Drug Gene Type Source bisindolylmaleimide i CHEK1 Text_Mining(Inhibitor) TTD bisindolylmaleimide i PRKCG Text_Mining(Inhibitor) TTD bisindolylmaleimide i MAPK12 Text_Mining(Inhibitor) TTD bisindolylmaleimide i MAPK8 Text_Mining(Inhibitor) TTD bisindolylmaleimide i AKT1 Text_Mining(Inhibitor) TTD bisindolylmaleimide i AKT2 Text_Mining(Inhibitor) TTD bisindolylmaleimide i AKT3 Text_Mining(Inhibitor) TTD bisindolylmaleimide i GSK3B Text_Mining(Inhibitor) TTD bisindolylmaleimide i CDK1 Text_Mining(Inhibitor) TTD bisindolylmaleimide i MAPK14 Text_Mining(Inhibitor) TTD bisindolylmaleimide i ROCK1 Text_Mining(Inhibitor) TTD bisindolylmaleimide i CCNB1 Text_Mining(Inhibitor) TTD bisindolylmaleimide i PDPK1 Text_Mining(Inhibitor) TTD bisindolylmaleimide i MAPK11 Text_Mining(Inhibitor) TTD bisindolylmaleimide i MAPK1 Text_Mining(Inhibitor) TTD bisindolylmaleimide i PRKCZ Text_Mining(Inhibitor) TTD bisindolylmaleimide i SGK1 Text_Mining(Inhibitor) TTD bisindolylmaleimide i PRKCE Text_Mining(Inhibitor) TTD bisindolylmaleimide i PRKCD Text_Mining(Inhibitor) TTD bisindolylmaleimide i LCK Text_Mining(Inhibitor) TTD bisindolylmaleimide i CYP1A2 None=None(uM) D4 PubChem bisindolylmaleimide i CYP1A2 AC50=7943.28(nM) D4 ChEMBL bisindolylmaleimide i CYP3A4 Potency=12.5893(uM) D4 PubChem bisindolylmaleimide i CYP3A4 None=None(uM) D4 PubChem bisindolylmaleimide i CYP3A4 AC50=12589.2(nM) D4 ChEMBL bisindolylmaleimide i CYP3A4 Potency=12589.3(nM) D4 ChEMBL bisindolylmaleimide i EHMT2 Potency=14.1254(uM) D4 PubChem bisindolylmaleimide i EHMT2 Potency=17.7828(uM) D4 PubChem bisindolylmaleimide i EHMT2 Potency=17782.8(nM) D4 ChEMBL bisindolylmaleimide i EHMT2 Potency=14125.4(nM) D4 ChEMBL bisindolylmaleimide i MAPK1 Potency=0.7943(uM) D4 PubChem bisindolylmaleimide i MAPK1 Potency=1.2589(uM) D4 PubChem bisindolylmaleimide i MAPK1 Potency=794.3(nM) D4 ChEMBL bisindolylmaleimide i MAPK1 Potency=1258.9(nM) D4 ChEMBL bisindolylmaleimide i MAPT Potency=12.5893(uM) D4 PubChem bisindolylmaleimide i MAPT None=None(uM) D4 PubChem bisindolylmaleimide i MAPT Potency=28183.8(nM) D4 ChEMBL bisindolylmaleimide i MAPT Potency=12589.3(nM) D4 ChEMBL bisindolylmaleimide i MAPT Potency=19952.6(nM) D4 ChEMBL bisindolylmaleimide i RECQL Potency=28183.8(nM) D4 ChEMBL bisindolylmaleimide i TDP1 Potency=23.715(uM) D4 PubChem bisindolylmaleimide i USP1 Potency=50.1187(uM) D4 PubChem