Drug Gene Type Source Tyrphostin AG 538 EGFR Text_Mining(Inhibitor) TTD Tyrphostin AG 538 ADRBK1 None=None(uM) D4 PubChem Tyrphostin AG 538 ALOX15 Potency=3.9811(uM) D4 PubChem Tyrphostin AG 538 ALOX15 Potency=3981.1(nM) D4 ChEMBL Tyrphostin AG 538 ALPI IC50_Mean=2.68(uM) D4 PubChem Tyrphostin AG 538 ALPI IC50_Mean=4.41(uM) D4 PubChem Tyrphostin AG 538 ALPI EC50_Mean=6.36(uM) D4 PubChem Tyrphostin AG 538 ALPI None=None(uM) D4 PubChem Tyrphostin AG 538 ALPI IC50=2680.0(nM) D4 ChEMBL Tyrphostin AG 538 ALPI IC50=4410.0(nM) D4 ChEMBL Tyrphostin AG 538 ALPI EC50=6360.0(nM) D4 ChEMBL Tyrphostin AG 538 ALPL IC50_Mean=9.49(uM) D4 PubChem Tyrphostin AG 538 ALPL IC50=9490.0(nM) D4 ChEMBL Tyrphostin AG 538 ALPPL2 IC50_Mean=5.59(uM) D4 PubChem Tyrphostin AG 538 ALPPL2 EC50_Mean=8.03(uM) D4 PubChem Tyrphostin AG 538 ALPPL2 IC50=5590.0(nM) D4 ChEMBL Tyrphostin AG 538 ALPPL2 EC50=8030.0(nM) D4 ChEMBL Tyrphostin AG 538 APEX1 Potency=281.8(nM) D4 ChEMBL Tyrphostin AG 538 APEX1 Potency=199.5(nM) D4 ChEMBL Tyrphostin AG 538 APLNR None=None(uM) D4 PubChem Tyrphostin AG 538 BAZ2B Potency=2.2387(uM) D4 PubChem Tyrphostin AG 538 BAZ2B Potency=2238.7(nM) D4 ChEMBL Tyrphostin AG 538 BLM Potency=8.9125(uM) D4 PubChem Tyrphostin AG 538 BLM Potency=8912.5(nM) D4 ChEMBL Tyrphostin AG 538 CASP6 None=None(uM) D4 PubChem Tyrphostin AG 538 CBX1 Potency=0.5012(uM) D4 PubChem Tyrphostin AG 538 CBX1 Potency=501.2(nM) D4 ChEMBL Tyrphostin AG 538 CCR6 None=None(uM) D4 PubChem Tyrphostin AG 538 CYP1A2 None=None(uM) D4 PubChem Tyrphostin AG 538 CYP3A4 Potency=15.8489(uM) D4 PubChem Tyrphostin AG 538 CYP3A4 None=None(uM) D4 PubChem Tyrphostin AG 538 CYP3A4 AC50=15848.9(nM) D4 ChEMBL Tyrphostin AG 538 CYP3A4 Potency=15848.9(nM) D4 ChEMBL Tyrphostin AG 538 EHMT2 Potency=2.2387(uM) D4 PubChem Tyrphostin AG 538 EHMT2 Potency=5.0119(uM) D4 PubChem Tyrphostin AG 538 EHMT2 Potency=15.8489(uM) D4 PubChem Tyrphostin AG 538 EHMT2 Potency=5011.9(nM) D4 ChEMBL Tyrphostin AG 538 EHMT2 Potency=15848.9(nM) D4 ChEMBL Tyrphostin AG 538 EHMT2 Potency=2238.7(nM) D4 ChEMBL Tyrphostin AG 538 ESR1 None=None(uM) D4 PubChem Tyrphostin AG 538 EZH2 None=None(uM) D4 PubChem Tyrphostin AG 538 FEN1 Potency=0.7519(uM) D4 PubChem Tyrphostin AG 538 FEN1 Potency=1.4125(uM) D4 PubChem Tyrphostin AG 538 FEN1 Potency=751.9(nM) D4 ChEMBL Tyrphostin AG 538 GFER None=None(uM) D4 PubChem Tyrphostin AG 538 HIF1A Potency=7.9433(uM) D4 PubChem Tyrphostin AG 538 HIF1A Potency=7943.3(nM) D4 ChEMBL