Drug Gene Type Source PD 98059 CHEK1 Text_Mining(Inhibitor) TTD PD 98059 MAPK12 Text_Mining(Inhibitor) TTD PD 98059 MAPK8 Text_Mining(Inhibitor) TTD PD 98059 AKT1 Text_Mining(Inhibitor) TTD PD 98059 AKT2 Text_Mining(Inhibitor) TTD PD 98059 AKT3 Text_Mining(Inhibitor) TTD PD 98059 RPS6KB1 Text_Mining(Inhibitor) TTD PD 98059 GSK3B Text_Mining(Inhibitor) TTD PD 98059 PRKCA Text_Mining(Inhibitor) TTD PD 98059 MAPK14 Text_Mining(Inhibitor) TTD PD 98059 ROCK1 Text_Mining(Inhibitor) TTD PD 98059 RAF1 Text_Mining(Inhibitor) TTD PD 98059 MAP3K1 Text_Mining(Inhibitor) TTD PD 98059 MAP2K1 Text_Mining(Inhibitor) TTD PD 98059 MAP3K2 Text_Mining(Inhibitor) TTD PD 98059 MAPK11 Text_Mining(Inhibitor) TTD PD 98059 MAPK1 Text_Mining(Inhibitor) TTD PD 98059 SGK1 Text_Mining(Inhibitor) TTD PD 98059 LCK Text_Mining(Inhibitor) TTD PD 98059 ATAD5 Potency=2.9081(uM) D4 PubChem PD 98059 ATAD5 Potency=2908.1(nM) D4 ChEMBL PD 98059 CYP1A2 None=None(uM) D4 PubChem PD 98059 CYP1A2 AC50=199.53(nM) D4 ChEMBL PD 98059 CYP2C19 Potency=6.3096(uM) D4 PubChem PD 98059 CYP2C19 None=None(uM) D4 PubChem PD 98059 CYP2C19 AC50=6309.57(nM) D4 ChEMBL PD 98059 CYP2C19 Potency=6309.6(nM) D4 ChEMBL PD 98059 CYP2C9 Potency=31.6228(uM) D4 PubChem PD 98059 CYP2C9 None=None(uM) D4 PubChem PD 98059 CYP2C9 AC50=31622.8(nM) D4 ChEMBL PD 98059 CYP2C9 Potency=31622.8(nM) D4 ChEMBL PD 98059 CYP2D6 Potency=7.9433(uM) D4 PubChem PD 98059 CYP2D6 None=None(uM) D4 PubChem PD 98059 CYP2D6 AC50=7943.28(nM) D4 ChEMBL PD 98059 CYP2D6 Potency=7943.3(nM) D4 ChEMBL PD 98059 CYP3A4 Potency=7.9433(uM) D4 PubChem PD 98059 CYP3A4 None=None(uM) D4 PubChem PD 98059 CYP3A4 AC50=7943.28(nM) D4 ChEMBL PD 98059 CYP3A4 Potency=7943.3(nM) D4 ChEMBL PD 98059 HPGD Potency=6.3096(uM) D4 PubChem PD 98059 HPGD Potency=12.5893(uM) D4 PubChem PD 98059 HPGD Potency=12589.3(nM) D4 ChEMBL PD 98059 HPGD Potency=6309.6(nM) D4 ChEMBL PD 98059 MAPK1 Potency=3.1623(uM) D4 PubChem PD 98059 MAPK1 Potency=3.9811(uM) D4 PubChem PD 98059 MAPK1 Potency=5.0119(uM) D4 PubChem PD 98059 MAPK1 Potency=3981.1(nM) D4 ChEMBL PD 98059 MAPK1 Inhibition=None(Unspecified) D4 ChEMBL PD 98059 MAPK1 Potency=3162.3(nM) D4 ChEMBL PD 98059 MAPK1 Potency=5011.9(nM) D4 ChEMBL PD 98059 MAPK3 Inhibition=None(Unspecified) D4 ChEMBL PD 98059 MAPT Potency=15.8489(uM) D4 PubChem PD 98059 MAPT Potency=15848.9(nM) D4 ChEMBL PD 98059 NPC1 Potency=2.3109(uM) D4 PubChem PD 98059 NPC1 Potency=2310.9(nM) D4 ChEMBL PD 98059 PKM Potency=15.8489(uM) D4 PubChem PD 98059 PKM Potency=15848.9(nM) D4 ChEMBL PD 98059 RAB9A Potency=2.0596(uM) D4 PubChem PD 98059 RAB9A Potency=2059.6(nM) D4 ChEMBL PD 98059 SMN1; SMN2 Potency=7943.3(nM) D4 ChEMBL PD 98059 SMN1; SMN2 Potency=8912.5(nM) D4 ChEMBL PD 98059 SMN1; SMN2 Potency=11220.2(nM) D4 ChEMBL PD 98059 SMN2 Potency=7.9433(uM) D4 PubChem PD 98059 SMN2 Potency=8.9125(uM) D4 PubChem PD 98059 SMN2 Potency=11.2202(uM) D4 PubChem PD 98059 TDP1 Potency=29.8554(uM) D4 PubChem PD 98059 THPO Potency=0.3981(uM) D4 PubChem PD 98059 THPO Potency=398.1(nM) D4 ChEMBL PD 98059 TP53 Potency=5.0119(uM) D4 PubChem PD 98059 TP53 Potency=7.9433(uM) D4 PubChem PD 98059 TP53 Potency=5011.9(nM) D4 ChEMBL PD 98059 TP53 Potency=7943.3(nM) D4 ChEMBL