Drug Gene Type Source nimesulide ABCB1 Text_Mining(decreases(expression)) CTD nimesulide ABCB1 Text_Mining(increases(expression)) CTD nimesulide ABCC1 Text_Mining(increases(expression)) CTD nimesulide ABCG2 Text_Mining(decreases(activity)) CTD nimesulide ABCG2 Text_Mining(decreases(expression)) CTD nimesulide ANGPTL4 Text_Mining(increases(expression)) CTD nimesulide AREG Text_Mining(decreases(reaction)) CTD nimesulide AREG Text_Mining(increases(expression)) CTD nimesulide BAK1 Text_Mining(decreases(reaction)) CTD nimesulide BAK1 Text_Mining(increases(activity)) CTD nimesulide BAX Text_Mining(affects(localization)) CTD nimesulide BAX Text_Mining(decreases(reaction)) CTD nimesulide BAX Text_Mining(increases(activity)) CTD nimesulide BCL2 Text_Mining(decreases(expression)) CTD nimesulide BID Text_Mining(decreases(reaction)) CTD nimesulide BID Text_Mining(increases(activity)) CTD nimesulide BID Text_Mining(increases(cleavage)) CTD nimesulide BIRC5 Text_Mining(decreases(expression)) CTD nimesulide C1QB Text_Mining(decreases(reaction)) CTD nimesulide C1QB Text_Mining(increases(expression)) CTD nimesulide CASP3 Text_Mining(decreases(reaction)) CTD nimesulide CASP3 Text_Mining(increases(activity)) CTD nimesulide CASP3 Text_Mining(increases(cleavage)) CTD nimesulide CASP3 Text_Mining(increases(expression)) CTD nimesulide CASP8 Text_Mining(decreases(reaction)) CTD nimesulide CASP8 Text_Mining(increases(activity)) CTD nimesulide CASP8 Text_Mining(increases(cleavage)) CTD nimesulide CASP9 Text_Mining(decreases(reaction)) CTD nimesulide CASP9 Text_Mining(increases(activity)) CTD nimesulide CASP9 Text_Mining(increases(cleavage)) CTD nimesulide CAT Text_Mining(decreases(expression)) CTD nimesulide CAV1 Text_Mining(increases(expression)) CTD nimesulide CCL2 Text_Mining(decreases(expression)) CTD nimesulide CCND1 Text_Mining(affects(cotreatment)) CTD nimesulide CCND1 Text_Mining(decreases(reaction)) CTD nimesulide CCND1 Text_Mining(increases(expression)) CTD nimesulide CDKN1A Text_Mining(decreases(reaction)) CTD nimesulide CDKN1A Text_Mining(increases(expression)) CTD nimesulide CDKN1B Text_Mining(increases(expression)) CTD nimesulide CDKN2C Text_Mining(decreases(expression)) CTD nimesulide CDKN2C Text_Mining(decreases(reaction)) CTD nimesulide CTNNB1 Text_Mining(affects(localization)) CTD nimesulide CXCL8 Text_Mining(affects(expression)) CTD nimesulide CXCL8 Text_Mining(decreases(reaction)) CTD nimesulide CXCL8 Text_Mining(increases(expression)) CTD nimesulide CYP19A1 Text_Mining(decreases(activity)) CTD nimesulide CYP19A1 Text_Mining(decreases(expression)) CTD nimesulide EDNRB Text_Mining(decreases(reaction)) CTD nimesulide EDNRB Text_Mining(increases(activity)) CTD nimesulide EREG Text_Mining(decreases(reaction)) CTD nimesulide EREG Text_Mining(increases(expression)) CTD nimesulide F2 Text_Mining(decreases(activity)) CTD nimesulide GPX1 Text_Mining(decreases(expression)) CTD nimesulide GSK3B Text_Mining(decreases(activity)) CTD nimesulide H2AFX Text_Mining(decreases(reaction)) CTD nimesulide H2AFX Text_Mining(increases(phosphorylation)) CTD nimesulide HRAS Text_Mining(affects(cotreatment)) CTD nimesulide HRAS Text_Mining(decreases(reaction)) CTD nimesulide HRAS Text_Mining(increases(expression)) CTD nimesulide ICAM1 Text_Mining(affects(cotreatment)) CTD nimesulide ICAM1 Text_Mining(decreases(expression)) CTD nimesulide IFNG Text_Mining(affects(cotreatment)) CTD nimesulide IFNG Text_Mining(increases(response to substance)) CTD nimesulide IL10 Text_Mining(affects(cotreatment)) CTD nimesulide IL10 Text_Mining(decreases(expression)) CTD nimesulide IL1A Text_Mining(affects(cotreatment)) CTD nimesulide IL1A Text_Mining(increases(response to substance)) CTD nimesulide IL1B Text_Mining(affects(cotreatment)) CTD nimesulide IL1B Text_Mining(decreases(expression)) CTD nimesulide IL1B Text_Mining(decreases(reaction)) CTD nimesulide IL1B Text_Mining(increases(activity)) CTD nimesulide IL1B Text_Mining(increases(expression)) CTD nimesulide IL6 Text_Mining(decreases(reaction)) CTD nimesulide IL6 Text_Mining(increases(expression)) CTD nimesulide ITGA5 Text_Mining(decreases(expression)) CTD nimesulide ITGA5 Text_Mining(decreases(reaction)) CTD