Drug Gene Type Source GUANFACINE GH1 Text_Mining(increases(expression)) CTD GUANFACINE REN Text_Mining(decreases(activity)) CTD GUANFACINE SLC22A2 Text_Mining(decreases(reaction)) CTD GUANFACINE SLC22A2 Text_Mining(increases(uptake)) CTD GUANFACINE CYP2C19 Potency=0.2512(uM) D4 PubChem GUANFACINE CYP2C19 None=None(uM) D4 PubChem GUANFACINE CYP2C19 AC50=251.19(nM) D4 ChEMBL GUANFACINE CYP2C19 Potency=251.2(nM) D4 ChEMBL GUANFACINE CYP2D6 Potency=0.1259(uM) D4 PubChem GUANFACINE CYP2D6 None=None(uM) D4 PubChem GUANFACINE CYP2D6 AC50=125.89(nM) D4 ChEMBL GUANFACINE CYP2D6 Potency=125.9(nM) D4 ChEMBL GUANFACINE CYP3A4 Potency=12.5893(uM) D4 PubChem GUANFACINE CYP3A4 None=None(uM) D4 PubChem GUANFACINE CYP3A4 AC50=12589.2(nM) D4 ChEMBL GUANFACINE CYP3A4 Potency=12589.3(nM) D4 ChEMBL GUANFACINE EHMT2 Potency=12.5893(uM) D4 PubChem GUANFACINE EHMT2 Potency=12589.3(nM) D4 ChEMBL