Drug Gene Type Source Rifampicin AADAC Text_Mining(affects(reaction)) CTD Rifampicin AADAC Text_Mining(increases(expression)) CTD Rifampicin AADAC Text_Mining(decreases(acetylation)) CTD Rifampicin AADAC Text_Mining(increases(hydrolysis)) CTD Rifampicin AADAC Text_Mining(decreases(reaction)) CTD Rifampicin ABCA1 Text_Mining(decreases(expression)) CTD Rifampicin ABCA1 Text_Mining(increases(expression)) CTD Rifampicin ABCB1 Text_Mining(decreases(reaction)) CTD Rifampicin ABCB1 Text_Mining(increases(expression)) CTD Rifampicin ABCB1 Text_Mining(increases(reaction)) CTD Rifampicin ABCB1 Text_Mining(affects(activity)) CTD Rifampicin ABCB1 Text_Mining(affects(binding)) CTD Rifampicin ABCB1 Text_Mining(decreases(uptake)) CTD Rifampicin ABCB1 Text_Mining(increases(activity)) CTD Rifampicin ABCB11 Text_Mining(decreases(reaction)) CTD Rifampicin ABCB11 Text_Mining(increases(transport)) CTD Rifampicin ABCB11 Text_Mining(decreases(activity)) CTD Rifampicin ABCB11 Text_Mining(decreases(expression)) CTD Rifampicin ABCC1 Text_Mining(increases(expression)) CTD Rifampicin ABCC2 Text_Mining(affects(export)) CTD Rifampicin ABCC2 Text_Mining(affects(cotreatment)) CTD Rifampicin ABCC2 Text_Mining(increases(expression)) CTD Rifampicin ABCC3 Text_Mining(affects(cotreatment)) CTD Rifampicin ABCC3 Text_Mining(increases(expression)) CTD Rifampicin ABCC3 Text_Mining(decreases(reaction)) CTD Rifampicin ABCC3 Text_Mining(increases(activity)) CTD Rifampicin ABCG1 Text_Mining(increases(expression)) CTD Rifampicin ABCG2 Text_Mining(increases(expression)) CTD Rifampicin ADH1C Text_Mining(increases(expression)) CTD Rifampicin AHR Text_Mining(affects(cotreatment)) CTD Rifampicin AHR Text_Mining(decreases(expression)) CTD Rifampicin AHR Text_Mining(increases(expression)) CTD Rifampicin ANGPTL4 Text_Mining(affects(cotreatment)) CTD Rifampicin ANGPTL4 Text_Mining(increases(expression)) CTD Rifampicin AQP3 Text_Mining(affects(cotreatment)) CTD Rifampicin AQP3 Text_Mining(increases(expression)) CTD Rifampicin BAX Text_Mining(decreases(expression)) CTD Rifampicin BCL2 Text_Mining(increases(expression)) CTD Rifampicin BCL2L1 Text_Mining(increases(expression)) CTD Rifampicin BHLHE40 Text_Mining(affects(cotreatment)) CTD Rifampicin BHLHE40 Text_Mining(increases(expression)) CTD Rifampicin BMP4 Text_Mining(affects(cotreatment)) CTD Rifampicin BMP4 Text_Mining(increases(expression)) CTD Rifampicin CASP3 Text_Mining(decreases(reaction)) CTD Rifampicin CASP3 Text_Mining(increases(activity)) CTD Rifampicin CASP8 Text_Mining(decreases(reaction)) CTD Rifampicin CASP8 Text_Mining(increases(activity)) CTD Rifampicin CCR6 Text_Mining(affects(cotreatment)) CTD Rifampicin CCR6 Text_Mining(increases(expression)) CTD Rifampicin CCR7 Text_Mining(affects(cotreatment)) CTD Rifampicin CCR7 Text_Mining(increases(expression)) CTD Rifampicin CDKN2B Text_Mining(affects(cotreatment)) CTD Rifampicin CDKN2B Text_Mining(increases(expression)) CTD Rifampicin CES1 Text_Mining(increases(expression)) CTD Rifampicin CES2 Text_Mining(decreases(reaction)) CTD Rifampicin