Tyrphostin AG 538 HPGD Potency=7.9433(uM) D4 PubChem Tyrphostin AG 538 HPGD Potency=7943.3(nM) D4 ChEMBL Tyrphostin AG 538 HSD17B10 Potency=1584.9(nM) D4 ChEMBL Tyrphostin AG 538 HSP90AA1 None=None(uM) D4 PubChem Tyrphostin AG 538 KDM4A Potency=707.9(nM) D4 ChEMBL Tyrphostin AG 538 KDM4E Potency=2511.9(nM) D4 ChEMBL Tyrphostin AG 538 L3MBTL1 Potency=0.0752(uM) D4 PubChem Tyrphostin AG 538 L3MBTL1 Potency=0.5012(uM) D4 PubChem Tyrphostin AG 538 L3MBTL1 Potency=501.2(nM) D4 ChEMBL Tyrphostin AG 538 MBD2 None=None(uM) D4 PubChem Tyrphostin AG 538 MPHOSPH8 Potency=1.4125(uM) D4 PubChem Tyrphostin AG 538 MPHOSPH8 Potency=2.9935(uM) D4 PubChem Tyrphostin AG 538 MPHOSPH8 Potency=2993.5(nM) D4 ChEMBL Tyrphostin AG 538 MPHOSPH8 Potency=1412.5(nM) D4 ChEMBL Tyrphostin AG 538 PAFAH1B2 None=None(uM) D4 PubChem Tyrphostin AG 538 PAFAH1B3 None=None(uM) D4 PubChem Tyrphostin AG 538 PAFAH2 None=None(uM) D4 PubChem Tyrphostin AG 538 PIN1 Potency=1.6944(uM) D4 PubChem Tyrphostin AG 538 PIN1 Potency=1694.4(nM) D4 ChEMBL Tyrphostin AG 538 PLA2G7 None=None(uM) D4 PubChem Tyrphostin AG 538 POLB Potency=0.0631(uM) D4 PubChem Tyrphostin AG 538 POLB Potency=63.1(nM) D4 ChEMBL Tyrphostin AG 538 POLH Potency=0.1259(uM) D4 PubChem Tyrphostin AG 538 POLH Potency=0.6746(uM) D4 PubChem Tyrphostin AG 538 POLI Potency=0.1122(uM) D4 PubChem Tyrphostin AG 538 POLI Potency=0.7519(uM) D4 PubChem Tyrphostin AG 538 POLI Potency=1.122(uM) D4 PubChem Tyrphostin AG 538 POLK Potency=0.3359(uM) D4 PubChem Tyrphostin AG 538 POLK Potency=0.3769(uM) D4 PubChem Tyrphostin AG 538 POLK Potency=0.7943(uM) D4 PubChem Tyrphostin AG 538 PRMT1 None=None(uM) D4 PubChem Tyrphostin AG 538 PSIP1 IC50=0.07955(uM) D4 PubChem Tyrphostin AG 538 PSIP1 IC50=8.046(uM) D4 PubChem Tyrphostin AG 538 PSIP1 None=None(uM) D4 PubChem Tyrphostin AG 538 RECQL Potency=281.8(nM) D4 ChEMBL Tyrphostin AG 538 RECQL Potency=1584.9(nM) D4 ChEMBL Tyrphostin AG 538 RGS4 Potency=26.6795(uM) D4 PubChem Tyrphostin AG 538 SENP6 None=None(uM) D4 PubChem Tyrphostin AG 538 SENP8 None=None(uM) D4 PubChem Tyrphostin AG 538 STK33 EC50_uM=44.89(uM) D4 PubChem Tyrphostin AG 538 STK33 None=None(uM) D4 PubChem Tyrphostin AG 538 TRA None=None(uM) D4 PubChem Tyrphostin AG 538 UHRF1 None=None(uM) D4 PubChem Tyrphostin AG 538 USP2 Potency=1.1668(uM) D4 PubChem Tyrphostin AG 538 USP2 Potency=1166.8(nM) D4 ChEMBL Tyrphostin AG 538 VDR Potency=50.1187(uM) D4 PubChem Tyrphostin AG 538 WRN Potency=0.1683(uM) D4 PubChem