Drug Gene Type Source pimozide DRD2 Text_Mining(Antagonist) TTD pimozide DRD2 Text_Mining(Drug(s)) TTD pimozide ABCB1 None=None(uM) D4 PubChem pimozide ADRB2 None=None(uM) D4 PubChem pimozide APAF1 None=None(uM) D4 PubChem pimozide AR Potency-Replicate_1=13.8006(uM) D4 PubChem pimozide AR AR Potency (uM)=23.4203(uM) D4 PubChem pimozide ATAD5 Potency=11.5774(uM) D4 PubChem pimozide ATAD5 Potency=11577.4(nM) D4 ChEMBL pimozide ATXN2 Potency=31.6228(uM) D4 PubChem pimozide CACNA1H None=None(uM) D4 PubChem pimozide CBX1 Potency=35.4813(uM) D4 PubChem pimozide CBX1 Potency=35481.3(nM) D4 ChEMBL pimozide CHRM1 None=None(uM) D4 PubChem pimozide CYP19A1 Potency-Replicate_1=30.6379(uM) D4 PubChem pimozide CYP1A2 None=None(uM) D4 PubChem pimozide CYP2C19 Potency=10.0(uM) D4 PubChem pimozide CYP2C19 Potency=10000.0(nM) D4 ChEMBL pimozide CYP2D6 Potency=3.1623(uM) D4 PubChem pimozide CYP2D6 Potency=10.0(uM) D4 PubChem pimozide CYP2D6 None=None(uM) D4 PubChem pimozide CYP2D6 AC50=3162.28(nM) D4 ChEMBL pimozide CYP2D6 Potency=3162.3(nM) D4 ChEMBL pimozide CYP2D6 Potency=10000.0(nM) D4 ChEMBL pimozide CYP3A4 Potency=3.1623(uM) D4 PubChem pimozide CYP3A4 Potency=5.0119(uM) D4 PubChem pimozide CYP3A4 Potency=3162.3(nM) D4 ChEMBL pimozide CYP3A4 Potency=5011.9(nM) D4 ChEMBL pimozide DRD2 None=None(uM) D4 PubChem pimozide DRD3 None=None(uM) D4 PubChem pimozide HIF1A Potency=2.5119(uM) D4 PubChem pimozide HIF1A Potency=5.0119(uM) D4 PubChem pimozide HIF1A Potency=5011.9(nM) D4 ChEMBL pimozide HIF1A Potency=2511.9(nM) D4 ChEMBL pimozide HTR1A None=None(uM) D4 PubChem pimozide HTR2A None=None(uM) D4 PubChem pimozide IDH1 Potency=16.3601(uM) D4 PubChem pimozide IL1B None=None(uM) D4 PubChem pimozide KCNH2 Potency=0.0562(uM) D4 PubChem pimozide KDM4A Potency=39810.7(nM) D4 ChEMBL pimozide MAP4K2 None=None(uM) D4 PubChem pimozide MAPK1 Potency=25.1189(uM) D4 PubChem pimozide MAPK1 Potency=25118.9(nM) D4 ChEMBL pimozide MDM2 None=None(uM) D4 PubChem pimozide MDM4 None=None(uM) D4 PubChem pimozide MMP14 EC50=None(uM) D4 PubChem pimozide MPHOSPH8 Potency=22.3872(uM) D4 PubChem pimozide MPHOSPH8 Potency=22387.2(nM) D4 ChEMBL pimozide MTOR Potency=16.4816(uM) D4 PubChem pimozide MTOR Potency=16481.6(nM) D4 ChEMBL pimozide NPSR1 Potency=6.3096(uM) D4 PubChem pimozide NPSR1 Potency=12.5893(uM) D4 PubChem pimozide NPSR1 Potency=12589.3(nM) D4 ChEMBL pimozide NPSR1 Potency=6309.6(nM) D4 ChEMBL pimozide NTSR1 None=None(uM) D4 PubChem pimozide PPARD Potency-Replicate_1=33.4889(uM) D4 PubChem pimozide PPARG Potency-Replicate_1=34.6654(uM) D4 PubChem pimozide RXRA Potency=17.7828(uM) D4 PubChem pimozide STK33 None=None(uM) D4 PubChem pimozide TDP1 Potency=6.6838(uM) D4 PubChem pimozide TDP1 Potency=14.581(uM) D4 PubChem pimozide TDP1 Potency=25.4789(uM) D4 PubChem pimozide TDP1 Potency=32.076(uM) D4 PubChem pimozide THPO Potency=10.0(uM) D4 PubChem pimozide THPO Potency=10000.0(nM) D4 ChEMBL pimozide TP53 Potency=15.8489(uM) D4 PubChem pimozide TP53 Potency=25.1189(uM) D4 PubChem pimozide TP53 Potency=15848.9(nM) D4 ChEMBL pimozide TP53 Potency=25118.9(nM) D4 ChEMBL pimozide XBP1 Absolute IC50 (XBP1)=10.0(uM) D4 PubChem pimozide XBP1 IC50=10000.0(nM) D4 ChEMBL