Drug Gene Type Source melphalan ABCC1 Text_Mining(affects(export)) CTD melphalan ABHD17C Text_Mining(decreases(expression)) CTD melphalan ABT1 Text_Mining(increases(expression)) CTD melphalan ACKR3 Text_Mining(increases(expression)) CTD melphalan ACVR1C Text_Mining(decreases(expression)) CTD melphalan AHRR Text_Mining(decreases(expression)) CTD melphalan ALAD Text_Mining(decreases(activity)) CTD melphalan AMMECR1L Text_Mining(increases(expression)) CTD melphalan ANKAR Text_Mining(decreases(expression)) CTD melphalan ANKRD10 Text_Mining(increases(expression)) CTD melphalan ANKRD28 Text_Mining(decreases(expression)) CTD melphalan ANKRD34A Text_Mining(decreases(expression)) CTD melphalan AR Text_Mining(decreases(expression)) CTD melphalan ARHGAP12 Text_Mining(decreases(expression)) CTD melphalan ARHGAP18 Text_Mining(decreases(expression)) CTD melphalan ARHGAP20 Text_Mining(decreases(expression)) CTD melphalan ARHGAP24 Text_Mining(decreases(expression)) CTD melphalan ARID5A Text_Mining(increases(expression)) CTD melphalan ATG16L1 Text_Mining(increases(expression)) CTD melphalan ATP1A1-AS1 Text_Mining(decreases(expression)) CTD melphalan ATP2B1 Text_Mining(decreases(expression)) CTD melphalan B3GNT2 Text_Mining(increases(expression)) CTD melphalan B3GNT5 Text_Mining(increases(expression)) CTD melphalan BAK1 Text_Mining(increases(expression)) CTD melphalan BAX Text_Mining(decreases(localization)) CTD melphalan BAX Text_Mining(increases(expression)) CTD melphalan BCHE Text_Mining(affects(cotreatment)) CTD melphalan BCHE Text_Mining(decreases(expression)) CTD melphalan BCL2 Text_Mining(decreases(expression)) CTD melphalan BCL2A1 Text_Mining(increases(expression)) CTD melphalan BICC1 Text_Mining(decreases(expression)) CTD melphalan BIRC5 Text_Mining(affects(response to substance)) CTD melphalan BIRC5 Text_Mining(affects(reaction)) CTD melphalan BNC2 Text_Mining(decreases(expression)) CTD melphalan BTG2 Text_Mining(increases(expression)) CTD melphalan C10ORF2 Text_Mining(increases(expression)) CTD melphalan C6ORF165 Text_Mining(decreases(expression)) CTD melphalan CABLES1 Text_Mining(decreases(expression)) CTD melphalan CASP3 Text_Mining(increases(activity)) CTD melphalan CASP9 Text_Mining(increases(activity)) CTD melphalan CASP9 Text_Mining(increases(cleavage)) CTD melphalan CAT Text_Mining(decreases(activity)) CTD melphalan CC2D2A Text_Mining(decreases(expression)) CTD melphalan CCDC110 Text_Mining(decreases(expression)) CTD melphalan CCDC171 Text_Mining(decreases(expression)) CTD melphalan CCDC64B Text_Mining(increases(expression)) CTD melphalan CCL20 Text_Mining(increases(expression)) CTD melphalan CCNJ Text_Mining(increases(expression)) CTD melphalan CD34 Text_Mining(affects(cotreatment)) CTD melphalan CD34 Text_Mining(decreases(expression)) CTD melphalan CDA Text_Mining(decreases(response to substance)) CTD melphalan CDC14B Text_Mining(decreases(expression)) CTD melphalan CDC42EP3 Text_Mining(decreases(expression)) CTD melphalan CHUK Text_Mining(affects(phosphorylation)) CTD melphalan CIITA Text_Mining(decreases(expression)) CTD melphalan CITED4 Text_Mining(increases(expression)) CTD melphalan CNKSR3 Text_Mining(decreases(expression)) CTD melphalan CPNE8 Text_Mining(decreases(expression)) CTD melphalan CREB5 Text_Mining(decreases(expression)) CTD melphalan CUL3 Text_Mining(increases(expression)) CTD