CES2 Text_Mining(increases(expression)) CTD Rifampicin CES2 Text_Mining(increases(reaction)) CTD Rifampicin CFLAR Text_Mining(decreases(reaction)) CTD Rifampicin CFLAR Text_Mining(increases(expression)) CTD Rifampicin CRP Text_Mining(affects(cotreatment)) CTD Rifampicin CRP Text_Mining(increases(expression)) CTD Rifampicin CYP1A1 Text_Mining(affects(cotreatment)) CTD Rifampicin CYP1A1 Text_Mining(increases(expression)) CTD Rifampicin CYP1A1 Text_Mining(increases(activity)) CTD Rifampicin CYP1A1 Text_Mining(decreases(reaction)) CTD Rifampicin CYP1A2 Text_Mining(decreases(reaction)) CTD Rifampicin CYP1A2 Text_Mining(increases(activity)) CTD Rifampicin CYP1A2 Text_Mining(increases(expression)) CTD Rifampicin CYP24A1 Text_Mining(increases(expression)) CTD Rifampicin CYP24A1 Text_Mining(increases(reaction)) CTD Rifampicin CYP24A1 Text_Mining(affects(binding)) CTD Rifampicin CYP24A1 Text_Mining(increases(activity)) CTD Rifampicin CYP26A1 Text_Mining(affects(cotreatment)) CTD Rifampicin CYP26A1 Text_Mining(increases(expression)) CTD Rifampicin CYP27A1 Text_Mining(affects(binding)) CTD Rifampicin CYP27A1 Text_Mining(increases(reaction)) CTD Rifampicin CYP27A1 Text_Mining(increases(expression)) CTD Rifampicin CYP2A13 Text_Mining(decreases(expression)) CTD Rifampicin CYP2A13 Text_Mining(increases(expression)) CTD Rifampicin CYP2A6 Text_Mining(affects(binding)) CTD Rifampicin CYP2A6 Text_Mining(increases(reaction)) CTD Rifampicin CYP2A6 Text_Mining(increases(expression)) CTD Rifampicin CYP2B6 Text_Mining(affects(reaction)) CTD Rifampicin CYP2B6 Text_Mining(increases(expression)) CTD Rifampicin CYP2B6 Text_Mining(increases(reaction)) CTD Rifampicin CYP2B6 Text_Mining(decreases(reaction)) CTD Rifampicin CYP2B6 Text_Mining(increases(activity)) CTD Rifampicin CYP2B6 Text_Mining(affects(cotreatment)) CTD Rifampicin CYP2C18 Text_Mining(decreases(expression)) CTD Rifampicin CYP2C19 Text_Mining(increases(activity)) CTD Rifampicin CYP2C19 Text_Mining(increases(expression)) CTD Rifampicin CYP2C8 Text_Mining(affects(binding)) CTD Rifampicin CYP2C8 Text_Mining(increases(activity)) CTD Rifampicin CYP2C8 Text_Mining(increases(expression)) CTD Rifampicin CYP2C9 Text_Mining(affects(cotreatment)) CTD Rifampicin CYP2C9 Text_Mining(increases(expression)) CTD Rifampicin CYP2C9 Text_Mining(increases(reaction)) CTD Rifampicin CYP2C9 Text_Mining(affects(reaction)) CTD Rifampicin CYP2C9 Text_Mining(increases(activity)) CTD Rifampicin CYP2D6 Text_Mining(increases(expression)) CTD Rifampicin CYP2E1 Text_Mining(affects(cotreatment)) CTD Rifampicin CYP2E1 Text_Mining(increases(activity)) CTD Rifampicin CYP2E1 Text_Mining(increases(expression)) CTD Rifampicin CYP2E1 Text_Mining(decreases(expression)) CTD Rifampicin CYP2F1 Text_Mining(decreases(expression)) CTD Rifampicin CYP2S1 Text_Mining(affects(cotreatment)) CTD Rifampicin CYP2S1 Text_Mining(increases(expression)) CTD Rifampicin CYP3A Text_Mining(increases(expression)) CTD Rifampicin CYP3A4 Text_Mining(affects(reaction)) CTD Rifampicin CYP3A4 Text_Mining(increases(expression)) CTD