Drug Gene Type Source NSC 95397 CDC25B Text_Mining(Inhibitor) TTD NSC 95397 CDC25A Text_Mining(Inhibitor) TTD NSC 95397 ABHD5 None=None(uM) D4 PubChem NSC 95397 AHR None=None(uM) D4 PubChem NSC 95397 ALDH1A1 Potency=17.7828(uM) D4 PubChem NSC 95397 ALDH1A1 Potency=17782.8(nM) D4 ChEMBL NSC 95397 APAF1 IC50_Mean=12.7(uM) D4 PubChem NSC 95397 APAF1 None=None(uM) D4 PubChem NSC 95397 APOBEC3G Potency=4.7318(uM) D4 PubChem NSC 95397 APOBEC3G None=None(uM) D4 PubChem NSC 95397 ATG4B IC50_Mean=12.8(uM) D4 PubChem NSC 95397 ATG4B None=None(uM) D4 PubChem NSC 95397 ATG4B IC50=12800.0(nM) D4 ChEMBL NSC 95397 ATXN2 Potency=4.4668(uM) D4 PubChem NSC 95397 ATXN2 Potency=15.8489(uM) D4 PubChem NSC 95397 BLM Potency=7.0795(uM) D4 PubChem NSC 95397 BLM Potency=8.9125(uM) D4 PubChem NSC 95397 BLM Potency=28.1838(uM) D4 PubChem NSC 95397 BLM Potency=7079.5(nM) D4 ChEMBL NSC 95397 BLM Potency=8912.5(nM) D4 ChEMBL NSC 95397 BLM Potency=28183.8(nM) D4 ChEMBL NSC 95397 CASP1 Potency=15.8489(uM) D4 PubChem NSC 95397 CASP1 Potency=15848.9(nM) D4 ChEMBL NSC 95397 CASP3 IC50_Mean=9.83(uM) D4 PubChem NSC 95397 CASP9 IC50_Mean=9.83(uM) D4 PubChem NSC 95397 CBX1 Potency=10.0(uM) D4 PubChem NSC 95397 CBX1 Potency=10000.0(nM) D4 ChEMBL NSC 95397 CCR6 None=None(uM) D4 PubChem NSC 95397 CFTR None=None(uM) D4 PubChem NSC 95397 CHRM4 None=None(uM) D4 PubChem NSC 95397 CHRM5 None=None(uM) D4 PubChem NSC 95397 CXCR6 None=None(uM) D4 PubChem NSC 95397 CYP1A2 None=None(uM) D4 PubChem NSC 95397 CYP1A2 AC50=630.96(nM) D4 ChEMBL NSC 95397 CYP2C19 Potency=0.0794(uM) D4 PubChem NSC 95397 CYP2C19 Potency=0.5012(uM) D4 PubChem NSC 95397 CYP2C19 None=None(uM) D4 PubChem NSC 95397 CYP2C19 Potency=79.4(nM) D4 ChEMBL NSC 95397 CYP2C19 AC50=79.43(nM) D4 ChEMBL NSC 95397 CYP2C19 Potency=501.2(nM) D4 ChEMBL NSC 95397 CYP2C9 Potency=5.0119(uM) D4 PubChem NSC 95397 CYP2C9 Potency=12.5893(uM) D4 PubChem NSC 95397 CYP2C9 None=None(uM) D4 PubChem NSC 95397 CYP2C9 AC50=5011.87(nM) D4 ChEMBL NSC 95397 CYP2C9 Potency=12589.3(nM) D4 ChEMBL NSC 95397 CYP2C9 Potency=5011.9(nM) D4 ChEMBL NSC 95397 CYP2D6 Potency=7.9433(uM) D4 PubChem NSC 95397 CYP2D6 Potency=7943.3(nM) D4 ChEMBL NSC 95397 CYP3A4 Potency=25.1189(uM) D4 PubChem NSC 95397 CYP3A4 None=None(uM) D4 PubChem NSC 95397 CYP3A4 AC50=25118.9(nM) D4 ChEMBL NSC 95397 CYP3A4 Potency=25118.9(nM) D4 ChEMBL NSC 95397 DNMT1 None=None(uM) D4 PubChem NSC 95397 DRD1 Potency=11.2202(uM) D4 PubChem NSC 95397 DRD1 None=None(uM) D4 PubChem NSC 95397 DRD1 Potency=11220.2(nM) D4 ChEMBL NSC 95397 DRD3 None=None(uM) D4 PubChem NSC 95397 EHMT2 Potency=1.2589(uM) D4 PubChem NSC 95397 EHMT2 Potency=1258.9(nM) D4 ChEMBL NSC 95397 EPAS1 None=None(uM) D4 