Drug Gene Type Source Spectrum_001666 ADD1 Text_Mining(decreases(expression)) CTD Spectrum_001666 AGER Text_Mining(decreases(reaction)) CTD Spectrum_001666 AGER Text_Mining(increases(expression)) CTD Spectrum_001666 AHR Text_Mining(decreases(expression)) CTD Spectrum_001666 AKT1 Text_Mining(decreases(phosphorylation)) CTD Spectrum_001666 AR Text_Mining(decreases(expression)) CTD Spectrum_001666 BACH1 Text_Mining(increases(expression)) CTD Spectrum_001666 BAP1 Text_Mining(increases(expression)) CTD Spectrum_001666 BRAF Text_Mining(decreases(expression)) CTD Spectrum_001666 CASP8 Text_Mining(decreases(expression)) CTD Spectrum_001666 CAT Text_Mining(increases(expression)) CTD Spectrum_001666 CCND1 Text_Mining(decreases(reaction)) CTD Spectrum_001666 CCND1 Text_Mining(increases(expression)) CTD Spectrum_001666 CCND1 Text_Mining(decreases(expression)) CTD Spectrum_001666 CCNE1 Text_Mining(decreases(expression)) CTD Spectrum_001666 CCNE1 Text_Mining(increases(expression)) CTD Spectrum_001666 CDK1 Text_Mining(decreases(expression)) CTD Spectrum_001666 CDK4 Text_Mining(decreases(expression)) CTD Spectrum_001666 CDK5 Text_Mining(decreases(expression)) CTD Spectrum_001666 CDK7 Text_Mining(decreases(expression)) CTD Spectrum_001666 CDK9 Text_Mining(decreases(expression)) CTD Spectrum_001666 CDKN1A Text_Mining(decreases(reaction)) CTD Spectrum_001666 CDKN1A Text_Mining(increases(expression)) CTD Spectrum_001666 CHGA Text_Mining(increases(expression)) CTD Spectrum_001666 CHGB Text_Mining(decreases(expression)) CTD Spectrum_001666 CRB1 Text_Mining(decreases(expression)) CTD Spectrum_001666 CYP3A4 Text_Mining(increases(activity)) CTD Spectrum_001666 DDB2 Text_Mining(increases(expression)) CTD Spectrum_001666 EIF4G1 Text_Mining(increases(expression)) CTD Spectrum_001666 ESR1 Text_Mining(decreases(reaction)) CTD Spectrum_001666 ESR1 Text_Mining(increases(activity)) CTD Spectrum_001666 ESR1 Text_Mining(increases(expression)) CTD Spectrum_001666 ESR2 Text_Mining(decreases(reaction)) CTD Spectrum_001666 ESR2 Text_Mining(increases(activity)) CTD Spectrum_001666 FANCC Text_Mining(decreases(expression)) CTD Spectrum_001666 FANCF Text_Mining(decreases(expression)) CTD Spectrum_001666 FASLG Text_Mining(decreases(expression)) CTD Spectrum_001666 FOS Text_Mining(increases(expression)) CTD Spectrum_001666 GJA4 Text_Mining(decreases(expression)) CTD Spectrum_001666 GJA5 Text_Mining(decreases(expression)) CTD Spectrum_001666 GJA5 Text_Mining(increases(expression)) CTD Spectrum_001666 GPX4 Text_Mining(decreases(expression)) CTD Spectrum_001666 HMGB1 Text_Mining(decreases(reaction)) CTD Spectrum_001666 HMGB1 Text_Mining(increases(expression)) CTD Spectrum_001666 HMGB1 Text_Mining(increases(secretion)) CTD Spectrum_001666 HMGB1 Text_Mining(decreases(response to substance)) CTD Spectrum_001666 ICAM1 Text_Mining(decreases(reaction)) CTD Spectrum_001666 ICAM1 Text_Mining(increases(expression)) CTD Spectrum_001666 IGF1 Text_Mining(decreases(reaction)) CTD Spectrum_001666 IGF1 Text_Mining(increases(expression)) CTD Spectrum_001666 IGF1 Text_Mining(increases(phosphorylation)) CTD Spectrum_001666 IGF1 Text_Mining(decreases(expression)) CTD Spectrum_001666 IGF1R Text_Mining(decreases(expression)) CTD Spectrum_001666 IGFBP2 Text_Mining(increases(expression)) CTD Spectrum_001666 IVL Text_Mining(decreases(expression)) CTD Spectrum_001666 JAK1 Text_Mining(increases(expression)) CTD Spectrum_001666 JUN Text_Mining(decreases(expression)) CTD Spectrum_001666 KIF2A Text_Mining(increases(expression)) CTD Spectrum_001666 KPNA2 Text_Mining(increases(expression)) CTD Spectrum_001666 