Rifampicin CYP3A4 Text_Mining(decreases(reaction)) CTD Rifampicin CYP3A4 Text_Mining(increases(activity)) CTD Rifampicin CYP3A4 Text_Mining(increases(reaction)) CTD Rifampicin CYP3A4 Text_Mining(affects(cotreatment)) CTD Rifampicin CYP3A4 Text_Mining(decreases(expression)) CTD Rifampicin CYP3A4 Text_Mining(affects(activity)) CTD Rifampicin CYP3A4 Text_Mining(affects(binding)) CTD Rifampicin CYP3A4 Text_Mining(increases(metabolic processing)) CTD Rifampicin CYP3A5 Text_Mining(increases(expression)) CTD Rifampicin CYP3A7 Text_Mining(increases(expression)) CTD Rifampicin CYP7A1 Text_Mining(decreases(expression)) CTD Rifampicin CYP7A1 Text_Mining(increases(reaction)) CTD Rifampicin CYP8B1 Text_Mining(affects(cotreatment)) CTD Rifampicin CYP8B1 Text_Mining(decreases(expression)) CTD Rifampicin CYR61 Text_Mining(affects(cotreatment)) CTD Rifampicin CYR61 Text_Mining(increases(expression)) CTD Rifampicin DHCR24 Text_Mining(increases(activity)) CTD Rifampicin DHCR24 Text_Mining(increases(expression)) CTD Rifampicin EDN1 Text_Mining(affects(cotreatment)) CTD Rifampicin EDN1 Text_Mining(increases(expression)) CTD Rifampicin EGR1 Text_Mining(affects(cotreatment)) CTD Rifampicin EGR1 Text_Mining(increases(expression)) CTD Rifampicin EGR2 Text_Mining(affects(cotreatment)) CTD Rifampicin EGR2 Text_Mining(increases(expression)) CTD Rifampicin EGR4 Text_Mining(affects(cotreatment)) CTD Rifampicin EGR4 Text_Mining(increases(expression)) CTD Rifampicin EPAS1 Text_Mining(affects(cotreatment)) CTD Rifampicin EPAS1 Text_Mining(increases(expression)) CTD Rifampicin EPHX1 Text_Mining(increases(expression)) CTD Rifampicin FAS Text_Mining(decreases(reaction)) CTD Rifampicin FAS Text_Mining(increases(activity)) CTD Rifampicin FAS Text_Mining(increases(expression)) CTD Rifampicin FASLG Text_Mining(decreases(reaction)) CTD Rifampicin FASLG Text_Mining(increases(expression)) CTD Rifampicin FASLG Text_Mining(decreases(expression)) CTD Rifampicin FGF19 Text_Mining(affects(binding)) CTD Rifampicin FGF19 Text_Mining(increases(activity)) CTD Rifampicin FGF19 Text_Mining(increases(expression)) CTD Rifampicin FIGF Text_Mining(affects(cotreatment)) CTD Rifampicin FIGF Text_Mining(increases(expression)) CTD Rifampicin FOXA1 Text_Mining(affects(cotreatment)) CTD Rifampicin FOXA1 Text_Mining(decreases(expression)) CTD Rifampicin GADD45B Text_Mining(increases(expression)) CTD Rifampicin GADD45B Text_Mining(increases(reaction)) CTD Rifampicin GATA5 Text_Mining(affects(cotreatment)) CTD Rifampicin GATA5 Text_Mining(decreases(expression)) CTD Rifampicin GPT Text_Mining(affects(cotreatment)) CTD Rifampicin GPT Text_Mining(decreases(activity)) CTD Rifampicin GSTA1 Text_Mining(increases(expression)) CTD Rifampicin GSTP1 Text_Mining(affects(cotreatment)) CTD Rifampicin GSTP1 Text_Mining(increases(expression)) CTD Rifampicin GSTT1 Text_Mining(affects(cotreatment)) CTD Rifampicin GSTT1 Text_Mining(affects(response to substance)) CTD Rifampicin GSTT1 Text_Mining(increases(response to substance)) CTD Rifampicin HBEGF Text_Mining(affects(cotreatment)) CTD