression)TCF20
D000638
CTDincreases(expression)TCF7
D000638
CTDincreases(expression)TCL1B
D000638
CTDincreases(expression)TDO2
D000638
CTDincreases(expression)TEF
D000638
CTDincreases(expression)TERF1
D000638
CTDincreases(expression)TFAP2C
D000638
CTDincreases(expression)TFG
D000638
CTDdecreases(expression)TG
D000638
CTDincreases(expression)TGOLN2
D000638
CTDaffects(binding)THRA
D000638
CTDaffects(binding)THRB
D000638
CTDincreases(expression)THRB
D000638
CTDincreases(expression)TIGD6
D000638
CTDincreases(expression)TIMM13
D000638
CTDincreases(expression)TIMM17A
D000638
CTDincreases(expression)TINAG
D000638
CTDincreases(expression)TKTL1
D000638
CTDincreases(expression)TMCC2
D000638
CTDincreases(expression)TMEM161B
D000638
CTDincreases(expression)TMEM31
D000638
CTDincreases(expression)TMEM68
D000638
CTDincreases(expression)TMLHE
D000638
CTDincreases(expression)TMPRSS9
D000638
CTDincreases(expression)TMUB2
D000638
CTDincreases(activity)TNF
D000638
CTDincreases(reaction)TNF
D000638
CTDaffects(cotreatment)TNF
D000638
CTDincreases(expression)TNF
D000638
CTDincreases(secretion)TNF
D000638
CTDdecreases(reaction)TNF
D000638
CTDincreases(expression)TNF
D000638
CTDdecreases(reaction)TNF
D000638
CTDincreases(activity)TNF
D000638
CTDincreases(expression)TNF
D000638
CTDaffects(cotreatment)TNF
D000638
CTDincreases(response to substance)TNF
D000638
CTDdecreases(reaction)TNF
D000638
CTDincreases(expression)TNFAIP3
D000638
CTDincreases(expression)TNFRSF10B
D000638
CTDdecreases(reaction)TNFRSF10B
D000638
CTDincreases(response to substance)TNFSF10
D000638
CTDaffects(cotreatment)TNFSF10
D000638
CTDincreases(cleavage)TNFSF10
D000638
CTDincreases(expression)TNNT1
D000638
CTDincreases(expression)TNRC6A
D000638
CTDincreases(expression)TOM1L1
D000638
CTDdecreases(expression)TPO
D000638
CTDincreases(expression)TREX1
D000638
CTDincreases(expression)TRIB3
D000638
CTDincreases(expression)TRIM36
D000638
CTDincreases(expression)TRIM61
D000638
CTDincreases(expression)TRMT10B
D000638
CTDincreases(expression)TRNT1
D000638
CTDincreases(expression)TRPV2
D000638
CTDincreases(expression)TSGA10
D000638
CTDincreases(expression)TSHB
D000638
CTDincreases(expression)TSLP
D000638
CTDincreases(expression)TSPYL2
D000638
CTDincreases(expression)TTBK2
D000638
CTDincreases(expression)TTLL3
D000638
CTDincreases(expression)TUSC3
D000638
CTDincreases(expression)UBE2D2
D000638
CTDincreases(expression)UBE2D3
D000638
CTDincreases(expression)UBXN10
D000638
CTDincreases(expression)UBXN11
D000638
CTDincreases(expression)ULK3
D000638
CTDincreases(expression)USF1
D000638
CTDincreases(expression)USP2
D000638
CTDincreases(expression)USP25
D000638
CTDincreases(expression)UTS2
D000638
CTDincreases(expression)VCAM1
D000638
CTDincreases(expression)VEGFA
D000638
CTDincreases(expression)VMAC
D000638
CTDincreases(expression)VPS11
D000638
CTDincreases(expression)VPS13B
D000638
CTDincreases(expression)VPS16
D000638
CTDincreases(expression)WBSCR16
D000638
CTDincreases(expression)WBSCR17
D000638
CTDincreases(expression)WIPI1
D000638
CTDincreases(expression)WNK1
D000638
CTDincreases(expression)WTAP
D000638
CTDincreases(expression)XBP1
D000638
CTDincreases(expression)XK
D000638
CTDincreases(expression)XPNPEP2
D000638
CTDincreases(expression)ZBED3
D000638
CTDincreases(expression)ZBTB49
D000638
CTDincreases(expression)ZC3HAV1
D000638
CTDincreases(expression)ZDHHC15
D000638
CTDincreases(expression)ZFP36
D000638
CTDincreases(expression)ZMYND10
D000638
CTDincreases(expression)ZNF101
D000638
CTDincreases(expression)ZNF121
D000638
CTDincreases(expression)ZNF197
D000638
CTDincreases(expression)ZNF205
D000638
CTDincreases(expression)ZNF225
D000638
CTDincreases(expression)ZNF311
D000638
CTDincreases(expression)ZNF420
D000638
CTDincreases(expression)ZNF497
D000638
CTDincreases(expression)ZNF554
D000638
CTDincreases(expression)ZNF584
D000638
CTDincreases(expression)ZNF592
D000638
CTDincreases(expression)ZNF624
D000638
CTDincreases(expression)ZNF676
D000638
CTDincreases(expression)ZNF683
D000638
CTDincreases(expression)ZNF703
D000638
CTDincreases(expression)ZNF704
D000638
CTDincreases(expression)ZNF710
D000638
CTDincreases(expression)ZNF771
D000638
CTDincreases(expression)ZNHIT2
D000638
CTDincreases(expression)ZSCAN20
D000638
CTDincreases(expression)ZXDA
D000638
PubChem PotencyuM44.668CBX1-GI(Protien) :
PubChem NoneuMCYP1A2-GI(Protien) :
PubChem PotencyuM31.623CYP2D6-GI(Protien) :
PubChem NoneuMCYP2D6-GI(Protien) :
PubChem PotencyuM12.995GMNN-GI(Protien) :
PubChem PotencyuM20.596GMNN-GI(Protien) :
PubChem PotencyuM13.092MTOR-GI(Protien) :
ChEMBLPotencynM44668.400CBX1
-Target : CHEMBL1741193
ChEMBLInhibition-CYP1A2
-Target : CHEMBL3356
ChEMBLInhibition-CYP2C19
-Target : CHEMBL3622
ChEMBLInhibition-CYP2C9
-Target : CHEMBL3397
ChEMBLAC50nM31622.800CYP2D6
-Target : CHEMBL289
ChEMBLPotencynM31622.800CYP2D6
-Target : CHEMBL289
ChEMBLPotencynM13091.800MTOR
-Target : CHEMBL2842
ChEMBLIC50-SQLE
-Target : CHEMBL3592
Download gene sets gmt, text, Detailed text
Contact us
Tan Lab , Mail Stop 8117
12801 East 17th Avenue
Division of Medical Oncology , Department of Medicine
University of Colorado School of Medicine
Aurora, CO 80045, USA

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