Drug Gene Type Source zaprinast PDE1A Text_Mining(Inhibitor) TTD zaprinast PDE1B Text_Mining(Inhibitor) TTD zaprinast PDE1C Text_Mining(Inhibitor) TTD zaprinast PDE5A Text_Mining(Inhibitor) TTD zaprinast PDE4D Text_Mining(Inhibitor) TTD zaprinast ALDH1A1 Potency=19.9526(uM) D4 PubChem zaprinast ALDH1A1 Potency=22.3872(uM) D4 PubChem zaprinast ALDH1A1 Potency=19952.6(nM) D4 ChEMBL zaprinast ALDH1A1 Potency=22387.2(nM) D4 ChEMBL zaprinast ALOX15 Potency=15.8489(uM) D4 PubChem zaprinast ALOX15 Potency=15848.9(nM) D4 ChEMBL zaprinast CYP1A2 None=None(uM) D4 PubChem zaprinast CYP1A2 AC50=3981.07(nM) D4 ChEMBL zaprinast CYP1A2 AC50=5011.87(nM) D4 ChEMBL zaprinast EHMT2 Potency=14.1254(uM) D4 PubChem zaprinast EHMT2 Potency=14125.4(nM) D4 ChEMBL zaprinast GPR35 Activity=None(Unspecified) D4 ChEMBL zaprinast HIF1A Potency=5.0119(uM) D4 PubChem zaprinast HIF1A Potency=5011.9(nM) D4 ChEMBL zaprinast HPGD Potency=6.3096(uM) D4 PubChem zaprinast HPGD Potency=8.9125(uM) D4 PubChem zaprinast HPGD Potency=15.8489(uM) D4 PubChem zaprinast HPGD Potency=15848.9(nM) D4 ChEMBL zaprinast HPGD Potency=8912.5(nM) D4 ChEMBL zaprinast HPGD Potency=6309.6(nM) D4 ChEMBL zaprinast USP2 Potency=1.5849(uM) D4 PubChem zaprinast USP2 Potency=10.0(uM) D4 PubChem zaprinast USP2 Potency=10000.0(nM) D4 ChEMBL zaprinast USP2 Potency=1584.9(nM) D4 ChEMBL