PubChem NSC 95397 ERG Potency=12.5893(uM) D4 PubChem NSC 95397 ERG Potency=50.1187(uM) D4 PubChem NSC 95397 EYA2 Potency=50.1187(uM) D4 PubChem NSC 95397 EYA2 Potency=50118.7(nM) D4 ChEMBL NSC 95397 GALK1 Potency=18.8181(uM) D4 PubChem NSC 95397 GALK1 Potency=25.1189(uM) D4 PubChem NSC 95397 GALK1 Potency=18818.1(nM) D4 ChEMBL NSC 95397 GALK1 Potency=25118.9(nM) D4 ChEMBL NSC 95397 GAPDH Potency=3.9811(uM) D4 PubChem NSC 95397 GAPDH None=None(uM) D4 PubChem NSC 95397 GAPDH Potency=3981.1(nM) D4 ChEMBL NSC 95397 GLS Potency=10.0(uM) D4 PubChem NSC 95397 GMNN Potency=3.9811(uM) D4 PubChem NSC 95397 GMNN Potency=3981.1(nM) D4 ChEMBL NSC 95397 GNA15 None=None(uM) D4 PubChem NSC 95397 GNAI1 None=None(uM) D4 PubChem NSC 95397 GSTO1 None=None(uM) D4 PubChem NSC 95397 HCRTR1 None=None(uM) D4 PubChem NSC 95397 HKDC1 IC50_Mean=3.15(uM) D4 PubChem NSC 95397 HKDC1 IC50_Mean=8.11(uM) D4 PubChem NSC 95397 HKDC1 None=None(uM) D4 PubChem NSC 95397 HKDC1 IC50=3150.0(nM) D4 ChEMBL NSC 95397 HKDC1 IC50=8110.0(nM) D4 ChEMBL NSC 95397 HNF4A None=None(uM) D4 PubChem NSC 95397 HPGD Potency=2.8184(uM) D4 PubChem NSC 95397 HPGD Potency=2818.4(nM) D4 ChEMBL NSC 95397 HSD17B10 Potency=12589.3(nM) D4 ChEMBL NSC 95397 HSP90AA1 None=None(uM) D4 PubChem NSC 95397 HTR5A None=None(uM) D4 PubChem NSC 95397 IDE None=None(uM) D4 PubChem NSC 95397 IL1B None=None(uM) D4 PubChem NSC 95397 KCNK3 None=None(uM) D4 PubChem NSC 95397 KDM4A Potency=8912.5(nM) D4 ChEMBL NSC 95397 KMT2A Potency=39.7828(uM) D4 PubChem NSC 95397 KMT2A Potency=39782.8(nM) D4 ChEMBL NSC 95397 LYPLA2 None=None(uM) D4 PubChem NSC 95397 MAPK1 Potency=15.8489(uM) D4 PubChem NSC 95397 MAPK1 Potency=15848.9(nM) D4 ChEMBL NSC 95397 MAPT Potency=1.122(uM) D4 PubChem NSC 95397 MAPT Potency=2.5119(uM) D4 PubChem NSC 95397 MAPT Potency=14.1254(uM) D4 PubChem NSC 95397 MAPT None=None(uM) D4 PubChem NSC 95397 MAPT Potency=1995.3(nM) D4 ChEMBL NSC 95397 MAPT Potency=2511.9(nM) D4 ChEMBL NSC 95397 MAPT Potency=1122.0(nM) D4 ChEMBL NSC 95397 MAPT Potency=14125.4(nM) D4 ChEMBL NSC 95397 MBNL1 Potency=5.0119(uM) D4 PubChem NSC 95397 MBNL1 Potency=10.0(uM) D4 PubChem NSC 95397 MBNL1 Potency=10000.0(nM) D4 ChEMBL NSC 95397 MBNL1 Potency=5011.9(nM) D4 ChEMBL NSC 95397 MC4R None=None(uM) D4 PubChem NSC 95397 MDM2 None=None(uM) D4 PubChem NSC 95397 MDM4 None=None(uM) D4 PubChem NSC 95397 MEN1 Potency=39.7828(uM) D4 PubChem NSC 95397 MEN1 Potency=39782.8(nM) D4 ChEMBL NSC 95397 MITF None=None(uM) D4 PubChem NSC 95397 MRGPRX1 None=None(uM) D4 PubChem NSC 95397 MTOR Potency=3.6898(uM) D4 PubChem NSC 95397 MTOR Potency=3689.8(nM) D4 ChEMBL NSC 95397 NFE2L2 Potency=25.929(uM) D4 PubChem NSC 95397 NFE2L2 