Drug Gene Type Source sertraline ABCB1 Text_Mining(increases(activity)) CTD sertraline ASAH1 Text_Mining(increases(expression)) CTD sertraline ASNS Text_Mining(increases(expression)) CTD sertraline ATF2 Text_Mining(increases(expression)) CTD sertraline ATF4 Text_Mining(increases(expression)) CTD sertraline BCL2 Text_Mining(decreases(expression)) CTD sertraline C10ORF10 Text_Mining(increases(expression)) CTD sertraline CASP3 Text_Mining(decreases(reaction)) CTD sertraline CASP3 Text_Mining(increases(activity)) CTD sertraline CASP3 Text_Mining(increases(cleavage)) CTD sertraline CASP4 Text_Mining(decreases(reaction)) CTD sertraline CASP4 Text_Mining(increases(cleavage)) CTD sertraline CASP7 Text_Mining(decreases(reaction)) CTD sertraline CASP7 Text_Mining(increases(activity)) CTD sertraline CASP9 Text_Mining(increases(activity)) CTD sertraline CASP9 Text_Mining(increases(cleavage)) CTD sertraline CD14 Text_Mining(decreases(expression)) CTD sertraline CRYAA Text_Mining(increases(expression)) CTD sertraline CUL1 Text_Mining(decreases(expression)) CTD sertraline CYP2B6 Text_Mining(decreases(methylation)) CTD sertraline CYP2B6 Text_Mining(increases(metabolic processing)) CTD sertraline CYP2C19 Text_Mining(affects(metabolic processing)) CTD sertraline CYP2C19 Text_Mining(decreases(amination)) CTD sertraline CYP2C19 Text_Mining(increases(metabolic processing)) CTD sertraline CYP2C19 Text_Mining(decreases(methylation)) CTD sertraline CYP2C9 Text_Mining(decreases(methylation)) CTD sertraline CYP2C9 Text_Mining(increases(metabolic processing)) CTD sertraline CYP2C9 Text_Mining(affects(metabolic processing)) CTD sertraline CYP2C9 Text_Mining(decreases(reaction)) CTD sertraline CYP2D6 Text_Mining(decreases(methylation)) CTD sertraline CYP2D6 Text_Mining(increases(metabolic processing)) CTD sertraline CYP3A4 Text_Mining(decreases(amination)) CTD sertraline CYP3A4 Text_Mining(increases(metabolic processing)) CTD sertraline CYP3A4 Text_Mining(decreases(methylation)) CTD sertraline CYP3A4 Text_Mining(increases(oxidation)) CTD sertraline CYP3A4 Text_Mining(increases(reaction)) CTD sertraline DDIT3 Text_Mining(decreases(reaction)) CTD sertraline DDIT3 Text_Mining(increases(expression)) CTD sertraline DNAJC5 Text_Mining(increases(expression)) CTD sertraline DUSP1 Text_Mining(increases(expression)) CTD sertraline DUSP10 Text_Mining(increases(expression)) CTD sertraline DUSP14 Text_Mining(increases(expression)) CTD sertraline DUSP16 Text_Mining(increases(expression)) CTD sertraline DUSP8 Text_Mining(increases(expression)) CTD sertraline EGFR Text_Mining(increases(expression)) CTD sertraline EIF2AK3 Text_Mining(decreases(reaction)) CTD sertraline EIF2AK3 Text_Mining(increases(phosphorylation)) CTD sertraline EIF2AK3 Text_Mining(increases(expression)) CTD sertraline EIF2S1 Text_Mining(increases(phosphorylation)) CTD sertraline ERN1 Text_Mining(increases(expression)) CTD sertraline FABP1 Text_Mining(increases(expression)) CTD sertraline FNDC4 Text_Mining(increases(expression)) CTD sertraline FOS Text_Mining(increases(expression)) CTD sertraline GADD45A Text_Mining(increases(expression)) CTD sertraline GADD45B Text_Mining(increases(expression)) CTD sertraline GDPD3 Text_Mining(increases(expression)) CTD sertraline HERPUD1 Text_Mining(increases(expression)) CTD sertraline HPN Text_Mining(increases(expression)) CTD sertraline HSPA1A Text_Mining(increases(expression)) CTD sertraline HSPA1B Text_Mining(increases(expression)) CTD sertraline HSPA6 Text_Mining(increases(expression)) CTD sertraline HSPA8 Text_Mining(decreases(expression)) CTD sertraline INHBE Text_Mining(increases(expression)) CTD sertraline JUN Text_Mining(increases(expression)) CTD sertraline JUN Text_Mining(increases(phosphorylation)) CTD sertraline JUND Text_Mining(increases(expression)) CTD sertraline LSS Text_Mining(increases(expression)) CTD sertraline MAOA Text_Mining(decreases(amination)) CTD sertraline MAOA Text_Mining(increases(metabolic processing)) CTD sertraline MAOB Text_Mining(decreases(amination)) CTD sertraline MAOB Text_Mining(increases(metabolic processing)) CTD sertraline MAP3K13 Text_Mining(increases(expression)) CTD