Drug Gene Type Source NSC25485 A2M Text_Mining(affects(expression)) CTD NSC25485 ABCB1 Text_Mining(decreases(reaction)) CTD NSC25485 ABCB1 Text_Mining(increases(expression)) CTD NSC25485 ABCB1 Text_Mining(decreases(response to substance)) CTD NSC25485 ACAA2 Text_Mining(affects(expression)) CTD NSC25485 ACTA2 Text_Mining(affects(expression)) CTD NSC25485 ADH1C Text_Mining(affects(expression)) CTD NSC25485 ANXA1 Text_Mining(affects(expression)) CTD NSC25485 ANXA2 Text_Mining(affects(expression)) CTD NSC25485 ARAF Text_Mining(decreases(expression)) CTD NSC25485 ARIH1 Text_Mining(decreases(expression)) CTD NSC25485 ARPC5 Text_Mining(affects(expression)) CTD NSC25485 ARRB1 Text_Mining(increases(expression)) CTD NSC25485 ASAH1 Text_Mining(affects(expression)) CTD NSC25485 ATP12A Text_Mining(affects(cotreatment)) CTD NSC25485 ATP12A Text_Mining(decreases(reaction)) CTD NSC25485 ATP12A Text_Mining(increases(uptake)) CTD NSC25485 ATP1A1 Text_Mining(decreases(reaction)) CTD NSC25485 ATP1A1 Text_Mining(increases(expression)) CTD NSC25485 ATP1A1 Text_Mining(affects(binding)) CTD NSC25485 ATP1A2 Text_Mining(decreases(reaction)) CTD NSC25485 ATP1A2 Text_Mining(increases(expression)) CTD NSC25485 ATP1A2 Text_Mining(affects(binding)) CTD NSC25485 ATP1A3 Text_Mining(affects(binding)) CTD NSC25485 ATP1A3 Text_Mining(increases(expression)) CTD NSC25485 ATP4B Text_Mining(affects(cotreatment)) CTD NSC25485 ATP4B Text_Mining(decreases(reaction)) CTD NSC25485 ATP4B Text_Mining(increases(uptake)) CTD NSC25485 ATP5A1 Text_Mining(affects(expression)) CTD NSC25485 BAHD1 Text_Mining(decreases(expression)) CTD NSC25485 BAX Text_Mining(affects(localization)) CTD NSC25485 BAX Text_Mining(affects(binding)) CTD NSC25485 BAX Text_Mining(decreases(reaction)) CTD NSC25485 BAX Text_Mining(increases(expression)) CTD NSC25485 CALML5 Text_Mining(affects(expression)) CTD NSC25485 CANX Text_Mining(increases(expression)) CTD NSC25485 CASP3 Text_Mining(increases(activity)) CTD NSC25485 CASP3 Text_Mining(increases(expression)) CTD NSC25485 CCDC14 Text_Mining(decreases(expression)) CTD NSC25485 CCNA1 Text_Mining(decreases(expression)) CTD NSC25485 CCNA2 Text_Mining(decreases(expression)) CTD NSC25485 CDK2 Text_Mining(decreases(expression)) CTD NSC25485 CDKN1A Text_Mining(decreases(expression)) CTD NSC25485 CDKN1A Text_Mining(increases(expression)) CTD NSC25485 CLDN1 Text_Mining(decreases(expression)) CTD NSC25485 CNPY2 Text_Mining(affects(expression)) CTD NSC25485 CYC1 Text_Mining(affects(localization)) CTD NSC25485 CYC1 Text_Mining(decreases(expression)) CTD NSC25485 DDOST Text_Mining(decreases(expression)) CTD NSC25485 DRD1 Text_Mining(decreases(expression)) CTD NSC25485 DRD1 Text_Mining(increases(phosphorylation)) CTD NSC25485 DSG1 Text_Mining(affects(expression)) CTD NSC25485 DUT Text_Mining(affects(expression)) CTD NSC25485 ECE1 Text_Mining(increases(expression)) CTD NSC25485 ECHS1 Text_Mining(affects(expression)) CTD NSC25485 EIF3K Text_Mining(affects(expression)) CTD NSC25485 ERCC4 Text_Mining(decreases(expression)) CTD NSC25485 FANCD2 Text_Mining(affects(ubiquitination)) CTD NSC25485 FANCD2 Text_Mining(decreases(reaction)) CTD NSC25485 FANCD2 Text_Mining(increases(expression)) CTD NSC25485 FANCD2 Text_Mining(decreases(expression)) CTD NSC25485 FANCF Text_Mining(decreases(expression)) CTD NSC25485 FANCI Text_Mining(affects(ubiquitination)) CTD NSC25485 FANCI Text_Mining(decreases(reaction)) CTD NSC25485 FANCI