Drug Gene Type Source metyrapone ABCC3 Text_Mining(increases(activity)) CTD metyrapone ABCC3 Text_Mining(increases(expression)) CTD metyrapone ATF6 Text_Mining(increases(expression)) CTD metyrapone ATF6 Text_Mining(increases(reaction)) CTD metyrapone CASP4 Text_Mining(affects(cotreatment)) CTD metyrapone CASP4 Text_Mining(affects(localization)) CTD metyrapone CYP3A4 Text_Mining(increases(activity)) CTD metyrapone CYP3A4 Text_Mining(increases(expression)) CTD metyrapone DDIT3 Text_Mining(affects(cotreatment)) CTD metyrapone DDIT3 Text_Mining(increases(expression)) CTD metyrapone DDIT3 Text_Mining(increases(reaction)) CTD metyrapone DHRS7 Text_Mining(increases(reduction)) CTD metyrapone HSD11B1 Text_Mining(decreases(activity)) CTD metyrapone HSD11B2 Text_Mining(decreases(activity)) CTD metyrapone HSPA5 Text_Mining(increases(expression)) CTD metyrapone HSPA5 Text_Mining(increases(reaction)) CTD metyrapone MAP1LC3B Text_Mining(affects(cotreatment)) CTD metyrapone MAP1LC3B Text_Mining(increases(expression)) CTD metyrapone NR1I2 Text_Mining(increases(activity)) CTD metyrapone NR1I2 Text_Mining(increases(expression)) CTD metyrapone NR1I3 Text_Mining(increases(activity)) CTD metyrapone POMC Text_Mining(increases(expression)) CTD metyrapone CYP1A2 None=None(uM) D4 PubChem metyrapone CYP3A4 Potency=1.2589(uM) D4 PubChem metyrapone CYP3A4 None=None(uM) D4 PubChem metyrapone CYP3A4 Potency=1258.9(nM) D4 ChEMBL metyrapone CYP3A4 AC50=1258.93(nM) D4 ChEMBL