nimesulide JUN Text_Mining(decreases(expression)) CTD nimesulide KCNH2 Text_Mining(decreases(activity)) CTD nimesulide LHB Text_Mining(decreases(reaction)) CTD nimesulide LHB Text_Mining(increases(expression)) CTD nimesulide MAPK1 Text_Mining(decreases(reaction)) CTD nimesulide MAPK1 Text_Mining(increases(phosphorylation)) CTD nimesulide MAPK1 Text_Mining(decreases(expression)) CTD nimesulide MAPK3 Text_Mining(decreases(reaction)) CTD nimesulide MAPK3 Text_Mining(increases(phosphorylation)) CTD nimesulide MAPK3 Text_Mining(decreases(expression)) CTD nimesulide MAPK9 Text_Mining(decreases(phosphorylation)) CTD nimesulide MMP9 Text_Mining(decreases(expression)) CTD nimesulide MPO Text_Mining(affects(activity)) CTD nimesulide MPO Text_Mining(affects(cotreatment)) CTD nimesulide MPO Text_Mining(increases(oxidation)) CTD nimesulide MPO Text_Mining(increases(chemical synthesis)) CTD nimesulide NFE2L2 Text_Mining(affects(localization)) CTD nimesulide NFE2L2 Text_Mining(affects(reaction)) CTD nimesulide PARP1 Text_Mining(increases(cleavage)) CTD nimesulide PAWR Text_Mining(increases(expression)) CTD nimesulide PLIN2 Text_Mining(increases(expression)) CTD nimesulide PPARA Text_Mining(decreases(reaction)) CTD nimesulide PPARA Text_Mining(increases(expression)) CTD nimesulide PPARA Text_Mining(increases(reaction)) CTD nimesulide PPARA Text_Mining(decreases(expression)) CTD nimesulide PPARD Text_Mining(increases(expression)) CTD nimesulide PPARG Text_Mining(affects(binding)) CTD nimesulide PPARG Text_Mining(decreases(reaction)) CTD nimesulide PPARG Text_Mining(increases(reaction)) CTD nimesulide PPARG Text_Mining(affects(cotreatment)) CTD nimesulide PPARG Text_Mining(increases(expression)) CTD nimesulide PPARG Text_Mining(decreases(expression)) CTD nimesulide PSEN2 Text_Mining(decreases(activity)) CTD nimesulide PTGS1 Text_Mining(increases(expression)) CTD nimesulide PTGS2 Text_Mining(affects(expression)) CTD nimesulide PTGS2 Text_Mining(affects(cotreatment)) CTD nimesulide PTGS2 Text_Mining(decreases(reaction)) CTD nimesulide PTGS2 Text_Mining(increases(expression)) CTD nimesulide PTGS2 Text_Mining(increases(reaction)) CTD nimesulide PTGS2 Text_Mining(affects(abundance)) CTD nimesulide PTGS2 Text_Mining(affects(chemical synthesis)) CTD nimesulide PTGS2 Text_Mining(increases(metabolic processing)) CTD nimesulide PTGS2 Text_Mining(decreases(expression)) CTD nimesulide PTGS2 Text_Mining(decreases(activity)) CTD nimesulide PTGS2 Text_Mining(decreases(abundance)) CTD nimesulide SELE Text_Mining(affects(cotreatment)) CTD nimesulide SELE Text_Mining(decreases(expression)) CTD nimesulide SELL Text_Mining(decreases(expression)) CTD nimesulide SOD2 Text_Mining(decreases(expression)) CTD nimesulide SP1 Text_Mining(increases(expression)) CTD nimesulide SULT1A1 Text_Mining(decreases(activity)) CTD nimesulide TNF Text_Mining(affects(cotreatment)) CTD nimesulide TNF Text_Mining(increases(response to substance)) CTD nimesulide TNF Text_Mining(decreases(expression)) CTD nimesulide VCAM1 Text_Mining(affects(cotreatment)) CTD nimesulide VCAM1 Text_Mining(decreases(expression)) CTD nimesulide VEGFA Text_Mining(affects(secretion)) CTD nimesulide VEGFA Text_Mining(affects(cotreatment)) CTD nimesulide VEGFA Text_Mining(decreases(expression)) CTD nimesulide VEGFA Text_Mining(increases(expression)) CTD nimesulide VEGFC Text_Mining(decreases(expression)) CTD nimesulide ABCB1 None=None(uM) D4 PubChem nimesulide APEX1 Potency=39810.7(nM) D4 ChEMBL nimesulide CFTR None=None(uM) D4 PubChem nimesulide CYP1A2 None=None(uM) D4 PubChem nimesulide CYP1A2 Inhibition=None(Unspecified) D4 ChEMBL nimesulide CYP2C19 Inhibition=None(Unspecified) D4 ChEMBL nimesulide CYP2C9 Potency=3.1623(uM) D4 PubChem nimesulide CYP2C9 Potency=10.0(uM) D4 PubChem nimesulide CYP2C9 None=None(uM) D4 PubChem nimesulide CYP2C9 Inhibition=None(Unspecified) D4 ChEMBL nimesulide CYP2C9 Potency=3162.3(nM) D4 ChEMBL nimesulide CYP2C9 Potency=10000.0(nM) D4 ChEMBL nimesulide CYP2C9 AC50=3162.28(nM) D4 ChEMBL nimesulide CYP2D6 Inhibition=None(Unspecified) D4 ChEMBL nimesulide EHMT2 Potency=31.6228(uM) D4 PubChem nimesulide PPARG None=None(uM) D4 PubChem nimesulide TDP1 Potency=8912.5(nM) D4 ChEMBL