Drug Gene Type Source terfenadine ABCB1 Text_Mining(affects(transport)) CTD terfenadine ABCB1 Text_Mining(decreases(activity)) CTD terfenadine ABCB11 Text_Mining(decreases(reaction)) CTD terfenadine ABCB11 Text_Mining(increases(transport)) CTD terfenadine ABCB11 Text_Mining(decreases(activity)) CTD terfenadine AKT1 Text_Mining(decreases(phosphorylation)) CTD terfenadine AKT1 Text_Mining(decreases(reaction)) CTD terfenadine BAX Text_Mining(increases(expression)) CTD terfenadine BCL2 Text_Mining(decreases(expression)) CTD terfenadine CASP2 Text_Mining(increases(activity)) CTD terfenadine CASP3 Text_Mining(increases(activity)) CTD terfenadine CASP3 Text_Mining(increases(reaction)) CTD terfenadine CASP3 Text_Mining(increases(cleavage)) CTD terfenadine CASP6 Text_Mining(increases(activity)) CTD terfenadine CASP8 Text_Mining(increases(activity)) CTD terfenadine CASP8 Text_Mining(increases(cleavage)) CTD terfenadine CASP9 Text_Mining(increases(activity)) CTD terfenadine CASP9 Text_Mining(increases(cleavage)) CTD terfenadine CD82 Text_Mining(decreases(reaction)) CTD terfenadine CD82 Text_Mining(increases(expression)) CTD terfenadine CDKN1A Text_Mining(increases(expression)) CTD terfenadine CDKN1B Text_Mining(increases(expression)) CTD terfenadine CYP2J2 Text_Mining(decreases(activity)) CTD terfenadine CYP3A Text_Mining(affects(metabolic processing)) CTD terfenadine CYP3A4 Text_Mining(affects(metabolic processing)) CTD terfenadine CYP3A4 Text_Mining(increases(degradation)) CTD terfenadine CYP3A4 Text_Mining(increases(metabolic processing)) CTD terfenadine CYP3A4 Text_Mining(decreases(reaction)) CTD terfenadine CYP3A4 Text_Mining(increases(expression)) CTD terfenadine CYP3A4 Text_Mining(increases(oxidation)) CTD terfenadine CYP3A4 Text_Mining(increases(reaction)) CTD terfenadine CYP3A5 Text_Mining(affects(metabolic processing)) CTD terfenadine EGFR Text_Mining(decreases(phosphorylation)) CTD terfenadine EGFR Text_Mining(decreases(reaction)) CTD terfenadine IL10 Text_Mining(decreases(reaction)) CTD terfenadine IL10 Text_Mining(increases(expression)) CTD terfenadine IL13 Text_Mining(decreases(reaction)) CTD terfenadine IL13 Text_Mining(increases(expression)) CTD terfenadine IL2 Text_Mining(decreases(expression)) CTD terfenadine IL2 Text_Mining(decreases(reaction)) CTD terfenadine IL4 Text_Mining(decreases(expression)) CTD terfenadine IL4 Text_Mining(decreases(reaction)) CTD terfenadine IL4 Text_Mining(increases(expression)) CTD terfenadine IL5 Text_Mining(decreases(reaction)) CTD terfenadine IL5 Text_Mining(increases(expression)) CTD terfenadine IL5 Text_Mining(decreases(expression)) CTD terfenadine IL6 Text_Mining(decreases(reaction)) CTD terfenadine IL6 Text_Mining(increases(expression)) CTD terfenadine KCNA5 Text_Mining(decreases(activity)) CTD terfenadine KCNE1 Text_Mining(decreases(reaction)) CTD terfenadine KCNE1 Text_Mining(increases(response to substance)) CTD terfenadine KCNH2 Text_Mining(decreases(reaction)) CTD terfenadine KCNH2 Text_Mining(increases(transport)) CTD terfenadine KCNH2 Text_Mining(decreases(activity)) CTD terfenadine KCNH2 Text_Mining(affects(binding)) CTD terfenadine KCNH2 Text_Mining(increases(reaction)) CTD terfenadine KCNH2 Text_Mining(affects(cotreatment)) CTD terfenadine KCNQ1 Text_Mining(decreases(reaction)) CTD terfenadine KCNQ1 Text_Mining(increases(response to substance)) CTD terfenadine NME1 Text_Mining(decreases(reaction)) CTD terfenadine NME1 Text_Mining(increases(expression)) CTD terfenadine PTH Text_Mining(decreases(expression)) CTD terfenadine RPS6 Text_Mining(decreases(expression)) CTD terfenadine TNF Text_Mining(decreases(expression)) CTD terfenadine TNF Text_Mining(decreases(reaction)) CTD terfenadine TP53 Text_Mining(increases(expression)) CTD terfenadine ABCB1 None=None(uM) D4 PubChem terfenadine ADRB2 None=None(uM) D4 PubChem terfenadine APAF1 None=None(uM) D4 PubChem terfenadine CACNA1H None=None(uM) D4 PubChem terfenadine CYP19A1 Potency-Replicate_1=29.8493(uM) D4 PubChem terfenadine DRD1 None=None(uM) D4 PubChem terfenadine DRD3 None=None(uM) D4 PubChem terfenadine EPAS1 None=None(uM) D4 PubChem terfenadine GMNN Potency=11.2202(uM) D4 PubChem terfenadine GMNN Potency=11220.2(nM) D4 ChEMBL terfenadine HIF1A None=None(uM) D4 PubChem terfenadine HTT Potency=22.3872(uM) D4 PubChem terfenadine HTT Potency=28.1838(uM) D4 PubChem terfenadine HTT Potency=22387.2(nM) D4 ChEMBL terfenadine HTT Potency=28183.8(nM) D4 ChEMBL terfenadine KCNH2 Potency=0.3981(uM) D4 PubChem terfenadine MAP1LC3A None=None(uM) D4 PubChem terfenadine MAP4K2 None=None(uM) D4 PubChem terfenadine MDM2 None=None(uM) D4 PubChem terfenadine MDM4 None=None(uM) D4 PubChem terfenadine MITF None=None(uM) D4 PubChem terfenadine MMP14 EC50=None(uM) D4 PubChem terfenadine MTOR Potency=7.3621(uM) D4 PubChem terfenadine MTOR Potency=18.4927(uM) D4 PubChem terfenadine MTOR Potency=18492.7(nM) D4 ChEMBL terfenadine MTOR Potency=7362.1(nM) D4 ChEMBL terfenadine S1PR4 None=None(uM) D4 PubChem terfenadine STK33 None=None(uM) D4 PubChem terfenadine TDP1 Potency=2.6609(uM) D4 PubChem terfenadine TDP1 Potency=2.9855(uM) D4 PubChem terfenadine TDP1 Potency=3.3498(uM) D4 PubChem terfenadine TDP1 Potency=4.6109(uM) D4 PubChem terfenadine TDP1 Potency=5.8048(uM) D4 PubChem terfenadine THPO Potency=2.5119(uM) D4 PubChem terfenadine THPO Potency=2511.9(nM) D4 ChEMBL terfenadine TNFRSF10B None=None(uM) D4 PubChem terfenadine UBE2N None=None(uM) D4 PubChem