Tan Lab | DSigDB

Gene Set: D4 : CTD - dasatinib

Collection

D4 : CTD

Chemical Name

dasatinib ( From PubChem : DASATINIB )

FDA	NPC	WHO	Indian	Australia	China	Traditional Herbal	Clinical Trail
Approved	Not	Not	Not	Not	Not	Not	Not

Molecular Weight	Hydrogen Bond Donor Count	Hydrogen Bond Acceptor Count	cLogP	Lipinski Rule
488.006 g/mol	3	9	3.4624	True

Structure

InChI

InChI=1S/C22H26ClN7O2S/c1-14-4-3-5-16(23)20(14)28-21(32)17-13-24-22(33-17)27-18-12-19(26-15(2)25-18)30-8-6-29(7-9-30)10-11-31/h3-5,12-13,31H,6-11H2,1-2H3,(H,28,32)(H,24,25,26,27)

InChIKey

ZBNZXTGUTAYRHI-UHFFFAOYSA-N

Links

Gene (502 / 642)

⊖ Less

Source	Type	Unit	Value	Gene	PMID	Other
CTD	increases(expression)			A2M		C488369
CTD	increases(expression)			ABCA1		C488369
CTD	decreases(activity)			ABCB11		C488369
CTD	increases(expression)			ABCC3		C488369
CTD	increases(expression)			ABHD4		C488369
CTD	affects(binding)			ABL1		C488369
CTD	affects(cotreatment)			ABL1		C488369
CTD	decreases(expression)			ABL1		C488369
CTD	decreases(phosphorylation)			ABL1		C488369
CTD	decreases(reaction)			ABL1		C488369
CTD	increases(phosphorylation)			ABL1		C488369
CTD	decreases(reaction)			ABL1		C488369
CTD	increases(phosphorylation)			ABL1		C488369
CTD	decreases(activity)			ABL1		C488369
CTD	decreases(phosphorylation)			ABL1		C488369
CTD	affects(binding)			ABL2		C488369
CTD	increases(expression)			ACAN		C488369
CTD	increases(expression)			ACTA2		C488369
CTD	increases(expression)			ACTC1		C488369
CTD	increases(expression)			ACTG2		C488369
CTD	increases(expression)			ADAMTS5		C488369
CTD	affects(localization)			AIFM1		C488369
CTD	affects(cotreatment)			AIFM1		C488369
CTD	decreases(expression)			AK5		C488369
CTD	increases(expression)			AKR1C3		C488369
CTD	affects(binding)			AKT1		C488369
CTD	affects(cotreatment)			AKT1		C488369
CTD	decreases(reaction)			AKT1		C488369
CTD	increases(reaction)			AKT1		C488369
CTD	increases(expression)			ALDH1A1		C488369
CTD	increases(expression)			ALDH1L2		C488369
CTD	increases(expression)			ALDH2		C488369
CTD	increases(expression)			ALPK2		C488369
CTD	increases(expression)			AMIGO2		C488369
CTD	increases(expression)			ANGPTL2		C488369
CTD	increases(expression)			ANKH		C488369
CTD	decreases(expression)			ANLN		C488369
CTD	decreases(reaction)			ANPEP		C488369
CTD	increases(expression)			ANPEP		C488369
CTD	decreases(expression)			ANPEP		C488369
CTD	increases(expression)			ANTXR1		C488369
CTD	decreases(expression)			AOX1		C488369
CTD	decreases(expression)			APOBEC3B		C488369
CTD	decreases(expression)			ARHGAP11A		C488369
CTD	decreases(expression)			ARHGAP18		C488369
CTD	decreases(expression)			ARHGAP22		C488369
CTD	increases(expression)			ARMC9		C488369
CTD	decreases(expression)			ARNTL2		C488369
CTD	decreases(expression)			ASF1B		C488369
CTD	increases(expression)			ASNS		C488369
CTD	decreases(expression)			ASPM		C488369
CTD	decreases(expression)			ATAD2		C488369
CTD	decreases(expression)			ATAD5		C488369
CTD	decreases(expression)			AURKA		C488369
CTD	decreases(expression)			AURKB		C488369
CTD	affects(binding)			BAX		C488369
CTD	affects(cotreatment)			BAX		C488369
CTD	decreases(reaction)			BAX		C488369
CTD	increases(reaction)			BAX		C488369
CTD	increases(cleavage)			BAX		C488369
CTD	affects(binding)			BCL2		C488369
CTD	affects(cotreatment)			BCL2		C488369
CTD	decreases(reaction)			BCL2		C488369
CTD	increases(reaction)			BCL2		C488369
CTD	decreases(expression)			BCL2		C488369
CTD	decreases(expression)			BCL2		C488369
CTD	decreases(expression)			BCL2		C488369
CTD	decreases(expression)			BCL2L1		C488369
