Drug Gene Type Source staurosporine CDK2 Text_Mining(Inhibitor) TTD staurosporine PIK3CG Text_Mining(Inhibitor) TTD staurosporine SYK Text_Mining(Inhibitor) TTD staurosporine GSK3B Text_Mining(Inhibitor) TTD staurosporine PRKCQ Text_Mining(Inhibitor) TTD staurosporine PDPK1 Text_Mining(Inhibitor) TTD staurosporine ITK Text_Mining(Inhibitor) TTD staurosporine IKBKB Text_Mining(Inhibitor) TTD staurosporine LCK Text_Mining(Inhibitor) TTD staurosporine AAK1 None=1.2(uM) D4 PubChem staurosporine APAF1 None=None(uM) D4 PubChem staurosporine APP None=None(uM) D4 PubChem staurosporine ATAD5 Potency=0.5174(uM) D4 PubChem staurosporine AXL None=6.8(uM) D4 PubChem staurosporine BMP2K None=5.6(uM) D4 PubChem staurosporine BRSK2 None=3.5(uM) D4 PubChem staurosporine CAMK1D None=1.1(uM) D4 PubChem staurosporine CAMK2A None=0.16(uM) D4 PubChem staurosporine CAMK2B None=1.3(uM) D4 PubChem staurosporine CAMK2G None=0.55(uM) D4 PubChem staurosporine CAMKK1 None=0.039(uM) D4 PubChem staurosporine CAMKK2 None=0.16(uM) D4 PubChem staurosporine CASP1 None=None(uM) D4 PubChem staurosporine CASP3 Activity=None(Unspecified) D4 ChEMBL staurosporine CDK2 None=7.0(uM) D4 PubChem staurosporine CHEK1 None=3.2(uM) D4 PubChem staurosporine CLK2 None=8.2(uM) D4 PubChem staurosporine CLK3 None=None(uM) D4 PubChem staurosporine CLK4 None=9.6(uM) D4 PubChem staurosporine CSNK2A2 None=6.5(uM) D4 PubChem staurosporine DAPK1 None=1.4(uM) D4 PubChem staurosporine DAPK2 None=1.6(uM) D4 PubChem staurosporine DAPK3 None=1.0(uM) D4 PubChem staurosporine DIRAS1 None=None(uM) D4 PubChem staurosporine DMPK None=3.5(uM) D4 PubChem staurosporine EGFR Potency=0.0056(uM) D4 PubChem staurosporine EGFR Potency=0.0398(uM) D4 PubChem staurosporine EGFR Potency=0.3548(uM) D4 PubChem staurosporine EGFR Potency=0.3981(uM) D4 PubChem staurosporine EGFR EGFR IC50=0.4467(uM) D4 PubChem staurosporine EGFR Potency=39.8(nM) D4 ChEMBL staurosporine EGFR Potency=5.6(nM) D4 ChEMBL staurosporine EGFR Potency=354.8(nM) D4 ChEMBL staurosporine EGFR Potency=398.1(nM) D4 ChEMBL staurosporine FLT3 None=2.1(uM) D4 PubChem staurosporine FLT3 None=2.4(uM) D4 PubChem staurosporine FLT3 None=2.5(uM) D4 PubChem staurosporine FLT3 None=2.9(uM) D4 PubChem staurosporine GPR55 IC50=3.18033(uM) D4 PubChem staurosporine IKBKE None=5.1(uM) D4 PubChem staurosporine JAK2 irf1 Inhibition [HEL cells] (IC50)=0.0044(uM) D4 PubChem staurosporine JAK2 irf1 Inhibition [Ba/F3 cells] (IC50)=0.028(uM) D4 PubChem staurosporine JAK2 JAK2V617F Inhibition (IC50)=8.9(uM) D4 PubChem staurosporine JAK2 None=None(uM) D4 PubChem staurosporine JAK3 None=10.0(uM) D4 PubChem staurosporine KCNJ1 None=None(uM) D4 PubChem staurosporine KCNQ1 None=None(uM) D4 PubChem staurosporine KIT None=0.64(uM) D4 PubChem staurosporine KIT None=9.5(uM) D4 PubChem staurosporine KLF5 None=None(uM) D4 PubChem staurosporine MAP2K1 Potency=0.1(uM) D4 PubChem staurosporine MAP2K1 Potency=100.0(nM) D4 ChEMBL staurosporine MAP2K3 None=5.0(uM) D4 PubChem staurosporine MAP2K6 None=3.4(uM) D4 PubChem staurosporine MAP3K5 None=None(uM) D4 PubChem staurosporine MAP3K9 None=10.0(uM) D4 PubChem staurosporine MAP4K1 None=4.3(uM) D4 PubChem staurosporine MAP4K2 None=None(uM) D4 PubChem staurosporine MAP4K3 None=8.2(uM) D4 PubChem staurosporine MARK1 None=4.0(uM) D4 PubChem staurosporine MARK2 None=0.7(uM) D4 PubChem staurosporine MARK3 None=3.0(uM) D4 PubChem staurosporine MARK4 None=5.4(uM) D4 PubChem staurosporine MCL1 