Drug Gene Type Source pyrimethamine CASP3 Text_Mining(increases(activity)) CTD pyrimethamine CASP3 Text_Mining(increases(reaction)) CTD pyrimethamine CASP3 Text_Mining(affects(cotreatment)) CTD pyrimethamine CASP3 Text_Mining(increases(cleavage)) CTD pyrimethamine CASP7 Text_Mining(increases(activity)) CTD pyrimethamine CASP7 Text_Mining(increases(reaction)) CTD pyrimethamine CASP8 Text_Mining(increases(activity)) CTD pyrimethamine CASP9 Text_Mining(increases(activity)) CTD pyrimethamine CTSB Text_Mining(increases(activity)) CTD pyrimethamine CYP2C9 Text_Mining(decreases(activity)) CTD pyrimethamine FOS Text_Mining(increases(expression)) CTD pyrimethamine GSTP1 Text_Mining(affects(metabolic processing)) CTD pyrimethamine GSTP1 Text_Mining(decreases(activity)) CTD pyrimethamine GSTP1 Text_Mining(decreases(reaction)) CTD pyrimethamine H2AFX Text_Mining(increases(phosphorylation)) CTD pyrimethamine HEXB Text_Mining(affects(binding)) CTD pyrimethamine SLC46A1 Text_Mining(decreases(activity)) CTD pyrimethamine AR Potency-Replicate_1=4.2163(uM) D4 PubChem pyrimethamine AR Ratio Potency (uM)=5.35378(uM) D4 PubChem pyrimethamine AR Potency-Replicate_1=39.4861(uM) D4 PubChem pyrimethamine AR Potency-Replicate_1=49.2994(uM) D4 PubChem pyrimethamine AR AR Potency (uM)=57.4789(uM) D4 PubChem pyrimethamine CYP19A1 Potency-Replicate_1=55.3148(uM) D4 PubChem pyrimethamine CYP1A2 None=None(uM) D4 PubChem pyrimethamine EPAS1 None=None(uM) D4 PubChem pyrimethamine ESR1 Potency-Replicate_1=23.7101(uM) D4 PubChem pyrimethamine ESR1 ER Potency (uM)=26.6032(uM) D4 PubChem pyrimethamine ESR1 None=None(uM) D4 PubChem pyrimethamine HIF1A None=None(uM) D4 PubChem pyrimethamine IDH1 Potency=0.8199(uM) D4 PubChem pyrimethamine IDH1 Potency=3.1623(uM) D4 PubChem pyrimethamine JAK2 None=None(uM) D4 PubChem pyrimethamine MDM2 None=None(uM) D4 PubChem pyrimethamine MDM4 None=None(uM) D4 PubChem pyrimethamine MRGPRX1 None=None(uM) D4 PubChem pyrimethamine NFE2L2 Ratio Potency (uM)=8.1191(uM) D4 PubChem pyrimethamine NFKB1 None=None(uM) D4 PubChem pyrimethamine RELA None=None(uM) D4 PubChem pyrimethamine TDP1 Potency=0.2818(uM) D4 PubChem pyrimethamine TDP1 Potency=0.4611(uM) D4 PubChem pyrimethamine TDP1 Potency=0.5309(uM) D4 PubChem pyrimethamine TDP1 Potency=0.6513(uM) D4 PubChem pyrimethamine TDP1 Potency=0.7943(uM) D4 PubChem pyrimethamine TDP1 Potency=0.9441(uM) D4 PubChem pyrimethamine TDP1 Potency=1.2995(uM) D4 PubChem pyrimethamine TDP1 Potency=3.1623(uM) D4 PubChem pyrimethamine TNFRSF10B None=None(uM) D4 PubChem