CTD	affects(binding)			BCR		C488369
CTD	affects(cotreatment)			BCR		C488369
CTD	decreases(expression)			BCR		C488369
CTD	decreases(phosphorylation)			BCR		C488369
CTD	decreases(reaction)			BCR		C488369
CTD	increases(phosphorylation)			BCR		C488369
CTD	decreases(activity)			BCR		C488369
CTD	decreases(phosphorylation)			BCR		C488369
CTD	increases(expression)			BGN		C488369
CTD	decreases(expression)			BIRC5		C488369
CTD	decreases(expression)			BORA		C488369
CTD	decreases(expression)			BRCA1		C488369
CTD	decreases(expression)			BRCA2		C488369
CTD	affects(binding)			BTK		C488369
CTD	decreases(activity)			BTK		C488369
CTD	affects(binding)			BTK		C488369
CTD	decreases(phosphorylation)			BTK		C488369
CTD	decreases(expression)			BUB1		C488369
CTD	decreases(expression)			BUB1B		C488369
CTD	increases(expression)			C10ORF10		C488369
CTD	decreases(expression)			C18ORF54		C488369
CTD	decreases(expression)			C1ORF112		C488369
CTD	increases(expression)			C1ORF198		C488369
CTD	increases(expression)			C1R		C488369
CTD	increases(expression)			C1S		C488369
CTD	increases(expression)			C9ORF3		C488369
CTD	increases(expression)			CACNA1C		C488369
CTD	increases(expression)			CALCOCO1		C488369
CTD	increases(activity)			CASP3		C488369
CTD	increases(reaction)			CASP3		C488369
CTD	increases(activity)			CASP3		C488369
CTD	increases(cleavage)			CASP3		C488369
CTD	increases(cleavage)			CASP7		C488369
CTD	increases(activity)			CASP8		C488369
CTD	increases(cleavage)			CASP8		C488369
CTD	increases(activity)			CASP9		C488369
CTD	increases(cleavage)			CASP9		C488369
CTD	decreases(expression)			CCL1		C488369
CTD	decreases(expression)			CCL2		C488369
CTD	decreases(expression)			CCL3		C488369
CTD	decreases(expression)			CCL4		C488369
CTD	decreases(expression)			CCL5		C488369
CTD	decreases(expression)			CCND1		C488369
CTD	affects(cotreatment)			CCND1		C488369
CTD	decreases(expression)			CCND1		C488369
CTD	decreases(expression)			CCND3		C488369
CTD	decreases(reaction)			CD164		C488369
CTD	increases(expression)			CD164		C488369
CTD	decreases(expression)			CD164		C488369
CTD	decreases(expression)			CD274		C488369
CTD	increases(expression)			CD302		C488369
CTD	decreases(expression)			CD38		C488369
CTD	decreases(reaction)			CD63		C488369
CTD	increases(expression)			CD63		C488369
CTD	decreases(expression)			CD63		C488369
CTD	decreases(expression)			CD69		C488369
CTD	decreases(expression)			CDC20		C488369
CTD	decreases(expression)			CDC25A		C488369
CTD	decreases(expression)			CDC25C		C488369
CTD	decreases(expression)			CDC45		C488369
CTD	decreases(expression)			CDC6		C488369
CTD	decreases(expression)			CDC7		C488369
CTD	decreases(expression)			CDCA2		C488369
CTD	decreases(expression)			CDCA3		C488369
CTD	decreases(expression)			CDCA5		C488369
CTD	decreases(expression)			CDCA8		C488369
CTD	decreases(expression)			CDK1		C488369
CTD	decreases(expression)			CDK2		C488369
CTD	affects(cotreatment)			CDK4		C488369
CTD	decreases(expression)			CDK4		C488369
CTD	affects(cotreatment)			CDK6		C488369
CTD	decreases(expression)			CDK6		C488369
CTD	increases(expression)			CDKN1A		C488369
CTD	affects(cotreatment)			CDKN1A		C488369
CTD	increases(expression)			CDKN1A		C488369
CTD	increases(expression)			CDKN1B		C488369
CTD	decreases(expression)			CDKN3		C488369
CTD	decreases(expression)			CENPA		C488369
CTD	decreases(expression)			CENPE		C488369
CTD	decreases(expression)			CENPF		C488369
CTD	decreases(expression)			CENPH		C488369
CTD	decreases(expression)			CENPI		C488369
CTD	decreases(expression)			CENPK		C488369
CTD	decreases(expression)			CENPL		C488369