sertraline MAP3K8 Text_Mining(increases(expression)) CTD sertraline MAP4K4 Text_Mining(decreases(reaction)) CTD sertraline MAP4K4 Text_Mining(increases(cleavage)) CTD sertraline MAP4K4 Text_Mining(increases(expression)) CTD sertraline MAP4K4 Text_Mining(increases(phosphorylation)) CTD sertraline MAP4K4 Text_Mining(decreases(expression)) CTD sertraline MAPK1 Text_Mining(decreases(reaction)) CTD sertraline MAPK1 Text_Mining(increases(phosphorylation)) CTD sertraline MAPK3 Text_Mining(increases(phosphorylation)) CTD sertraline MAPK8IP3 Text_Mining(increases(expression)) CTD sertraline MCL1 Text_Mining(decreases(expression)) CTD sertraline MYC Text_Mining(increases(expression)) CTD sertraline NFE2L2 Text_Mining(increases(expression)) CTD sertraline NFKB1 Text_Mining(increases(expression)) CTD sertraline NFKB2 Text_Mining(increases(expression)) CTD sertraline NR0B2 Text_Mining(increases(expression)) CTD sertraline NUPR1 Text_Mining(increases(expression)) CTD sertraline PECAM1 Text_Mining(decreases(expression)) CTD sertraline PF4 Text_Mining(decreases(expression)) CTD sertraline PHYH Text_Mining(increases(expression)) CTD sertraline PPBP Text_Mining(decreases(expression)) CTD sertraline PPP1R15A Text_Mining(increases(expression)) CTD sertraline PTGS2 Text_Mining(decreases(expression)) CTD sertraline RBX1 Text_Mining(decreases(expression)) CTD sertraline RELB Text_Mining(increases(expression)) CTD sertraline RPS6KA3 Text_Mining(decreases(expression)) CTD sertraline SEC61G Text_Mining(decreases(expression)) CTD sertraline SELE Text_Mining(decreases(expression)) CTD sertraline SELP Text_Mining(decreases(expression)) CTD sertraline VIMP Text_Mining(increases(expression)) CTD sertraline SERPINA3 Text_Mining(increases(expression)) CTD sertraline SKP1 Text_Mining(decreases(expression)) CTD sertraline SLC2A3 Text_Mining(decreases(expression)) CTD sertraline SLC6A4 Text_Mining(decreases(reaction)) CTD sertraline SLC6A4 Text_Mining(increases(expression)) CTD sertraline SLC6A4 Text_Mining(increases(response to substance)) CTD sertraline SLC6A4 Text_Mining(affects(response to substance)) CTD sertraline SSR2 Text_Mining(increases(expression)) CTD sertraline STAT3 Text_Mining(decreases(expression)) CTD sertraline STMN1 Text_Mining(decreases(expression)) CTD sertraline SYVN1 Text_Mining(increases(expression)) CTD sertraline TAGLN Text_Mining(decreases(expression)) CTD sertraline TAOK2 Text_Mining(increases(expression)) CTD sertraline TNF Text_Mining(decreases(secretion)) CTD sertraline TNF Text_Mining(increases(expression)) CTD sertraline TXNDC5 Text_Mining(decreases(expression)) CTD sertraline UBE2D4 Text_Mining(decreases(expression)) CTD sertraline UBE2G1 Text_Mining(decreases(expression)) CTD sertraline UBE4B Text_Mining(decreases(expression)) CTD sertraline UBQLN1 Text_Mining(increases(expression)) CTD sertraline UGT2B7 Text_Mining(increases(glucuronidation)) CTD sertraline UGT2B7 Text_Mining(increases(metabolic processing)) CTD sertraline VCAM1 Text_Mining(increases(expression)) CTD sertraline WIPI1 Text_Mining(increases(expression)) CTD sertraline XBP1 Text_Mining(increases(splicing)) CTD sertraline APAF1 None=None(uM) D4 PubChem sertraline ATXN2 Potency=14.1254(uM) D4 PubChem sertraline ATXN2 Potency=25.1189(uM) D4 PubChem sertraline CDK1 Activity=None(Unspecified) D4 ChEMBL sertraline CFL1 Inhibition=None(Unspecified) D4 ChEMBL sertraline CFL1 Activity=None(Unspecified) D4 ChEMBL sertraline DRD1 Potency=10.0(uM) D4 PubChem sertraline DRD1 Potency=11.2202(uM) D4 PubChem sertraline DRD1 None=None(uM) D4 PubChem sertraline DRD1 Potency=11220.2(nM) D4 ChEMBL sertraline DRD1 Potency=10000.0(nM) D4 ChEMBL sertraline IDH1 Potency=10.3225(uM) D4 PubChem sertraline JUN Activity=None(Unspecified) D4 ChEMBL sertraline MCHR1 None=None(uM) D4 PubChem sertraline MDM2 None=None(uM) D4 PubChem sertraline MDM4 None=None(uM) D4 PubChem sertraline NPBWR1 None=None(uM) D4 PubChem sertraline SLC5A7 None=None(uM) D4 PubChem sertraline STK33 None=None(uM) D4 PubChem sertraline TAAR1 None=None(uM) D4 PubChem sertraline TP53 Activity=None(Unspecified) D4 ChEMBL sertraline UBE2N None=None(uM) D4 PubChem