Drug Gene Type Source ticlopidine ABCB11 Text_Mining(decreases(activity)) CTD ticlopidine ABCC2 Text_Mining(decreases(activity)) CTD ticlopidine CASP3 Text_Mining(increases(activity)) CTD ticlopidine CASP3 Text_Mining(increases(reaction)) CTD ticlopidine CASP7 Text_Mining(increases(activity)) CTD ticlopidine CASP7 Text_Mining(increases(reaction)) CTD ticlopidine CYP1A2 Text_Mining(increases(cleavage)) CTD ticlopidine CYP1A2 Text_Mining(increases(oxidation)) CTD ticlopidine CYP1A2 Text_Mining(decreases(reaction)) CTD ticlopidine CYP1A2 Text_Mining(decreases(activity)) CTD ticlopidine CYP2B6 Text_Mining(affects(metabolic processing)) CTD ticlopidine CYP2B6 Text_Mining(decreases(reaction)) CTD ticlopidine CYP2B6 Text_Mining(increases(metabolic processing)) CTD ticlopidine CYP2B6 Text_Mining(decreases(activity)) CTD ticlopidine CYP2C19 Text_Mining(increases(cleavage)) CTD ticlopidine CYP2C19 Text_Mining(increases(oxidation)) CTD ticlopidine CYP2C19 Text_Mining(decreases(reaction)) CTD ticlopidine CYP2C19 Text_Mining(increases(hydroxylation)) CTD ticlopidine CYP2C19 Text_Mining(increases(metabolic processing)) CTD ticlopidine CYP2C19 Text_Mining(decreases(activity)) CTD ticlopidine CYP2C8 Text_Mining(increases(cleavage)) CTD ticlopidine CYP2C8 Text_Mining(increases(oxidation)) CTD ticlopidine CYP2C9 Text_Mining(increases(cleavage)) CTD ticlopidine CYP2C9 Text_Mining(increases(oxidation)) CTD ticlopidine CYP2D6 Text_Mining(increases(cleavage)) CTD ticlopidine CYP2D6 Text_Mining(increases(oxidation)) CTD ticlopidine CYP2D6 Text_Mining(decreases(activity)) CTD ticlopidine CYP3A4 Text_Mining(increases(degradation)) CTD ticlopidine CYP3A4 Text_Mining(increases(cleavage)) CTD ticlopidine CYP3A4 Text_Mining(increases(oxidation)) CTD ticlopidine CYP3A4 Text_Mining(increases(response to substance)) CTD ticlopidine CYP3A4 Text_Mining(decreases(reaction)) CTD ticlopidine CYP3A4 Text_Mining(increases(reaction)) CTD ticlopidine CYP3A5 Text_Mining(increases(cleavage)) CTD ticlopidine CYP3A5 Text_Mining(increases(oxidation)) CTD ticlopidine HMOX1 Text_Mining(affects(cotreatment)) CTD ticlopidine HMOX1 Text_Mining(decreases(reaction)) CTD ticlopidine HMOX1 Text_Mining(increases(expression)) CTD ticlopidine HMOX1 Text_Mining(increases(reaction)) CTD ticlopidine THBS1 Text_Mining(affects(expression)) CTD ticlopidine UGT1A1 Text_Mining(increases(expression)) CTD ticlopidine CYP1A2 None=None(uM) D4 PubChem ticlopidine CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL ticlopidine CYP1A2 AC50=501.19(nM) D4 ChEMBL ticlopidine CYP2C19 Potency=0.0398(uM) D4 PubChem ticlopidine CYP2C19 None=None(uM) D4 PubChem ticlopidine CYP2C19 AC50=39.81(nM) D4 ChEMBL ticlopidine CYP2C19 Potency=39.8(nM) D4 ChEMBL ticlopidine CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL ticlopidine CYP2D6 Potency=0.3981(uM) D4 PubChem ticlopidine CYP2D6 None=None(uM) D4 PubChem ticlopidine CYP2D6 AC50=398.11(nM) D4 ChEMBL ticlopidine CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL ticlopidine CYP2D6 Potency=398.1(nM) D4 ChEMBL ticlopidine CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL ticlopidine ESR1 Potency-Replicate_1=11.8832(uM) D4 PubChem ticlopidine ESR1 Ratio Potency (uM)=21.2929(uM) D4 PubChem ticlopidine ESR1 Potency-Replicate_1=23.8911(uM) D4 PubChem ticlopidine MAP3K3 None=None(uM) D4 PubChem ticlopidine MAP4K2 None=None(uM) D4 PubChem