Drug Gene Type Source U-0126 CHEK1 Text_Mining(Inhibitor) TTD U-0126 MAPK12 Text_Mining(Inhibitor) TTD U-0126 MAPK8 Text_Mining(Inhibitor) TTD U-0126 AKT1 Text_Mining(Inhibitor) TTD U-0126 AKT2 Text_Mining(Inhibitor) TTD U-0126 AKT3 Text_Mining(Inhibitor) TTD U-0126 RPS6KB1 Text_Mining(Inhibitor) TTD U-0126 GSK3B Text_Mining(Inhibitor) TTD U-0126 PRKCA Text_Mining(Inhibitor) TTD U-0126 MAPK14 Text_Mining(Inhibitor) TTD U-0126 ROCK1 Text_Mining(Inhibitor) TTD U-0126 RAF1 Text_Mining(Inhibitor) TTD U-0126 MAP2K7 Text_Mining(Inhibitor) TTD U-0126 MAP2K1 Text_Mining(Inhibitor) TTD U-0126 MAPK11 Text_Mining(Inhibitor) TTD U-0126 MAPK1 Text_Mining(Inhibitor) TTD U-0126 SGK1 Text_Mining(Inhibitor) TTD U-0126 MAP2K2 Text_Mining(Inhibitor) TTD U-0126 LCK Text_Mining(Inhibitor) TTD U-0126 ALOX15 Potency=12589.3(nM) D4 ChEMBL U-0126 ALOX15 Potency=12.5893(uM) D4 PubChem U-0126 CYP1A2 AC50=12589.2(nM) D4 ChEMBL U-0126 CYP1A2 AC50=31622.8(nM) D4 ChEMBL U-0126 CYP1A2 None=None(uM) D4 PubChem U-0126 CYP2D6 AC50=19.95(nM) D4 ChEMBL U-0126 CYP2D6 Potency=20.0(nM) D4 ChEMBL U-0126 CYP2D6 Potency=0.02(uM) D4 PubChem U-0126 CYP2D6 None=None(uM) D4 PubChem U-0126 CYP3A4 AC50=3162.28(nM) D4 ChEMBL U-0126 CYP3A4 AC50=316.23(nM) D4 ChEMBL U-0126 CYP3A4 Potency=316.2(nM) D4 ChEMBL U-0126 CYP3A4 Potency=3162.3(nM) D4 ChEMBL U-0126 CYP3A4 Potency=0.3162(uM) D4 PubChem U-0126 CYP3A4 Potency=3.1623(uM) D4 PubChem U-0126 CYP3A4 None=None(uM) D4 PubChem U-0126 EGFR EGFR IC50=100.0(uM) D4 PubChem U-0126 EHMT2 Potency=8.9125(uM) D4 PubChem U-0126 EHMT2 Potency=12.5893(uM) D4 PubChem U-0126 EHMT2 Potency=12589.3(nM) D4 ChEMBL U-0126 EHMT2 Potency=8912.5(nM) D4 ChEMBL U-0126 HPGD Potency=28183.8(nM) D4 ChEMBL U-0126 HPGD Potency=28.1838(uM) D4 PubChem U-0126 HSD17B10 Potency=31622.8(nM) D4 ChEMBL U-0126 HSD17B10 Potency=25118.9(nM) D4 ChEMBL U-0126 MAPK1 Potency=199.5(nM) D4 ChEMBL U-0126 MAPK1 Potency=891.3(nM) D4 ChEMBL U-0126 MAPK1 Potency=501.2(nM) D4 ChEMBL U-0126 MAPK1 Potency=0.1995(uM) D4 PubChem U-0126 MAPK1 Potency=0.5012(uM) D4 PubChem U-0126 MAPK1 Potency=0.8913(uM) D4 PubChem U-0126 MAPT Potency=14.1254(uM) D4 PubChem U-0126 MAPT Potency=25.1189(uM) D4 PubChem U-0126 MAPT Potency=35481.3(nM) D4 ChEMBL U-0126 MAPT Potency=25118.9(nM) D4 ChEMBL U-0126 MAPT Potency=17782.8(nM) D4 ChEMBL U-0126 MAPT Potency=14125.4(nM) D4 ChEMBL U-0126 MAPT Potency=35.4813(uM) D4 PubChem U-0126 STK33 None=None(uM) D4 PubChem U-0126 TDP1 Potency=4.042(uM) D4 PubChem U-0126 TDP1 Potency=4.6109(uM) D4 PubChem U-0126 TDP1 Potency=6.4062(uM) D4 PubChem U-0126 TDP1 Potency=6.5131(uM) D4 PubChem U-0126 TDP1 Potency=26.6086(uM) D4 PubChem U-0126 VDR Potency=39.8107(uM) D4 PubChem U-0126 VDR Potency=8.9125(uM) D4 PubChem