melphalan CXCL12 Text_Mining(decreases(expression)) CTD melphalan CXORF57 Text_Mining(decreases(expression)) CTD melphalan CYP1A1 Text_Mining(decreases(reaction)) CTD melphalan CYP1A1 Text_Mining(increases(activity)) CTD melphalan CYP1A2 Text_Mining(decreases(reaction)) CTD melphalan CYP1A2 Text_Mining(increases(activity)) CTD melphalan CYP27B1 Text_Mining(increases(expression)) CTD melphalan DBF4 Text_Mining(increases(expression)) CTD melphalan DENND4C Text_Mining(decreases(expression)) CTD melphalan DIEXF Text_Mining(increases(expression)) CTD melphalan DLG3 Text_Mining(decreases(expression)) CTD melphalan DOCK9-AS2 Text_Mining(increases(expression)) CTD melphalan DST Text_Mining(decreases(expression)) CTD melphalan DUSP2 Text_Mining(increases(expression)) CTD melphalan EAF1 Text_Mining(increases(expression)) CTD melphalan EBF1 Text_Mining(decreases(expression)) CTD melphalan EDN1 Text_Mining(increases(expression)) CTD melphalan EEPD1 Text_Mining(decreases(expression)) CTD melphalan EFNA2 Text_Mining(increases(expression)) CTD melphalan EFNA5 Text_Mining(decreases(expression)) CTD melphalan EMX2 Text_Mining(decreases(expression)) CTD melphalan ENOX1 Text_Mining(decreases(expression)) CTD melphalan EPHA5 Text_Mining(decreases(expression)) CTD melphalan EXOC6 Text_Mining(decreases(expression)) CTD melphalan FABP5 Text_Mining(increases(expression)) CTD melphalan FAM110B Text_Mining(decreases(expression)) CTD melphalan FAM175A Text_Mining(decreases(expression)) CTD melphalan FAM49A Text_Mining(decreases(expression)) CTD melphalan FAM65B Text_Mining(decreases(expression)) CTD melphalan FAM90A1 Text_Mining(decreases(expression)) CTD melphalan FANCC Text_Mining(increases(response to substance)) CTD melphalan FANCG Text_Mining(increases(response to substance)) CTD melphalan FAT4 Text_Mining(decreases(expression)) CTD melphalan FGD4 Text_Mining(decreases(expression)) CTD melphalan FGD6 Text_Mining(decreases(expression)) CTD melphalan FGF5 Text_Mining(decreases(expression)) CTD melphalan FIGN Text_Mining(decreases(expression)) CTD melphalan FMN2 Text_Mining(decreases(expression)) CTD melphalan FOSB Text_Mining(increases(expression)) CTD melphalan FOXP2 Text_Mining(decreases(expression)) CTD melphalan FRMD4A Text_Mining(decreases(expression)) CTD melphalan FRMD4B Text_Mining(decreases(expression)) CTD melphalan FRY Text_Mining(decreases(expression)) CTD melphalan FUT10 Text_Mining(decreases(expression)) CTD melphalan GAB1 Text_Mining(decreases(expression)) CTD melphalan GAREM Text_Mining(decreases(expression)) CTD melphalan GAS1 Text_Mining(decreases(expression)) CTD melphalan GCNT1 Text_Mining(decreases(expression)) CTD melphalan GLI3 Text_Mining(decreases(expression)) CTD melphalan GRIN2C Text_Mining(increases(expression)) CTD melphalan GRK5 Text_Mining(decreases(expression)) CTD melphalan GSTM1 Text_Mining(decreases(response to substance)) CTD melphalan GSTP1 Text_Mining(affects(cotreatment)) CTD melphalan GSTP1 Text_Mining(increases(response to substance)) CTD melphalan GSTP1 Text_Mining(decreases(reaction)) CTD melphalan GSTP1 Text_Mining(increases(metabolic processing)) CTD melphalan CYCSP39 Text_Mining(increases(expression)) CTD melphalan HECW2 Text_Mining(decreases(expression)) CTD melphalan HGF Text_Mining(decreases(expression)) CTD melphalan HMGA2 Text_Mining(decreases(expression)) CTD