Drug Gene Type Source astemizole ABCB11 Text_Mining(decreases(reaction)) CTD astemizole ABCB11 Text_Mining(increases(transport)) CTD astemizole ABCB11 Text_Mining(decreases(activity)) CTD astemizole CYP2J2 Text_Mining(decreases(methylation)) CTD astemizole CYP2J2 Text_Mining(decreases(reaction)) CTD astemizole CYP2J2 Text_Mining(increases(metabolic processing)) CTD astemizole CYP3A4 Text_Mining(increases(degradation)) CTD astemizole HRH1 Text_Mining(affects(cotreatment)) CTD astemizole HRH1 Text_Mining(decreases(activity)) CTD astemizole HRH1 Text_Mining(decreases(reaction)) CTD astemizole ICAM1 Text_Mining(decreases(reaction)) CTD astemizole ICAM1 Text_Mining(increases(expression)) CTD astemizole IGF1 Text_Mining(decreases(reaction)) CTD astemizole IGF1 Text_Mining(increases(activity)) CTD astemizole IL1B Text_Mining(decreases(reaction)) CTD astemizole IL1B Text_Mining(increases(expression)) CTD astemizole KCNH1 Text_Mining(affects(binding)) CTD astemizole KCNH1 Text_Mining(decreases(activity)) CTD astemizole KCNH1 Text_Mining(decreases(reaction)) CTD astemizole KCNH1 Text_Mining(increases(activity)) CTD astemizole KCNH2 Text_Mining(affects(localization)) CTD astemizole KCNH2 Text_Mining(affects(binding)) CTD astemizole KCNH2 Text_Mining(decreases(activity)) CTD astemizole KCNH2 Text_Mining(decreases(reaction)) CTD astemizole KCNH2 Text_Mining(decreases(metabolic processing)) CTD astemizole KCNH2 Text_Mining(increases(transport)) CTD astemizole KCNH2 Text_Mining(increases(reaction)) CTD astemizole KCNQ2 Text_Mining(affects(cotreatment)) CTD astemizole KCNQ2 Text_Mining(decreases(activity)) CTD astemizole KCNQ2 Text_Mining(decreases(reaction)) CTD astemizole KCNQ3 Text_Mining(affects(cotreatment)) CTD astemizole KCNQ3 Text_Mining(decreases(activity)) CTD astemizole KCNQ3 Text_Mining(decreases(reaction)) CTD astemizole MAPT Text_Mining(affects(binding)) CTD astemizole VCAM1 Text_Mining(decreases(reaction)) CTD astemizole VCAM1 Text_Mining(increases(expression)) CTD astemizole ABCB1 None=None(uM) D4 PubChem astemizole APAF1 None=None(uM) D4 PubChem astemizole APLNR None=None(uM) D4 PubChem astemizole AR Potency-Replicate_1=12.464(uM) D4 PubChem astemizole AR Potency-Replicate_1=18.9959(uM) D4 PubChem astemizole AVPR1A None=None(uM) D4 PubChem astemizole CACNA1H None=None(uM) D4 PubChem astemizole CYP19A1 Potency-Replicate_1=6.2468(uM) D4 PubChem astemizole CYP19A1 Potency-Replicate_1=21.1317(uM) D4 PubChem astemizole CYP2D6 Potency=7.9433(uM) D4 PubChem astemizole CYP2D6 None=None(uM) D4 PubChem astemizole CYP2D6 AC50=7943.28(nM) D4 ChEMBL astemizole CYP2D6 Potency=7943.3(nM) D4 ChEMBL astemizole DRD1 None=None(uM) D4 PubChem astemizole GMNN Potency=3.6626(uM) D4 PubChem astemizole GMNN Potency=4.6109(uM) D4 PubChem astemizole GMNN Potency=23.715(uM) D4 PubChem astemizole GNA15 None=None(uM) D4 PubChem astemizole HPSE Activity=None(Unspecified) D4 ChEMBL astemizole IDH1 Potency=14.581(uM) D4 PubChem astemizole IL1B None=None(uM) D4 PubChem astemizole ITGA4 None=None(uM) D4 PubChem astemizole JAK2 None=None(uM) D4 PubChem astemizole MAP4K2 None=None(uM) D4 PubChem astemizole MDM2 None=None(uM) D4 PubChem astemizole MDM4 None=None(uM) D4 PubChem astemizole MITF None=None(uM) D4 PubChem astemizole MMP14 EC50=None(uM) D4 PubChem astemizole OXTR None=None(uM) D4 PubChem astemizole PAX8 None=None(uM) D4 PubChem astemizole PPARD Potency-Replicate_1=29.847(uM) D4 PubChem astemizole PPARG Potency-Replicate_1=29.847(uM) D4 PubChem astemizole STK33 None=None(uM) D4 PubChem astemizole TAAR1 None=None(uM) D4 PubChem astemizole TDP1 Potency=2.6609(uM) D4 PubChem astemizole TDP1 Potency=3.7586(uM) D4 PubChem astemizole TDP1 Potency=7.3078(uM) D4 PubChem astemizole TDP1 Potency=10.3225(uM) D4 PubChem astemizole TDP1 Potency=14.581(uM) D4 PubChem astemizole TDP1 Potency=16.3601(uM) D4 PubChem astemizole TP53 Potency=12.5893(uM) D4 PubChem astemizole TP53 Potency=12589.3(nM) D4 ChEMBL astemizole UBE2N None=None(uM) D4 PubChem