Drug Gene Type Source purvalanol A CDK2 Text_Mining(Inhibitor) TTD purvalanol A CDK1 Text_Mining(Inhibitor) TTD purvalanol A PCNA Text_Mining(Inhibitor) TTD purvalanol A CCNA2 Text_Mining(Inhibitor) TTD purvalanol A SRC Text_Mining(Inhibitor) TTD purvalanol A CLK3 None=None(uM) D4 PubChem purvalanol A CSNK1G2 None=None(uM) D4 PubChem purvalanol A CYP1A2 None=None(uM) D4 PubChem purvalanol A CYP1A2 AC50=316.23(nM) D4 ChEMBL purvalanol A CYP2C9 Potency=7.9433(uM) D4 PubChem purvalanol A CYP2C9 Potency=7943.3(nM) D4 ChEMBL purvalanol A CYP3A4 Potency=12.5893(uM) D4 PubChem purvalanol A CYP3A4 None=None(uM) D4 PubChem purvalanol A CYP3A4 AC50=12589.2(nM) D4 ChEMBL purvalanol A CYP3A4 Potency=12589.3(nM) D4 ChEMBL purvalanol A HIF1A Potency=10.0(uM) D4 PubChem purvalanol A HIF1A Potency=10000.0(nM) D4 ChEMBL purvalanol A HSD17B10 Potency=31622.8(nM) D4 ChEMBL purvalanol A JAK2 irf1 Inhibition [Ba/F3 cells] (IC50)=0.84(uM) D4 PubChem purvalanol A JAK2 JAK2V617F Inhibition (IC50)=0.91(uM) D4 PubChem purvalanol A JAK2 irf1 Inhibition [HEL cells] (IC50)=1.13(uM) D4 PubChem purvalanol A JAK2 None=None(uM) D4 PubChem purvalanol A JAK2 Activity=1.13(um) D4 ChEMBL purvalanol A JAK2 Activity=0.91(um) D4 ChEMBL purvalanol A JAK2 Activity=0.84(um) D4 ChEMBL purvalanol A PAK4 None=None(uM) D4 PubChem purvalanol A PAK6 None=None(uM) D4 PubChem purvalanol A PAK7 None=None(uM) D4 PubChem purvalanol A STAT6 Potency=5.0119(uM) D4 PubChem purvalanol A STAT6 Potency=5011.9(nM) D4 ChEMBL purvalanol A STK16 None=None(uM) D4 PubChem purvalanol A TDP1 Potency=9.4411(uM) D4 PubChem