None=None(uM) D4 PubChem staurosporine MDM2 None=None(uM) D4 PubChem staurosporine MDM4 None=None(uM) D4 PubChem staurosporine MITF None=None(uM) D4 PubChem staurosporine MRGPRX1 None=None(uM) D4 PubChem staurosporine NFKB1 None=None(uM) D4 PubChem staurosporine NLRP1 None=None(uM) D4 PubChem staurosporine NLRP3 None=None(uM) D4 PubChem staurosporine NPBWR1 None=None(uM) D4 PubChem staurosporine NPSR1 Potency=6.3096(uM) D4 PubChem staurosporine NPY1R None=None(uM) D4 PubChem staurosporine NPY2R None=None(uM) D4 PubChem staurosporine NTRK1 None=4.0(uM) D4 PubChem staurosporine NTRK2 None=3.8(uM) D4 PubChem staurosporine NUAK1 None=4.4(uM) D4 PubChem staurosporine NUAK2 None=0.086(uM) D4 PubChem staurosporine PAK1 None=0.57(uM) D4 PubChem staurosporine PAK2 None=3.1(uM) D4 PubChem staurosporine PAK3 None=7.1(uM) D4 PubChem staurosporine PAK4 None=6.3(uM) D4 PubChem staurosporine PAK4 None=None(uM) D4 PubChem staurosporine PAK6 None=0.57(uM) D4 PubChem staurosporine PAK6 None=None(uM) D4 PubChem staurosporine PAK7 None=1.2(uM) D4 PubChem staurosporine PAK7 None=None(uM) D4 PubChem staurosporine PDGFRA None=10.0(uM) D4 PubChem staurosporine PDGFRB None=1.8(uM) D4 PubChem staurosporine PDPK1 None=1.7(uM) D4 PubChem staurosporine PHKG1 None=0.65(uM) D4 PubChem staurosporine PHKG2 None=0.14(uM) D4 PubChem staurosporine PIM1 None=3.2(uM) D4 PubChem staurosporine PIM1 None=None(uM) D4 PubChem staurosporine PIM2 None=1.9(uM) D4 PubChem staurosporine PIM2 None=None(uM) D4 PubChem staurosporine PIM3 None=0.51(uM) D4 PubChem staurosporine PKN1 None=1.3(uM) D4 PubChem staurosporine PKN2 None=2.5(uM) D4 PubChem staurosporine PLA2G7 None=None(uM) D4 PubChem staurosporine PPME1 None=None(uM) D4 PubChem staurosporine PREPL None=None(uM) D4 PubChem staurosporine PRKACA AC50_uM=0.126(uM) D4 PubChem staurosporine PRKCD None=1.5(uM) D4 PubChem staurosporine PRKCE None=0.25(uM) D4 PubChem staurosporine PRKCH None=4.8(uM) D4 PubChem staurosporine PRKCQ None=8.5(uM) D4 PubChem staurosporine PRKD1 DR_IC50uM_Run1=0.1(uM) D4 PubChem staurosporine PRKD1 None=None(uM) D4 PubChem staurosporine PTBP1 None=None(uM) D4 PubChem staurosporine PTK2B None=3.5(uM) D4 PubChem staurosporine RECQL Potency=35481.3(nM) D4 ChEMBL staurosporine RGS4 None=None(uM) D4 PubChem staurosporine RPS6KA2 None=8.9(uM) D4 PubChem staurosporine S1PR1 IC50=0.662(uM) D4 PubChem staurosporine S1PR1 None=None(uM) D4 PubChem staurosporine S1PR3 None=None(uM) D4 PubChem staurosporine S1PR4 IC50=0.183(uM) D4 PubChem staurosporine S1PR4 None=None(uM) D4 PubChem staurosporine SELE None=None(uM) D4 PubChem staurosporine SIK1 None=2.2(uM) D4 PubChem staurosporine SIK2 None=1.1(uM) D4 PubChem staurosporine SLC5A7 None=None(uM) D4 PubChem staurosporine SLK None=0.024(uM) D4 PubChem staurosporine SLK None=None(uM) D4 PubChem staurosporine SRPK1 None=5.5(uM) D4 PubChem staurosporine STAT1 None=None(uM) D4 PubChem staurosporine STAT3 None=None(uM) D4 PubChem staurosporine STK16 None=None(uM) D4 PubChem staurosporine STK3 None=0.18(uM) D4 PubChem staurosporine STK33 None=None(uM) D4 PubChem staurosporine STK33 None=1.8(uM) D4 PubChem staurosporine STK4 None=0.19(uM) D4 PubChem staurosporine TNFSF10 None=None(uM) D4 PubChem staurosporine TNIK None=4.7(uM) D4 PubChem staurosporine TNK1 None=2.5(uM) D4 PubChem staurosporine VCP None=None(uM) D4 PubChem staurosporine XBP1 Absolute IC50 (XBP1)=0.66(uM) D4 PubChem staurosporine YWHAB None=None(uM) D4 PubChem