Drug Gene Type Source Tozasertib AURKA Text_Mining(Multitarget) TTD Tozasertib AURKA Text_Mining(Inhibitor) TTD Tozasertib AURKA Text_Mining(Drug(s)) TTD Tozasertib AURKB Text_Mining(Multitarget) TTD Tozasertib AURKB Text_Mining(Inhibitor) TTD Tozasertib AURKB Text_Mining(Drug(s)) TTD Tozasertib LCK Text_Mining(Multitarget) TTD Tozasertib LCK Text_Mining(Inhibitor) TTD Tozasertib LCK Text_Mining(Drug(s)) TTD Tozasertib ABL1 None=6.3(uM) D4 PubChem Tozasertib ABL1 None=9.1(uM) D4 PubChem Tozasertib ABL1 None=9.4(uM) D4 PubChem Tozasertib ABL2 None=4.0(uM) D4 PubChem Tozasertib ABL2 Activity=None(Unspecified) D4 ChEMBL Tozasertib AURKA None=4.1(uM) D4 PubChem Tozasertib AURKA Activity=None(Unspecified) D4 ChEMBL Tozasertib AURKB None=7.4(uM) D4 PubChem Tozasertib AURKB Activity=None(Unspecified) D4 ChEMBL Tozasertib CSNK2A1 Activity=None(Unspecified) D4 ChEMBL Tozasertib EPAS1 None=None(uM) D4 PubChem Tozasertib FLT3 None=4.3(uM) D4 PubChem Tozasertib FLT3 None=6.5(uM) D4 PubChem Tozasertib GMNN Potency=0.2593(uM) D4 PubChem Tozasertib KCNH2 None=None(uM) D4 PubChem Tozasertib KCNQ1 None=None(uM) D4 PubChem Tozasertib MAP4K2 None=None(uM) D4 PubChem Tozasertib MAP4K5 Activity=None(Unspecified) D4 ChEMBL Tozasertib MDM2 None=None(uM) D4 PubChem Tozasertib MDM4 None=None(uM) D4 PubChem Tozasertib MRGPRX1 None=None(uM) D4 PubChem Tozasertib MYLK Activity=None(Unspecified) D4 ChEMBL Tozasertib PLK4 Activity=None(Unspecified) D4 ChEMBL Tozasertib RET Activity=None(Unspecified) D4 ChEMBL Tozasertib STK11 Activity=None(Unspecified) D4 ChEMBL Tozasertib TNK1 Activity=None(Unspecified) D4 ChEMBL Tozasertib YES1 Potency=0.0972(uM) D4 PubChem Tozasertib YES1 Potency=0.4873(uM) D4 PubChem