Text_Mining(increases(expression)) CTD NSC25485 FANCI Text_Mining(decreases(expression)) CTD NSC25485 FARS2 Text_Mining(increases(expression)) CTD NSC25485 FH Text_Mining(affects(expression)) CTD NSC25485 FKBP7 Text_Mining(increases(expression)) CTD NSC25485 GC Text_Mining(affects(expression)) CTD NSC25485 GLRB Text_Mining(increases(expression)) CTD NSC25485 GTPBP6 Text_Mining(increases(expression)) CTD NSC25485 HIF1A Text_Mining(affects(localization)) CTD NSC25485 HIF1A Text_Mining(decreases(reaction)) CTD NSC25485 HIF1A Text_Mining(increases(phosphorylation)) CTD NSC25485 HIF1A Text_Mining(increases(activity)) CTD NSC25485 HIF1A Text_Mining(increases(expression)) CTD NSC25485 HNRNPA2B1 Text_Mining(affects(expression)) CTD NSC25485 HNRNPDL Text_Mining(decreases(expression)) CTD NSC25485 HPCAL1 Text_Mining(affects(expression)) CTD NSC25485 HRG Text_Mining(affects(expression)) CTD NSC25485 HSPD1 Text_Mining(affects(expression)) CTD NSC25485 HSPD1 Text_Mining(affects(binding)) CTD NSC25485 HSPD1 Text_Mining(decreases(reaction)) CTD NSC25485 HSPD1 Text_Mining(affects(localization)) CTD NSC25485 HSPD1 Text_Mining(decreases(expression)) CTD NSC25485 IL2RA Text_Mining(decreases(expression)) CTD NSC25485 IL2RB Text_Mining(decreases(expression)) CTD NSC25485 KCND2 Text_Mining(increases(expression)) CTD NSC25485 KCNH2 Text_Mining(decreases(reaction)) CTD NSC25485 KCNH2 Text_Mining(increases(transport)) CTD NSC25485 KCNH2 Text_Mining(decreases(activity)) CTD NSC25485 KCNH2 Text_Mining(decreases(expression)) CTD NSC25485 LGALS1 Text_Mining(affects(expression)) CTD NSC25485 LGALS1 Text_Mining(increases(expression)) CTD NSC25485 LSS Text_Mining(increases(abundance)) CTD NSC25485 MAPK7 Text_Mining(decreases(reaction)) CTD NSC25485 MAPK7 Text_Mining(increases(activity)) CTD NSC25485 MAPK7 Text_Mining(increases(phosphorylation)) CTD NSC25485 MDH2 Text_Mining(affects(expression)) CTD NSC25485 MYC Text_Mining(decreases(expression)) CTD NSC25485 MYC Text_Mining(increases(expression)) CTD NSC25485 MYL12A Text_Mining(increases(expression)) CTD NSC25485 NPC2 Text_Mining(decreases(expression)) CTD NSC25485 PARP1 Text_Mining(increases(cleavage)) CTD NSC25485 PARP1 Text_Mining(increases(reaction)) CTD NSC25485 PCNA Text_Mining(decreases(expression)) CTD NSC25485 PDCD6 Text_Mining(increases(expression)) CTD NSC25485 PFDN5 Text_Mining(affects(expression)) CTD NSC25485 PFN1 Text_Mining(affects(expression)) CTD NSC25485 PFN1 Text_Mining(decreases(expression)) CTD NSC25485 PPT2 Text_Mining(decreases(expression)) CTD NSC25485 PSMB6 Text_Mining(affects(expression)) CTD NSC25485 PTPN2 Text_Mining(decreases(expression)) CTD NSC25485 RAB11B Text_Mining(increases(expression)) CTD NSC25485 ROCK1 Text_Mining(decreases(reaction)) CTD NSC25485 ROCK1 Text_Mining(increases(cleavage)) CTD NSC25485 ROCK2 Text_Mining(decreases(reaction)) CTD NSC25485 ROCK2 Text_Mining(increases(cleavage)) CTD NSC25485 RPA3 Text_Mining(affects(expression)) CTD NSC25485 RPGRIP1L Text_Mining(decreases(expression)) CTD NSC25485 S100A13 Text_Mining(affects(expression)) CTD NSC25485 SGK1 Text_Mining(decreases(reaction)) CTD NSC25485 SGK1 Text_Mining(increases(transport)) CTD NSC25485 SGK2 Text_Mining(decreases(reaction)) CTD NSC25485 SGK2 Text_Mining(increases(transport)) CTD NSC25485 SGK3 Text_Mining(decreases(reaction)) CTD NSC25485 SGK3 Text_Mining(increases(transport)) CTD NSC25485 SLC5A5 Text_Mining(decreases(reaction)) CTD NSC25485 SLC5A5 