Drug Gene Type Source THIORPHAN AKT1 Text_Mining(affects(activity)) CTD THIORPHAN AKT1 Text_Mining(decreases(activity)) CTD THIORPHAN AKT1 Text_Mining(decreases(phosphorylation)) CTD THIORPHAN IGFBP5 Text_Mining(affects(expression)) CTD THIORPHAN MAPK1 Text_Mining(affects(phosphorylation)) CTD THIORPHAN MAPK3 Text_Mining(affects(phosphorylation)) CTD THIORPHAN MME Text_Mining(decreases(activity)) CTD THIORPHAN MME Text_Mining(affects(activity)) CTD THIORPHAN CFTR None=None(uM) D4 PubChem THIORPHAN ESR1 None=None(uM) D4 PubChem THIORPHAN MRGPRX1 None=None(uM) D4 PubChem THIORPHAN NFE2L2 Potency=10.3225(uM) D4 PubChem THIORPHAN NFE2L2 Potency=10322.5(nM) D4 ChEMBL