LDLR Text_Mining(increases(expression)) CTD Spectrum_001666 LIPA Text_Mining(increases(expression)) CTD Spectrum_001666 MAP2K1 Text_Mining(increases(expression)) CTD Spectrum_001666 MAP2K2 Text_Mining(decreases(expression)) CTD Spectrum_001666 MAP2K4 Text_Mining(decreases(expression)) CTD Spectrum_001666 MAP2K6 Text_Mining(decreases(expression)) CTD Spectrum_001666 MAPK14 Text_Mining(decreases(expression)) CTD Spectrum_001666 MAPK14 Text_Mining(increases(expression)) CTD Spectrum_001666 MAPK3 Text_Mining(decreases(expression)) CTD Spectrum_001666 MAPK8 Text_Mining(decreases(expression)) CTD Spectrum_001666 MGAT2 Text_Mining(increases(expression)) CTD Spectrum_001666 MICA Text_Mining(increases(expression)) CTD Spectrum_001666 MLH1 Text_Mining(increases(expression)) CTD Spectrum_001666 MSH2 Text_Mining(increases(expression)) CTD Spectrum_001666 MSH6 Text_Mining(increases(expression)) CTD Spectrum_001666 NOS1 Text_Mining(decreases(expression)) CTD Spectrum_001666 NUP214 Text_Mining(decreases(expression)) CTD Spectrum_001666 PLA2G2A Text_Mining(decreases(reaction)) CTD Spectrum_001666 PLA2G2A Text_Mining(increases(expression)) CTD Spectrum_001666 PLA2G2A Text_Mining(increases(secretion)) CTD Spectrum_001666 PRKDC Text_Mining(decreases(expression)) CTD Spectrum_001666 RAD50 Text_Mining(increases(expression)) CTD Spectrum_001666 RASSF7 Text_Mining(increases(expression)) CTD Spectrum_001666 RB1 Text_Mining(decreases(activity)) CTD Spectrum_001666 RB1 Text_Mining(decreases(reaction)) CTD Spectrum_001666 RB1 Text_Mining(increases(phosphorylation)) CTD Spectrum_001666 RB1 Text_Mining(decreases(phosphorylation)) CTD Spectrum_001666 RDX Text_Mining(decreases(expression)) CTD Spectrum_001666 RPS6KA1 Text_Mining(decreases(expression)) CTD Spectrum_001666 RPS6KA3 Text_Mining(decreases(expression)) CTD Spectrum_001666 RRM2 Text_Mining(increases(expression)) CTD Spectrum_001666 SELE Text_Mining(decreases(reaction)) CTD Spectrum_001666 SELE Text_Mining(increases(expression)) CTD Spectrum_001666 SEPP1 Text_Mining(decreases(expression)) CTD Spectrum_001666 SMAD3 Text_Mining(increases(expression)) CTD Spectrum_001666 SMC1A Text_Mining(decreases(expression)) CTD Spectrum_001666 STAT3 Text_Mining(increases(expression)) CTD Spectrum_001666 TFF1 Text_Mining(decreases(expression)) CTD Spectrum_001666 TFPI2 Text_Mining(decreases(expression)) CTD Spectrum_001666 TGFA Text_Mining(increases(expression)) CTD Spectrum_001666 TLR2 Text_Mining(decreases(reaction)) CTD Spectrum_001666 TLR2 Text_Mining(increases(expression)) CTD Spectrum_001666 TLR4 Text_Mining(decreases(reaction)) CTD Spectrum_001666 TLR4 Text_Mining(increases(expression)) CTD Spectrum_001666 TNF Text_Mining(decreases(reaction)) CTD Spectrum_001666 TNF Text_Mining(increases(expression)) CTD Spectrum_001666 TNF Text_Mining(increases(secretion)) CTD Spectrum_001666 TP53 Text_Mining(decreases(expression)) CTD Spectrum_001666 VCAM1 Text_Mining(decreases(reaction)) CTD Spectrum_001666 VCAM1 Text_Mining(increases(expression)) CTD Spectrum_001666 VCP Text_Mining(increases(expression)) CTD Spectrum_001666 WRB Text_Mining(decreases(expression)) CTD Spectrum_001666 ZNF138 Text_Mining(increases(expression)) CTD Spectrum_001666 AR Ratio Potency (uM)=19.7391(uM) D4 PubChem Spectrum_001666 EHMT2 Potency=19.9526(uM) D4 PubChem Spectrum_001666 EHMT2 Potency=19952.6(nM) D4 ChEMBL Spectrum_001666 ESR1 Potency-Replicate_1=6.6824(uM) D4 PubChem Spectrum_001666 ESR1 Potency-Replicate_1=7.5624(uM) D4 PubChem Spectrum_001666 ESR1 Ratio Potency (uM)=13.9605(uM) D4 PubChem Spectrum_001666 GMNN Potency=18.8375(uM) D4 PubChem