Rifampicin HBEGF Text_Mining(increases(expression)) CTD Rifampicin HDAC5 Text_Mining(affects(cotreatment)) CTD Rifampicin HDAC5 Text_Mining(decreases(expression)) CTD Rifampicin HEY1 Text_Mining(affects(cotreatment)) CTD Rifampicin HEY1 Text_Mining(increases(expression)) CTD Rifampicin HIF1A Text_Mining(affects(cotreatment)) CTD Rifampicin HIF1A Text_Mining(increases(expression)) CTD Rifampicin HMOX1 Text_Mining(increases(expression)) CTD Rifampicin HNF4A Text_Mining(affects(cotreatment)) CTD Rifampicin HNF4A Text_Mining(increases(expression)) CTD Rifampicin HNF4A Text_Mining(increases(reaction)) CTD Rifampicin HNF4A Text_Mining(decreases(expression)) CTD Rifampicin HNF4A Text_Mining(affects(binding)) CTD Rifampicin HNF4A Text_Mining(decreases(reaction)) CTD Rifampicin HNF4A Text_Mining(increases(activity)) CTD Rifampicin IGFBP1 Text_Mining(affects(cotreatment)) CTD Rifampicin IGFBP1 Text_Mining(increases(expression)) CTD Rifampicin IGFBP3 Text_Mining(affects(cotreatment)) CTD Rifampicin IGFBP3 Text_Mining(increases(expression)) CTD Rifampicin IGFBP4 Text_Mining(affects(cotreatment)) CTD Rifampicin IGFBP4 Text_Mining(increases(expression)) CTD Rifampicin IL6 Text_Mining(decreases(expression)) CTD Rifampicin JUN Text_Mining(affects(cotreatment)) CTD Rifampicin JUN Text_Mining(increases(expression)) CTD Rifampicin KLF2 Text_Mining(affects(cotreatment)) CTD Rifampicin KLF2 Text_Mining(increases(expression)) CTD Rifampicin KLF5 Text_Mining(affects(cotreatment)) CTD Rifampicin KLF5 Text_Mining(increases(expression)) CTD Rifampicin KLF6 Text_Mining(affects(cotreatment)) CTD Rifampicin KLF6 Text_Mining(increases(expression)) CTD Rifampicin LEFTY1 Text_Mining(affects(cotreatment)) CTD Rifampicin LEFTY1 Text_Mining(increases(expression)) CTD Rifampicin MAFF Text_Mining(affects(cotreatment)) CTD Rifampicin MAFF Text_Mining(increases(expression)) CTD Rifampicin MAPKAPK2 Text_Mining(increases(phosphorylation)) CTD Rifampicin MED1 Text_Mining(affects(binding)) CTD Rifampicin MED1 Text_Mining(increases(activity)) CTD Rifampicin MED1 Text_Mining(increases(reaction)) CTD Rifampicin ABCC5 Text_Mining(increases(expression)) CTD Rifampicin NCOA1 Text_Mining(affects(binding)) CTD Rifampicin NCOA1 Text_Mining(increases(activity)) CTD Rifampicin NCOA1 Text_Mining(increases(reaction)) CTD Rifampicin NCOA1 Text_Mining(increases(expression)) CTD Rifampicin NCOA2 Text_Mining(affects(binding)) CTD Rifampicin NCOA2 Text_Mining(increases(reaction)) CTD Rifampicin NCOA6 Text_Mining(affects(cotreatment)) CTD Rifampicin NCOA6 Text_Mining(increases(expression)) CTD Rifampicin NCOA6 Text_Mining(increases(reaction)) CTD Rifampicin NCOA6 Text_Mining(affects(binding)) CTD Rifampicin NCOR1 Text_Mining(affects(binding)) CTD Rifampicin NCOR1 Text_Mining(decreases(activity)) CTD Rifampicin NCOR1 Text_Mining(decreases(reaction)) CTD Rifampicin NCOR2 Text_Mining(affects(binding)) CTD Rifampicin NCOR2 Text_Mining(decreases(activity)) CTD Rifampicin NCOR2 Text_Mining(decreases(reaction)) CTD Rifampicin NPAS1 