CTD	decreases(expression)			CENPN		C488369
CTD	decreases(expression)			CENPO		C488369
CTD	decreases(expression)			CENPU		C488369
CTD	decreases(expression)			CENPW		C488369
CTD	decreases(expression)			CEP128		C488369
CTD	decreases(expression)			CEP152		C488369
CTD	increases(expression)			CES1		C488369
CTD	increases(expression)			CHAC1		C488369
CTD	increases(expression)			CHI3L1		C488369
CTD	decreases(expression)			CKAP2L		C488369
CTD	decreases(expression)			CKS1B		C488369
CTD	decreases(expression)			CKS2		C488369
CTD	decreases(expression)			CLSPN		C488369
CTD	increases(expression)			CLU		C488369
CTD	increases(expression)			CNN1		C488369
CTD	increases(expression)			CNNM2		C488369
CTD	increases(expression)			COL11A1		C488369
CTD	increases(expression)			COL3A1		C488369
CTD	increases(expression)			COL4A1		C488369
CTD	increases(expression)			COL4A2		C488369
CTD	decreases(expression)			CPA4		C488369
CTD	increases(expression)			CPQ		C488369
CTD	increases(expression)			CRISPLD2		C488369
CTD	affects(cotreatment)			CRKL		C488369
CTD	decreases(phosphorylation)			CRKL		C488369
CTD	decreases(reaction)			CRKL		C488369
CTD	increases(phosphorylation)			CRKL		C488369
CTD	decreases(reaction)			CRKL		C488369
CTD	increases(phosphorylation)			CRKL		C488369
CTD	increases(expression)			CRYAB		C488369
CTD	decreases(expression)			CSF2		C488369
CTD	affects(binding)			CSK		C488369
CTD	decreases(expression)			CXCL1		C488369
CTD	decreases(expression)			CXCL10		C488369
CTD	increases(expression)			CXCL10		C488369
CTD	decreases(expression)			CXCL12		C488369
CTD	decreases(expression)			CXCL8		C488369
CTD	increases(expression)			CYP1B1		C488369
CTD	increases(expression)			DACT1		C488369
CTD	decreases(expression)			DCBLD2		C488369
CTD	decreases(expression)			DDIAS		C488369
CTD	increases(expression)			DDIT4		C488369
CTD	decreases(expression)			DDX39A		C488369
CTD	decreases(expression)			DEPDC1		C488369
CTD	decreases(expression)			DEPDC1B		C488369
CTD	increases(expression)			DEPTOR		C488369
CTD	decreases(expression)			DHFR		C488369
CTD	increases(expression)			DHRS3		C488369
CTD	affects(localization)			DIABLO		C488369
CTD	affects(cotreatment)			DIABLO		C488369
CTD	decreases(expression)			DIAPH3		C488369
CTD	decreases(expression)			DKK1		C488369
CTD	decreases(expression)			DLEU2		C488369
CTD	decreases(expression)			DLGAP5		C488369
CTD	decreases(expression)			DNA2		C488369
CTD	increases(expression)			DPP4		C488369
CTD	decreases(expression)			DSN1		C488369
CTD	decreases(expression)			DTL		C488369
CTD	decreases(expression)			E2F7		C488369
CTD	increases(expression)			ECH1		C488369
CTD	decreases(expression)			ECT2		C488369
CTD	increases(expression)			EDIL3		C488369
CTD	increases(expression)			EFEMP1		C488369
CTD	decreases(reaction)			EGF		C488369
CTD	increases(phosphorylation)			EGF		C488369
CTD	decreases(reaction)			EGFR		C488369
CTD	increases(phosphorylation)			EGFR		C488369
CTD	decreases(phosphorylation)			EGFR		C488369
CTD	increases(response to substance)			EGFR		C488369
CTD	decreases(phosphorylation)			EGFR		C488369
CTD	increases(expression)			ELN		C488369
CTD	decreases(expression)			ELOVL6		C488369
CTD	decreases(expression)			ENPP1		C488369
CTD	decreases(reaction)			ENPP3		C488369
CTD	increases(expression)			ENPP3		C488369
CTD	decreases(expression)			ENPP3		C488369
CTD	increases(expression)			EPAS1		C488369
CTD	affects(binding)			EPHA5		C488369
CTD	affects(binding)			EPHB4		C488369
CTD	increases(expression)			EPHX1		C488369
CTD	decreases(expression)			EXO1		C488369
CTD	decreases(expression)			EZH2		C488369
