Drug Gene Type Source 1,2-Benzisothiazol-3(2H)-one E2F1 Text_Mining(decreases(reaction)) CTD 1,2-Benzisothiazol-3(2H)-one E2F1 Text_Mining(increases(expression)) CTD 1,2-Benzisothiazol-3(2H)-one ESR1 Text_Mining(decreases(reaction)) CTD 1,2-Benzisothiazol-3(2H)-one ESR1 Text_Mining(increases(activity)) CTD 1,2-Benzisothiazol-3(2H)-one ESR1 Text_Mining(decreases(activity)) CTD 1,2-Benzisothiazol-3(2H)-one MAFF Text_Mining(increases(expression)) CTD 1,2-Benzisothiazol-3(2H)-one MT2A Text_Mining(increases(expression)) CTD 1,2-Benzisothiazol-3(2H)-one NQO1 Text_Mining(increases(expression)) CTD 1,2-Benzisothiazol-3(2H)-one TXN Text_Mining(increases(expression)) CTD 1,2-Benzisothiazol-3(2H)-one ABHD5 None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one APBA1 IC50=12200.0(nM) D4 ChEMBL 1,2-Benzisothiazol-3(2H)-one AR Potency-Replicate_1=27.306(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one BAZ2B Potency=50.1187(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one BAZ2B Potency=50118.7(nM) D4 ChEMBL 1,2-Benzisothiazol-3(2H)-one CACNA1B IC50=12.2(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one CACNA1B IC50=12200.0(nM) D4 ChEMBL 1,2-Benzisothiazol-3(2H)-one CYP19A1 Potency-Replicate_1=30.6379(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one EHMT2 Potency=1.7783(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one EHMT2 Potency=1778.3(nM) D4 ChEMBL 1,2-Benzisothiazol-3(2H)-one HNF4A None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one HSPB1 Ratio Potency (uM)=54.941(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one IL1B None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one KAT2A Potency=8.9125(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one KAT2A Potency=8912.5(nM) D4 ChEMBL 1,2-Benzisothiazol-3(2H)-one KCNJ1 None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one KCNQ1 None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one KDM4A Potency=31622.8(nM) D4 ChEMBL 1,2-Benzisothiazol-3(2H)-one MAPT Potency=11.2202(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one MAPT Potency=25.1189(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one MAPT Potency=25118.9(nM) D4 ChEMBL 1,2-Benzisothiazol-3(2H)-one MAPT Potency=11220.2(nM) D4 ChEMBL 1,2-Benzisothiazol-3(2H)-one NFE2L2 Potency=27.306(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one NR1H4 Potency=44.6684(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one NR2E3 None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one PLIN5 None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one PLK1 Potency=5.3233(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one POLI Potency=25.1189(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one PRMT1 None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one RXRA Potency=19.9526(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one S1PR4 None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one SMARCA2 None=None(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one TDP1 Potency=0.6513(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one TDP1 Potency=1.2995(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one THRB Potency=15.8489(uM) D4 PubChem 1,2-Benzisothiazol-3(2H)-one WRN Potency=31.6228(uM) D4 PubChem