Drug Gene Type Source sulfinpyrazone ABCB11 Text_Mining(decreases(reaction)) CTD sulfinpyrazone ABCB11 Text_Mining(increases(transport)) CTD sulfinpyrazone ABCB11 Text_Mining(decreases(activity)) CTD sulfinpyrazone ABCC1 Text_Mining(decreases(activity)) CTD sulfinpyrazone ABCC2 Text_Mining(decreases(activity)) CTD sulfinpyrazone CYP2B6 Text_Mining(increases(expression)) CTD sulfinpyrazone CYP2C8 Text_Mining(decreases(activity)) CTD sulfinpyrazone CYP2C9 Text_Mining(affects(metabolic processing)) CTD sulfinpyrazone CYP2C9 Text_Mining(decreases(reaction)) CTD sulfinpyrazone CYP3A4 Text_Mining(increases(activity)) CTD sulfinpyrazone CYP3A4 Text_Mining(increases(expression)) CTD sulfinpyrazone GSTM1 Text_Mining(decreases(reaction)) CTD sulfinpyrazone GSTM1 Text_Mining(decreases(response to substance)) CTD sulfinpyrazone GSTP1 Text_Mining(decreases(reaction)) CTD sulfinpyrazone GSTP1 Text_Mining(decreases(response to substance)) CTD sulfinpyrazone NR1I2 Text_Mining(affects(binding)) CTD sulfinpyrazone NR1I2 Text_Mining(increases(activity)) CTD sulfinpyrazone SLC22A12 Text_Mining(decreases(reaction)) CTD sulfinpyrazone SLC22A12 Text_Mining(increases(uptake)) CTD sulfinpyrazone ABCB1 None=None(uM) D4 PubChem sulfinpyrazone ALDH1A1 Potency=0.7943(uM) D4 PubChem sulfinpyrazone ALDH1A1 Potency=794.3(nM) D4 ChEMBL sulfinpyrazone CYP3A4 Potency=12.5893(uM) D4 PubChem sulfinpyrazone CYP3A4 Potency=12589.3(nM) D4 ChEMBL sulfinpyrazone EHMT2 Potency=7.0795(uM) D4 PubChem sulfinpyrazone EHMT2 Potency=7079.5(nM) D4 ChEMBL sulfinpyrazone FPR1 IC50_MICROM=14.4(uM) D4 PubChem sulfinpyrazone FPR1 None=None(uM) D4 PubChem sulfinpyrazone HPGD Potency=10.0(uM) D4 PubChem sulfinpyrazone HPGD Potency=12.5893(uM) D4 PubChem sulfinpyrazone HPGD Potency=22.3872(uM) D4 PubChem sulfinpyrazone HPGD Potency=12589.3(nM) D4 ChEMBL sulfinpyrazone HPGD Potency=22387.2(nM) D4 ChEMBL sulfinpyrazone HPGD Potency=10000.0(nM) D4 ChEMBL sulfinpyrazone ITGA4 None=None(uM) D4 PubChem sulfinpyrazone KDM4E Potency=17782.8(nM) D4 ChEMBL sulfinpyrazone PRMT1 None=None(uM) D4 PubChem sulfinpyrazone VDR Potency=28.1838(uM) D4 PubChem