CTD	decreases(expression)			FAM111B		C488369
CTD	increases(expression)			FAM150A		C488369
CTD	decreases(expression)			FAM180A		C488369
CTD	increases(expression)			FAM198B		C488369
CTD	decreases(expression)			FAM64A		C488369
CTD	decreases(expression)			FAM72D		C488369
CTD	decreases(expression)			FANCA		C488369
CTD	decreases(expression)			FANCD2		C488369
CTD	decreases(expression)			FANCI		C488369
CTD	decreases(expression)			FANCM		C488369
CTD	increases(expression)			FBLN5		C488369
CTD	increases(expression)			FBXO32		C488369
CTD	decreases(expression)			FBXO5		C488369
CTD	decreases(expression)			FEN1		C488369
CTD	decreases(expression)			FGF5		C488369
CTD	increases(expression)			FGF9		C488369
CTD	increases(expression)			FGL2		C488369
CTD	affects(binding)			FGR		C488369
CTD	increases(expression)			FHL1		C488369
CTD	decreases(expression)			FIGNL1		C488369
CTD	decreases(phosphorylation)			FIP1L1		C488369
CTD	decreases(phosphorylation)			FLT3		C488369
CTD	decreases(expression)			FOXM1		C488369
CTD	affects(binding)			FRK		C488369
CTD	affects(binding)			FYN		C488369
CTD	decreases(expression)			G0S2		C488369
CTD	decreases(expression)			GAS2L3		C488369
CTD	decreases(expression)			GEN1		C488369
CTD	decreases(expression)			GINS1		C488369
CTD	decreases(expression)			GINS2		C488369
CTD	decreases(expression)			GINS4		C488369
CTD	increases(expression)			GLIPR2		C488369
CTD	increases(expression)			GPC4		C488369
CTD	increases(expression)			GPNMB		C488369
CTD	increases(expression)			GREM2		C488369
CTD	increases(expression)			GSTM5		C488369
CTD	decreases(expression)			H2AFZ		C488369
CTD	increases(expression)			HAPLN3		C488369
CTD	decreases(expression)			HAS2		C488369
CTD	decreases(expression)			HBEGF		C488369
CTD	decreases(phosphorylation)			HCK		C488369
CTD	increases(expression)			HEG1		C488369
CTD	decreases(expression)			HELLS		C488369
CTD	increases(expression)			HEPH		C488369
CTD	decreases(expression)			HERC2P10		C488369
CTD	decreases(expression)			HERC4		C488369
CTD	decreases(expression)			HIST1H1A		C488369
CTD	decreases(expression)			HIST1H1B		C488369
CTD	decreases(expression)			HIST1H1E		C488369
CTD	decreases(expression)			HIST1H2BB		C488369
CTD	decreases(expression)			HIST1H2BH		C488369
CTD	decreases(expression)			HIST1H2BM		C488369
CTD	decreases(expression)			HIST2H2AB		C488369
CTD	decreases(expression)			HJURP		C488369
CTD	increases(expression)			HMCN1		C488369
CTD	decreases(expression)			HMGA2		C488369
CTD	decreases(expression)			HMGB2		C488369
CTD	decreases(expression)			HMMR		C488369
CTD	affects(binding)			HSPA8		C488369
CTD	increases(expression)			HTR2B		C488369
CTD	increases(expression)			HTRA1		C488369
CTD	increases(expression)			IFIT3		C488369
CTD	decreases(expression)			IFNG		C488369
CTD	increases(expression)			IGF2		C488369
CTD	increases(expression)			IGFBP5		C488369
CTD	increases(expression)			IGFBP7		C488369
CTD	decreases(response to substance)			IGH		C488369
CTD	decreases(expression)			IL1R1		C488369
CTD	decreases(expression)			IL2		C488369
CTD	decreases(expression)			IL5		C488369
CTD	decreases(expression)			IL6		C488369
CTD	increases(expression)			IL6		C488369
CTD	decreases(expression)			IQGAP3		C488369
CTD	increases(expression)			ITGA11		C488369
CTD	decreases(expression)			ITGA6		C488369
CTD	decreases(reaction)			ITGAM		C488369
CTD	increases(expression)			ITGAM		C488369
CTD	increases(expression)			ITGAV		C488369
CTD	decreases(expression)			ITGB3BP		C488369
CTD	increases(expression)			ITPR1		C488369
CTD	increases(expression)			JAG1		C488369
CTD	increases(expression)			JMY		C488369
CTD	decreases(expression)			KCNK2		C488369
