Drug Gene Type Source loratadine ABCB1 Text_Mining(increases(export)) CTD loratadine ABCB11 Text_Mining(decreases(reaction)) CTD loratadine ABCB11 Text_Mining(increases(transport)) CTD loratadine ABCB11 Text_Mining(decreases(activity)) CTD loratadine ABCC1 Text_Mining(decreases(response to substance)) CTD loratadine ABCC2 Text_Mining(decreases(reaction)) CTD loratadine ABCC2 Text_Mining(increases(export)) CTD loratadine ALOX5 Text_Mining(decreases(activity)) CTD loratadine AP1S1 Text_Mining(decreases(expression)) CTD loratadine ASNS Text_Mining(increases(expression)) CTD loratadine CASP3 Text_Mining(increases(activity)) CTD loratadine CASP3 Text_Mining(increases(reaction)) CTD loratadine CASP3 Text_Mining(increases(cleavage)) CTD loratadine CASP7 Text_Mining(increases(activity)) CTD loratadine CASP7 Text_Mining(increases(reaction)) CTD loratadine CASP8 Text_Mining(increases(cleavage)) CTD loratadine CASP9 Text_Mining(increases(cleavage)) CTD loratadine CYP2C8 Text_Mining(decreases(activity)) CTD loratadine CYP2D6 Text_Mining(affects(metabolic processing)) CTD loratadine CYP3A4 Text_Mining(decreases(activity)) CTD loratadine FABP1 Text_Mining(increases(expression)) CTD loratadine GDPD3 Text_Mining(increases(expression)) CTD loratadine HPN Text_Mining(increases(expression)) CTD loratadine HRH1 Text_Mining(affects(binding)) CTD loratadine INHBE Text_Mining(increases(expression)) CTD loratadine KCNH2 Text_Mining(affects(activity)) CTD loratadine KCNH2 Text_Mining(affects(binding)) CTD loratadine KCNH2 Text_Mining(decreases(activity)) CTD loratadine KCNH2 Text_Mining(decreases(reaction)) CTD loratadine KCNH2 Text_Mining(increases(transport)) CTD loratadine LSS Text_Mining(increases(expression)) CTD loratadine NR0B2 Text_Mining(increases(expression)) CTD loratadine NUPR1 Text_Mining(increases(expression)) CTD loratadine RPS6 Text_Mining(decreases(expression)) CTD loratadine SERPINA3 Text_Mining(increases(expression)) CTD loratadine SLC2A3 Text_Mining(decreases(expression)) CTD loratadine TAGLN Text_Mining(decreases(expression)) CTD loratadine AR Potency-Replicate_1=17.3739(uM) D4 PubChem loratadine AR AR Potency (uM)=27.644(uM) D4 PubChem loratadine AR Potency-Replicate_1=61.1306(uM) D4 PubChem loratadine CACNA1H None=None(uM) D4 PubChem loratadine CYP2C19 Potency=0.3981(uM) D4 PubChem loratadine CYP2C19 Potency=398.1(nM) D4 ChEMBL loratadine CYP2C9 Potency=15.8489(uM) D4 PubChem loratadine CYP2C9 None=None(uM) D4 PubChem loratadine CYP2C9 Potency=15848.9(nM) D4 ChEMBL loratadine CYP2C9 AC50=15848.9(nM) D4 ChEMBL loratadine CYP2D6 Potency=31.6228(uM) D4 PubChem loratadine CYP2D6 Potency=31622.8(nM) D4 ChEMBL loratadine DRD3 None=None(uM) D4 PubChem loratadine ESR1 Ratio Potency (uM)=22.5767(uM) D4 PubChem loratadine ESR1 Potency-Replicate_1=26.8325(uM) D4 PubChem loratadine ESR1 Potency-Replicate_1=61.1306(uM) D4 PubChem loratadine ESR1 ER Potency (uM)=61.1306(uM) D4 PubChem loratadine GMNN Potency=23.1093(uM) D4 PubChem loratadine HIF1A Potency=15.8489(uM) D4 PubChem loratadine HIF1A Potency=15848.9(nM) D4 ChEMBL loratadine MAPK1 Potency=19.9526(uM) D4 PubChem loratadine MAPK1 Potency=19952.6(nM) D4 ChEMBL loratadine NFE2L2 Ratio Potency (uM)=6.18824(uM) D4 PubChem loratadine NFE2L2 Ratio Potency (uM)=6.60073(uM) D4 PubChem loratadine NPSR1 Potency=7.9433(uM) D4 PubChem loratadine NPSR1 Potency=12.5893(uM) D4 PubChem loratadine NPSR1 Potency=7943.3(nM) D4 ChEMBL loratadine NPSR1 Potency=12589.3(nM) D4 ChEMBL loratadine PHOSPHO1 IC50=None(uM) D4 PubChem loratadine PPARD Ratio Potency (uM)=59.3239(uM) D4 PubChem loratadine PPARG Potency-Replicate_1=13.3322(uM) D4 PubChem loratadine PPARG None=None(uM) D4 PubChem loratadine TDP1 Potency=2.6609(uM) D4 PubChem loratadine TDP1 Potency=11.8856(uM) D4 PubChem loratadine TDP1 Potency=12.9953(uM) D4 PubChem loratadine TDP1 Potency=14.9631(uM) D4 PubChem loratadine TDP1 Potency=20.5962(uM) D4 PubChem loratadine TSHR Potency=39.8107(uM) D4 PubChem loratadine TSHR Potency=39810.7(nM) D4 ChEMBL