Drug Gene Type Source thiostrepton BAX Text_Mining(increases(expression)) CTD thiostrepton BCL2 Text_Mining(decreases(expression)) CTD thiostrepton BCL2L1 Text_Mining(decreases(expression)) CTD thiostrepton CCL3 Text_Mining(decreases(expression)) CTD thiostrepton CCL4 Text_Mining(decreases(expression)) CTD thiostrepton CCND1 Text_Mining(decreases(expression)) CTD thiostrepton CDKN1A Text_Mining(increases(expression)) CTD thiostrepton CRYAB Text_Mining(increases(expression)) CTD thiostrepton CYP1A1 Text_Mining(decreases(expression)) CTD thiostrepton CYP2E1 Text_Mining(decreases(expression)) CTD thiostrepton DDIT3 Text_Mining(increases(expression)) CTD thiostrepton DNAJA1 Text_Mining(increases(expression)) CTD thiostrepton DNAJB4 Text_Mining(increases(expression)) CTD thiostrepton EIF2S1 Text_Mining(increases(expression)) CTD thiostrepton GADD45A Text_Mining(increases(expression)) CTD thiostrepton GDF15 Text_Mining(increases(expression)) CTD thiostrepton GSR Text_Mining(increases(expression)) CTD thiostrepton GSTP1 Text_Mining(decreases(reaction)) CTD thiostrepton GSTP1 Text_Mining(increases(metabolic processing)) CTD thiostrepton HMOX1 Text_Mining(increases(expression)) CTD thiostrepton HSP90AA2P Text_Mining(increases(expression)) CTD thiostrepton HSP90AB1 Text_Mining(increases(expression)) CTD thiostrepton HSPA1A Text_Mining(increases(expression)) CTD thiostrepton HSPA1L Text_Mining(increases(expression)) CTD thiostrepton HSPA2 Text_Mining(increases(expression)) CTD thiostrepton HSPA4 Text_Mining(increases(expression)) CTD thiostrepton HSPA5 Text_Mining(increases(expression)) CTD thiostrepton HSPA6 Text_Mining(increases(expression)) CTD thiostrepton HSPA8 Text_Mining(increases(expression)) CTD thiostrepton HSPB1 Text_Mining(increases(expression)) CTD thiostrepton HSPD1 Text_Mining(increases(expression)) CTD thiostrepton HSPH1 Text_Mining(increases(expression)) CTD thiostrepton IL1A Text_Mining(decreases(expression)) CTD thiostrepton IL1B Text_Mining(decreases(expression)) CTD thiostrepton MCL1 Text_Mining(decreases(expression)) CTD thiostrepton MCL1 Text_Mining(increases(expression)) CTD thiostrepton NFKB1 Text_Mining(decreases(expression)) CTD thiostrepton PMAIP1 Text_Mining(increases(expression)) CTD thiostrepton PTGS1 Text_Mining(increases(expression)) CTD thiostrepton SOD1 Text_Mining(increases(expression)) CTD thiostrepton TP53 Text_Mining(decreases(expression)) CTD thiostrepton XRCC2 Text_Mining(decreases(expression)) CTD thiostrepton AR AR Potency (uM)=10.5196(uM) D4 PubChem thiostrepton NR3C1 None=None(uM) D4 PubChem thiostrepton PPARG Ratio Potency (uM)=4.06451(uM) D4 PubChem thiostrepton TDP1 Potency=4.1095(uM) D4 PubChem thiostrepton TDP1 Potency=5.0807(uM) D4 PubChem thiostrepton TDP1 Potency=5.1735(uM) D4 PubChem thiostrepton TDP1 Potency=7.1767(uM) D4 PubChem