CTD	decreases(expression)			KIAA0101		C488369
CTD	decreases(expression)			KIAA1524		C488369
CTD	decreases(expression)			KIF20B		C488369
CTD	decreases(expression)			KIF23		C488369
CTD	decreases(expression)			KIF2C		C488369
CTD	decreases(expression)			KIF4A		C488369
CTD	decreases(expression)			KIFC1		C488369
CTD	affects(binding)			KIT		C488369
CTD	decreases(phosphorylation)			KIT		C488369
CTD	decreases(expression)			KNSTRN		C488369
CTD	decreases(expression)			KNTC1		C488369
CTD	decreases(expression)			KPNA2		C488369
CTD	increases(expression)			LAMB1		C488369
CTD	increases(expression)			LBH		C488369
CTD	decreases(activity)			LCK		C488369
CTD	increases(expression)			LIMCH1		C488369
CTD	increases(expression)			LINC00312		C488369
CTD	increases(expression)			LMCD1		C488369
CTD	decreases(expression)			LMNB1		C488369
CTD	increases(expression)			LMOD1		C488369
CTD	decreases(expression)			LPXN		C488369
CTD	increases(expression)			LRP1		C488369
CTD	decreases(expression)			LRR1		C488369
CTD	increases(expression)			LSAMP		C488369
CTD	increases(expression)			LUM		C488369
CTD	affects(binding)			LYN		C488369
CTD	decreases(phosphorylation)			LYN		C488369
CTD	decreases(activity)			LYN		C488369
CTD	decreases(activity)			LYN		C488369
CTD	decreases(phosphorylation)			LYN		C488369
CTD	decreases(expression)			MAD2L1		C488369
CTD	decreases(expression)			MALL		C488369
CTD	increases(expression)			MAMDC2		C488369
CTD	decreases(reaction)			MAP2K1		C488369
CTD	increases(phosphorylation)			MAP2K1		C488369
CTD	decreases(reaction)			MAPK1		C488369
CTD	increases(phosphorylation)			MAPK1		C488369
CTD	decreases(phosphorylation)			MAPK1		C488369
CTD	affects(cotreatment)			MAPK1		C488369
CTD	decreases(phosphorylation)			MAPK1		C488369
CTD	affects(binding)			MAPK14		C488369
CTD	decreases(reaction)			MAPK3		C488369
CTD	increases(phosphorylation)			MAPK3		C488369
CTD	decreases(phosphorylation)			MAPK3		C488369
CTD	affects(cotreatment)			MAPK3		C488369
CTD	decreases(phosphorylation)			MAPK3		C488369
CTD	decreases(expression)			MARCH3		C488369
CTD	decreases(expression)			MASTL		C488369
CTD	increases(expression)			MCAM		C488369
CTD	decreases(expression)			MCL1		C488369
CTD	decreases(expression)			MCM10		C488369
CTD	decreases(expression)			MCM6		C488369
CTD	decreases(expression)			MCM7		C488369
CTD	decreases(expression)			MCM8		C488369
CTD	increases(expression)			MDGA1		C488369
CTD	decreases(expression)			MELK		C488369
CTD	decreases(phosphorylation)			MET		C488369
CTD	affects(cotreatment)			MET		C488369
CTD	increases(expression)			MFAP4		C488369
CTD	increases(expression)			MFGE8		C488369
CTD	decreases(expression)			MGME1		C488369
CTD	increases(expression)			MGP		C488369
CTD	increases(expression)			MIR143HG		C488369
CTD	decreases(expression)			MIS18A		C488369
CTD	decreases(expression)			MIS18BP1		C488369
CTD	decreases(expression)			MKI67		C488369
CTD	decreases(expression)			MKI67		C488369
CTD	decreases(expression)			MMP1		C488369
CTD	decreases(expression)			MMS22L		C488369
CTD	decreases(expression)			MND1		C488369
CTD	increases(expression)			MRVI1		C488369
CTD	decreases(expression)			MSH2		C488369
CTD	decreases(expression)			MTBP		C488369
CTD	decreases(expression)			MTFR2		C488369
CTD	decreases(phosphorylation)			MTOR		C488369
CTD	decreases(expression)			MYBL1		C488369
CTD	decreases(expression)			MYBL2		C488369
CTD	decreases(expression)			MYC		C488369
CTD	increases(expression)			MYH10		C488369
CTD	increases(expression)			MYH11		C488369
CTD	increases(expression)			MYLK		C488369
CTD	decreases(expression)			MYPN		C488369