melphalan HOXD1 Text_Mining(increases(expression)) CTD melphalan ICAM1 Text_Mining(increases(expression)) CTD melphalan IER3 Text_Mining(increases(expression)) CTD melphalan IKBKE Text_Mining(decreases(expression)) CTD melphalan IKZF2 Text_Mining(decreases(expression)) CTD melphalan IL12A Text_Mining(increases(expression)) CTD melphalan IL16 Text_Mining(decreases(expression)) CTD melphalan IL1B Text_Mining(increases(expression)) CTD melphalan IL7 Text_Mining(decreases(expression)) CTD melphalan IRF2 Text_Mining(decreases(expression)) CTD melphalan JADE2 Text_Mining(decreases(expression)) CTD melphalan JAK2 Text_Mining(decreases(expression)) CTD melphalan JAKMIP3 Text_Mining(decreases(expression)) CTD melphalan KALRN Text_Mining(decreases(expression)) CTD melphalan KBTBD3 Text_Mining(decreases(expression)) CTD melphalan KIAA0922 Text_Mining(decreases(expression)) CTD melphalan KIAA1107 Text_Mining(decreases(expression)) CTD melphalan KITLG Text_Mining(decreases(expression)) CTD melphalan KLF12 Text_Mining(decreases(expression)) CTD melphalan KLHL42 Text_Mining(increases(expression)) CTD melphalan LINC00312 Text_Mining(increases(expression)) CTD melphalan LRIG3 Text_Mining(decreases(expression)) CTD melphalan LURAP1 Text_Mining(decreases(expression)) CTD melphalan LYST Text_Mining(decreases(expression)) CTD melphalan MAPK1 Text_Mining(increases(activity)) CTD melphalan MAPK1 Text_Mining(increases(phosphorylation)) CTD melphalan MAPK3 Text_Mining(increases(activity)) CTD melphalan MAPK3 Text_Mining(increases(phosphorylation)) CTD melphalan MBOAT1 Text_Mining(decreases(expression)) CTD melphalan MEOX2 Text_Mining(decreases(expression)) CTD melphalan MESDC1 Text_Mining(increases(expression)) CTD melphalan MEX3A Text_Mining(increases(expression)) CTD melphalan MEX3B Text_Mining(increases(expression)) CTD melphalan MFSD2A Text_Mining(increases(expression)) CTD melphalan MGST2 Text_Mining(decreases(response to substance)) CTD melphalan MIR17HG Text_Mining(increases(expression)) CTD melphalan MITF Text_Mining(decreases(expression)) CTD melphalan MKL2 Text_Mining(decreases(expression)) CTD melphalan MLLT3 Text_Mining(decreases(expression)) CTD melphalan MMS22L Text_Mining(decreases(expression)) CTD melphalan MTA3 Text_Mining(decreases(expression)) CTD melphalan MTCL1 Text_Mining(decreases(expression)) CTD melphalan MYO1B Text_Mining(decreases(expression)) CTD melphalan NEAT1 Text_Mining(decreases(expression)) CTD melphalan NEBL Text_Mining(increases(expression)) CTD melphalan NFIA Text_Mining(decreases(expression)) CTD melphalan NHS Text_Mining(decreases(expression)) CTD melphalan NKRF Text_Mining(increases(expression)) CTD melphalan NOP56 Text_Mining(increases(expression)) CTD melphalan NPPB Text_Mining(increases(expression)) CTD melphalan NR4A3 Text_Mining(increases(expression)) CTD melphalan NRG2 Text_Mining(decreases(expression)) CTD melphalan NRP1 Text_Mining(decreases(expression)) CTD melphalan NUAK1 Text_Mining(decreases(expression)) CTD melphalan OSBPL10 Text_Mining(decreases(expression)) CTD melphalan PAG1 Text_Mining(decreases(expression)) CTD melphalan PDLIM5 Text_Mining(decreases(expression)) CTD melphalan PHF21A Text_Mining(decreases(expression)) CTD melphalan PHF3 Text_Mining(decreases(expression)) CTD melphalan PHLDA1 Text_Mining(increases(expression)) CTD melphalan