Drug Gene Type Source Canertinib dihydrochloride ERBB4 Text_Mining(Multitarget) TTD Canertinib dihydrochloride ERBB4 Text_Mining(Inhibitor) TTD Canertinib dihydrochloride ERBB4 Text_Mining(Drug(s)) TTD Canertinib dihydrochloride AKT1 Text_Mining(Multitarget) TTD Canertinib dihydrochloride AKT2 Text_Mining(Multitarget) TTD Canertinib dihydrochloride AKT3 Text_Mining(Multitarget) TTD Canertinib dihydrochloride AKT1 Text_Mining(Inhibitor) TTD Canertinib dihydrochloride AKT2 Text_Mining(Inhibitor) TTD Canertinib dihydrochloride AKT3 Text_Mining(Inhibitor) TTD Canertinib dihydrochloride AKT1 Text_Mining(Drug(s)) TTD Canertinib dihydrochloride AKT2 Text_Mining(Drug(s)) TTD Canertinib dihydrochloride AKT3 Text_Mining(Drug(s)) TTD Canertinib dihydrochloride ERBB2 Text_Mining(Multitarget) TTD Canertinib dihydrochloride ERBB2 Text_Mining(Inhibitor) TTD Canertinib dihydrochloride ERBB2 Text_Mining(Drug(s)) TTD Canertinib dihydrochloride EGFR Text_Mining(Multitarget) TTD Canertinib dihydrochloride EGFR Text_Mining(Inhibitor) TTD Canertinib dihydrochloride EGFR Text_Mining(Drug(s)) TTD Canertinib dihydrochloride AR Ratio Potency (uM)=3.01065(uM) D4 PubChem Canertinib dihydrochloride BMX Activity=None(Unspecified) D4 ChEMBL Canertinib dihydrochloride EGFR Inhibition=None(Unspecified) D4 ChEMBL Canertinib dihydrochloride EGFR None=0.13(uM) D4 PubChem Canertinib dihydrochloride EGFR None=0.17(uM) D4 PubChem Canertinib dihydrochloride EGFR None=0.19(uM) D4 PubChem Canertinib dihydrochloride EGFR None=0.22(uM) D4 PubChem Canertinib dihydrochloride EGFR None=0.24(uM) D4 PubChem Canertinib dihydrochloride EGFR None=0.26(uM) D4 PubChem Canertinib dihydrochloride ESR1 Potency-Replicate_1=23.9145(uM) D4 PubChem Canertinib dihydrochloride ESR1 Ratio Potency (uM)=25.3067(uM) D4 PubChem Canertinib dihydrochloride ESR1 Potency-Replicate_1=29.8493(uM) D4 PubChem Canertinib dihydrochloride HSPB1 Ratio Potency (uM)=17.7787(uM) D4 PubChem Canertinib dihydrochloride MTOR Potency=11.5305(uM) D4 PubChem Canertinib dihydrochloride NFE2L2 Ratio Potency (uM)=2.66011(uM) D4 PubChem Canertinib dihydrochloride NR1H4 None=None(uM) D4 PubChem Canertinib dihydrochloride NR3C1 Potency-Replicate_1=3.0107(uM) D4 PubChem Canertinib dihydrochloride TDP1 Potency=4.7318(uM) D4 PubChem Canertinib dihydrochloride TDP1 Potency=5.3091(uM) D4 PubChem Canertinib dihydrochloride YES1 Potency=0.1729(uM) D4 PubChem