Potency=25929.0(nM) D4 ChEMBL NSC 95397 NOD2 None=None(uM) D4 PubChem NSC 95397 NPSR1 Potency=12.5893(uM) D4 PubChem NSC 95397 NPSR1 Potency=12589.3(nM) D4 ChEMBL NSC 95397 NR5A1 None=None(uM) D4 PubChem NSC 95397 NR5A2 None=None(uM) D4 PubChem NSC 95397 PADI4 None=None(uM) D4 PubChem NSC 95397 PAFAH1B2 None=None(uM) D4 PubChem NSC 95397 PAFAH1B3 None=None(uM) D4 PubChem NSC 95397 PAFAH2 None=None(uM) D4 PubChem NSC 95397 PAX8 None=None(uM) D4 PubChem NSC 95397 PLIN5 None=None(uM) D4 PubChem NSC 95397 PLK1 Potency=2.1192(uM) D4 PubChem NSC 95397 POLH Potency=15.8489(uM) D4 PubChem NSC 95397 POLH Potency=23.9341(uM) D4 PubChem NSC 95397 POLH Potency=31.6228(uM) D4 PubChem NSC 95397 POLI Potency=1.122(uM) D4 PubChem NSC 95397 POLI Potency=3.5481(uM) D4 PubChem NSC 95397 POLI Potency=23.7781(uM) D4 PubChem NSC 95397 PPME1 None=None(uM) D4 PubChem NSC 95397 PRMT1 None=None(uM) D4 PubChem NSC 95397 PRNP None=None(uM) D4 PubChem NSC 95397 PSIP1 None=None(uM) D4 PubChem NSC 95397 PTGER2 None=None(uM) D4 PubChem NSC 95397 RACGAP1 IC50=32.49(uM) D4 PubChem NSC 95397 RGS12 None=None(uM) D4 PubChem NSC 95397 RGS4 Potency=3.3587(uM) D4 PubChem NSC 95397 RIPK2 None=None(uM) D4 PubChem NSC 95397 SENP6 None=None(uM) D4 PubChem NSC 95397 SENP7 None=None(uM) D4 PubChem NSC 95397 SENP8 None=None(uM) D4 PubChem NSC 95397 SMAD3 Potency=3.1623(uM) D4 PubChem NSC 95397 SMAD3 Potency=7.0795(uM) D4 PubChem NSC 95397 STAT6 Potency=6.3096(uM) D4 PubChem NSC 95397 STAT6 Potency=6309.6(nM) D4 ChEMBL NSC 95397 STK33 None=None(uM) D4 PubChem NSC 95397 TAAR1 None=None(uM) D4 PubChem NSC 95397 TDP1 Potency=0.0517(uM) D4 PubChem NSC 95397 TDP1 Potency=0.1636(uM) D4 PubChem NSC 95397 TDP1 Potency=0.3981(uM) D4 PubChem NSC 95397 TDP1 Potency=0.5623(uM) D4 PubChem NSC 95397 TDP1 Potency=0.631(uM) D4 PubChem NSC 95397 TDP1 Potency=0.7499(uM) D4 PubChem NSC 95397 TDP2 None=None(uM) D4 PubChem NSC 95397 THPO Potency=1.2589(uM) D4 PubChem NSC 95397 THPO Potency=1258.9(nM) D4 ChEMBL NSC 95397 THRB Potency=14.1254(uM) D4 PubChem NSC 95397 THRB Potency=14125.4(nM) D4 ChEMBL NSC 95397 TLR9 IC50=1.869(uM) D4 PubChem NSC 95397 TLR9 None=None(uM) D4 PubChem NSC 95397 TP53 Potency=0.631(uM) D4 PubChem NSC 95397 TP53 Potency=0.7943(uM) D4 PubChem NSC 95397 TP53 Potency=631.0(nM) D4 ChEMBL NSC 95397 TP53 Potency=794.3(nM) D4 ChEMBL NSC 95397 TSHR Potency=3.3808(uM) D4 PubChem NSC 95397 TSHR Potency=25.1189(uM) D4 PubChem NSC 95397 TSHR None=None(uM) D4 PubChem NSC 95397 TSHR Potency=25118.9(nM) D4 ChEMBL NSC 95397 USP1 Potency=6.3096(uM) D4 PubChem NSC 95397 USP1 Potency=15.8489(uM) D4 PubChem NSC 95397 VDR Potency=5.6234(uM) D4 PubChem NSC 95397 WRN Potency=79.4328(uM) D4 PubChem