Text_Mining(affects(cotreatment)) CTD Rifampicin NPAS1 Text_Mining(increases(expression)) CTD Rifampicin NPPB Text_Mining(affects(cotreatment)) CTD Rifampicin NPPB Text_Mining(increases(expression)) CTD Rifampicin NR0B2 Text_Mining(increases(expression)) CTD Rifampicin NR1H3 Text_Mining(decreases(reaction)) CTD Rifampicin NR1H3 Text_Mining(increases(expression)) CTD Rifampicin NR1I2 Text_Mining(affects(cotreatment)) CTD Rifampicin NR1I2 Text_Mining(increases(activity)) CTD Rifampicin NR1I2 Text_Mining(increases(reaction)) CTD Rifampicin NR1I2 Text_Mining(decreases(reaction)) CTD Rifampicin NR1I2 Text_Mining(affects(reaction)) CTD Rifampicin NR1I2 Text_Mining(increases(expression)) CTD Rifampicin NR1I2 Text_Mining(affects(response to substance)) CTD Rifampicin NR1I2 Text_Mining(decreases(expression)) CTD Rifampicin NR1I2 Text_Mining(increases(abundance)) CTD Rifampicin NR1I2 Text_Mining(affects(binding)) CTD Rifampicin NR1I2 Text_Mining(decreases(uptake)) CTD Rifampicin NR1I2 Text_Mining(decreases(activity)) CTD Rifampicin NR1I3 Text_Mining(affects(cotreatment)) CTD Rifampicin NR1I3 Text_Mining(increases(expression)) CTD Rifampicin NR3C1 Text_Mining(affects(reaction)) CTD Rifampicin NR3C1 Text_Mining(increases(expression)) CTD Rifampicin NR3C1 Text_Mining(increases(reaction)) CTD Rifampicin PIP4K2A Text_Mining(affects(cotreatment)) CTD Rifampicin PIP4K2A Text_Mining(increases(expression)) CTD Rifampicin POU2F1 Text_Mining(decreases(expression)) CTD Rifampicin PPARA Text_Mining(affects(cotreatment)) CTD Rifampicin PPARA Text_Mining(decreases(expression)) CTD Rifampicin PPARGC1A Text_Mining(affects(binding)) CTD Rifampicin PPARGC1A Text_Mining(increases(reaction)) CTD Rifampicin RXRA Text_Mining(affects(cotreatment)) CTD Rifampicin RXRA Text_Mining(increases(activity)) CTD Rifampicin RXRA Text_Mining(increases(reaction)) CTD Rifampicin RXRA Text_Mining(decreases(reaction)) CTD Rifampicin RXRA Text_Mining(decreases(expression)) CTD Rifampicin RXRA Text_Mining(affects(binding)) CTD Rifampicin RXRA Text_Mining(increases(expression)) CTD Rifampicin SCARB1 Text_Mining(decreases(expression)) CTD Rifampicin SERPINA4 Text_Mining(affects(cotreatment)) CTD Rifampicin SERPINA4 Text_Mining(decreases(expression)) CTD Rifampicin SERPINB1 Text_Mining(affects(cotreatment)) CTD Rifampicin SERPINB1 Text_Mining(increases(expression)) CTD Rifampicin SERPINB8 Text_Mining(affects(cotreatment)) CTD Rifampicin SERPINB8 Text_Mining(increases(expression)) CTD Rifampicin SERPINB9 Text_Mining(affects(cotreatment)) CTD Rifampicin SERPINB9 Text_Mining(increases(expression)) CTD Rifampicin SERPINE1 Text_Mining(affects(cotreatment)) CTD Rifampicin SERPINE1 Text_Mining(increases(expression)) CTD Rifampicin SGK2 Text_Mining(affects(cotreatment)) CTD Rifampicin SGK2 Text_Mining(increases(expression)) CTD Rifampicin SLC10A1 Text_Mining(decreases(expression)) CTD Rifampicin SLC22A7 Text_Mining(decreases(expression)) CTD Rifampicin SLCO1B1 Text_Mining(decreases(reaction)) CTD Rifampicin SLCO1B1 Text_Mining(increases(response to substance)) CTD