Drug Gene Type Source Melatonin ACAN Text_Mining(increases(expression)) CTD Melatonin ADIPOQ Text_Mining(decreases(expression)) CTD Melatonin AKT1 Text_Mining(increases(phosphorylation)) CTD Melatonin ALPL Text_Mining(increases(expression)) CTD Melatonin APP Text_Mining(affects(binding)) CTD Melatonin APP Text_Mining(affects(reaction)) CTD Melatonin APP Text_Mining(decreases(reaction)) CTD Melatonin APP Text_Mining(increases(secretion)) CTD Melatonin ATF2 Text_Mining(decreases(reaction)) CTD Melatonin ATF2 Text_Mining(increases(expression)) CTD Melatonin BAD Text_Mining(affects(binding)) CTD Melatonin BAD Text_Mining(increases(reaction)) CTD Melatonin BAD Text_Mining(increases(phosphorylation)) CTD Melatonin BAK1 Text_Mining(affects(cotreatment)) CTD Melatonin BAK1 Text_Mining(increases(expression)) CTD Melatonin BAX Text_Mining(affects(cotreatment)) CTD Melatonin BAX Text_Mining(increases(expression)) CTD Melatonin BAX Text_Mining(affects(binding)) CTD Melatonin BAX Text_Mining(decreases(reaction)) CTD Melatonin BAX Text_Mining(increases(reaction)) CTD Melatonin BAX Text_Mining(decreases(expression)) CTD Melatonin BAX Text_Mining(increases(activity)) CTD Melatonin BCL2 Text_Mining(affects(cotreatment)) CTD Melatonin BCL2 Text_Mining(decreases(expression)) CTD Melatonin BCL2 Text_Mining(affects(localization)) CTD Melatonin BCL2 Text_Mining(increases(reaction)) CTD Melatonin BCL2 Text_Mining(increases(expression)) CTD Melatonin BCL2L1 Text_Mining(decreases(expression)) CTD Melatonin BCL2L1 Text_Mining(increases(reaction)) CTD Melatonin BGLAP Text_Mining(increases(expression)) CTD Melatonin BID Text_Mining(affects(binding)) CTD Melatonin BID Text_Mining(increases(reaction)) CTD Melatonin BID Text_Mining(increases(expression)) CTD Melatonin CASP3 Text_Mining(affects(cotreatment)) CTD Melatonin CASP3 Text_Mining(increases(expression)) CTD Melatonin CASP3 Text_Mining(decreases(reaction)) CTD Melatonin CASP3 Text_Mining(increases(activity)) CTD Melatonin CASP3 Text_Mining(increases(reaction)) CTD Melatonin CASP8 Text_Mining(increases(activity)) CTD Melatonin CASP8 Text_Mining(increases(reaction)) CTD Melatonin CASP9 Text_Mining(decreases(reaction)) CTD Melatonin CASP9 Text_Mining(increases(activity)) CTD Melatonin CASP9 Text_Mining(increases(reaction)) CTD Melatonin CAT Text_Mining(affects(cotreatment)) CTD Melatonin CAT Text_Mining(increases(activity)) CTD Melatonin CAT Text_Mining(decreases(activity)) CTD Melatonin CAT Text_Mining(decreases(reaction)) CTD Melatonin CCNB1 Text_Mining(decreases(expression)) CTD Melatonin CCND1 Text_Mining(decreases(expression)) CTD Melatonin CDK1 Text_Mining(decreases(expression)) CTD Melatonin CDK4 Text_Mining(decreases(expression)) CTD Melatonin CDKN1A Text_Mining(increases(expression)) CTD Melatonin CTSB Text_Mining(affects(cotreatment)) CTD Melatonin CTSB Text_Mining(decreases(reaction)) CTD Melatonin CTSB Text_Mining(increases(expression)) CTD Melatonin CTSD Text_Mining(decreases(reaction)) CTD Melatonin CTSD Text_Mining(increases(expression)) CTD Melatonin CYP19A1 Text_Mining(decreases(expression)) CTD Melatonin CYP1A1 Text_Mining(increases(hydroxylation)) CTD Melatonin CYP1A1 Text_Mining(decreases(activity)) CTD Melatonin CYP1A2 Text_Mining(affects(metabolic processing)) CTD Melatonin CYP1A2 Text_Mining(decreases(methylation)) CTD Melatonin CYP1A2 Text_Mining(increases(hydroxylation)) CTD Melatonin CYP1A2 Text_Mining(increases(metabolic processing)) CTD Melatonin CYP1A2 Text_Mining(decreases(reaction)) CTD Melatonin CYP1A2 Text_Mining(increases(hydrolysis)) CTD Melatonin CYP1A2 Text_Mining(decreases(activity)) CTD Melatonin CYP1B1 Text_Mining(decreases(reaction)) CTD