DSigDB Home
Search Gene
Collections
Browse Gene Sets
Download
Help

Gene Set: D4 : CTD - saracatinib

Collection D4 : CTD
Chemical Name saracatinib ( From PubChem : SARACATINIB )
FDA NPC WHO Indian Australia China Traditional
Herbal		 Clinical
Trail
NotNotNotNotNotNotNotNot
Molecular
Weight		 Hydrogen Bond
Donor Count		 Hydrogen Bond
Acceptor Count		 cLogP Lipinski Rule
542.026 g/mol 1 9 3.8883 False(3/4)
Structure
InChI InChI=1S/C27H32ClN5O5/c1-32-6-8-33(9-7-32)10-13-35-19-14-21-24(23(15-19)38-18-4-11-34-12-5-18)27(30-16-29-21)31-25-20(28)2-3-22-26(25)37-17-36-22/h2-3,14-16,18H,4-13,17H2,1H3,(H,29,30,31)
InChIKey OUKYUETWWIPKQR-UHFFFAOYSA-N
Links

Gene (5 / 12)


⊖ Less
Source Type Unit Value Gene PMID Assay Other
CTDdecreases(expression)CSK
C515233
CTDdecreases(reaction)CSK
C515233
CTDdecreases(activity)CSK
C515233
CTDdecreases(reaction)CYP24A1
C515233
CTDincreases(expression)CYP24A1
C515233
CTDdecreases(expression)CYP7A1
C515233
CTDdecreases(reaction)CYP7A1
C515233
CTDincreases(expression)CYP7A1
C515233
CTDdecreases(reaction)VDR
C515233
CTDincreases(phosphorylation)VDR
C515233
PubChem PotencyuM0.000YES1GI(Protien) :
PubChem PotencyuM0.006YES1-GI(Protien) :
Download gene sets gmt, text, Detailed text
Contact us
Tan Lab , Mail Stop 8117
12801 East 17th Avenue
Division of Medical Oncology , Department of Medicine
University of Colorado School of Medicine
Aurora, CO 80045, USA

* Best viewed in the latest version of Chrome (42+), Safari (8+), IE (11+) or Firefox (35+).