CTD	decreases(expression)			NCAPD2		C488369
CTD	decreases(expression)			NCAPD3		C488369
CTD	decreases(expression)			NCAPG		C488369
CTD	decreases(expression)			NCAPG2		C488369
CTD	decreases(expression)			NCAPH		C488369
CTD	decreases(expression)			NCEH1		C488369
CTD	decreases(expression)			NDC1		C488369
CTD	decreases(expression)			NDC80		C488369
CTD	decreases(expression)			NEFM		C488369
CTD	increases(expression)			NEO1		C488369
CTD	increases(expression)			NNMT		C488369
CTD	increases(expression)			NREP		C488369
CTD	increases(expression)			NRP2		C488369
CTD	increases(expression)			NRXN3		C488369
CTD	increases(expression)			NUAK1		C488369
CTD	decreases(expression)			NUSAP1		C488369
CTD	decreases(expression)			ORC1		C488369
CTD	decreases(expression)			ORC6		C488369
CTD	decreases(expression)			PARPBP		C488369
CTD	decreases(expression)			PBK		C488369
CTD	increases(expression)			PBX1		C488369
CTD	increases(expression)			PCK2		C488369
CTD	increases(expression)			PCMTD1		C488369
CTD	increases(expression)			PDE3A		C488369
CTD	decreases(phosphorylation)			PDGFRA		C488369
CTD	decreases(phosphorylation)			PDGFRB		C488369
CTD	increases(expression)			PDGFRB		C488369
CTD	decreases(expression)			PLAU		C488369
CTD	increases(expression)			PLEKHH2		C488369
CTD	decreases(expression)			PLK1		C488369
CTD	decreases(expression)			PLK4		C488369
CTD	increases(expression)			PLN		C488369
CTD	increases(expression)			PLSCR4		C488369
CTD	increases(expression)			PLXDC2		C488369
CTD	increases(expression)			PODN		C488369
CTD	increases(expression)			PODNL1		C488369
CTD	decreases(expression)			POLA1		C488369
CTD	decreases(expression)			POLA2		C488369
CTD	decreases(expression)			POLE2		C488369
CTD	decreases(expression)			POLQ		C488369
CTD	decreases(expression)			POLR3G		C488369
CTD	affects(binding)			PPAT		C488369
CTD	increases(expression)			PPP1R3C		C488369
CTD	decreases(expression)			PRC1		C488369
CTD	decreases(expression)			PRIM1		C488369
CTD	decreases(expression)			PRIM2		C488369
CTD	decreases(expression)			PRR11		C488369
CTD	increases(expression)			PSAT1		C488369
CTD	decreases(expression)			PSMC3IP		C488369
CTD	increases(expression)			PTGIS		C488369
CTD	decreases(phosphorylation)			PTK2		C488369
CTD	decreases(expression)			PTTG1		C488369
CTD	decreases(expression)			PTX3		C488369
CTD	decreases(phosphorylation)			PXN		C488369
CTD	decreases(expression)			RACGAP1		C488369
CTD	decreases(expression)			RAD51		C488369
CTD	increases(expression)			RASSF2		C488369
CTD	increases(expression)			RAVER2		C488369
CTD	increases(expression)			RDH10		C488369
CTD	increases(expression)			RECK		C488369
CTD	decreases(expression)			RFC2		C488369
CTD	decreases(expression)			RFC3		C488369
CTD	decreases(expression)			RFC4		C488369
CTD	decreases(expression)			RFC5		C488369
CTD	decreases(expression)			RFWD3		C488369
CTD	decreases(expression)			RFX8		C488369
CTD	decreases(expression)			RGMB		C488369
CTD	decreases(expression)			RGS4		C488369
CTD	decreases(expression)			RNASEH2A		C488369
CTD	decreases(expression)			RNU5F-1		C488369
CTD	increases(expression)			ROR1		C488369
CTD	decreases(phosphorylation)			RPS6		C488369
CTD	decreases(expression)			RPSAP52		C488369
CTD	decreases(expression)			RRM1		C488369
CTD	decreases(expression)			RRM2		C488369
CTD	increases(expression)			SDC2		C488369
CTD	decreases(expression)			SEMA3A		C488369
CTD	increases(expression)			SEPP1		C488369
CTD	decreases(expression)			SERPINB2		C488369
CTD	decreases(expression)			SERPINB7		C488369
CTD	decreases(expression)			SGOL1		C488369
CTD	decreases(expression)			SGOL2		C488369
