Drug Gene Type Source 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide RELA Text_Mining(Inhibitor) TTD 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide APLNR None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide APOBEC3G Potency=7.0795(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide APOBEC3G Average IC50=100.0(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide APP None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ARNT None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide BAZ2B Potency=6.3096(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide BAZ2B Potency=6309.6(nM) D4 ChEMBL 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide CCR6 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide CFTR None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide CHRM4 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide CHRM5 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide CXCR6 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide CYP2C9 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide DRD3 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide GSTO1 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide HSP90AA1 AC50_uM=0.195(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide HTR1A None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide IDH1 Potency=0.5623(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide IL1B None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide ITGA4 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide KCNQ1 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide KDM4A Potency=5623.4(nM) D4 ChEMBL 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide L3MBTL1 Potency=2.9935(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide L3MBTL1 Potency=11.2202(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide L3MBTL1 Potency=11220.2(nM) D4 ChEMBL 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide MDM2 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide MDM4 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide MITF None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide MMP14 EC50=24.6(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide MPI IC50=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NAE1 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NFE2L2 Potency=7.0795(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NFKBIA None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NLRP3 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NOD1 EC50=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NOD2 EC50=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NOD2 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NPSR1 Potency=3.1623(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NPSR1 Potency=4.4668(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NPSR1 Potency=4466.8(nM) D4 ChEMBL 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NPSR1 Potency=3162.3(nM) D4 ChEMBL 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NR2E3 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide NR5A1 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide OPRK1 IC50=1.3(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide OPRK1 IC50=1300.0(nM) D4 ChEMBL 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide PLA2G7 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide RBBP8 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide RELA None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide RIPK2 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide S1PR1 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide S1PR4 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide SIX1 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide SLC12A5 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide SMAD3 Potency=1.2589(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide TACC3 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide TDP1 Potency=1.1582(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide TDP1 Potency=1.4581(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide TLR9 None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide TNF None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide UBE2M None=None(uM) D4 PubChem 5H-quinolino[8,7-c][1,2]benzothiazine 6,6-dioxide VCP None=None(uM) D4 PubChem