PHLDB2 Text_Mining(decreases(expression)) CTD melphalan PIK3R1 Text_Mining(decreases(expression)) CTD melphalan PIK3R3 Text_Mining(decreases(expression)) CTD melphalan PLCL2 Text_Mining(decreases(expression)) CTD melphalan PLEKHA2 Text_Mining(decreases(expression)) CTD melphalan PLEKHA5 Text_Mining(decreases(expression)) CTD melphalan PLK3 Text_Mining(increases(expression)) CTD melphalan PPIF Text_Mining(increases(expression)) CTD melphalan PPM1H Text_Mining(decreases(expression)) CTD melphalan PPP2R2B Text_Mining(decreases(expression)) CTD melphalan PPP2R5A Text_Mining(decreases(expression)) CTD melphalan PRUNE2 Text_Mining(decreases(expression)) CTD melphalan PSD3 Text_Mining(decreases(expression)) CTD melphalan PTGS2 Text_Mining(increases(expression)) CTD melphalan PTPRG Text_Mining(decreases(expression)) CTD melphalan PXK Text_Mining(decreases(expression)) CTD melphalan RAD54B Text_Mining(decreases(expression)) CTD melphalan RARB Text_Mining(decreases(expression)) CTD melphalan RASD1 Text_Mining(increases(expression)) CTD melphalan RASL10A Text_Mining(increases(expression)) CTD melphalan RASL11B Text_Mining(increases(expression)) CTD melphalan RBM24 Text_Mining(increases(expression)) CTD melphalan REV3L Text_Mining(decreases(expression)) CTD melphalan RGL1 Text_Mining(decreases(expression)) CTD melphalan RGMB Text_Mining(decreases(expression)) CTD melphalan RGS16 Text_Mining(increases(expression)) CTD melphalan RGS2 Text_Mining(increases(expression)) CTD melphalan RNF128 Text_Mining(decreases(expression)) CTD melphalan RNF144B Text_Mining(decreases(expression)) CTD melphalan ROR1 Text_Mining(decreases(expression)) CTD melphalan RPL27A Text_Mining(increases(expression)) CTD melphalan RRAD Text_Mining(increases(expression)) CTD melphalan RSPO2 Text_Mining(decreases(expression)) CTD melphalan RUNX1T1 Text_Mining(decreases(expression)) CTD melphalan SCN8A Text_Mining(decreases(expression)) CTD melphalan SEMA6D Text_Mining(decreases(expression)) CTD melphalan SERPINB2 Text_Mining(increases(expression)) CTD melphalan SGK1 Text_Mining(increases(expression)) CTD melphalan SGMS1 Text_Mining(decreases(expression)) CTD melphalan SHANK2 Text_Mining(decreases(expression)) CTD melphalan SHROOM3 Text_Mining(decreases(expression)) CTD melphalan SIK1 Text_Mining(increases(expression)) CTD melphalan SLC14A1 Text_Mining(decreases(expression)) CTD melphalan SLC19A2 Text_Mining(increases(expression)) CTD melphalan SMAD2 Text_Mining(decreases(reaction)) CTD melphalan SMAD2 Text_Mining(increases(phosphorylation)) CTD melphalan SMAD3 Text_Mining(decreases(expression)) CTD melphalan SNHG15 Text_Mining(increases(expression)) CTD melphalan SNORA70 Text_Mining(increases(expression)) CTD melphalan SNORD14E Text_Mining(increases(expression)) CTD melphalan SNORD22 Text_Mining(increases(expression)) CTD melphalan SNTB1 Text_Mining(decreases(expression)) CTD melphalan SNX29 Text_Mining(decreases(expression)) CTD melphalan SOCS5 Text_Mining(decreases(expression)) CTD melphalan SPATA17 Text_Mining(decreases(expression)) CTD melphalan SPATA7 Text_Mining(decreases(expression)) CTD melphalan SPRED1 Text_Mining(decreases(expression)) CTD melphalan SPTY2D1 Text_Mining(increases(expression)) CTD melphalan SRGAP2 Text_Mining(decreases(expression)) CTD melphalan STAC Text_Mining(decreases(expression)) CTD melphalan