Drug Gene Type Source phloretin CYP1A1 Text_Mining(decreases(reaction)) CTD phloretin CYP1A1 Text_Mining(increases(activity)) CTD phloretin CYP1A1 Text_Mining(increases(expression)) CTD phloretin ESR1 Text_Mining(affects(binding)) CTD phloretin ESR1 Text_Mining(increases(activity)) CTD phloretin ESR2 Text_Mining(affects(binding)) CTD phloretin ESR2 Text_Mining(increases(activity)) CTD phloretin GSK3B Text_Mining(decreases(activity)) CTD phloretin IL1B Text_Mining(decreases(reaction)) CTD phloretin IL1B Text_Mining(increases(secretion)) CTD phloretin INS Text_Mining(decreases(reaction)) CTD phloretin INS Text_Mining(increases(activity)) CTD phloretin INS Text_Mining(increases(secretion)) CTD phloretin NOS3 Text_Mining(decreases(reaction)) CTD phloretin NOS3 Text_Mining(increases(expression)) CTD phloretin NOS3 Text_Mining(decreases(expression)) CTD phloretin SLC2A1 Text_Mining(affects(transport)) CTD phloretin SLC2A1 Text_Mining(decreases(reaction)) CTD phloretin SLC2A1 Text_Mining(decreases(activity)) CTD phloretin SLC9A1 Text_Mining(affects(cotreatment)) CTD phloretin SLC9A1 Text_Mining(affects(transport)) CTD phloretin SLC9A1 Text_Mining(decreases(reaction)) CTD phloretin SLC9A1 Text_Mining(decreases(activity)) CTD phloretin SLC9B2 Text_Mining(decreases(activity)) CTD phloretin UGT1A10 Text_Mining(increases(glucuronidation)) CTD phloretin UGT1A7 Text_Mining(increases(glucuronidation)) CTD phloretin UGT1A8 Text_Mining(increases(glucuronidation)) CTD phloretin AR Ratio Potency (uM)=48.2028(uM) D4 PubChem phloretin ARSA Potency=2.6855(uM) D4 PubChem phloretin ATM Potency=28.1838(uM) D4 PubChem phloretin ATM Potency=28183.8(nM) D4 ChEMBL phloretin CYP1A2 None=None(uM) D4 PubChem phloretin CYP1A2 AC50=6309.57(nM) D4 ChEMBL phloretin CYP2C19 Potency=3.9811(uM) D4 PubChem phloretin CYP2C19 Potency=3981.1(nM) D4 ChEMBL phloretin CYP2C9 Potency=2.5119(uM) D4 PubChem phloretin CYP2C9 Potency=12.5893(uM) D4 PubChem phloretin CYP2C9 None=None(uM) D4 PubChem phloretin CYP2C9 AC50=12589.2(nM) D4 ChEMBL phloretin CYP2C9 Potency=2511.9(nM) D4 ChEMBL phloretin CYP2C9 Potency=12589.3(nM) D4 ChEMBL phloretin CYP3A4 Potency=1.9953(uM) D4 PubChem phloretin CYP3A4 Potency=10.0(uM) D4 PubChem phloretin CYP3A4 Potency=15.8489(uM) D4 PubChem phloretin CYP3A4 None=None(uM) D4 PubChem phloretin CYP3A4 AC50=10000.0(nM) D4 ChEMBL phloretin CYP3A4 Potency=10000.0(nM) D4 ChEMBL phloretin CYP3A4 Potency=1995.3(nM) D4 ChEMBL phloretin CYP3A4 Potency=15848.9(nM) D4 ChEMBL phloretin ESR1 Potency-Replicate_1=4.9646(uM) D4 PubChem phloretin ESR1 Potency-Replicate_1=14.1169(uM) D4 PubChem phloretin ESR1 Ratio Potency (uM)=19.1784(uM) D4 PubChem phloretin FGF22 AbsAC1_uM=1.74(uM) D4 PubChem phloretin FGF22 AbsAC0.54_uM=2.95(uM) D4 PubChem phloretin FGF22 None=None(uM) D4 PubChem phloretin GAA Potency=31.3814(uM) D4 PubChem phloretin GAA Potency=31381.4(nM) D4 ChEMBL phloretin GBA Potency=17.7828(uM) D4 PubChem phloretin GBA Potency=17782.8(nM) D4 ChEMBL phloretin GSTO1 None=None(uM) D4 PubChem phloretin HPGD Potency=25.1189(uM) D4 PubChem phloretin HPGD Potency=35.4813(uM) D4 PubChem phloretin HPGD Potency=25118.9(nM) D4 ChEMBL phloretin HPGD Potency=35481.3(nM) D4 ChEMBL phloretin HSD17B10 Potency=25118.9(nM) D4 ChEMBL phloretin KDM4E Potency=31622.8(nM) D4 ChEMBL phloretin NFE2L2 Potency-Replicate_1=31.3246(uM) D4 PubChem phloretin NFE2L2 Ratio Potency (uM)=39.4353(uM) D4 PubChem phloretin PAFAH1B2 None=None(uM) D4 PubChem phloretin POLB Potency=7.0795(uM) D4 PubChem phloretin POLB Potency=7079.5(nM) D4 ChEMBL phloretin PPARG None=None(uM) D4 PubChem phloretin RECQL Potency=12589.3(nM) D4 ChEMBL phloretin RGS4 Potency=18.8876(uM) D4 PubChem phloretin STK33 EC50_uM=21.41(uM) D4 PubChem phloretin STK33 None=None(uM) D4 PubChem