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Gene Set: D1 - Approved - 5-AZACYTIDINE

Collection D1 : Approved
Chemical Name 5-AZACYTIDINE
FDA NPC WHO Indian Australia China Traditional
Herbal		 Clinical
Trail
ApprovedNotNotNotNotNotNotNot
Molecular
Weight		 Hydrogen Bond
Donor Count		 Hydrogen Bond
Acceptor Count		 cLogP Lipinski Rule
244.205 g/mol 4 9 -2.5868 True
Structure
InChI InChI=1S/C8H12N4O5/c9-7-10-2-12(8(16)11-7)6-5(15)4(14)3(1-13)17-6/h2-6,13-15H,1H2,(H2,9,11,16)/t3-,4-,5-,6-/m1/s1
InChIKey NMUSYJAQQFHJEW-KVTDHHQDSA-N
Links

Gene (29 / 80)


⊖ Less
Source Type Unit Value Gene PMID Assay Other
PubChem PotencyuM22.387ALDH1A1-GI(Protien) :
PubChem PotencyuM1.096AR-GI(Protien) :
PubChem AR Potency (uM)uM2.342AR-GI(Protien) :
PubChem PotencyuM2.731AR-GI(Protien) :
PubChem PotencyuM3.378AR-GI(Protien) :
PubChem PotencyuM5.956AR-GI(Protien) :
PubChem PotencyuM1.254ATAD5-GI(Protien) :
PubChem PotencyuM2.818ATAD5-GI(Protien) :
PubChem PotencyuM5.601ATAD5-GI(Protien) :
PubChem PotencyuM8.196ATAD5-GI(Protien) :
PubChem PotencyuM15.785ATAD5-GI(Protien) :
PubChem uMBARD1-GI(Protien) :
PubChem uMBRCA1-GI(Protien) :
PubChem PotencyuM8.635CYP19A1-GI(Protien) :
PubChem PotencyuM13.333CYP19A1-GI(Protien) :
PubChem uMDNMT1-GI(Protien) :
PubChem uMDNMT3A-GI(Protien) :
PubChem IC50_1_GAPDH 24hruM0.557GAPDH-GI(Protien) :
PubChem IC50_1_GAPDH 6hruM2.732GAPDH-GI(Protien) :
PubChem IC50_PEG-3_MeanuMGAPDH-GI(Protien) :
PubChem PotencyuM3.162GMNN-GI(Protien) :
PubChem PotencyuM1.259HBB-GI(Protien) :
PubChem PotencyuM12.589HTT-GI(Protien) :
PubChem PotencyuM1.636IDH1-GI(Protien) :
PubChem uMMDM2-GI(Protien) :
PubChem uMMDM2-GI(Protien) :
PubChem uMMDM4-GI(Protien) :
PubChem uMMDM4-GI(Protien) :
PubChem uMMITF-GI(Protien) :
PubChem uMNCOA1-GI(Protien) :
PubChem uMNCOA3-GI(Protien) :
PubChem uMNCOA3-GI(Protien) :
PubChem PotencyuM1.369NFE2L2-GI(Protien) :
PubChem PotencyuM1.536NFE2L2-GI(Protien) :
PubChem Ratio Potency (uM)uM1.790NFE2L2-GI(Protien) :
PubChem PotencyuM1.883NFE2L2-GI(Protien) :
PubChem PotencyuM2.660NFE2L2-GI(Protien) :
PubChem Ratio Potency (uM)uM3.223NFE2L2-GI(Protien) :
PubChem uMNR1H4-GI(Protien) :
PubChem PotencyuM1.738NR3C1-GI(Protien) :
PubChem PotencyuM3.011NR3C1-GI(Protien) :
PubChem PotencyuM5.623NR3C1-GI(Protien) :
PubChem PotencyuM7.943NR3C1-GI(Protien) :
PubChem uMNR3C1-GI(Protien) :
PubChem uMNR5A1-GI(Protien) :
PubChem uMNR5A2-GI(Protien) :
PubChem uMNR5A2-GI(Protien) :
PubChem uMPRNP-GI(Protien) :
PubChem PotencyuM3.349RORC-GI(Protien) :
PubChem PotencyuM11.220SMAD3-GI(Protien) :
PubChem PotencyuM2.512TDP1-GI(Protien) :
PubChem PotencyuM3.162TDP1-GI(Protien) :
PubChem PotencyuM6.684TDP1-GI(Protien) :
PubChem PotencyuM7.308TDP1-GI(Protien) :
PubChem PotencyuM7.499TDP1-GI(Protien) :
PubChem PotencyuM8.200TDP1-GI(Protien) :
PubChem PotencyuM3.162THPO-GI(Protien) :
PubChem PotencyuM2.113TP53-GI(Protien) :
PubChem Ratio Potency (uM)uM3.254TP53-GI(Protien) :
PubChem PotencyuM4.856TP53-GI(Protien) :
PubChem Ratio Potency (uM)uM5.661TP53-GI(Protien) :
PubChem PotencyuM6.310TP53-GI(Protien) :
ChEMBLPotencynM22387.200ALDH1A1
-Target : CHEMBL3577
ChEMBLPotencynM15785.000ATAD5
-Target : CHEMBL1741209
ChEMBLPotencynM2818.400ATAD5
-Target : CHEMBL1741209
ChEMBLPotencynM8196.100ATAD5
-Target : CHEMBL1741209
ChEMBLPotencynM5600.700ATAD5
-Target : CHEMBL1741209
ChEMBLPotencynM1253.800ATAD5
-Target : CHEMBL1741209
ChEMBLPotencynM3162.300GMNN
-Target : CHEMBL1293278
ChEMBLPotencynM1258.900HBB
-Target : CHEMBL4331
ChEMBLPotencynM12589.300HTT
-Target : CHEMBL5514
ChEMBLPotencynM1636.000IDH1
-Target : CHEMBL2007625
ChEMBLPotencynM1883.400NFE2L2
-Target : CHEMBL1075094
ChEMBLPotencynM1368.500NFE2L2
-Target : CHEMBL1075094
ChEMBLPotencynM5623.400NR3C1
-Target : CHEMBL2034
ChEMBLPotencynM7943.300NR3C1
-Target : CHEMBL2034
ChEMBLPotencynM3349.100RORC
-Target : CHEMBL1741186
ChEMBLPotencynM11220.200SMAD3
-Target : CHEMBL1293258
ChEMBLPotencynM3162.300THPO
-Target : CHEMBL1293256
ChEMBLPotencynM6309.600TP53
-Target : CHEMBL4096
Download gene sets gmt, text, Detailed text
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