Rifampicin SLCO1B1 Text_Mining(increases(uptake)) CTD Rifampicin SLCO1B1 Text_Mining(decreases(activity)) CTD Rifampicin SLCO1B1 Text_Mining(increases(expression)) CTD Rifampicin SLCO1B1 Text_Mining(affects(uptake)) CTD Rifampicin SLCO1B3 Text_Mining(decreases(reaction)) CTD Rifampicin SLCO1B3 Text_Mining(increases(import)) CTD Rifampicin SLCO1B3 Text_Mining(increases(uptake)) CTD Rifampicin SLCO2A1 Text_Mining(decreases(reaction)) CTD Rifampicin SLCO2A1 Text_Mining(increases(expression)) CTD Rifampicin SLCO2B1 Text_Mining(decreases(reaction)) CTD Rifampicin SLCO2B1 Text_Mining(increases(uptake)) CTD Rifampicin SMAD9 Text_Mining(affects(cotreatment)) CTD Rifampicin SMAD9 Text_Mining(increases(expression)) CTD Rifampicin SOCS3 Text_Mining(affects(cotreatment)) CTD Rifampicin SOCS3 Text_Mining(increases(expression)) CTD Rifampicin STAT5A Text_Mining(affects(cotreatment)) CTD Rifampicin STAT5A Text_Mining(decreases(expression)) CTD Rifampicin SULT1E1 Text_Mining(affects(cotreatment)) CTD Rifampicin SULT1E1 Text_Mining(decreases(expression)) CTD Rifampicin SULT1E1 Text_Mining(affects(binding)) CTD Rifampicin SULT1E1 Text_Mining(decreases(reaction)) CTD Rifampicin SULT1E1 Text_Mining(increases(activity)) CTD Rifampicin TNF Text_Mining(decreases(expression)) CTD Rifampicin UGDH Text_Mining(affects(cotreatment)) CTD Rifampicin UGDH Text_Mining(decreases(expression)) CTD Rifampicin UGDH Text_Mining(increases(expression)) CTD Rifampicin UGT1A1 Text_Mining(affects(expression)) CTD Rifampicin UGT1A1 Text_Mining(affects(cotreatment)) CTD Rifampicin UGT1A1 Text_Mining(increases(expression)) CTD Rifampicin UGT1A6 Text_Mining(increases(expression)) CTD Rifampicin XIAP Text_Mining(increases(expression)) CTD Rifampicin ABCB1 None=None(uM) D4 PubChem Rifampicin AR Ratio Potency (uM)=19.7221(uM) D4 PubChem Rifampicin AR Ratio Potency (uM)=22.1476(uM) D4 PubChem Rifampicin AR Potency-Replicate_1=23.9145(uM) D4 PubChem Rifampicin AR Potency-Replicate_1=31.2574(uM) D4 PubChem Rifampicin AR Ratio Potency (uM)=36.2333(uM) D4 PubChem Rifampicin AR Potency-Replicate_1=39.1238(uM) D4 PubChem Rifampicin CFTR None=None(uM) D4 PubChem Rifampicin CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL Rifampicin CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL Rifampicin CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL Rifampicin CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL Rifampicin CYP3A4 Inhibition=None(Unspecified) D4 ChEMBL Rifampicin EHMT2 Potency=19.9526(uM) D4 PubChem Rifampicin GSTO1 None=None(uM) D4 PubChem Rifampicin MLLT3 None=None(uM) D4 PubChem Rifampicin NFE2L2 Potency=4.1095(uM) D4 PubChem Rifampicin NFE2L2 Potency=4.6109(uM) D4 PubChem Rifampicin NFE2L2 Potency=54.4827(uM) D4 PubChem Rifampicin NR1I2 Activity=None(Unspecified) D4 ChEMBL Rifampicin NR1I2 Potency-Replicate_1=5.6234(uM) D4 PubChem Rifampicin NR3C1 Potency-Replicate_1=21.3138(uM) D4 PubChem Rifampicin NR3C1 None=None(uM) D4 PubChem Rifampicin TDP1 Potency=18.8375(uM) D4 PubChem Rifampicin TDP1 Potency=23.715(uM) D4 PubChem