CTD	decreases(expression)			SHCBP1		C488369
CTD	decreases(expression)			SKA1		C488369
CTD	decreases(expression)			SKA3		C488369
CTD	decreases(expression)			SLC16A6		C488369
CTD	increases(expression)			SLC1A4		C488369
CTD	decreases(expression)			SLC20A1		C488369
CTD	increases(expression)			SLC40A1		C488369
CTD	increases(expression)			SLC6A6		C488369
CTD	decreases(expression)			SLFN11		C488369
CTD	decreases(expression)			SMC2		C488369
CTD	decreases(expression)			SMC4		C488369
CTD	decreases(expression)			SNORD14E		C488369
CTD	decreases(expression)			SNORD30		C488369
CTD	decreases(expression)			SNORD50B		C488369
CTD	decreases(localization)			SOX17		C488369
CTD	increases(expression)			SOX4		C488369
CTD	decreases(expression)			SPRY2		C488369
CTD	affects(binding)			SRC		C488369
CTD	decreases(activity)			SRC		C488369
CTD	decreases(activity)			SRC		C488369
CTD	decreases(phosphorylation)			SRC		C488369
CTD	decreases(phosphorylation)			SRC		C488369
CTD	decreases(phosphorylation)			SRC		C488369
CTD	decreases(reaction)			STAT1		C488369
CTD	increases(phosphorylation)			STAT1		C488369
CTD	affects(localization)			STAT1		C488369
CTD	increases(expression)			STAT1		C488369
CTD	decreases(phosphorylation)			STAT3		C488369
CTD	decreases(phosphorylation)			STAT3		C488369
CTD	increases(response to substance)			STAT3		C488369
CTD	decreases(expression)			STC1		C488369
CTD	decreases(expression)			STEAP1		C488369
CTD	decreases(expression)			STEAP1B		C488369
CTD	decreases(expression)			STIL		C488369
CTD	increases(expression)			STK38L		C488369
CTD	decreases(expression)			STMN1		C488369
CTD	increases(expression)			SULF1		C488369
CTD	increases(expression)			SULF2		C488369
CTD	increases(expression)			SVEP1		C488369
CTD	increases(expression)			SYNPO2		C488369
CTD	increases(expression)			SYT15		C488369
CTD	decreases(expression)			TACC3		C488369
CTD	decreases(expression)			TCF19		C488369
CTD	increases(expression)			TCP11L2		C488369
CTD	decreases(expression)			TDP1		C488369
CTD	affects(binding)			TEC		C488369
CTD	decreases(activity)			TEC		C488369
CTD	affects(binding)			TEC		C488369
CTD	decreases(expression)			TEX30		C488369
CTD	increases(expression)			TGFB2		C488369
CTD	increases(expression)			THBS2		C488369
CTD	increases(expression)			THBS3		C488369
CTD	decreases(expression)			TICRR		C488369
CTD	decreases(expression)			TIMELESS		C488369
CTD	decreases(expression)			TIPIN		C488369
CTD	decreases(expression)			TK1		C488369
CTD	increases(expression)			TM6SF1		C488369
CTD	increases(expression)			TMEM155		C488369
CTD	decreases(expression)			TMEM194A		C488369
CTD	decreases(expression)			TMPO		C488369
CTD	decreases(reaction)			TNF		C488369
CTD	increases(secretion)			TNF		C488369
CTD	decreases(expression)			TNF		C488369
CTD	decreases(secretion)			TNF		C488369
CTD	increases(expression)			TNS3		C488369
CTD	decreases(expression)			TOP2A		C488369
CTD	increases(expression)			TP53INP1		C488369
CTD	increases(expression)			TPD52L1		C488369
CTD	decreases(expression)			TPX2		C488369
CTD	decreases(expression)			TRIP13		C488369
CTD	decreases(expression)			TRPA1		C488369
CTD	increases(expression)			TSPAN2		C488369
CTD	decreases(expression)			TTK		C488369
CTD	increases(expression)			TXNIP		C488369
CTD	decreases(expression)			UBE2S		C488369
CTD	decreases(expression)			UBE2T		C488369
CTD	decreases(expression)			UHRF1		C488369
CTD	decreases(expression)			VEPH1		C488369
CTD	increases(expression)			VLDLR		C488369
CTD	decreases(expression)			VRK1		C488369
CTD	decreases(expression)			WDHD1		C488369
CTD	decreases(expression)			WDR76		C488369
