Drug Gene Type Source cisapride ABCB11 Text_Mining(decreases(activity)) CTD cisapride CYP2C9 Text_Mining(decreases(activity)) CTD cisapride CYP3A4 Text_Mining(decreases(reaction)) CTD cisapride CYP3A4 Text_Mining(increases(oxidation)) CTD cisapride CYP3A4 Text_Mining(decreases(activity)) CTD cisapride CYP3A4 Text_Mining(affects(chemical synthesis)) CTD cisapride CYP3A4 Text_Mining(affects(metabolic processing)) CTD cisapride KCNH2 Text_Mining(decreases(activity)) CTD cisapride KCNH2 Text_Mining(decreases(reaction)) CTD cisapride KCNH2 Text_Mining(affects(localization)) CTD cisapride KCNH2 Text_Mining(affects(binding)) CTD cisapride KCNH2 Text_Mining(increases(transport)) CTD cisapride SCN5A Text_Mining(increases(localization)) CTD cisapride SLC22A2 Text_Mining(decreases(reaction)) CTD cisapride SLC22A2 Text_Mining(increases(uptake)) CTD cisapride ABCB1 None=None(uM) D4 PubChem cisapride CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL cisapride CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL cisapride CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL cisapride CYP2D6 Potency=0.2512(uM) D4 PubChem cisapride CYP2D6 None=None(uM) D4 PubChem cisapride CYP2D6 Potency=251.2(nM) D4 ChEMBL cisapride CYP2D6 AC50=251.19(nM) D4 ChEMBL cisapride CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL cisapride CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL cisapride DRD3 None=None(uM) D4 PubChem cisapride HPSE Activity=None(Unspecified) D4 ChEMBL cisapride HTR4 None=None(uM) D4 PubChem cisapride KCNH2 Activity=None(Unspecified) D4 ChEMBL cisapride LYPLA2 None=None(uM) D4 PubChem cisapride PREPL None=None(uM) D4 PubChem cisapride UBE2N None=None(uM) D4 PubChem