Drug Gene Type Source ketoconazole CYP51A1 Text_Mining(Inhibitor) TTD ketoconazole CYP51A1 Text_Mining(Drug(s)) TTD ketoconazole ABCB1 None=None(uM) D4 PubChem ketoconazole AHR AhR Potency (uM)=0.485577(uM) D4 PubChem ketoconazole AHR Potency-Replicate_1=6.6824(uM) D4 PubChem ketoconazole AR Potency-Replicate_1=9.77(uM) D4 PubChem ketoconazole AR Potency-Replicate_1=30.6379(uM) D4 PubChem ketoconazole BAZ2B Potency=17.7828(uM) D4 PubChem ketoconazole BAZ2B Potency=35.4813(uM) D4 PubChem ketoconazole CBX1 Potency=39.8107(uM) D4 PubChem ketoconazole CYP19A1 Potency-Replicate_1=30.6379(uM) D4 PubChem ketoconazole CYP1A2 None=None(uM) D4 PubChem ketoconazole CYP2C19 Potency=12.5893(uM) D4 PubChem ketoconazole CYP2C19 None=None(uM) D4 PubChem ketoconazole CYP2C9 Potency=12.5893(uM) D4 PubChem ketoconazole CYP2C9 None=None(uM) D4 PubChem ketoconazole CYP3A4 Potency=0.1259(uM) D4 PubChem ketoconazole CYP3A4 None=None(uM) D4 PubChem ketoconazole EHMT2 Potency=10.0(uM) D4 PubChem ketoconazole EHMT2 Potency=25.1189(uM) D4 PubChem ketoconazole EHMT2 Potency=39.8107(uM) D4 PubChem ketoconazole ESR1 Potency-Replicate_1=13.3332(uM) D4 PubChem ketoconazole ESR1 ER Potency (uM)=26.6032(uM) D4 PubChem ketoconazole HSP90AA1 AC50_uM=0.435(uM) D4 PubChem ketoconazole HSPB1 Ratio Potency (uM)=43.6412(uM) D4 PubChem ketoconazole MPHOSPH8 Potency=39.8107(uM) D4 PubChem ketoconazole NFE2L2 Ratio Potency (uM)=2.34203(uM) D4 PubChem ketoconazole NFE2L2 Potency=18.3564(uM) D4 PubChem ketoconazole NFE2L2 Potency=30.6379(uM) D4 PubChem ketoconazole NR1H4 Potency-Replicate_1=43.6412(uM) D4 PubChem ketoconazole NR1H4 Potency=44.6684(uM) D4 PubChem ketoconazole PLA2G7 None=None(uM) D4 PubChem ketoconazole PREPL None=None(uM) D4 PubChem ketoconazole SLC6A3 None=None(uM) D4 PubChem ketoconazole TDP1 Potency=6.3096(uM) D4 PubChem ketoconazole TDP1 Potency=6.5131(uM) D4 PubChem ketoconazole TDP1 Potency=11.8856(uM) D4 PubChem ketoconazole TDP1 Potency=20.5962(uM) D4 PubChem ketoconazole VDR Potency=44.6684(uM) D4 PubChem