Text_Mining(increases(uptake)) CTD NSC25485 SLC5A6 Text_Mining(decreases(reaction)) CTD NSC25485 SLC5A6 Text_Mining(increases(transport)) CTD NSC25485 TPI1 Text_Mining(affects(expression)) CTD NSC25485 TPT1 Text_Mining(affects(expression)) CTD NSC25485 TXN Text_Mining(affects(expression)) CTD NSC25485 ZFHX3 Text_Mining(decreases(expression)) CTD NSC25485 APP None=None(uM) D4 PubChem NSC25485 AR Ratio Potency (uM)=0.022421(uM) D4 PubChem NSC25485 AR Ratio Potency (uM)=0.0393847(uM) D4 PubChem NSC25485 AR Potency-Replicate_1=0.0465(uM) D4 PubChem NSC25485 AR Potency-Replicate_1=0.19(uM) D4 PubChem NSC25485 AR Potency-Replicate_1=0.2131(uM) D4 PubChem NSC25485 AR AR Potency (uM)=0.779114(uM) D4 PubChem NSC25485 AR Potency-Replicate_1=0.8413(uM) D4 PubChem NSC25485 AR AR Potency (uM)=1.01922(uM) D4 PubChem NSC25485 ATAD5 Potency=0.092(uM) D4 PubChem NSC25485 ATAD5 Potency=0.1636(uM) D4 PubChem NSC25485 ATAD5 Potency=92.0(nM) D4 ChEMBL NSC25485 ATAD5 Potency=163.6(nM) D4 ChEMBL NSC25485 CFTR AC50_uM=3.38(uM) D4 PubChem NSC25485 CFTR None=None(uM) D4 PubChem NSC25485 CYP19A1 None=None(uM) D4 PubChem NSC25485 EPAS1 None=None(uM) D4 PubChem NSC25485 ESR1 Potency-Replicate_1=0.1634(uM) D4 PubChem NSC25485 ESR1 ER Potency (uM)=0.249293(uM) D4 PubChem NSC25485 ESR1 ER Potency (uM)=0.455268(uM) D4 PubChem NSC25485 ESR1 Potency-Replicate_1=0.5308(uM) D4 PubChem NSC25485 GALR3 None=None(uM) D4 PubChem NSC25485 GMNN Potency=6.5131(uM) D4 PubChem NSC25485 GMNN Potency=0.2593(uM) D4 PubChem NSC25485 HTR5A None=None(uM) D4 PubChem NSC25485 IDH1 Potency=0.13(uM) D4 PubChem NSC25485 IL1B None=None(uM) D4 PubChem NSC25485 KLF5 IC50=0.02973(uM) D4 PubChem NSC25485 KLF5 IC50=0.05532(uM) D4 PubChem NSC25485 KLF5 IC50=0.16455(uM) D4 PubChem NSC25485 KLF5 None=None(uM) D4 PubChem NSC25485 KLF5 IC50=164.55(nM) D4 ChEMBL NSC25485 MC4R None=None(uM) D4 PubChem NSC25485 MDM2 None=None(uM) D4 PubChem NSC25485 MDM4 None=None(uM) D4 PubChem NSC25485 MITF None=None(uM) D4 PubChem NSC25485 NCOA1 None=None(uM) D4 PubChem NSC25485 NCOA2 None=None(uM) D4 PubChem NSC25485 NCOA3 None=None(uM) D4 PubChem NSC25485 NFE2L2 Potency=0.0326(uM) D4 PubChem NSC25485 NFE2L2 Potency=0.058(uM) D4 PubChem NSC25485 NOD1 EC50=None(uM) D4 PubChem NSC25485 NOD2 EC50=None(uM) D4 PubChem NSC25485 NPY1R None=None(uM) D4 PubChem NSC25485 NPY2R None=None(uM) D4 PubChem NSC25485 NR2F2 None=None(uM) D4 PubChem NSC25485 NR3C1 Potency-Replicate_1=0.2683(uM) D4 PubChem NSC25485 NR5A1 None=None(uM) D4 PubChem NSC25485 NR5A2 None=None(uM) D4 PubChem NSC25485 OPRD1 None=None(uM) D4 PubChem NSC25485 OPRM1 None=None(uM) D4 PubChem NSC25485 PLA2G3 None=None(uM) D4 PubChem NSC25485 PTBP1 None=None(uM) D4 PubChem NSC25485 S1PR4 None=None(uM) D4 PubChem NSC25485 SLC6A3 None=None(uM) D4 PubChem NSC25485 SMAD3 Potency=0.206(uM) D4 PubChem NSC25485 SMAD3 Potency=1.122(uM) D4 PubChem NSC25485 SMAD3 Potency=3.6626(uM) D4 PubChem NSC25485 STAT3 IC50=1.154(uM) D4 PubChem NSC25485 STAT3 None=None(uM) D4 PubChem NSC25485 STAT3 IC50=1154.0(nM) D4 ChEMBL NSC25485 STK33 None=None(uM) D4 PubChem NSC25485 TDP1 Potency=2.0596(uM) D4 PubChem NSC25485 TDP1 Potency=2.3109(uM) D4 PubChem NSC25485 TDP1 Potency=0.2371(uM) D4 PubChem NSC25485 TDP1 Potency=0.2661(uM) D4 PubChem NSC25485 TDP1 Potency=0.9441(uM) D4 PubChem NSC25485 TDP1 Potency=1.6789(uM) D4 PubChem NSC25485 TNF None=None(uM) D4 PubChem NSC25485 TNFRSF10B None=None(uM) D4 PubChem NSC25485 TNFSF10 None=None(uM) D4 PubChem