Drug Gene Type Source methapyrilene PDCD4 Text_Mining(decreases(expression)) CTD methapyrilene TNFAIP3 Text_Mining(increases(expression)) CTD methapyrilene TPD52 Text_Mining(decreases(expression)) CTD methapyrilene TPD52 Text_Mining(increases(expression)) CTD methapyrilene CYP1A2 None=None(uM) D4 PubChem methapyrilene CYP2D6 Potency=0.5012(uM) D4 PubChem methapyrilene CYP2D6 Potency=1.5849(uM) D4 PubChem methapyrilene CYP2D6 None=None(uM) D4 PubChem methapyrilene CYP2D6 AC50=1584.89(nM) D4 ChEMBL methapyrilene CYP2D6 AC50=501.19(nM) D4 ChEMBL methapyrilene CYP2D6 Potency=501.2(nM) D4 ChEMBL methapyrilene CYP2D6 Potency=1584.9(nM) D4 ChEMBL methapyrilene HTT None=None(uM) D4 PubChem