Drug Gene Type Source triamterene SCNN1A Text_Mining(Drug(s)) TTD triamterene SCNN1A Text_Mining(Blocker) TTD triamterene AHR AhR Potency (uM)=11.5149(uM) D4 PubChem triamterene AHR AhR Potency (uM)=29.8145(uM) D4 PubChem triamterene AR Potency-Replicate_1=21.3138(uM) D4 PubChem triamterene AR Potency=44.6684(uM) D4 PubChem triamterene AR Potency-Replicate_1=48.9722(uM) D4 PubChem triamterene AR Potency-Replicate_1=49.5119(uM) D4 PubChem triamterene CBFB IC50=None(uM) D4 PubChem triamterene CYP1A2 None=None(uM) D4 PubChem triamterene CYP1A2 AC50=5011.87(nM) D4 ChEMBL triamterene ESR1 Potency=35.4813(uM) D4 PubChem triamterene ESR1 Potency-Replicate_1=68.5896(uM) D4 PubChem triamterene GAA Potency=39.8107(uM) D4 PubChem triamterene GAA Potency=39810.7(nM) D4 ChEMBL triamterene HIF1A Potency=10.0(uM) D4 PubChem triamterene HIF1A Potency=10000.0(nM) D4 ChEMBL triamterene HSD17B10 Potency=3162.3(nM) D4 ChEMBL triamterene HSD17B10 Potency=5011.9(nM) D4 ChEMBL triamterene HSD17B10 Potency=1258.9(nM) D4 ChEMBL triamterene HSD17B10 Potency=7943.3(nM) D4 ChEMBL triamterene HSPB1 Potency-Replicate_1=24.5442(uM) D4 PubChem triamterene HSPB1 Potency-Replicate_1=29.847(uM) D4 PubChem triamterene HSPB1 Potency-Replicate_1=49.5119(uM) D4 PubChem triamterene IDH1 Potency=2.3109(uM) D4 PubChem triamterene JAK2 IC50=4.613(uM) D4 PubChem triamterene JAK2 None=None(uM) D4 PubChem triamterene JAK2 IC50=4613.0(nM) D4 ChEMBL triamterene KLK7 None=None(uM) D4 PubChem triamterene NFE2L2 Potency-Replicate_1=23.7083(uM) D4 PubChem triamterene NFE2L2 Potency-Replicate_1=30.6379(uM) D4 PubChem triamterene NFE2L2 Potency-Replicate_1=30.9809(uM) D4 PubChem triamterene NFE2L2 Potency=33.4915(uM) D4 PubChem triamterene NFE2L2 Potency=54.4827(uM) D4 PubChem triamterene NR1H4 Potency-Replicate_1=21.13(uM) D4 PubChem triamterene NR1H4 Potency-Replicate_1=49.5119(uM) D4 PubChem triamterene NR3C1 Potency-Replicate_1=48.9722(uM) D4 PubChem triamterene PPARD Potency-Replicate_1=23.7083(uM) D4 PubChem triamterene PPARD Potency-Replicate_1=24.5442(uM) D4 PubChem triamterene PPARG Potency-Replicate_1=23.9145(uM) D4 PubChem triamterene RUNX1 IC50=None(uM) D4 PubChem triamterene TDP1 Potency=2.0596(uM) D4 PubChem triamterene TDP1 Potency=6.6838(uM) D4 PubChem triamterene TDP1 Potency=8.1995(uM) D4 PubChem triamterene TDP1 Potency=14.9631(uM) D4 PubChem triamterene TDP1 Potency=15.8489(uM) D4 PubChem triamterene TDP1 Potency=17.7828(uM) D4 PubChem triamterene TDP1 Potency=18.3564(uM) D4 PubChem triamterene THRB Potency=22.3872(uM) D4 PubChem triamterene TNFRSF10B None=None(uM) D4 PubChem triamterene TP53 Potency=12.5893(uM) D4 PubChem triamterene TP53 Potency=12589.3(nM) D4 ChEMBL