Drug Gene Type Source pyrilamine HRH1 Text_Mining(Antagonist) TTD pyrilamine HRH1 Text_Mining(Antagonist) TTD pyrilamine HRH1 Text_Mining(Drug(s)) TTD pyrilamine ALOX5 Text_Mining(Inhibitor) TTD pyrilamine ALOX5 Text_Mining(Drug(s)) TTD pyrilamine AR AR Potency (uM)=70.8978(uM) D4 PubChem pyrilamine CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL pyrilamine CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL pyrilamine CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL pyrilamine CYP2D6 Potency=0.1(uM) D4 PubChem pyrilamine CYP2D6 Potency=0.1259(uM) D4 PubChem pyrilamine CYP2D6 Potency=0.5012(uM) D4 PubChem pyrilamine CYP2D6 None=None(uM) D4 PubChem pyrilamine CYP2D6 Potency=100.0(nM) D4 ChEMBL pyrilamine CYP2D6 AC50=100.0(nM) D4 ChEMBL pyrilamine CYP2D6 AC50=125.89(nM) D4 ChEMBL pyrilamine CYP2D6 Potency=501.2(nM) D4 ChEMBL pyrilamine CYP2D6 Potency=125.9(nM) D4 ChEMBL pyrilamine CYP2D6 AC50=501.19(nM) D4 ChEMBL pyrilamine CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL pyrilamine HRH1 Activity=None(Unspecified) D4 ChEMBL pyrilamine KCNH2 Potency=12.5893(uM) D4 PubChem