STAMBPL1 Text_Mining(decreases(expression)) CTD melphalan TACC2 Text_Mining(decreases(expression)) CTD melphalan TBC1D12 Text_Mining(decreases(expression)) CTD melphalan TBL1XR1 Text_Mining(decreases(expression)) CTD melphalan TET1 Text_Mining(decreases(expression)) CTD melphalan TEX30 Text_Mining(increases(expression)) CTD melphalan TFPI2 Text_Mining(increases(expression)) CTD melphalan THSD4 Text_Mining(decreases(expression)) CTD melphalan TIGD2 Text_Mining(decreases(expression)) CTD melphalan TLR4 Text_Mining(decreases(expression)) CTD melphalan TMEM133 Text_Mining(decreases(expression)) CTD melphalan TMEM200A Text_Mining(decreases(expression)) CTD melphalan TMEM26 Text_Mining(decreases(expression)) CTD melphalan TMEM88 Text_Mining(increases(expression)) CTD melphalan TNF Text_Mining(increases(expression)) CTD melphalan TNFRSF19 Text_Mining(decreases(expression)) CTD melphalan TNNI3 Text_Mining(increases(expression)) CTD melphalan TNRC6B Text_Mining(decreases(expression)) CTD melphalan TOX Text_Mining(decreases(expression)) CTD melphalan TP63 Text_Mining(decreases(expression)) CTD melphalan TRERF1 Text_Mining(decreases(expression)) CTD melphalan TRIB1 Text_Mining(increases(expression)) CTD melphalan TRMT10C Text_Mining(increases(expression)) CTD melphalan TTC30B Text_Mining(decreases(expression)) CTD melphalan TUFT1 Text_Mining(increases(expression)) CTD melphalan UBAP1L Text_Mining(increases(expression)) CTD melphalan USP36 Text_Mining(increases(expression)) CTD melphalan USP53 Text_Mining(decreases(expression)) CTD melphalan VDAC1 Text_Mining(increases(expression)) CTD melphalan VDAC1 Text_Mining(increases(response to substance)) CTD melphalan YOD1 Text_Mining(increases(expression)) CTD melphalan YPEL2 Text_Mining(decreases(expression)) CTD melphalan YRDC Text_Mining(increases(expression)) CTD melphalan ZBTB20 Text_Mining(decreases(expression)) CTD melphalan ZC3H12A Text_Mining(increases(expression)) CTD melphalan ZFHX4 Text_Mining(decreases(expression)) CTD melphalan ZNF214 Text_Mining(decreases(expression)) CTD melphalan ZNF277 Text_Mining(decreases(expression)) CTD melphalan ZNF438 Text_Mining(decreases(expression)) CTD melphalan ZNF521 Text_Mining(decreases(expression)) CTD melphalan ZNF618 Text_Mining(decreases(expression)) CTD melphalan ZSWIM5 Text_Mining(decreases(expression)) CTD melphalan ABCB1 None=None(uM) D4 PubChem melphalan AR AR Potency (uM)=26.6032(uM) D4 PubChem melphalan AR Ratio Potency (uM)=26.8325(uM) D4 PubChem melphalan AR Potency-Replicate_1=29.8493(uM) D4 PubChem melphalan AR Potency-Replicate_1=30.1065(uM) D4 PubChem melphalan CYP3A4 Potency=3.1623(uM) D4 PubChem melphalan CYP3A4 Potency=3162.3(nM) D4 ChEMBL melphalan EHMT2 Potency=7.9433(uM) D4 PubChem melphalan EHMT2 Potency=7943.3(nM) D4 ChEMBL melphalan ESR1 ER Potency (uM)=17.4947(uM) D4 PubChem melphalan ESR1 Potency-Replicate_1=23.3296(uM) D4 PubChem melphalan MDM2 None=None(uM) D4 PubChem melphalan MDM4 None=None(uM) D4 PubChem melphalan NFE2L2 Potency=42.1632(uM) D4 PubChem melphalan NFE2L2 Potency=54.4827(uM) D4 PubChem melphalan NR1H4 Potency=39.8107(uM) D4 PubChem melphalan NR1I2 Potency-Replicate_1=44.6684(uM) D4 PubChem melphalan STK33 None=None(uM) D4 PubChem melphalan TDP1 Potency=0.2311(uM) D4 PubChem melphalan TDP1 Potency=0.2593(uM) D4 PubChem melphalan TDP1 Potency=0.5309(uM) D4 PubChem