Melatonin CYP1B1 Text_Mining(increases(hydroxylation)) CTD Melatonin CYP1B1 Text_Mining(decreases(activity)) CTD Melatonin CYP2C19 Text_Mining(decreases(methylation)) CTD Melatonin CYP2C19 Text_Mining(increases(hydroxylation)) CTD Melatonin EIF4EBP1 Text_Mining(increases(phosphorylation)) CTD Melatonin EIF4EBP1 Text_Mining(increases(reaction)) CTD Melatonin ESR1 Text_Mining(decreases(reaction)) CTD Melatonin ESR1 Text_Mining(increases(activity)) CTD Melatonin FABP4 Text_Mining(decreases(expression)) CTD Melatonin HMOX1 Text_Mining(decreases(reaction)) CTD Melatonin HMOX1 Text_Mining(increases(expression)) CTD Melatonin IL2 Text_Mining(increases(activity)) CTD Melatonin LEP Text_Mining(decreases(expression)) CTD Melatonin LPL Text_Mining(decreases(expression)) CTD Melatonin MAPK10 Text_Mining(increases(expression)) CTD Melatonin MAPK8 Text_Mining(increases(expression)) CTD Melatonin MAPK9 Text_Mining(increases(expression)) CTD Melatonin MAPT Text_Mining(decreases(reaction)) CTD Melatonin MAPT Text_Mining(increases(phosphorylation)) CTD Melatonin MCL1 Text_Mining(decreases(expression)) CTD Melatonin MCL1 Text_Mining(decreases(reaction)) CTD Melatonin MKI67 Text_Mining(decreases(expression)) CTD Melatonin MTNR1A Text_Mining(affects(binding)) CTD Melatonin MTNR1B Text_Mining(affects(binding)) CTD Melatonin MTOR Text_Mining(increases(phosphorylation)) CTD Melatonin MTOR Text_Mining(increases(reaction)) CTD Melatonin MTOR Text_Mining(increases(activity)) CTD Melatonin NES Text_Mining(decreases(expression)) CTD Melatonin NOS3 Text_Mining(decreases(expression)) CTD Melatonin NOS3 Text_Mining(decreases(reaction)) CTD Melatonin NOS3 Text_Mining(increases(reaction)) CTD Melatonin NQO2 Text_Mining(decreases(reaction)) CTD Melatonin NQO2 Text_Mining(increases(oxidation)) CTD Melatonin NQO2 Text_Mining(increases(reduction)) CTD Melatonin NR3C1 Text_Mining(decreases(reaction)) CTD Melatonin NR3C1 Text_Mining(increases(activity)) CTD Melatonin NR3C1 Text_Mining(decreases(expression)) CTD Melatonin NR3C1 Text_Mining(increases(reaction)) CTD Melatonin PCNA Text_Mining(decreases(expression)) CTD Melatonin PGR Text_Mining(decreases(reaction)) CTD Melatonin PGR Text_Mining(increases(expression)) CTD Melatonin POMC Text_Mining(decreases(reaction)) CTD Melatonin POMC Text_Mining(increases(abundance)) CTD Melatonin POMC Text_Mining(decreases(response to substance)) CTD Melatonin PPARG Text_Mining(decreases(expression)) CTD Melatonin PTGS2 Text_Mining(decreases(reaction)) CTD Melatonin PTGS2 Text_Mining(increases(expression)) CTD Melatonin RARA Text_Mining(affects(cotreatment)) CTD Melatonin RARA Text_Mining(increases(activity)) CTD Melatonin RARA Text_Mining(increases(reaction)) CTD Melatonin RUNX2 Text_Mining(increases(expression)) CTD Melatonin SIRT1 Text_Mining(decreases(expression)) CTD Melatonin SLC22A2 Text_Mining(decreases(reaction)) CTD Melatonin SLC22A2 Text_Mining(increases(uptake)) CTD Melatonin SOD2 Text_Mining(decreases(reaction)) CTD Melatonin SOD2 Text_Mining(increases(expression)) CTD Melatonin TGFB1 Text_Mining(affects(cotreatment)) CTD Melatonin TGFB1 Text_Mining(increases(expression)) CTD Melatonin TP53 Text_Mining(increases(expression)) CTD Melatonin YWHAB Text_Mining(affects(binding)) CTD Melatonin YWHAB Text_Mining(increases(reaction)) CTD Melatonin AHR AhR Potency (uM)=49.2994(uM) D4 PubChem Melatonin CYP1A2 None=None(uM) D4 PubChem Melatonin CYP1A2 AC50=5011.87(nM) D4 ChEMBL Melatonin CYP3A4 Potency=19.9526(uM) D4 PubChem Melatonin CYP3A4 Potency=19952.6(nM) D4 ChEMBL Melatonin ESR1 Potency-Replicate_1=55.3148(uM) D4 PubChem Melatonin HTR2B None=None(uM) D4 PubChem Melatonin MAP4K2 None=None(uM) D4 PubChem