Drug Gene Type Source methotrexate DHFR Text_Mining(Inhibitor) TTD methotrexate PDF Text_Mining(Inhibitor) TTD methotrexate APEX1 Potency=19952.6(nM) D4 ChEMBL methotrexate CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL methotrexate CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL methotrexate CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL methotrexate CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL methotrexate CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL methotrexate EHMT2 Potency=7.5193(uM) D4 PubChem methotrexate EHMT2 Potency=7.9433(uM) D4 PubChem methotrexate EHMT2 Potency=7943.3(nM) D4 ChEMBL methotrexate EHMT2 Potency=7519.3(nM) D4 ChEMBL methotrexate HSD17B10 Potency=31622.8(nM) D4 ChEMBL methotrexate IDH1 Potency=0.0052(uM) D4 PubChem methotrexate KLK7 None=None(uM) D4 PubChem methotrexate MDM2 None=None(uM) D4 PubChem methotrexate MDM4 None=None(uM) D4 PubChem methotrexate MPHOSPH8 Potency=79.4328(uM) D4 PubChem methotrexate MPHOSPH8 Potency=79432.8(nM) D4 ChEMBL methotrexate NCOA1 None=None(uM) D4 PubChem methotrexate NCOA3 IC50=0.21097(uM) D4 PubChem methotrexate NCOA3 None=None(uM) D4 PubChem methotrexate NFE2L2 Potency-Replicate_1=0.0097(uM) D4 PubChem methotrexate NFE2L2 Potency-Replicate_1=0.0596(uM) D4 PubChem methotrexate NFE2L2 Potency=0.1536(uM) D4 PubChem methotrexate NFE2L2 Potency=0.5805(uM) D4 PubChem methotrexate NFE2L2 Potency=1.4581(uM) D4 PubChem methotrexate NFE2L2 Potency=580.5(nM) D4 ChEMBL methotrexate NFE2L2 Potency=1458.1(nM) D4 ChEMBL methotrexate NR1H4 Potency-Replicate_1=0.3758(uM) D4 PubChem methotrexate NR5A1 None=None(uM) D4 PubChem methotrexate NR5A2 None=None(uM) D4 PubChem methotrexate POLB Potency=39.8107(uM) D4 PubChem methotrexate POLB Potency=39810.7(nM) D4 ChEMBL methotrexate POLH Potency=31.6228(uM) D4 PubChem methotrexate POLI Potency=31.6228(uM) D4 PubChem methotrexate PPARG Potency=0.4467(uM) D4 PubChem methotrexate TDP1 Potency=0.0103(uM) D4 PubChem methotrexate TDP1 Potency=0.0106(uM) D4 PubChem methotrexate TDP1 Potency=0.0211(uM) D4 PubChem methotrexate TDP1 Potency=0.0411(uM) D4 PubChem methotrexate TDP1 Potency=0.1259(uM) D4 PubChem methotrexate TNFRSF10B None=None(uM) D4 PubChem methotrexate VDR Potency=39.8107(uM) D4 PubChem