CTD	decreases(expression)			WHSC1		C488369
CTD	decreases(expression)			XRCC2		C488369
CTD	affects(binding)			YES1		C488369
CTD	affects(binding)			ZAK		C488369
CTD	increases(response to substance)			ZAP70		C488369
CTD	decreases(expression)			ZWILCH		C488369
CTD	decreases(expression)			ZWINT		C488369
PubChem	None	uM	0.530	ABL1	-	GI(Protien) :
PubChem	None	uM	0.720	ABL1	-	GI(Protien) :
PubChem	None	uM	0.960	ABL1	-	GI(Protien) :
PubChem	None	uM	1.100	ABL1	-	GI(Protien) :
PubChem	None	uM	1.200	ABL1	-	GI(Protien) :
PubChem	None	uM	2.100	ABL1	-	GI(Protien) :
PubChem	None	uM	0.170	ABL2	-	GI(Protien) :
PubChem	Potency-Replicate_1	uM	1.188	AHR	-	GI(Protien) :
PubChem	Ratio Potency (uM)	uM	10.682	AR	-	GI(Protien) :
PubChem	Potency-Replicate_1	uM	11.986	AR	-	GI(Protien) :
PubChem	Potency-Replicate_1	uM	26.603	AR	-	GI(Protien) :
PubChem	None	uM	0.210	BLK	-	GI(Protien) :
PubChem	None	uM	1.400	BMX	-	GI(Protien) :
PubChem	None	uM	1.400	BTK	-	GI(Protien) :
PubChem	None	uM	0.580	CSF1R	-	GI(Protien) :
PubChem	None	uM	1.000	CSK	-	GI(Protien) :
PubChem	Potency-Replicate_1	uM	1.333	CYP19A1	-	GI(Protien) :
PubChem	None	uM	0.690	DDR1	-	GI(Protien) :
PubChem	None	uM	3.200	DDR2	-	GI(Protien) :
PubChem	None	uM	4.100	EPHA1	-	GI(Protien) :
PubChem	None	uM	0.850	EPHA2	-	GI(Protien) :
PubChem	None	uM	0.093	EPHA3	-	GI(Protien) :
PubChem	None	uM	1.200	EPHA4	-	GI(Protien) :
PubChem	None	uM	0.240	EPHA5	-	GI(Protien) :
PubChem	None	uM	0.240	EPHA8	-	GI(Protien) :
PubChem	None	uM	0.450	EPHB1	-	GI(Protien) :
PubChem	None	uM	0.390	EPHB2	-	GI(Protien) :
PubChem	None	uM	6.900	EPHB3	-	GI(Protien) :
PubChem	None	uM	0.340	EPHB4	-	GI(Protien) :
PubChem	None	uM	0.500	FGR	-	GI(Protien) :
PubChem	None	uM	0.310	FRK	-	GI(Protien) :
PubChem	None	uM	0.790	FYN	-	GI(Protien) :
PubChem	None	uM	2.600	GAK	-	GI(Protien) :
PubChem	Potency	uM	16.789	GMNN	-	GI(Protien) :
PubChem	Potency	uM	18.837	GMNN	-	GI(Protien) :
PubChem	None	uM	0.350	HCK	-	GI(Protien) :
PubChem	None	uM	0.620	KIT	-	GI(Protien) :
PubChem	None	uM	0.680	KIT	-	GI(Protien) :
PubChem	None	uM	2.600	KIT	-	GI(Protien) :
PubChem	None	uM	2.700	KIT	-	GI(Protien) :
PubChem	None	uM	0.200	LCK	-	GI(Protien) :
PubChem	None	uM	0.570	LYN	-	GI(Protien) :
PubChem	None	uM		NR0B1	-	GI(Protien) :
PubChem	None	uM		NR2F2	-	GI(Protien) :
PubChem	None	uM		NR3C1	-	GI(Protien) :
PubChem	None	uM	0.470	PDGFRA	-	GI(Protien) :
PubChem	None	uM	0.630	PDGFRB	-	GI(Protien) :
PubChem	Potency-Replicate_1	uM	0.473	PPARD	-	GI(Protien) :
PubChem	None	uM		PPARG	-	GI(Protien) :
PubChem	None	uM		PRNP	-	GI(Protien) :
PubChem	None	uM	7.800	PTK6	-	GI(Protien) :
PubChem	None	uM	3.900	SIK1	-	GI(Protien) :
PubChem	None	uM	6.400	SIK2	-	GI(Protien) :
PubChem	Potency	uM	1.259	SMAD3	-	GI(Protien) :
PubChem	None	uM	0.210	SRC	-	GI(Protien) :
PubChem	Potency	uM	2.114	TDP1	-	GI(Protien) :
PubChem	Potency	uM	2.372	TDP1	-	GI(Protien) :
PubChem	Potency	uM	2.818	TDP1	-	GI(Protien) :
PubChem	Potency	uM	3.981	TDP1	-	GI(Protien) :
PubChem	None	uM	5.600	TNK2	-	GI(Protien) :
PubChem	None	uM	2.100	TXK	-	GI(Protien) :
PubChem	Potency	uM	0.002	YES1		GI(Protien) :
PubChem	None	uM	0.300	YES1	-	GI(Protien) :
ChEMBL	Activity	-		BTK	-	Target : CHEMBL5251
ChEMBL	Activity	-		BTK	-	Target : CHEMBL5251
ChEMBL	Activity	-		BTK	-	Target : CHEMBL5251
ChEMBL	Activity	-		BTK	-	Target : CHEMBL5251
ChEMBL	Activity	-		SRC	-	Target : CHEMBL267
ChEMBL	Activity	-		SRC	-	Target : CHEMBL267
ChEMBL	Activity	-		SRC	-	Target : CHEMBL267
ChEMBL	Activity	-		SRC	-	Target : CHEMBL267
ChEMBL	Activity	-		TEC	-	Target : CHEMBL4246

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