Drug Gene Type Source bromocriptine DRD3 IC50=0.000596(uM) D1 PubChem bromocriptine DRD2 IC50=0.00158(uM) D1 PubChem bromocriptine HTR2B IC50=0.00832(uM) D1 PubChem bromocriptine DRD2 Ki=0.01(uM) D1 PubChem bromocriptine ADRA2A IC50=0.015(uM) D1 PubChem bromocriptine HTR6 IC50=0.022(uM) D1 PubChem bromocriptine HTR1A Ki=0.024(uM) D1 PubChem bromocriptine ADRA1D IC50=0.03(uM) D1 PubChem bromocriptine ADRA2B IC50=0.035(uM) D1 PubChem bromocriptine HTR2A IC50=0.036(uM) D1 PubChem bromocriptine HTR6 Ki=0.05(uM) D1 PubChem bromocriptine DRD3 Ki=0.087(uM) D1 PubChem bromocriptine ADRA2C IC50=0.52(uM) D1 PubChem bromocriptine HTR2C IC50=0.532(uM) D1 PubChem bromocriptine CYP3A4 IC50=2.0(uM) D1 PubChem bromocriptine ADRB1 IC50=2.4(uM) D1 PubChem bromocriptine DRD1 IC50=2.889(uM) D1 PubChem bromocriptine DRD1 Potency=3.2643(uM) D1 PubChem bromocriptine TDP1 Potency=9.4411(uM) D1 PubChem bromocriptine ESR1 Potency=9.5205(uM) D1 PubChem bromocriptine ESR1 Ratio Potency (uM)=17.5925(uM) D1 PubChem bromocriptine TDP1 Potency=21.136(uM) D1 PubChem bromocriptine AR Potency=21.3138(uM) D1 PubChem bromocriptine AR Ratio Potency (uM)=22.1476(uM) D1 PubChem bromocriptine AR AR Potency (uM)=25.1151(uM) D1 PubChem bromocriptine AR Potency=26.6032(uM) D1 PubChem bromocriptine VDR Potency=28.1838(uM) D1 PubChem bromocriptine DRD3 - D1 PubChem bromocriptine HTR1A - D1 PubChem bromocriptine STK33 - D1 PubChem bromocriptine HTR1B - D1 PubChem bromocriptine HTR1D - D1 PubChem bromocriptine HTR6 - D1 PubChem bromocriptine HTR2B - D1 PubChem bromocriptine HTR2C - D1 PubChem bromocriptine HTR2A - D1 PubChem bromocriptine NR3C1 - D1 PubChem bromocriptine VDR Potency=28183.8(nM) D1 ChEMBL bromocriptine EHMT2 Potency=23778.1(nM) D1 ChEMBL bromocriptine EHMT2 Potency=14125.4(nM) D1 ChEMBL bromocriptine VDR Potency=17782.8(nM) D1 ChEMBL bromocriptine DRD1 Potency=3264.3(nM) D1 ChEMBL